1779Nc1nccn2c(nc(-c3cccc(OCc4ccccc4)c3)c12)C1CCC1 2579CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13 4078Oc1cc2c3c(oc(=O)c4cc(O)c(O)c(oc2=O)c34)c1O 4293Oc1ccc(\C=C(/C#N)C(=O)c2ccc(O)c(O)c2)cc1O 4814CCN(CC)CCNC(=O)c1c(C)[nH]c(\C=C2/C(=O)Nc3ccc(F)cc23)c1C 7460Oc1cc(O)c2c(c1)oc(-c1ccc(O)c(O)c1)c(O)c2=O 7657NS(=O)(=O)c1ccc(Nc2nccc(n2)-c2cnc3ccccn23)cc1 13534CN1CCN(CC1)c1cc(Nc2cc(C)n[nH]2)nc(Sc2ccc(NC(=O)C3CC3)cc2)n1 15015CCOC(=O)c1c(CC)c([nH]c1C=O)C(=O)OC(C)(C)C 22372C[C@@H](Cc1ccc(O)c(O)c1)[C@H](C)Cc1ccc(O)c(O)c1 24459COc1ccc2c(Oc3ccc(NC(=O)c4c(C)n(C)n(-c5ccccc5)c4=O)cc3F)ccnc2c1 24460CCCn1c(C)c(C(=O)Nc2ccc(Oc3ccnc4cc(OC)ccc34)c(F)c2)c(=O)n1-c1ccccc1 24461COc1ccc2c(Oc3ccc(NC(=O)c4c(C)n(CC(C)C)n(-c5ccccc5)c4=O)cc3F)ccnc2c1 24462COc1ccc2c(Oc3ccc(NC(=O)c4c(C)n(C[C@@H](C)O)n(-c5ccccc5)c4=O)cc3F)ccnc2c1 24463COc1ccc2c(Oc3ccc(NC(=O)c4c(C)n(C[C@H](C)O)n(-c5ccccc5)c4=O)cc3F)ccnc2c1 24465COc1ccc2c(Oc3ccc(NC(=O)c4c(C)n(CC(C)(C)O)n(-c5ccccc5)c4=O)cc3F)ccnc2c1 24466COc1ccc2c(Oc3ccc(NC(=O)c4c(C)n(CC(C)(C)O)n(-c5ccccc5)c4=O)nc3)ccnc2c1 27783COc1cc(ccc1Nc1nc(Nc2cccc(F)c2C(N)=O)c2cc[nH]c2n1)N1CCN(CC1)C(C)C 27799COc1cc2CCN(C(=O)CN(C)C)c2cc1Nc1nc(Nc2cccc(F)c2C(N)=O)c2cc[nH]c2n1 27817CNC(=O)c1c(F)cccc1Nc1nc(Nc2cc3N(CCc3cc2OC)C(=O)CN(C)C)nc2[nH]ccc12 27828COc1cc(ccc1Nc1nc(Nc2cc(F)ccc2C(N)=O)c2cc[nH]c2n1)N1CCN(CC1)C(C)C 27839COc1cc(ccc1Nc1nc(Nc2ccc(F)cc2C(N)=O)c2cc[nH]c2n1)N1CCN(CC1)C(C)C 27840COc1cc(ccc1Nc1nc(Nc2ccc(F)c(F)c2C(N)=O)c2cc[nH]c2n1)N1CCN(CC1)C(C)C 27841COc1cc(ccc1Nc1nc(Nc2cc(F)cc(F)c2C(N)=O)c2cc[nH]c2n1)N1CCN(CC1)C(C)C 27879Cc1cc(cc2[nH]c(nc12)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O)N1CCOCC1 27961Nc1ncnc2n(nc(-c3ccc4nc(Cc5ccccc5)[nH]c4c3)c12)[C@H]1CC[C@@H](CC1)N1CCOCC1 27962Nc1ncnc2n(nc(-c3ccc4nc(Cc5cccs5)[nH]c4c3)c12)[C@H]1CC[C@@H](CC1)N1CCOCC1 27963Nc1ncnc2n(nc(-c3ccc4nc(Cc5ccccc5Cl)[nH]c4c3)c12)[C@H]1CC[C@@H](CC1)N1CCOCC1 27964COc1ccccc1Cc1nc2ccc(cc2[nH]1)-c1nn([C@H]2CC[C@@H](CC2)N2CCOCC2)c2ncnc(N)c12 28104CCN1CCN(CCCOc2cc3ncc(C#N)c(Nc4ccc(Sc5nc(C)c(C)n5CC)c(Cl)c4)c3cc2OC)CC1 107003C[C@]1(CCCN1c1nc(Nc2cc([nH]n2)C2CC2)c2cccn2n1)C(=O)Nc1cnccn1 50059889CN[C@@H]1CC2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13 50130355CC(O)C(Nc1cc(O)c(NC(C(C)=O)C(O)=O)cc1O)C(O)=O 50130356CC(=O)C(Nc1c(O)cc(O)c(O)c1CC1CCCC2CCCCC12)C(O)=O 50150778Oc1c(Br)cc2CCNC(=O)C(Cc3ccc(Oc4cc(CC(N=O)C(=O)NC=Cc5ccc(Oc1c2)c(Br)c5)cc(Br)c4O)c(Br)c3)N=O 50181672CN1CCN(CCc2ccc(NC(=O)c3cc(c[nH]c3=O)-c3ccc4OCOc4c3)cc2)CC1 50182475COc1cc(cc(OC)c1OC)C1=C(C(=O)NC1=O)c1c[nH]c2ccccc12 50199623Nc1nccn2c(nc(-c3cccc(OCc4ccccc4)c3)c12)[C@H]1CC[C@H](CN2CCCC2)CC1 50199624Nc1nccn2c(nc(-c3cccc(OCc4ccccc4)c3)c12)[C@H]1CC[C@H](CN2CCOCC2)CC1 50199625Nc1nccn2c(nc(-c3cccc(OCc4cccc(F)c4)c3)c12)C1CCC1 50199626CN(C)C[C@H]1C[C@H](C1)c1nc(-c2cccc(OCc3ccccc3)c2)c2c(N)nccn12 50199627Nc1nccn2c(nc(-c3cccc(OCc4c(Cl)cccc4Cl)c3)c12)C1CCC1 50199628Nc1nccn2c(nc(-c3cccc(OCc4cc(F)cc(F)c4)c3)c12)C1CCC1 50199629NC(=O)[C@H]1C[C@@H](C1)c1nc(-c2cccc(OCc3ccccc3)c2)c2c(N)nccn12 50199630Nc1nccn2c(nc(-c3cccc(OCc4ccccc4F)c3)c12)C1CCC1 50199631NC[C@H]1CC[C@H](CC1)c1nc(-c2cccc(OCc3ccccc3)c2)c2c(N)nccn12 50199632Nc1nccn2c(nc(-c3cccc(OCc4ccccc4)c3)c12)[C@@H]1C[C@H](CN2CCCC2)C1 50199633Nc1nccn2c(nc(-c3cccc(OCc4ccc(F)c(F)c4)c3)c12)C1CCC1 50199634NC(=O)[C@H]1CC[C@H](CC1)c1nc(-c2cccc(OCc3ccccc3)c2)c2c(N)nccn12 50199636Nc1nccn2c(nc(-c3cccc(OCc4ccc(F)cc4)c3)c12)C1CCC1 50199638Nc1nccn2c(nc(-c3cccc(OCc4ccccc4)c3)c12)[C@@H]1C[C@H](CN2CCCCC2)C1 50199640NC[C@H]1CC[C@@H](CC1)c1nc(-c2cccc(OCc3ccccc3)c2)c2c(N)nccn12 50199641Nc1nccn2c(nc(-c3cccc(OCc4c(F)cccc4F)c3)c12)C1CCC1 50199642Nc1nccn2c(nc(-c3cccc(OC4CCCCC4)c3)c12)C1CCC1 50199643Nc1nccn2c(nc(-c3cccc(OCc4ccc(Cl)cc4)c3)c12)C1CCC1 50199644Nc1nccn2c(nc(-c3cccc(OCc4ccccc4)c3)c12)C1CCCCCC1 50199645Nc1nccn2c(nc(-c3cccc(OCc4ccccc4)c3)c12)C1CCCCC1 50199646CNC(=O)[C@H]1CC[C@@H](CC1)c1nc(-c2cccc(OCc3ccccc3)c2)c2c(N)nccn12 50199649NC(=O)[C@H]1C[C@H](C1)c1nc(-c2cccc(OCc3ccccc3)c2)c2c(N)nccn12 50199650CC(C)NC[C@H]1C[C@H](C1)c1nc(-c2cccc(OCc3ccccc3)c2)c2c(N)nccn12 50199652Nc1nccn2c(nc(-c3cccc(OCc4cccc(OC(F)F)c4)c3)c12)C1CCC1 50199653Nc1nccn2c(nc(-c3cccc(OCc4ccccc4OC(F)F)c3)c12)C1CCC1 50199654Nc1nccn2c(nc(-c3cccc(OCC4CCCCC4)c3)c12)C1CCC1 50199655Nc1nccn2c(nc(-c3ccc(O)c(OCc4ccccc4)c3)c12)C1CCC1 50199656Nc1nccn2c(nc(-c3cccc(OCc4cccc(F)c4F)c3)c12)C1CCC1 50199657COCCOc1cccc(c1)-c1nc(C2CCC2)n2ccnc(N)c12 50199658Nc1nccn2c(nc(-c3cccc(OCc4ccccc4)c3)c12)[C@H]1CC[C@@H](CC1)C(=O)N1CCCCC1 50199659NC[C@H]1C[C@H](C1)c1nc(-c2cccc(OCc3ccccc3)c2)c2c(N)nccn12 50199660Nc1nccn2c(nc(-c3ccc(OCc4ccccc4)cc3)c12)C1CCC1 50199661Nc1nccn2c(nc(-c3cccc(OCc4ccccc4)c3)c12)[C@H]1CC[C@H](CN2CCC2)CC1 50199662Nc1nccn2c(nc(-c3cccc(OCc4ccccc4)c3)c12)-c1ccccc1 50199663Nc1nccn2c(nc(-c3cccc(OCc4ccccc4)c3)c12)[C@H]1CC[C@@H](CC1)C(=O)Nc1ccccc1 50199665Nc1nccn2c(nc(-c3cccc(OCc4cc(F)ccc4F)c3)c12)C1CCC1 50199666Nc1nccn2c(nc(-c3cccc(OCc4ccccc4)c3)c12)[C@H]1C[C@H](CN2CCCC2)C1 50199667NC(=O)[C@H]1CC[C@@H](CC1)c1nc(-c2cccc(OCc3ccccc3)c2)c2c(N)nccn12 50199668CCN(CC)C[C@H]1CC[C@@H](CC1)c1nc(-c2cccc(OCc3ccccc3)c2)c2c(N)nccn12 50199669Nc1nccn2c(nc(-c3cccc(OCC4CC4)c3)c12)C1CCC1 50199671Nc1nccn2c(nc(-c3cccc(OCc4cccc(Cl)c4)c3)c12)C1CCC1 50199673Nc1nccn2c(nc(-c3cccc(OC4CCCC4)c3)c12)C1CCC1 50199675CN(C[C@H]1C[C@H](C1)C1=NC(C2N1C=CN=C2N)c1cccc(OCc2ccccc2)c1)N1CCNCC1 50199676Nc1nccn2c(nc(-c3cccc(OCc4c(F)cccc4Cl)c3)c12)C1CCC1 50199678Nc1nccn2c(nc(-c3cccc(OCc4ccccc4)c3)c12)[C@H]1CC[C@@H](CC1)C(=O)N1CCCC1 50199680COc1ccc(cc1OCc1ccccc1)-c1nc(C2CCC2)n2ccnc(N)c12 50199681Nc1nccn2c(nc(-c3cccc(OCc4ccc(OC(F)F)cc4)c3)c12)C1CCC1 50199682Nc1nccn2c(nc(-c3cccc(OCc4ccccn4)c3)c12)C1CCC1 50199683Nc1nccn2c(nc(-c3cccc(O)c3)c12)C1CCC1 50199685Nc1nccn2c(nc(-c3cccc(OCc4ccccc4)c3)c12)[C@H]1CC[C@@H](CC1)C(=O)NCc1ccccc1 50199686Nc1nccn2c(nc(-c3cccc(OCc4ccccc4)c3)c12)[C@@H]1C[C@H](CN2CCOCC2)C1 50199688Nc1nccn2c(nc(-c3cccc(OCc4ccccc4)c3)c12)C1CCCC1 50199689Nc1nccn2c(nc(-c3cccc(OCc4ccccc4Cl)c3)c12)C1CCC1 50200392FC(F)(F)c1cccc(Nc2ccnc(Nc3cccc(NC(=O)C4CC4)c3)n2)c1 50201120Cc1cc(cc2nc([nH]c12)-c1c(NCC(O)c2ccc(Cl)c(Cl)c2)cc[nH]c1=O)-n1ccnc1 50201121Cc1cc(cc2nc([nH]c12)-c1c(NCC(O)c2ccccc2)cc[nH]c1=O)-n1ccnc1 50201122CC(CNc1cc[nH]c(=O)c1-c1nc2cc(cc(C)c2[nH]1)-n1ccnc1)c1cccc(Br)c1 50201123Cc1ccc(cc1)C(O)CNc1cc[nH]c(=O)c1-c1nc2cc(cc(C)c2[nH]1)-n1ccnc1 50201124Cc1cc(cc2nc([nH]c12)-c1c(NCC(O)c2cccc(Cl)c2)cc[nH]c1=O)-n1ccnc1 50201125Cc1cc(cc2nc([nH]c12)-c1c(NCC(O)c2cccc(c2)C(F)(F)F)cc[nH]c1=O)-n1ccnc1 50201126Cc1cc(cc2nc([nH]c12)-c1c(NCC(O)c2cccc(c2)C#N)cc[nH]c1=O)-n1ccnc1 50201127Cc1cc(cc2nc([nH]c12)-c1ccc[nH]c1=O)-n1ccnc1 50201128Cc1cc(cc2nc([nH]c12)-c1c(NCC(O)c2cccc(NS(C)(=O)=O)c2)cc[nH]c1=O)-n1ccnc1 50201129Cc1cc(cc2nc([nH]c12)-c1c(NCC(O)c2cc(Cl)cc(Cl)c2)cc[nH]c1=O)-n1ccnc1 50201130Cc1cc(cc2nc([nH]c12)-c1c(NC[C@H](O)c2cccc(Cl)c2)cc[nH]c1=O)-n1ccnc1 50201131Cc1cc(cc2nc([nH]c12)-c1c(NCCO)cc[nH]c1=O)-n1ccnc1 50201132COc1ccc(cc1Cl)C(O)CNc1cc[nH]c(=O)c1-c1nc2cc(cc(C)c2[nH]1)-n1ccnc1 50201133Cc1cc(cc2nc([nH]c12)-c1c(NCC(O)c2cccc(O)c2)cc[nH]c1=O)-n1ccnc1 50201134Cc1cc(cc2nc([nH]c12)-c1c(NCC(O)c2cccc(F)c2)cc[nH]c1=O)-n1ccnc1 50201135Cc1cc(cc2nc([nH]c12)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O)-n1ccnc1 50201136Cc1cc(cc2nc([nH]c12)-c1c(NCC(O)c2ccc(NS(C)(=O)=O)cc2)cc[nH]c1=O)-n1ccnc1 50201137COc1ccc(cc1)C(O)CNc1cc[nH]c(=O)c1-c1nc2cc(cc(C)c2[nH]1)-n1ccnc1 50201138Cc1cc(cc2nc([nH]c12)-c1c(NCC(O)c2ccc(F)c(Cl)c2)cc[nH]c1=O)-n1ccnc1 50201139COC(CNc1cc[nH]c(=O)c1-c1nc2cc(cc(C)c2[nH]1)-n1ccnc1)c1cccc(Cl)c1 50201140Cc1cc(cc2nc([nH]c12)-c1c(NCCc2ccccc2)cc[nH]c1=O)-n1ccnc1 50201141Cc1cc(cc2nc([nH]c12)-c1c(NCC(O)c2ccccc2Cl)cc[nH]c1=O)-n1ccnc1 50201142Cc1cc(cc2nc([nH]c12)-c1c(NCC(O)c2ccccc2NS(C)(=O)=O)cc[nH]c1=O)-n1ccnc1 50201143Cc1cccc(c1)C(O)CNc1cc[nH]c(=O)c1-c1nc2cc(cc(C)c2[nH]1)-n1ccnc1 50201144Cc1cc(cc2nc([nH]c12)-c1c(NCC(O)c2cccc(Br)c2)cc[nH]c1=O)-n1ccnc1 50201145COc1cccc(c1)C(O)CNc1cc[nH]c(=O)c1-c1nc2cc(cc(C)c2[nH]1)-n1ccnc1 50201788COc1cc(C=C2SC(O)=NC2=O)cc(OC)c1O 50206118Cc1cc(cc2nc([nH]c12)-c1c(N[C@H](CO)Cc2ccccc2Br)cc[nH]c1=O)-n1ccnc1 50206120Cc1cc(cc2nc([nH]c12)-c1c(NCc2ccccn2)cc[nH]c1=O)-n1ccnc1 50206121Cc1cc(cc2nc([nH]c12)-c1c(N[C@H](CO)Cc2ccccn2)cc[nH]c1=O)-n1ccnc1 50206122Cc1cc(cc2nc([nH]c12)-c1c(N[C@H](CO)Cc2ccc(OC(C)(C)C)cc2)cc[nH]c1=O)-n1ccnc1 50206124Cc1cc(cc2nc([nH]c12)-c1c(N[C@H](CO)Cc2ccccc2Cl)cc[nH]c1=O)-n1ccnc1 50206125COc1cccc(C[C@@H](CO)Nc2cc[nH]c(=O)c2-c2nc3cc(cc(C)c3[nH]2)-n2ccnc2)c1 50206126Cc1cc(cc2nc([nH]c12)-c1c(N[C@H](CO)Cc2cccc(Cl)c2)cc[nH]c1=O)-n1ccnc1 50206127Cc1cc(cc2nc([nH]c12)-c1c(N[C@H](CO)Cc2cccc(c2)[N+]([O-])=O)cc[nH]c1=O)-n1ccnc1 50206128Cc1cc(cc2nc([nH]c12)-c1c(NCc2ccco2)cc[nH]c1=O)-n1ccnc1 50206129Cc1cc(cc2nc([nH]c12)-c1c(N[C@H](CO)Cc2ccc(Cl)cc2)cc[nH]c1=O)-n1ccnc1 50206130COc1ccccc1C[C@@H](CO)Nc1cc[nH]c(=O)c1-c1nc2cc(cc(C)c2[nH]1)-n1ccnc1 50206132Cc1cc(cc2nc([nH]c12)-c1c(NCCn2nccn2)cc[nH]c1=O)-n1ccnc1 50206134Cc1cc(cc2nc([nH]c12)-c1c(NCCc2cccs2)cc[nH]c1=O)-n1ccnc1 50206135COc1ccc(C[C@@H](CO)Nc2cc[nH]c(=O)c2-c2nc3cc(cc(C)c3[nH]2)-n2ccnc2)cc1 50206136Cc1cc(cc2nc([nH]c12)-c1c(N[C@H](CO)Cc2ccccc2)cc[nH]c1=O)-n1ccnc1 50206139Cc1cc(cc2nc([nH]c12)-c1c(N[C@H](CO)Cc2ccc(F)cc2)cc[nH]c1=O)-n1ccnc1 50206141Cc1cc(cc2nc([nH]c12)-c1c(NCCc2ccccn2)cc[nH]c1=O)-n1ccnc1 50206143Cc1cc(cc2nc([nH]c12)-c1c(N[C@H](CO)Cc2cccc(Br)c2)cc[nH]c1=O)-n1ccnc1 50206146Cc1cc(cc2nc([nH]c12)-c1c(NCc2cccs2)cc[nH]c1=O)-n1ccnc1 50206147Cc1cc(cc2nc([nH]c12)-c1c(N[C@H](CO)Cc2ccccc2OC(F)(F)F)cc[nH]c1=O)-n1ccnc1 50206148Cc1cc(cc2nc([nH]c12)-c1c(N[C@H](CO)Cc2ccccc2C#N)cc[nH]c1=O)-n1ccnc1 50206150Cc1ccccc1C[C@@H](CO)Nc1cc[nH]c(=O)c1-c1nc2cc(cc(C)c2[nH]1)-n1ccnc1 50206151Cc1cc(cc2nc([nH]c12)-c1c(N[C@H](CO)Cc2cccc(F)c2)cc[nH]c1=O)-n1ccnc1 50206152Cc1cc(cc2nc([nH]c12)-c1c(N[C@H](CO)Cc2cccc(c2)C(F)(F)F)cc[nH]c1=O)-n1ccnc1 50209378Cc1cccc2[nH]c(nc12)-c1c(NCC(O)c2cccc(Cl)c2)cc[nH]c1=O 50209379COc1ccc(cc1)-c1cc(C)c2nc([nH]c2c1)-c1c(N[C@H](CO)Cc2ccccc2)cc[nH]c1=O 50209380Cc1cc(Br)cc2[nH]c(nc12)-c1c(N[C@H](CO)Cc2ccccc2)cc[nH]c1=O 50209381Cc1cc(cc2[nH]c(nc12)-c1c(NCC(O)c2cccc(Cl)c2)cc[nH]c1=O)C(=O)NC1CCCC1 50209382CNC(=N)c1cc(C)c2nc([nH]c2c1)-c1c(NCC(O)c2cccc(Cl)c2)cc[nH]c1=O 50209383Cc1cc(cc2[nH]c(nc12)-c1c(N[C@H](CO)Cc2ccccc2)cc[nH]c1=O)-c1ccc(F)cc1 50209384CN(C)C(=O)c1cc(C)c2nc([nH]c2c1)-c1c(NCC(O)c2cccc(Cl)c2)cc[nH]c1=O 50209385CC1CNC(=N1)c1cc(C)c2nc([nH]c2c1)-c1c(NCC(O)c2cccc(Cl)c2)cc[nH]c1=O 50209386CNC(=O)c1cc(C)c2nc([nH]c2c1)-c1c(NCC(O)c2cccc(Cl)c2)cc[nH]c1=O 50209387Cc1cc(cc2[nH]c(nc12)-c1c(NCC(O)c2cccc(Cl)c2)cc[nH]c1=O)C1=NC(C)(C)CN1 50209388Cc1cc(cc2[nH]c(nc12)-c1c(N[C@H](CO)Cc2ccccc2)cc[nH]c1=O)-c1ccccc1 50209389Cc1cc(cc2[nH]c(nc12)-c1c(NCC(O)c2cccc(Cl)c2)cc[nH]c1=O)C1=NCCCN1 50209390Cc1cc(cc2[nH]c(nc12)-c1c(NCC(O)c2cccc(Cl)c2)cc[nH]c1=O)C(=O)NC1CCCCC1 50209391Cc1c[nH]c(n1)-c1cc(C)c2[nH]c(nc2c1)-c1c(NCC(O)c2cccc(Cl)c2)cc[nH]c1=O 50209392CN1CCN=C1c1cc(C)c2nc([nH]c2c1)-c1c(NCC(O)c2cccc(Cl)c2)cc[nH]c1=O 50209393Cc1cc(cc2[nH]c(nc12)-c1c(NCC(O)c2cccc(Cl)c2)cc[nH]c1=O)C(=O)NC1CC1 50209394Cc1cc(cc2[nH]c(nc12)-c1c(NCC(O)c2cccc(Cl)c2)cc[nH]c1=O)C(N)=O 50211912SC1=NC(=O)C(S1)=Cc1ccc(o1)-c1ccccc1Cl 50212955Oc1ccc(CCCCc2ccc(O)c(O)c2)cc1 50212956Oc1ccc(CCCCc2ccccc2)cc1O 50212957Oc1ccc(CCCCc2ccc(Cl)c(Cl)c2)cc1O 50212958Oc1ccc(CCCCc2ccc(O)c(O)c2)cc1O 50212959Cc1ccc(CCCCc2ccc(O)c(O)c2)cc1 50212960Oc1ccc(CCCCc2ccc(Cl)cc2)cc1O 50212961Oc1cc2CCCC(c3ccccc3)c2cc1O 50212962COc1ccc(CCCCc2ccc(O)c(O)c2)cc1 50219355Nc1ncnc2n(cc(-c3cccc(OCc4ccccc4)c3)c12)[C@H]1C[C@H](CN2CCCC2)C1 50219357Cc1ccccc1Cc1nc2ccc(cc2[nH]1)-c1nn([C@H]2CC[C@@H](CC2)N2CCOCC2)c2ncnc(N)c12 50219358Nc1ncnc2n(nc(-c3ccc4nc(Cc5ccccn5)[nH]c4c3)c12)[C@H]1CC[C@@H](CC1)N1CCOCC1 50219359Cc1cc(cc2[nH]c(Cc3ccccc3)nc12)-c1nn([C@H]2CC[C@@H](CC2)N2CCOCC2)c2ncnc(N)c12 50219361Nc1ncnc2n(nc(-c3ccc4nc(Cc5ccccc5F)[nH]c4c3)c12)[C@H]1CC[C@@H](CC1)N1CCOCC1 50219362Cn1c(Cc2ccccc2)nc2cc(ccc12)-c1nn([C@H]2CC[C@@H](CC2)N2CCOCC2)c2ncnc(N)c12 50219363Nc1ncnc2n(nc(-c3ccc4nc(Cc5cc(F)cc(F)c5)[nH]c4c3)c12)[C@H]1CC[C@@H](CC1)N1CCOCC1 50219364Nc1ncnc2n(nc(-c3ccc4nc(Cc5ccc(Cl)cc5)[nH]c4c3)c12)[C@H]1CC[C@@H](CC1)N1CCOCC1 50219365Nc1ncnc2n(nc(-c3ccc4nc(Cc5cccc(Cl)c5)[nH]c4c3)c12)[C@H]1CC[C@@H](CC1)N1CCOCC1 50219366Nc1ncnc2n(nc(-c3ccc4nc(Cc5cccc(Cl)c5Cl)[nH]c4c3)c12)[C@H]1CC[C@@H](CC1)N1CCOCC1 50219367Nc1ncnc2n(nc(-c3ccc4nc(Cc5c(F)cccc5Cl)[nH]c4c3)c12)[C@H]1CC[C@@H](CC1)N1CCOCC1 50219369Nc1ncnc2n(nc(-c3ccc4nc(Cc5ccc(Cl)c(Cl)c5)[nH]c4c3)c12)[C@H]1CC[C@@H](CC1)N1CCOCC1 50219370Cc1nc(Cc2nc3ccc(cc3[nH]2)-c2nn([C@H]3CC[C@@H](CC3)N3CCOCC3)c3ncnc(N)c23)cs1 50219371Nc1ncnc2n(nc(-c3ccc4nc(Cc5cccc(F)c5)[nH]c4c3)c12)[C@H]1CC[C@@H](CC1)N1CCOCC1 50219372Cc1cccc(Cc2nc3ccc(cc3[nH]2)-c2nn([C@H]3CC[C@@H](CC3)N3CCOCC3)c3ncnc(N)c23)c1 50219373Nc1ncnc2n(nc(-c3ccc4nc(Cc5cccc(F)c5F)[nH]c4c3)c12)[C@H]1CC[C@@H](CC1)N1CCOCC1 50219374Nc1ncnc2n(nc(-c3ccc4nc(Cc5c(Cl)cccc5Cl)[nH]c4c3)c12)[C@H]1CC[C@@H](CC1)N1CCOCC1 50219375Nc1ncnc2n(nc(-c3ccc4nc(CCc5ccccc5)[nH]c4c3)c12)[C@H]1CC[C@@H](CC1)N1CCOCC1 50219377Nc1ncnc2n(nc(-c3ccc4nc(Cc5ccsc5)[nH]c4c3)c12)[C@H]1CC[C@@H](CC1)N1CCOCC1 50219378Nc1ncnc2n(nc(-c3ccc4nc(Cc5ccc(F)cc5)[nH]c4c3)c12)[C@H]1CC[C@@H](CC1)N1CCOCC1 50219379Nc1ncnc2n(nc(-c3ccc4nc(Cc5c(F)cccc5F)[nH]c4c3)c12)[C@H]1CC[C@@H](CC1)N1CCOCC1 50219380Nc1ncnc2n(nc(-c3ccc4nc(Cc5ccccc5Br)[nH]c4c3)c12)[C@H]1CC[C@@H](CC1)N1CCOCC1 50219381Nc1ncnc2n(nc(-c3ccc4nc(Cc5ccc(F)c(F)c5)[nH]c4c3)c12)[C@H]1CC[C@@H](CC1)N1CCOCC1 50219382CN1CCN(CC1)[C@H]1C[C@H](C1)c1nc(-c2ccc3ccc(nc3c2)-c2ccccc2)c2c(N)nccn12 50219383Cc1ccc(Cc2nc3ccc(cc3[nH]2)-c2nn([C@H]3CC[C@@H](CC3)N3CCOCC3)c3ncnc(N)c23)cc1 50219384Nc1ncnc2n(nc(-c3ccc4nc(Cc5ccc6ccccc6c5)[nH]c4c3)c12)[C@H]1CC[C@@H](CC1)N1CCOCC1 50219385Nc1ncnc2n(nc(-c3ccc4nc([nH]c4c3)-c3ccccc3)c12)[C@H]1CC[C@@H](CC1)N1CCOCC1 50229085C[C@@H](N)C(=O)N1CCN(CC1)C(=O)c1cc(Sc2cnc(Nc3cccc(Br)n3)s2)ccc1C 50229087C[C@H](N)C(=O)N1CCN(CC1)C(=O)c1cc(Sc2cnc(Nc3cccc(Br)n3)s2)ccc1C 50230005COc1ccc(Cl)cc1NC(=O)Nc1cc(C)nc2ccccc12 50234501COCCn1cnc(CCNc2cc[nH]c(=O)c2-c2nc3c(C)cc(cc3[nH]2)N2CCOCC2)c1Cl 50234502Cc1ccn(CCNc2cc[nH]c(=O)c2-c2nc3c(C)cc(cc3[nH]2)N2CCOCC2)n1 50234503Cc1cc(cc2[nH]c(nc12)-c1c(NCCc2cn(C)cn2)cc[nH]c1=O)N1CCOCC1 50234504Cc1cc(cc2[nH]c(nc12)-c1c(NCCn2ncc(Br)c2CO)cc[nH]c1=O)N1CCOCC1 50234505CCn1cnc(CCNc2cc[nH]c(=O)c2-c2nc3c(C)cc(cc3[nH]2)N2CCOCC2)c1Cl 50234506Cc1cc(cc2[nH]c(nc12)-c1c(NCCn2cc(Br)cn2)cc[nH]c1=O)N1CCOCC1 50234507COCCn1cnc(CCNc2cc[nH]c(=O)c2-c2nc3c(C)cc(cc3[nH]2)N2CCOCC2)c1 50234508Cc1ccnn1CCNc1cc[nH]c(=O)c1-c1nc2c(C)cc(cc2[nH]1)N1CCOCC1 50234509Cc1cc(cc2[nH]c(nc12)-c1c(NCCc2ncn(C)c2Cl)cc[nH]c1=O)N1CCOCC1 50234510Cc1nn(CCNc2cc[nH]c(=O)c2-c2nc3c(C)cc(cc3[nH]2)N2CCOCC2)cc1Cl 50234511CCn1cnc(CCNc2cc[nH]c(=O)c2-c2nc3c(C)cc(cc3[nH]2)N2CCOCC2)c1 50234512Cc1cc(cc2[nH]c(nc12)-c1c(NCCn2cc(Br)c(CO)n2)cc[nH]c1=O)N1CCOCC1 50234513Cc1cc(cc2[nH]c(nc12)-c1c(NCCn2cc(Cl)cn2)cc[nH]c1=O)N1CCOCC1 50234514Cc1c(Cl)cnn1CCNc1cc[nH]c(=O)c1-c1nc2c(C)cc(cc2[nH]1)N1CCOCC1 50234515Cc1c(Br)cnn1CCNc1cc[nH]c(=O)c1-c1nc2c(C)cc(cc2[nH]1)N1CCOCC1 50234516Cc1cc(cc2[nH]c(nc12)-c1c(NCCn2cc(cn2)C#N)cc[nH]c1=O)N1CCOCC1 50234517CC(C)n1cnc(CCNc2cc[nH]c(=O)c2-c2nc3c(C)cc(cc3[nH]2)N2CCOCC2)c1Cl 50234518Cc1cc(cc2[nH]c(nc12)-c1c(NCCc2ncn(C)c2Br)cc[nH]c1=O)N1CCOCC1 50234519Cc1cc(cc2[nH]c(nc12)-c1c(NCCc2nc(Cl)n(C)c2Cl)cc[nH]c1=O)N1CCOCC1 50234520CC(C)n1cnc(CCNc2cc[nH]c(=O)c2-c2nc3c(C)cc(cc3[nH]2)N2CCOCC2)c1 50234521Cc1cnn(CCNc2cc[nH]c(=O)c2-c2nc3c(C)cc(cc3[nH]2)N2CCOCC2)c1 50234522COC(=O)c1cnn(CCNc2cc[nH]c(=O)c2-c2nc3c(C)cc(cc3[nH]2)N2CCOCC2)c1 50234523Cc1nc(CCNc2cc[nH]c(=O)c2-c2nc3c(C)cc(cc3[nH]2)N2CCOCC2)c(Cl)n1C 50234524CCOC(=O)c1cnn(CCNc2cc[nH]c(=O)c2-c2nc3c(C)cc(cc3[nH]2)N2CCOCC2)c1 50234525Cc1cc(cc2[nH]c(nc12)-c1c(NCCc2ncn(CCF)c2Cl)cc[nH]c1=O)N1CCOCC1 50234526Cc1cc(cc2[nH]c(nc12)-c1c(NCCn2cccn2)cc[nH]c1=O)N1CCOCC1 50234527Cc1nn(CCNc2cc[nH]c(=O)c2-c2nc3c(C)cc(cc3[nH]2)N2CCOCC2)cc1Br 50234528CCn1cnc(CCNc2cc[nH]c(=O)c2-c2nc3c(C)cc(cc3[nH]2)N2CCOCC2)c1C#C 50234529CCn1cnc(CCNc2cc[nH]c(=O)c2-c2nc3c(C)cc(cc3[nH]2)N2CCOCC2)c1Br 50242742COc1cc(ccc1Nc1ncc(Cl)c(Nc2ccccc2S(=O)(=O)C(C)C)n1)N1CCC(CC1)N1CCN(C)CC1 50243880COc1cc(cc(OC)c1OC)C1=C(CNC1=O)c1cn(COCC[Si](C)(C)C)c2ccccc12 50243930COc1cc(cc(OC)c1OC)C1=C(CNC1=O)c1cn(COC(C)(C)C)c2ccccc12 50246774NC(=N)SCCCn1c(=O)c2c(n3c(cc4ccccc34)c3cccc4ccn2c34)c1=O 50246815N=C(Nc1ccccc1)SCCCN1C(=O)C2=C(C1=O)n1ccc3cccc(C4Cc5ccccc5N24)c13 50248085Oc1ccc(NC(=S)NC(=O)c2ccc(cc2)[N+]([O-])=O)cc1-c1nc2ccccc2s1 50248148N(c1ccc(cc1)-c1nc2ccccc2s1)c1ncnc2[nH]ccc12 50248149COc1cc(Nc2ncnc3[nH]ccc23)ccc1-c1nc2ccccc2s1 50248150COc1nc(Nc2ccc(cc2)-c2nc3ccccc3s2)c2cc[nH]c2n1 50248182COc1nc(Nc2ccc(-c3nc4ccccc4s3)c(OC)c2)c2cc[nH]c2n1 50248230Clc1ccc2c(Nc3ccc(cc3)-c3nc4ccccc4s3)ccnc2c1 50248232Clc1ccc2c(Nc3ccc(-c4nc5ccccc5s4)c(Cl)c3)ncnc2c1 50248291Fc1cc(ccc1Nc1ncnc2cc(Cl)ccc12)-c1nc2ccccc2s1 50248292Cc1cc2c(Nc3ccc(cc3)-c3nc4ccccc4s3)ncnc2cc1Cl 50248351COc1cc2nc(Nc3cc(C)n[nH]3)nc(Nc3ccc(cc3)-c3nc4ccccc4s3)c2cc1OC 50248413Cc1cc(Nc2ccnc(Nc3cccc(c3)-c3nc4ccccc4s3)n2)[nH]n1 50248414COc1cc2nc(Nc3cc(C)n[nH]3)nc(Nc3cccc(c3)-c3nc4ccccc4s3)c2cc1OC 50248416N(c1cccc(c1)-c1nc2ccccc2s1)c1ncnc2nc[nH]c12 50248464COc1cc2ncnc(Nc3ccc(cc3)N3Cc4ccccc4C3)c2cc1OC 50249542COc1cc(Nc2ncc(F)c(Nc3ccc4OC(C)(C)C(=O)Nc4n3)n2)cc(OC)c1OC 50252094Cc1cc(cc2[nH]c(nc12)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O)N1CCC(O)CC1 50252142COC1CCN(CC1)c1cc(C)c2nc([nH]c2c1)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O 50252143COCCOC1CCN(CC1)c1cc(C)c2nc([nH]c2c1)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O 50252144Cc1cc(cc2[nH]c(nc12)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O)N1CCC(CC1)OCCO 50252193Cc1cc(cc2[nH]c(nc12)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O)N1CCC2(CC1)OCCO2 50252194CNC1CCN(CC1)c1cc(C)c2nc([nH]c2c1)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O 50252195CN(C)C1CCN(CC1)c1cc(C)c2nc([nH]c2c1)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O 50252235Cc1cc(cc2[nH]c(nc12)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O)N1CCC(CC1)N1CCCC1 50252236Cc1cc(cc2[nH]c(nc12)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O)N1CCC(CC1)NC(=O)C1CC1 50252237COC(=O)NC1CCN(CC1)c1cc(C)c2nc([nH]c2c1)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O 50252238COCCN(CCOC)C1CCN(CC1)c1cc(C)c2nc([nH]c2c1)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O 50252293Cc1cc(cc2[nH]c(nc12)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O)N1CCC(CC1)N1CCOCC1 50252294C[C@H]1CN(C[C@@H](C)O1)C1CCN(CC1)c1cc(C)c2nc([nH]c2c1)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O 50252295Cc1cc(cc2[nH]c(nc12)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O)N1CCC(CC1)N1C[C@@H]2C[C@@H]1CO2 50252296CN1CCN(CC1)C1CCN(CC1)c1cc(C)c2nc([nH]c2c1)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O 50252297CC(=O)N1CCN(CC1)C1CCN(CC1)c1cc(C)c2nc([nH]c2c1)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O 50252298COCC(=O)N1CCN(CC1)C1CCN(CC1)c1cc(C)c2nc([nH]c2c1)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O 50252299COCCOCC(=O)N1CCN(CC1)C1CCN(CC1)c1cc(C)c2nc([nH]c2c1)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O 50252300Cc1cc(cc2[nH]c(nc12)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O)N1CCC(CC1)N1CCN(CC1)C(=O)C1CC1 50252301COC(=O)N1CCN(CC1)C1CCN(CC1)c1cc(C)c2nc([nH]c2c1)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O 50252302COCCOC(=O)N1CCN(CC1)C1CCN(CC1)c1cc(C)c2nc([nH]c2c1)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O 50252303Cc1cc(cc2[nH]c(nc12)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O)N1CCC(CC1)N1CCN(CC1)C(=O)OCCO 50252304Cc1cc(cc2[nH]c(nc12)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O)N1CCC(CC1)N1CCN(CC1)C(=O)N1CCOCC1 50252305CN1CCN(CC1)C(=O)N1CCN(CC1)C1CCN(CC1)c1cc(C)c2nc([nH]c2c1)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O 50256410CN(C)CCCc1ccc(Nc2nccc(n2)-c2c(nc3ccccn23)-c2cccc(c2)C(=O)Nc2c(F)cccc2F)cc1 50256411Fc1cccc(F)c1C(=O)Nc1cccc(c1)-c1nc2ccccn2c1-c1ccnc(Nc2cccc(CN3CCCC3)c2)n1 50256412Fc1cccc(F)c1NC(=O)c1cccc(c1)-c1nc2ccccn2c1-c1ccnc(Nc2cccc(CN3CCCC3)c2)n1 50256413Nc1nccc(n1)-c1c(nc2ccccn12)-c1cccc(c1)C(=O)Nc1c(F)cccc1F 50256465Fc1cccc(Nc2nccc(n2)-c2c(nc3ccccn23)-c2cccc(c2)C(=O)Nc2c(F)cccc2F)c1 50256466Fc1cccc(F)c1NC(=O)c1cccc(c1)-c1nc2ccccn2c1-c1ccnc(Nc2ccc3OCCOc3c2)n1 50256467CN(C)CCOc1cccc(Nc2nccc(n2)-c2c(nc3ccccn23)-c2cccc(c2)C(=O)Nc2c(F)cccc2F)c1 50256468Fc1cccc(F)c1NC(=O)c1cccc(c1)-c1nc2ccccn2c1-c1ccnc(Nc2ccc(CCN3CCOCC3)cc2)n1 50256469CN(C)C[C@H](O)COc1cccc(Nc2nccc(n2)-c2c(nc3ccccn23)-c2cccc(c2)C(=O)Nc2c(F)cccc2F)c1 50256470Fc1cccc(F)c1NC(=O)c1cccc(c1)-c1nc2ccccn2c1-c1ccnc(Nc2ccc(cc2)N2CCC(CC2)N2CCCCC2)n1 50256471COc1cc(ccc1Nc1nccc(n1)-c1c(nc2ccccn12)-c1cccc(c1)C(=O)Nc1c(F)cccc1F)N1CCC(CC1)N1CCCCC1 50256472COc1cc(ccc1Nc1nccc(n1)-c1c(nc2ccccn12)-c1cccc(c1)C(=O)Nc1c(F)cccc1F)N1CCC(CC1)N1CCOCC1 50256473COc1cc(ccc1Nc1nccc(n1)-c1c(nc2ccccn12)-c1cccc(c1)C(=O)Nc1c(F)cccc1F)N1CCC(CC1)N1CCCC1 50256474COc1cc(ccc1Nc1nccc(n1)-c1c(nc2ccccn12)-c1cccc(c1)C(=O)Nc1c(F)cccc1F)N1CCC(CC1)N1CC[C@@H](F)C1 50256475COc1cc(ccc1Nc1nccc(n1)-c1c(nc2ccccn12)-c1cccc(c1)C(=O)Nc1c(F)cccc1F)N1CCC(CC1)N1CCN(C)CC1 50256476COc1cc(ccc1Nc1nccc(n1)-c1c(nc2ccccn12)-c1cccc(c1)C(=O)Nc1c(F)cccc1F)N1CCC(CC1)N1C[C@H](C)O[C@H](C)C1 50256477COc1cc(ccc1Nc1nccc(n1)-c1c(nc2ccccn12)-c1cccc(c1)C(=O)Nc1c(F)cccc1F)N1CCC(CC1)N1CCN(CC1)C(C)=O 50256478COc1cc(ccc1Nc1nccc(n1)-c1c(nc2ccccn12)-c1cccc(c1)C(=O)Nc1c(F)cccc1F)N1CCC(CC1)N1CCN(CC1)S(C)(=O)=O 50256479CCc1cc(Nc2nccc(n2)-c2c(nc3ccccn23)-c2cccc(c2)C(=O)Nc2c(F)cccc2F)c(OC)cc1N1CCC(CC1)N1CCN(CC1)S(C)(=O)=O 50256480CCc1cc(Nc2nccc(n2)-c2c(nc3ccccn23)-c2ccc(OC)c(c2)C(=O)Nc2c(F)cccc2F)c(OC)cc1N1CCC(CC1)N1CCN(CC1)S(C)(=O)=O 50265843COc1cc(ccc1Nc1nc(Nc2ccccc2-n2cccn2)c2cc[nH]c2n1)N1CCN(CC1)C(C)C 50265844COc1cc(ccc1Nc1nc(Nc2ccsc2C(N)=O)c2cc[nH]c2n1)N1CCN(CC1)C(C)C 50265846CCCN1CCC(CC1)c1ccc(Nc2nc(Nc3ccsc3C(N)=O)c3cc[nH]c3n2)c(OC)c1 50265847COc1cc2CCCN(C(=O)CN(C)C)c2cc1Nc1nc(Nc2ccoc2C(N)=O)c2cc[nH]c2n1 50265848COc1cc2CCN(C(=O)CN(C)C)c2cc1Nc1nc(N2CCc3ccccc23)c2cc[nH]c2n1 50265849COc1cc2CCCN(C(=O)CN(C)C)c2cc1Nc1nc(N2CCc3ccccc23)c2cc[nH]c2n1 50265850COc1cc2CCN(C(=O)CN(C)C)c2cc1Nc1nc(Nc2cccnc2C(N)=O)c2cc[nH]c2n1 50265867COc1cc(ccc1Nc1nc2[nH]ccc2c2nc3cccc(F)c3c(=O)n12)N1CCN(CC1)C(C)C 50265869COc1cc2CCN(C(=O)CN(C)C)c2cc1Nc1nc(Nc2ccsc2C(N)=O)c2cc[nH]c2n1 50265870COc1cc2CCCN(C(=O)CN(C)C)c2cc1Nc1nc(Nc2ccsc2C(N)=O)c2cc[nH]c2n1 50265871COc1cc2c(cc1Nc1nc(Nc3ccsc3C(N)=O)c3cc[nH]c3n1)N(CCC2(C)C)C(=O)CN(C)C 50265872COc1cc2CCCN(C(=O)CN(C)C)c2cc1Nc1nc(Nc2cccnc2C(N)=O)c2cc[nH]c2n1 50265873COc1cc2CCN(C(=O)CN(C)C)c2cc1Nc1nc(Nc2cccc3CNC(=O)c23)c2cc[nH]c2n1 50265887CNC(=O)c1cscc1Nc1nc(Nc2cc3N(CCc3cc2OC)C(=O)CN(C)C)nc2[nH]ccc12 50265888COc1cc2CCN(C(=O)CN(C)C)c2cc1Nc1nc(Nc2ccoc2C(N)=O)c2cc[nH]c2n1 50266295COc1cc(ccc1Nc1nc(Nc2ccccc2C#N)c2cc[nH]c2n1)N1CCN(CC(C)C)CC1 50266296COc1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCN(CC2)C(C)C)nc2[nH]ccc12 50266331COc1cc(ccc1Nc1nc(Nc2ccc3ncccc3c2)c2cc[nH]c2n1)N1CCN(CC1)C(C)C 50266332COc1cc(ccc1Nc1nc(Nc2cccc3ncccc23)c2cc[nH]c2n1)N1CCN(CC1)C(C)C 50266333COc1cc(ccc1Nc1nc(Nc2cccc3CCNc23)c2cc[nH]c2n1)N1CCN(CC1)C(C)C 50293528COc1ccc(cc1OC)-c1cnc2[nH]cc(-c3cccc(NC(=O)Nc4ccc(cc4F)C(F)(F)F)c3)c2c1 50293529Fc1cccc(c1)-c1cnc2[nH]cc(-c3cccc(NC(=O)Nc4ccc(cc4F)C(F)(F)F)c3)c2c1 50293530Nc1cccc(c1)-c1cnc2[nH]cc(-c3cccc(NC(=O)Nc4ccc(cc4F)C(F)(F)F)c3)c2c1 50293531Nc1ccc(cc1)-c1cnc2[nH]cc(-c3cccc(NC(=O)Nc4ccc(cc4F)C(F)(F)F)c3)c2c1 50293532NCc1ccc(cc1)-c1cnc2[nH]cc(-c3cccc(NC(=O)Nc4ccc(cc4F)C(F)(F)F)c3)c2c1 50293533CN1CCN(CC1)C(=O)c1cccc(c1)-c1cnc2[nH]cc(-c3cccc(NC(=O)Nc4ccc(cc4F)C(F)(F)F)c3)c2c1 50293534CN(C)CCNC(=O)c1cccc(c1)-c1cnc2[nH]cc(-c3cccc(NC(=O)Nc4ccc(cc4F)C(F)(F)F)c3)c2c1 50293535CN1CCN(CC1)C(=O)c1ccc(cc1)-c1cnc2[nH]cc(-c3cccc(NC(=O)Nc4ccc(cc4F)C(F)(F)F)c3)c2c1 50293536CN(C)CCNC(=O)c1ccc(cc1)-c1cnc2[nH]cc(-c3cccc(NC(=O)Nc4ccc(cc4F)C(F)(F)F)c3)c2c1 50293537Clc1cccc(NC(=O)Nc2cccc(c2)-c2c[nH]c3ncc(cc23)-c2ccccc2)c1 50293538NCc1ccc(cc1)-c1cnc2[nH]cc(-c3cccc(NC(=O)Nc4cccc(Cl)c4)c3)c2c1 50293539NCc1ccc(cc1)-c1cnc2[nH]cc(-c3cccc(NC(=O)Nc4ccccc4Oc4ccccc4)c3)c2c1 50293540CN(C)CCNC(=O)c1ccc(cc1)-c1cnc2[nH]cc(-c3cccc(NC(=O)Nc4ccccc4Oc4ccccc4)c3)c2c1 50293541CN(C)CCNC(=O)c1cccc(c1)-c1cnc2[nH]cc(-c3cccc(NC(=O)Nc4ccccc4Oc4ccccc4)c3)c2c1 50293542O=C(Nc1cccc(c1)-c1c[nH]c2ncc(cc12)-c1ccccc1)Nc1ccccc1Oc1ccccc1 50293543CN(C)C(=O)c1cccc(c1)-c1cnc2[nH]cc(-c3cccc(NC(=O)Nc4ccccc4Oc4ccccc4)c3)c2c1 50293544CN(C)S(=O)(=O)c1cccc(c1)-c1cnc2[nH]cc(-c3cccc(NC(=O)Nc4ccccc4Oc4ccccc4)c3)c2c1 50293545CN(C)C(=O)c1ccc(cc1)-c1cnc2[nH]cc(-c3cccc(NC(=O)Nc4ccccc4Oc4ccccc4)c3)c2c1 50293546OC(=O)c1cccc(c1)-c1cnc2[nH]cc(-c3cccc(NC(=O)Nc4ccccc4Oc4ccccc4)c3)c2c1 50293547OC(=O)CCc1ccc(cc1)-c1cnc2[nH]cc(-c3cccc(NC(=O)Nc4ccccc4Oc4ccccc4)c3)c2c1 50293548O=C(Nc1cccc(c1)-c1c[nH]c2ncc(cc12)-c1ccc[nH]1)Nc1ccccc1Oc1ccccc1 50293549CN(C)C(=O)c1cccc(c1)-c1cnc2[nH]cc(-c3cccc(NC(=O)Nc4ccccc4Nc4ccccc4)c3)c2c1 50293550CN(C)C(=O)c1cccc(c1)-c1cnc2[nH]cc(-c3cccc(NC(=O)Nc4ccccc4OCc4ccccc4)c3)c2c1 50293551CN(C)C(=O)c1cccc(c1)-c1cnc2[nH]cc(-c3cccc(NC(=O)Nc4ccccc4-c4ccccc4)c3)c2c1 50293552CN(C)C(=O)c1cccc(c1)-c1cnc2[nH]cc(-c3cccc(NC(=O)Nc4cccc(Oc5ccccc5)c4)c3)c2c1 50293553CN(C)C(=O)c1cccc(c1)-c1cnc2[nH]cc(-c3cccc(NC(=O)Nc4ccc(Oc5ccccc5)cc4)c3)c2c1 50293555O=C(Nc1ccccc1)Nc1cccc(c1)-c1c[nH]c2ncc(cc12)-c1ccccc1 50293556Fc1cc(ccc1NC(=O)Nc1cccc(c1)-c1c[nH]c2ncc(cc12)-c1ccccc1)C(F)(F)F 50294542COc1nc(C)cc2N(CCc3ccccc3)CCc3c([nH]c4cc(ccc34)N3CCN(C)CC3)-c12 50296347Nc1ncnc2n(cc(-c3cccc(OCc4ccccc4)c3)c12)[C@H]1C[C@@H](C1)N1CCCC1 50296348Nc1ncnc2n(cc(-c3cccc(OCc4ccccc4)c3)c12)[C@H]1C[C@@H](C1)N1CCC1 50296350Cc1cc(cc2[nH]c(nc12)-c1c(NC[C@@H](O)c2ccccc2Cl)cc[nH]c1=O)N1CCN(CCC#N)CC1 50296351Cc1cc(cc2[nH]c(nc12)-c1c(NC[C@H](O)c2ccccc2Cl)cc[nH]c1=O)N1CCOCC1 50296352CN1CCN(CC1)C1CC(C1)c1c(ccc2ccc(nc12)-c1ccccc1)-c1ncn2ccnc(N)c12 50296353Nc1nccn2cnc(-c3ccc4ccc(nc4c3C3CC(C3)N3CC3)-c3ccccc3)c12 50296354CN1CCN(CC1)c1ccc(cc1)C(=O)Nc1[nH]nc2CCN(Cc12)S(=O)(=O)c1cc(F)cc(F)c1 50296355CN1CCN(CC1)c1ccc(C(=O)Nc2[nH]nc3CCN(Cc23)S(=O)(=O)c2cc(F)cc(F)c2)c(NC(=O)c2ccc[nH]2)c1 50296356CN1CCN(CC1)c1ccc(cc1NC(=O)c1cc[nH]c1)C(=O)Nc1[nH]nc2c1CN(C2(C)C)S(=O)(=O)c1cc(F)cc(F)c1 50296357Oc1ccc(CN(Cc2ccc(O)c(O)c2)c2ccc3OCOc3c2)cc1O 50299138NC(=O)[C@@H]1CCCN1c1nc(Nc2cc([nH]n2)C2CC2)c2cccn2n1 50299139NC(=O)[C@H]1CCCN1c1nc(Nc2cc([nH]n2)C2CC2)c2cccn2n1 50299140O=C(Nc1ccccc1)[C@@H]1CCCN1c1nc(Nc2cc([nH]n2)C2CC2)c2cccn2n1 50299141Cc1ccc(NC(=O)[C@@H]2CCCN2c2nc(Nc3cc([nH]n3)C3CC3)c3cccn3n2)cc1 50299142CN(C(=O)[C@@H]1CCCN1c1nc(Nc2cc([nH]n2)C2CC2)c2cccn2n1)c1ccccc1 50299143O=C(Nc1nccs1)[C@@H]1CCCN1c1nc(Nc2cc([nH]n2)C2CC2)c2cccn2n1 50299144O=C(Nc1cccnc1)[C@@H]1CCCN1c1nc(Nc2cc([nH]n2)C2CC2)c2cccn2n1 50299145C[C@]1(CCCN1c1nc(Nc2cc([nH]n2)C2CC2)c2cccn2n1)C(=O)Nc1nccs1 50299146C[C@]1(CCCN1c1nc(Nc2cc([nH]n2)C2CC2)c2cccn2n1)C(=O)Nc1cccnc1 50299148C[C@]1(CCCN1c1nc(Nc2cc([nH]n2)C2CC2)c2cccn2n1)C(=O)Nc1ccc(F)nc1 50306682C[C@@H](Oc1cc(cnc1N)-c1cnn(c1)C1CCNCC1)c1c(Cl)ccc(F)c1Cl 50308341Brc1cc2OCOc2cc1\C=C1\SC(=O)NC1=O 50308342CCOc1cc(Br)cc(\C=C2/SC(=O)NC2=O)c1O 50308343COc1c(Br)cc(\C=C2/SC(=O)NC2=O)cc1Br 50308344CCOc1cc(\C=C2\SC(=O)NC2=O)cc(Br)c1O 50308345COc1cc(\C=C2\SC(=O)NC2=O)cc(I)c1O 50308346Brc1cccc(c1)-c1ccc(C=C2SC(=O)NC2=O)o1 50308347OC(=O)c1ccc(cc1)-c1ccc(C=C2SC(=S)NC2=O)o1 50308348Brc1ccc(cc1)-c1ccc(C=C2SC(=O)NC2=O)o1 50308349Fc1ccc(cc1)-c1ccc(C=C2SC(=O)NC2=O)o1 50308350Clc1cccc(-c2ccc(C=C3SC(=O)NC3=O)o2)c1Cl 50308351Clc1ccc(-c2ccc(C=C3SC(=O)NC3=O)o2)c(Cl)c1 50308352Cc1ccc(-c2ccc(C=C3SC(=O)NC3=O)o2)c(Br)c1 50308353Fc1ccc(cc1Cl)-c1ccc(C=C2SC(=O)NC2=O)o1 50308354Clc1ccc(cc1Cl)-c1ccc(C=C2SC(=O)NC2=O)o1 50308355OC(=O)c1cc(ccc1O)-c1ccc(C=C2SC(=O)NC2=O)o1 50308357[O-][N+](=O)c1ccccc1-c1ccc(\C=C2/SC(=O)NC2=O)o1 50308358Fc1ccccc1\C=C1/SC(=O)NC1=O 50308360CCC(C)COc1ccccc1\C=C1\SC(=O)NC1=O 50308361Clc1ccc(COc2cccc(\C=C3/SC(=O)NC3=O)c2)c(Cl)c1 50308362[O-][N+](=O)c1cccc(\C=C2\SC(=O)NC2=O)c1 50308365CCOc1cccc(\C=C2\SC(=O)NC2=O)c1O 50308367Clc1ccc(\C=C2\SC(=O)NC2=O)cc1Cl 50308378Cc1ccc(N2CCC(CC2)N2CCN(CC2)C(=O)N2CCOCC2)c2nc([nH]c12)-c1c(N[C@@H](CO)Cc2ccccc2Br)cc[nH]c1=O 50308379CCC(=O)c1cccc(Nc2ccc3C(=O)NC(=O)C(=CNc4ccc(cc4)N4CCN(C)CC4)c3c2)c1 50308380Nc1ncnc2n(nc(-c3ccc4CC(Cc5cccs5)=Cc4c3)c12)[C@H]1CC[C@@H](CC1)N1CCOCC1 50309547COc1cc(cc(OC)c1OC)C1=C(C(=O)NC1=O)c1c[nH]c2ccc(I)cc12 50309548COc1cc(cc(OC)c1OC)C1=C(C(=O)NC1=O)c1c[nH]c2ccc(Br)cc12 50309549COc1cc(cc(OC)c1OC)C1=C(C(=O)NC1=O)c1c[nH]c2ccc(F)cc12 50313554Cc1cc(cc2[nH]c(nc12)-c1c(NCCn2cc(cn2)C(N)=O)cc[nH]c1=O)N1CCOCC1 50313555CN(C)C(=O)c1cnn(CCNc2cc[nH]c(=O)c2-c2nc3c(C)cc(cc3[nH]2)N2CCOCC2)c1 50313556Cc1cc(cc2[nH]c(nc12)-c1c(NCCn2cc(cn2)C(O)=O)cc[nH]c1=O)N1CCOCC1 50313557Cc1cc(cc2[nH]c(nc12)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O)N1CCNCC1 50313558CN1CCN(CC1)c1cc(C)c2nc([nH]c2c1)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O 50313559Cc1cc(cc2[nH]c(nc12)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O)N1CCN(CCF)CC1 50313560Cc1cc(cc2[nH]c(nc12)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O)N1CC[C@@H](N)C1 50313561Cc1cc(cc2[nH]c(nc12)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O)N1CC[C@H](N)C1 50313562Cc1cc(cc2[nH]c(nc12)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O)N1CCC(CC1)NC(=O)OC(C)(C)C 50313563Cc1cc(cc2[nH]c(nc12)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O)N1CC[C@@H](C1)NC(=O)OC(C)(C)C 50313564Cc1cc(cc2[nH]c(nc12)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O)N1CCC(CC1)N1C[C@@H]2C[C@H]1CO2 50313567Cc1cc(cc2[nH]c(nc12)-c1c(NCCn2cc(CO)cn2)cc[nH]c1=O)N1CCOCC1 50313568CNC(=O)c1cnn(CCNc2cc[nH]c(=O)c2-c2nc3c(C)cc(cc3[nH]2)N2CCOCC2)c1 50313647COCCCN1CCC(CC1)[C@H]1CCC(CC1)n1nc(-c2ccc3nc(Cc4ccccc4Cl)[nH]c3c2)c2c(N)ncnc12 50313648COc1ccccc1Cc1nc2ccc(cc2[nH]1)-c1nn(C2CC[C@@H](CC2)C2CCN(C)CC2)c2ncnc(N)c12 50313651Nc1ncnc2n(cc(-c3ccc(OCc4ccccc4)cc3)c12)[C@@H]1C[C@H](CN2CCC2)C1 50315885CCN1CCN(CC1)c1ccc(Nc2nccc(n2)-c2c(nc3sccn23)-c2cccc(NC(=O)Cc3ccccc3)c2)cc1 50315886O=C(Cc1ccccc1)Nc1cccc(c1)-c1nc2sccn2c1-c1ccnc(Nc2ccc3CNCCc3c2)n1 50315887C[C@@]1(O)C[C@@H](C1)c1nc(-c2ccc3ccc(nc3c2)-c2ccccc2)c2c(N)nccn12 50315888O=C(Cc1ccccc1)Nc1cccc(c1)-c1nc2sccn2c1-c1ccnc(Nc2cccc(c2)N2CCOCC2)n1 50315889O=C(CC1CCCCC1)Nc1cccc(c1)-c1nc2sccn2c1-c1ccnc(Nc2ccc(cc2)N2CCOCC2)n1 50315890O=C(CC1CCCC1)Nc1cccc(c1)-c1nc2sccn2c1-c1ccnc(Nc2ccc(cc2)N2CCOCC2)n1 50315891O=C(Nc1ccccc1)Nc1cccc(c1)-c1nc2sccn2c1-c1ccnc(Nc2ccc(cc2)N2CCOCC2)n1 50315892O=C(Nc1cccc(c1)-c1nc2sccn2c1-c1ccnc(Nc2ccc(cc2)N2CCOCC2)n1)Oc1ccccc1 50315893O=C(Cc1ccccc1)Nc1cccc(c1)-c1nc2sccn2c1-c1ccnc(Nc2ccc(cc2)N2CCOCC2)n1 50315894Fc1cccc(F)c1C(=O)Nc1cccc(c1)-c1nc2sccn2c1-c1ccnc(Nc2cccc(c2)N2CCOCC2)n1 50315895CN(C)CCc1ccc(Nc2nccc(n2)-c2c(nc3sccn23)-c2cccc(NC(=O)c3c(F)cccc3F)c2)cc1 50315896CCN1CCN(CC1)c1ccc(Nc2nccc(n2)-c2c(nc3sccn23)-c2cccc(NC(=O)c3c(F)cccc3F)c2)cc1 50315897Fc1cccc(F)c1C(=O)Nc1cccc(c1)-c1nc2sccn2c1-c1ccnc(Nc2ccc3CNCCc3c2)n1 50315898CN1CCc2cc(Nc3nccc(n3)-c3c(nc4sccn34)-c3cccc(NC(=O)Cc4ccccc4)c3)ccc2C1 50315899CN(C)CCc1cccc(Nc2nccc(n2)-c2c(nc3sccn23)-c2cccc(NC(=O)Cc3ccccc3)c2)c1 50315905O=C(Nc1cccc(c1)-c1nc2sccn2c1-c1ccnc(Nc2ccc(cc2)N2CCOCC2)n1)c1ccccc1 50315906Fc1cccc(F)c1C(=O)Nc1cccc(c1)-c1nc2sccn2c1-c1ccnc(Nc2ccc(cc2)N2CCOCC2)n1 50316492CCn1cc(c(n1)-c1ccc(NC(=O)Nc2ccccc2)cc1)-c1ccnc2[nH]ccc12 50316775COc1ccc(cc1)-c1ccc(Cn2cc(CCN)c3cc(OCCc4ccc(O)cc4)ccc23)cc1 50316776NCCc1cn(Cc2ccc(cc2)-c2ccccc2)c2ccc(OCCc3ccc(O)cc3)cc12 50316777NCCc1c[nH]c2ccc(OCCc3ccc(O)cc3)cc12 50316779COc1ccc(CCOc2ccc3n(CCCCCc4ccc(SC)cc4)cc(CCN)c3c2)cc1 50316780CN(C)c1ccc(CCCCCn2c3CCC(N)Cc3c3cc(OCCc4ccc(O)cc4)ccc23)cc1 50316781COc1ccc(CCCCCn2c3CCC(N)Cc3c3cc(OCCc4ccc(O)cc4)ccc23)cc1 50316782NC1CCc2c(C1)c1cc(OCCc3ccc(O)cc3)ccc1n2CCCCCc1ccc(cc1)C(F)(F)F 50316783NC1CCc2c(C1)c1cc(OCCc3ccc(O)cc3)ccc1n2CCCCCc1ccccn1 50316784NC1CCc2c(C1)c1cc(OCCc3ccc(O)cc3)ccc1n2CCCc1ccccc1 50316787NCCc1cn(CCCCCc2ccccc2)c2ccc(OCCc3ccc(O)cc3)cc12 50316788NC1CCc2c(C1)c1cc(OCCc3ccc(O)cc3)ccc1n2CCCCCc1ccccc1 50316790COc1ccc(CCCCCn2cc(CCN)c3cc(OCCc4ccc(O)cc4)ccc23)cc1 50316791CSc1ccc(CCCCCn2cc(CCN)c3cc(OCCc4ccc(O)cc4)ccc23)cc1 50316792NCCc1cn(Cc2ccc(cc2)-c2cccc(c2)C(F)(F)F)c2ccc(OCCc3ccc(O)cc3)cc12 50318107CNC(=O)CN1CCN(CC1)c1cc(C)c2nc([nH]c2c1)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O 50318108Cc1cc(cc2[nH]c(nc12)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O)N1CCN(CC(=O)NCCF)CC1 50318109Cc1cc(cc2[nH]c(nc12)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O)N1CCN(CCCF)CC1 50318110Cc1cc(cc2[nH]c(nc12)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O)N1CCN(CC#N)CC1 50318111Cc1cc(cc2[nH]c(nc12)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O)N1CCN(CCC#N)CC1 50318112COCCN1CCN(CC1)c1cc(C)c2nc([nH]c2c1)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O 50318113CCN1CCN(CC1)c1cc(C)c2nc([nH]c2c1)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O 50318114CC(=O)N1CCN(CC1)c1cc(C)c2nc([nH]c2c1)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O 50318115COCC(=O)N1CCN(CC1)c1cc(C)c2nc([nH]c2c1)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O 50318116Cc1cc(cc2[nH]c(nc12)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O)N1CCN(CC1)C(=O)CCCF 50318117Cc1cc(cc2[nH]c(nc12)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O)N1CCN(CC1)C(=O)OC(C)(C)C 50318118COC(=O)N1CCN(CC1)c1cc(C)c2nc([nH]c2c1)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O 50318119CCOC(=O)N1CCN(CC1)c1cc(C)c2nc([nH]c2c1)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O 50318120Cc1cc(cc2[nH]c(nc12)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O)N1CCN(CC1)S(C)(=O)=O 50318121Cc1cc(cc2[nH]c(nc12)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O)N1CCN(CCO)CC1 50318122Cc1cc(cc2[nH]c(nc12)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O)N1CCN(CCCO)CC1 50325424Fc1ccc(NC(=O)[C@@H]2CCCN2c2nc(Nc3cc([nH]n3)C3CC3)c3cccn3n2)cn1 50325425Fc1ccc(cn1)C(=O)N1CCC[C@H]1c1nc(Nc2cc(n[nH]2)C2CC2)c2cccn2n1 50325426Fc1ccc(cn1)C(=O)N1CCC[C@@H]1c1nc(Nc2cc(n[nH]2)C2CC2)c2cccn2n1 50325427Fc1ccc(cn1)C(=O)N1[C@@H](CCC1=O)c1nc(Nc2cc(n[nH]2)C2CC2)c2cccn2n1 50325428Fc1ccc(NC(=O)[C@@H]2CCC[C@H]2c2nc(Nc3cc(n[nH]3)C3CC3)c3cccn3n2)cn1 50325429Fc1ccc(NC(=O)C2=C(CCC2)c2nc(Nc3cc(n[nH]3)C3CC3)c3cccn3n2)cn1 50325430Fc1ccc(cn1)C(=O)NCc1nc(Nc2cc(n[nH]2)C2CC2)c2cccn2n1 50326003Oc1ccc(CNc2ccc3OCOc3c2)cc1O 50326004Oc1ccc(CNc2ccc3cn[nH]c3c2)cc1O 50326005Oc1ccc(CN(Cc2ccc(O)c(O)c2)c2ccc3cn[nH]c3c2)cc1O 50326006Oc1ccc(CNc2ccc3ccccc3c2)cc1O 50326007Oc1ccc(CN(Cc2ccc(O)c(O)c2)c2ccc3ccccc3c2)cc1O 50326008CC(=O)Oc1ccc(CNc2ccc3OCOc3c2)cc1OC(C)=O 50326801Cc1cncc(Oc2ccc(NC(=O)Nc3cc(C)nc4ccccc34)cc2)n1 50326802COc1ccc(Cl)cc1NC(=O)Nc1cc(nc2ccccc12)C(F)(F)F 50326803COc1ccc(NC(=O)Nc2cc(nc3ccccc23)C(F)(F)F)cc1Cl 50326806FC(F)(F)Oc1ccc(NC(=O)Nc2cc(nc3ccccc23)C(F)(F)F)cc1 50326811Cc1cncc(Oc2ccc(NC(=O)Nc3cc(nc4ccccc34)C(F)(F)F)cc2)n1 50326820COc1ccc(Cl)cc1NC(=O)Nc1cc(=O)[nH]c2ccccc12 50327947CN1CCN(CC1)[C@H]1CC[C@@H](CC1)n1nc(-c2ccc(Nc3nc4cccc(Cl)c4o3)c(F)c2)c2c(N)ncnc12 50327948CN1CCN(CC1)[C@H]1CC[C@@H](CC1)n1nc(-c2ccc(Nc3nc4cccc(Cl)c4o3)cc2)c2c(N)ncnc12 50327949CN1CCN(CC1)[C@H]1CC[C@@H](CC1)n1nc(-c2ccc(Nc3nc4cccc(Cl)c4o3)cc2C)c2c(N)ncnc12 50327950CN1CCN(CC1)[C@H]1CC[C@@H](CC1)n1nc(-c2ccc(Nc3nc4cccc(Cl)c4o3)cc2Cl)c2c(N)ncnc12 50327951CN1CCN(CC1)[C@H]1CC[C@@H](CC1)n1nc(-c2ccc(Nc3nc4cccc(Cl)c4o3)c(Cl)c2)c2c(N)ncnc12 50327952COCCCN1CCC(CC1)N1CCC(CC1)n1nc(-c2ccc(Nc3nc4cccc(Cl)c4o3)cc2)c2c(N)ncnc12 50327953CC(C)N1CCC(CC1)N1CCC(CC1)n1nc(-c2ccc(Nc3nc4cccc(Cl)c4o3)cc2)c2c(N)ncnc12 50327954CN1CCC(CC1)N1CCC(CC1)n1nc(-c2ccc(Nc3nc4cccc(Cl)c4o3)cc2)c2c(N)ncnc12 50327955CN(C)C(=O)CN1CCN(CC1)[C@H]1CC[C@@H](CC1)n1nc(-c2ccc(Nc3nc4cccc(Cl)c4o3)cc2)c2c(N)ncnc12 50327956COCCCN1CCN(CC1)[C@H]1CC[C@H](CC1)n1nc(-c2ccc(Nc3nc4cccc(Cl)c4o3)cc2)c2c(N)ncnc12 50327957COCCCN1CCN(CC1)[C@H]1CC[C@@H](CC1)n1nc(-c2ccc(Nc3nc4cccc(Cl)c4o3)cc2)c2c(N)ncnc12 50327958CC(C)N1CCN(CC1)[C@H]1CC[C@H](CC1)n1nc(-c2ccc(Nc3nc4cccc(Cl)c4o3)cc2)c2c(N)ncnc12 50327959CC(C)N1CCN(CC1)[C@H]1CC[C@@H](CC1)n1nc(-c2ccc(Nc3nc4cccc(Cl)c4o3)cc2)c2c(N)ncnc12 50327960Nc1ncnc2n(nc(-c3ccc(Nc4nc5cccc(Cl)c5o4)cc3)c12)[C@H]1CC[C@@H](CC1)N1CCOCC1 50327961CN1CCN(CC1)[C@H]1CC[C@H](CC1)n1nc(-c2ccc(Nc3nc4cc(C)cc(Cl)c4o3)cc2)c2c(N)ncnc12 50327962CN1CCN(CC1)[C@H]1CC[C@H](CC1)n1nc(-c2ccc(Nc3nc4cccc(Cl)c4o3)c(F)c2)c2c(N)ncnc12 50327963CN1CCN(CC1)[C@H]1CC[C@H](CC1)n1nc(-c2ccc(Nc3nc4cccc(Cl)c4o3)cc2)c2c(N)ncnc12 50327964CN1CCN(CC1)[C@H]1CC[C@H](CC1)n1cc(-c2ccc(Nc3nc4cc(C)cc(Br)c4o3)c(F)c2)c2c(N)ncnc12 50327965CN1CCN(CC1)[C@H]1CC[C@H](CC1)n1nc(-c2ccc(Nc3nc4cc(C)cc(C)c4o3)c(F)c2)c2c(N)ncnc12 50327966CN1CCN(CC1)[C@H]1CC[C@@H](CC1)n1nc(-c2ccc(Nc3nc4cccc(Cl)c4o3)c(C)c2)c2c(N)ncnc12 50327967CN1CCN(CC1)[C@H]1CC[C@H](CC1)n1nc(-c2ccc(Nc3nc4cc(Cl)cc(Cl)c4o3)cc2)c2c(N)ncnc12 50327968CN1CCN(CC1)[C@H]1CC[C@H](CC1)n1nc(-c2ccc(Nc3nc4cc(Cl)ccc4o3)c(F)c2)c2c(N)ncnc12 50327969COC(=O)c1cccc2nc(Nc3ccc(cc3)-c3nn([C@@H]4CC[C@@H](CC4)N4CCN(C)CC4)c4ncnc(N)c34)oc12 50327970CN1CCN(CC1)[C@H]1CC[C@H](CC1)n1nc(-c2ccc(Nc3nc4cccc(C#N)c4o3)cc2)c2c(N)ncnc12 50327971CN1CCN(CC1)[C@H]1CC[C@H](CC1)n1nc(-c2ccc(Nc3nc4ccccc4o3)cc2)c2c(N)ncnc12 50331612COc1ccc(CNc2ccnc3oc4ccccc4c23)cc1 50331613Clc1ccc(CNc2ccnc3oc4ccccc4c23)cc1 50331615Clc1cccc(CNc2ccnc3oc4ccccc4c23)c1 50331616C(Nc1ccnc2oc3ccccc3c12)c1cccc2ccccc12 50331617C(Cc1ccccc1)Nc1ccnc2oc3ccccc3c12 50331618C(Nc1ccnc2oc3ccccc3c12)c1ccccc1 50332294Cc1cnc(Nc2ccc(OCCN3CCCC3)cc2)nc1Nc1cccc(c1)S(=O)(=O)NC(C)(C)C 50336315Nc1nccn2c(nc(-c3ccc4ccc(nc4c3F)-c3ccccc3)c12)[C@H]1CC[C@@H](CC1)C(=O)Nc1nc2ccccc2[nH]1 50336316Nc1nccn2c(nc(-c3ccc4ccc(nc4c3)-c3ccccc3)c12)[C@@H]1C[C@H](CN2CCC2)C1 50336317C[C@@]1(O)C[C@@H](C1)c1nc(-c2ccc3ccc(nc3c2F)-c2ccccc2)c2c(N)ncnn12 50336318Nc1nccn2c(nc(-c3ccc4ccc(nc4c3F)-c3ccccc3)c12)[C@H]1CC[C@H](CO)CC1 50336319Nc1nccn2c(nc(-c3ccc4ccc(nc4c3F)-c3ccccc3)c12)[C@H]1CC[C@@H](CC1)C(O)=O 50336320CN(C)C(=O)[C@H]1CC[C@@H](CC1)c1nc(-c2ccc3ccc(nc3c2F)-c2ccccc2)c2c(N)nccn12 50336321CNC(=O)[C@H]1CC[C@@H](CC1)c1nc(-c2ccc3ccc(nc3c2F)-c2ccccc2)c2c(N)nccn12 50336322NC(=O)[C@H]1CC[C@@H](CC1)c1nc(-c2ccc3ccc(nc3c2F)-c2ccccc2)c2c(N)nccn12 50336323Nc1nccn2c(nc(-c3ccc4ccc(nc4c3F)-c3ccccc3)c12)[C@H]1CC[C@@H](CC1)C(=O)Nc1nncs1 50336324Nc1nccn2c(nc(-c3ccc4ccc(nc4c3F)-c3ccccc3)c12)[C@H]1CC[C@@H](CC1)C(=O)Nc1ccn[nH]1 50336325Nc1nccn2c(nc(-c3ccc4ccc(nc4c3F)-c3ccccc3)c12)[C@H]1CC[C@@H](CC1)C(=O)Nc1nccs1 50336326Nc1nccn2c(nc(-c3ccc4ccc(nc4c3F)-c3ccccc3)c12)[C@H]1CC[C@@H](CC1)C(=O)Nc1nnc[nH]1 50336327Nc1nccn2c(nc(-c3ccc4ccc(nc4c3F)-c3ccccc3)c12)[C@H]1CC[C@@H](CC1)C(=O)Nc1ccccn1 50336328Nc1nccn2c(nc(-c3ccc4ccc(nc4c3F)-c3ccccc3)c12)[C@H]1CC[C@@H](CC1)C(=O)Nc1ccncn1 50336329Nc1ccccc1NC(=O)[C@H]1CC[C@@H](CC1)c1nc(-c2ccc3ccc(nc3c2F)-c2ccccc2)c2c(N)nccn12 50336330Nc1nccn2c(nc(-c3ccc4ccc(nc4c3F)-c3ccccc3)c12)[C@H]1CC[C@@H](CC1)C(=O)Nc1ccc2[nH]ccc2c1 50336331Cn1c(NC(=O)[C@H]2CC[C@@H](CC2)c2nc(-c3ccc4ccc(nc4c3F)-c3ccccc3)c3c(N)nccn23)nc2ccccc12 50338873COc1ccc(Cn2ncc(NC(=O)c3cc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)ccc3C)c2N)cc1 50339058Nc1ncnn2c(nc(-c3ccc4ccc(nc4c3)-c3ccccc3)c12)C1CCC1 50339059Nc1nccn2c(nc(-c3ccc4ccc(nc4c3)-c3ccccc3)c12)C1CCC1 50339060C[C@@]1(O)C[C@@H](C1)c1nc(-c2ccc3ccc(nc3c2)-c2ccccc2)c2c(N)ncnn12 50339061Nc1ncnn2c(nc(-c3ccc4ccc(nc4c3)-c3ccccc3)c12)[C@@H]1C[C@@H](C1)N1CCN(CC1)C=O 50339062Nc1ncnn2c(nc(-c3ccc4ccc(nc4c3F)-c3ccccc3)c12)[C@@H]1C[C@@H](C1)N1CCN(CC1)C=O 50339063CN1CCN(CC1)[C@H]1C[C@H](C1)c1nc(-c2ccc3ccc(nc3c2)-c2ccccc2)c2c(N)ncnn12 50339064CN1CCN(CC1)[C@H]1C[C@H](C1)c1nc(-c2ccc3ccc(nc3c2F)-c2ccccc2)c2c(N)ncnn12 50340118COc1cc(Nc2nccc(Nc3cccc(OC(F)(F)F)c3)n2)cc(OC)c1OC 50340119COc1cc(Nc2ncnc(Nc3cnc4ccccc4c3)n2)cc(OC)c1OC 50340120COc1cc(Nc2ncnc(Nc3ccc4ccccc4c3)n2)cc(OC)c1OC 50340121COc1cc(Nc2nccc(Nc3cnc4ccccc4c3)n2)cc(OC)c1OC 50340122COc1cc(Nc2nccc(Nc3ccc4ccccc4c3)n2)cc(OC)c1OC 50340123COc1cc(Nc2nccc(Nc3cc4ccccc4nc3C)n2)cc(OC)c1OC 50340124COc1cc(Nc2nccc(n2)N(C)c2cnc3ccccc3c2)cc(OC)c1OC 50340125COc1cc(Nc2nccc(Oc3cnc4ccccc4c3)n2)cc(OC)c1OC 50340126COc1cc(Nc2nccc(Nc3cnc4ccccc4c3)n2)ccc1N1CCOCC1 50340127COc1cc(Nc2nccc(Nc3cc4ccccc4cn3)n2)cc(OC)c1OC 50340128COc1cc(Nc2nccc(Nc3ccc4ncccc4c3)n2)cc(OC)c1OC 50340129COc1cc(Nc2nccc(Nc3ccc4nccnc4c3)n2)cc(OC)c1OC 50340130COc1cc(Nc2nccc(Nc3ccc4cn[nH]c4c3)n2)cc(OC)c1OC 50340131COc1cc(Nc2nccc(Nc3ccc4[nH]ncc4c3)n2)cc(OC)c1OC 50340132COc1cc(Nc2nccc(Nc3ccc4nc[nH]c4c3)n2)cc(OC)c1OC 50340133COc1cc(Nc2nccc(Nc3ccc4c(NCC4(C)C)c3)n2)cc(OC)c1OC 50340134COc1cc(Nc2nccc(Nc3ccccn3)n2)cc(OC)c1OC 50340135COc1ccc(Nc2nccc(Nc3cnc4ccccc4c3)n2)cc1OC 50340136COc1cc(Nc2nccc(Nc3cnc4ccccc4c3)n2)cc(OC)c1 50340137COc1ccc(Nc2nccc(Nc3cnc4ccccc4c3)n2)cc1 50340138COc1cccc(Nc2nccc(Nc3cnc4ccccc4c3)n2)c1 50340139FC(F)(F)Oc1cccc(Nc2nccc(Nc3cnc4ccccc4c3)n2)c1 50340140Clc1cccc(Nc2nccc(Nc3cnc4ccccc4c3)n2)c1 50340141COc1ccc(Nc2nccc(Nc3cnc4ccccc4c3)n2)cc1Cl 50340142C1CN(CCO1)c1ccc(Nc2nccc(Nc3cnc4ccccc4c3)n2)cc1 50340143C(COc1ccc(Nc2nccc(Nc3cnc4ccccc4c3)n2)cc1)CN1CCCCC1 50340144COc1cc(Nc2nccc(Nc3cnc4ccccc4c3)n2)ccc1OCCCN1CCCCC1 50340484Cc1c(O)n(-c2ccc(cc2)S(=O)(=O)C(F)(F)F)c(=O)n1Cc1ccnc2ccccc12 50340486CC1(C)N(Cc2ccnc(NS(C)(=O)=O)c2)C(=O)N(C1=O)c1ccc(SC(F)(F)F)cc1 50340487CN(C)c1cc(CN2C(=O)N(C(=O)C2(C)C)c2ccc(SC(F)(F)F)cc2)ccn1 50340488CC1(C)N(Cc2ccnc(c2)C(N)=O)C(=O)N(C1=O)c1ccc(SC(F)(F)F)cc1 50340489CC1(C)N(Cc2ccnc(F)c2)C(=O)N(C1=O)c1ccc(SC(F)(F)F)cc1 50340490CCOc1cc(CN2C(=O)N(C(=O)C2(C)C)c2ccc(SC(F)(F)F)cc2)ccn1 50340491CC1(C)N(Cc2ccnc(NC3CCCCC3)c2)C(=O)N(C1=O)c1ccc(SC(F)(F)F)cc1 50340492COc1ccc(CNc2cc(CN3C(=O)N(C(=O)C3(C)C)c3ccc(SC(F)(F)F)cc3)ccn2)cc1 50340493CC1(C)N(Cc2ccnc(Nc3ccccc3)c2)C(=O)N(C1=O)c1ccc(SC(F)(F)F)cc1 50340494CC1(C)N(Cc2ccnc(NCc3ccccc3)c2)C(=O)N(C1=O)c1ccc(SC(F)(F)F)cc1 50340495CC1(C)N(Cc2ccnc(Cl)c2)C(=O)N(C1=O)c1ccc(SC(F)(F)F)cc1 50340496CC(C)(C)OC(=O)Nc1cc(CN2C(=O)N(C(=O)C2(C)C)c2ccc(SC(F)(F)F)cc2)ccn1 50340497CNC(=O)c1cc(CN2C(=O)N(C(=O)C2(C)C)c2ccc(SC(F)(F)F)cc2)ccn1 50340498CCc1cc(CN2C(=O)N(C(=O)C2(C)C)c2ccc(SC(F)(F)F)cc2)ccn1 50340499CC(C)Nc1cc(CN2C(=O)N(C(=O)C2(C)C)c2ccc(SC(F)(F)F)cc2)ccn1 50340500CNc1cc(CN2C(=O)N(C(=O)C2(C)C)c2ccc(SC(F)(F)F)cc2)ccn1 50340501CCNc1cc(CN2C(=O)N(C(=O)C2(C)C)c2ccc(SC(F)(F)F)cc2)ccn1 50340502CC(=O)Nc1cc(CN2C(=O)N(C(=O)C2(C)C)c2ccc(SC(F)(F)F)cc2)ccn1 50340503CC1(C)N(Cc2ccnc(N)c2)C(=O)N(C1=O)c1ccc(SC(F)(F)F)cc1 50340504Cc1c(O)n(-c2ccc(cc2)S(=O)(=O)C(F)(F)F)c(=O)n1Cc1ccncc1 50340513COc1cc2c(cn(C)c2cc1OC)-c1cc2cccnc2[nH]1 50340514CC1(C)N(Cc2ccncc2)C(=O)N(C1=O)c1ccc(SC(F)(F)F)cc1 50340515Cc1c(O)n(-c2ccc(cc2)S(=O)C(F)(F)F)c(=O)n1Cc1ccnc2ccccc12 50340516Cc1c(O)n(-c2ccc(SC(F)(F)F)cc2)c(=O)n1Cc1ccnc2ccccc12 50340518Oc1cn(Cc2ccnc3ccccc23)c(=O)n1-c1ccc(cc1)S(=O)(=O)C(F)(F)F 50340520CC1(C)N(Cc2ccnc3ccccc23)C(=O)N(C1=O)c1ccc(cc1)S(=O)(=O)C(F)(F)F 50340954CC(=O)NC[C@H]1CC[C@@H](CC1)c1nc(-c2cc3ccccc3[nH]2)c2c(N)nccn12 50344664CC1(C)c2[nH]c3cc(ccc3c2C(=O)c2ccc(cc12)C1CCN(CC1)C1COC1)C#N 50346827CC(C)(C)c1ccc(cc1)C(=O)NNC(=O)C(=O)c1c[nH]c2ccccc12 50346828FC(F)(F)c1ccc(cc1)C(=O)NNC(=O)C(=O)c1c[nH]c2ccccc12 50346830Ic1ccc(cc1)C(=O)NNC(=O)C(=O)c1c[nH]c2ccccc12 50346832Cc1ccc(C)n1-c1ccc(cc1)C(=O)NNC(=O)C(=O)c1c[nH]c2ccccc12 50346835Fc1ccc(COc2ccccc2-c2ccc(cc2)C(=O)NNC(=O)C(=O)c2c[nH]c3ccccc23)cc1 50346836FC(F)(F)c1cccc(OCc2ccccc2-c2ccc(cc2)C(=O)NNC(=O)C(=O)c2c[nH]c3ccccc23)c1 50346837FC(F)(F)c1cccc(OCc2cccc(c2)-c2ccc(cc2)C(=O)NNC(=O)C(=O)c2c[nH]c3ccccc23)c1 50346838Cc1cc(ccc1OCc1cccc(c1)-c1ccc(cc1)C(=O)NNC(=O)C(=O)c1c[nH]c2ccccc12)C(C)(C)C 50346839CS(=O)(=O)NCc1cccc(c1)-c1ccc(cc1)C(=O)NNC(=O)C(=O)c1c[nH]c2ccccc12 50346843COCCc1ccc(OCc2cccc(c2)-c2ccc(cc2)C(=O)NNC(=O)C(=O)c2c[nH]c3ccccc23)cc1 50349687COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12)N1CCN(CC1)C(C)=O 50349688COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12)C1CCN(CC1)C(C)=O 50349689COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12)C1CCNCC1 50349690COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12)N1CCNC(=O)C1 50349691COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12)N1CCCN(CC1)C(C)=O 50349692COc1cc(OC2CCN(CC2)C(C)=O)ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12 50349693COc1cc(OC2CCNCC2)ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12 50349694COc1cc(OC2CN(C2)C(C)=O)ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12 50349695COc1cc(OC2CNC2)ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12 50349696COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12)N1CCOCC1 50349697COC(=O)N1CCN(CC1)c1ccc(Nc2ncc(Cl)c(n2)-c2cnc3ccccn23)c(OC)c1 50349698COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12)N1CCN(CC1)C(N)=O 50349699COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12)N1CCN(CC1)C(=O)N(C)C 50349700COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12)N1CCN(CC1)C(=O)CO 50349701COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12)N1CCN(CC1)C(=O)[C@H](C)O 50349702COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12)N1CCN(CC1)C(=O)[C@@H](C)O 50349703COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12)N1CCN(CC1)C(=O)CN 50349704CNCC(=O)N1CCN(CC1)c1ccc(Nc2ncc(Cl)c(n2)-c2cnc3ccccn23)c(OC)c1 50349705COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12)N1CCN(CC1)C(=O)[C@H](C)N 50349706COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12)N1CCN(CC1)C(=O)[C@@H](C)N 50349707COc1ccc(cc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12)N1CCN(CC1)C(C)=O 50349708COc1ccc(cc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12)N1CCNCC1 50349709COc1ccc(cc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12)N1CCOCC1 50349710COc1ccc(cc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12)C(=O)N1CCOCC1 50349711COc1cc(CN2CCOCC2)ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12 50349712COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12)C(=O)N1CCOCC1 50349713COc1cc(CC(=O)N2CCOCC2)ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12 50349714COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12)C(CO)CO 50349715COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12)N1CC2CNCC(C1)O2 50349716COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12)N1CC2CN(CCO)CC(C1)O2 50349717COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12)N1CC2COCC(C1)N2 50349718COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12)N1CCNCC1 50349719COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12)N1CCN(CCO)CC1 50349720COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12)N1CCN(CC(=O)N(C)C)CC1 50349721COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12)N1CCN(CCS(C)(=O)=O)CC1 50349722COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccccn12)N1CCN(CC1)S(C)(=O)=O 50349764COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2cc(ccn12)N1CCCC1)N1CCN(CC1)C(C)=O 50349765COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccc(F)cn12)N1CCN(CC1)C(C)=O 50349766COc1ccc2ncc(-c3nc(Nc4ccc(cc4OC)N4CCN(CC4)C(C)=O)ncc3Cl)n2c1 50349767COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccc(cn12)C#N)N1CCN(CC1)C(C)=O 50349768COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccc(cn12)N(C)C)N1CCN(CC1)C(C)=O 50349769COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2c(F)cc(F)cn12)N1CCN(CC1)C(C)=O 50349770CC(=O)N1CCN(CC1)c1ccc(Nc2nccc(n2)-c2cnc3ccccn23)cc1 50349771COc1cc(ccc1Nc1nccc(n1)-c1cnc2ccccn12)N1CCN(CC1)C(C)=O 50349772COc1cc(ccc1Nc1ncc(F)c(n1)-c1cnc2ccccn12)N1CCN(CC1)C(C)=O 50349773COc1cc(ccc1Nc1ncc(Br)c(n1)-c1cnc2ccccn12)N1CCN(CC1)C(C)=O 50349774COc1cc(ccc1Nc1ncc(C)c(n1)-c1cnc2ccccn12)N1CCN(CC1)C(C)=O 50349775COc1cc(ccc1Nc1ncc(c(n1)-c1cnc2ccccn12)C(F)(F)F)N1CCN(CC1)C(C)=O 50349776COc1cc(ccc1Nc1ncc(OC)c(n1)-c1cnc2ccccn12)N1CCN(CC1)C(C)=O 50349777COc1cc(ccc1Nc1ncc(C#N)c(n1)-c1cnc2ccccn12)N1CCN(CC1)C(C)=O 50349778COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2c(F)cccn12)N1CCN(CC1)C(C)=O 50349779COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2c(C)cccn12)N1CCN(CC1)C(C)=O 50349780COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2c(OC)cccn12)N1CCN(CC1)C(C)=O 50349781COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2c(N)cccn12)N1CCN(CC1)C(C)=O 50349782COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2c(CO)cccn12)N1CCN(CC1)C(C)=O 50349783COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2cc(F)ccn12)N1CCN(CC1)C(C)=O 50349784COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2cc(C)ccn12)N1CCN(CC1)C(C)=O 50349785COc1ccn2c(cnc2c1)-c1nc(Nc2ccc(cc2OC)N2CCN(CC2)C(C)=O)ncc1Cl 50349786COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2cc(CO)ccn12)N1CCN(CC1)C(C)=O 50349787COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2cc(ccn12)C#N)N1CCN(CC1)C(C)=O 50349788COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2cc(Cl)ccn12)N1CCN(CC1)C(C)=O 50349789COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2ccc(C)cn12)N1CCN(CC1)C(C)=O 50349790COc1cc(ccc1Nc1ncc(Cl)c(n1)-c1cnc2c(cccn12)C#N)N1CCN(CC1)C(C)=O 50350424Cc1c(O)c(O)cc2oc3cc(O)cc(O)c3c(=O)c12 50355496O=C(N1CCNCC1)c1ccc(\C=C\c2n[nH]c3ccccc23)cc1 50355499CN(C)CC(=O)N1CCC(CC1)c1ccc(NC(=O)c2ncc([nH]2)C#N)c(c1)C1=CCCCC1 50355502CN(C(=O)CN1CCN(C)CC1)c1ccc(cc1)N=C(C1C(=O)Nc2ccccc12)c1ccccc1 50355504COc1cc2c(Oc3ccc(NC(=O)C4(CC4)C(=O)NC4=CCC(F)C=C4)cc3F)ccnc2cc1OCCCN1CCOCC1 50358243CC(C)C\C=C\[C@@H](C)[C@H]1CC[C@H]2[C@H](CCc3cc(O)ccc3C)[C@@H](O)CC[C@]12C 50358244CC(C)C\C=C\[C@@H](C)[C@H]1CC[C@H]2[C@H](CCc3cc(O)ccc3C)C(=O)CC[C@]12C 50358245CC(C)C(=C)CC[C@@H](C)[C@H]1CC[C@H]2[C@H](CCc3cc(O)ccc3C)C(=O)CC[C@]12C 50358246CC(C)CCC[C@@H](C)[C@H]1CC[C@H]2[C@H](CCc3cc(O)ccc3C)C(=O)CC[C@]12C 50358247CC(C)CCC[C@@H](C)[C@H]1CC[C@H]2[C@H](CCc3cc(O)ccc3C)[C@H](O)CC[C@]12C 50375330Nc1nccn2c(nc(-c3ccc4ccc(nc4c3)-c3ccccc3)c12)[C@@H]1C[C@@H](C1)N1CCCCC1 50375331Nc1nccn2c(nc(-c3ccc4ccc(nc4c3)-c3ccccc3)c12)[C@H]1C[C@H](CN2CCOCC2)C1 50375332Nc1nccn2c(nc(-c3ccc4ccc(nc4c3)-c3ccccc3)c12)[C@@H]1C[C@@H](C1)N1CCC1 50375333CN(C)[C@H]1C[C@H](C1)c1nc(-c2ccc3ccc(nc3c2)-c2ccccc2)c2c(N)nccn12 50375334Nc1nccn2c(nc(-c3ccc4ccc(nc4c3)-c3ccccc3)c12)[C@@H]1C[C@H](CN2CCOCC2)C1 50375335Nc1nccn2c(nc(-c3ccc4ccc(nc4c3)-c3ccccc3)c12)[C@H]1C[C@H](CN2CCC2)C1 50375336CN(C)C[C@H]1C[C@@H](C1)c1nc(-c2ccc3ccc(nc3c2)-c2ccccc2)c2c(N)nccn12 50375337CN(C)C[C@H]1C[C@H](C1)c1nc(-c2ccc3ccc(nc3c2)-c2ccccc2)c2c(N)nccn12 50375338Cc1nc(-c2ccc3ccc(nc3c2)-c2ccccc2)c2c(N)nccn12 50375339Nc1nccn2c(nc(-c3ccc4ccc(nc4c3)-c3ccccc3)c12)[C@@H]1C[C@@H](C1)N1CCOCC1 50375340Nc1nccn2c(nc(-c3ccc4ccc(nc4c3)-c3ccccc3)c12)[C@@H]1C[C@@H](C1)N1CCSCC1 50375341Nc1nccn2c(nc(-c3ccc4ccc(nc4c3)-c3ccccc3)c12)[C@@H]1C[C@@H](C1)N1CCCC1 50378022COc1cc(ccc1Nc1nc(-n2[nH]c(=O)c3ccccc23)c2cc[nH]c2n1)N1CCN(CC1)C(C)C 50378023COc1cc(ccc1Nc1nc(N2CCc3ccccc23)c2cc[nH]c2n1)N1CCN(CC1)C(C)C 50378024COc1cc(ccc1Nc1nc(Nc2ccsc2C(N)=O)c2cc[nH]c2n1)N1CCC(CC1)N1CCN(CC1)S(C)(=O)=O 50378035O=C(Nc1cccc(c1)-c1c[nH]c2ncc(cc12)-c1ccoc1)Nc1ccccc1Oc1ccccc1 50381716Nc1ncc(-c2cnn(CCO)c2)c2scc(-c3ccc(NC(=O)Nc4cccc(F)c4)cc3)c12 50382640COc1cccc(Nc2nccc(n2)N2CCC[C@@H](C2)C(=O)NCc2ccc(C)cc2)c1 50382646COc1cc(Nc2nccc(n2)N2CCC[C@@H](C2)C(=O)NCc2ccc(C)cc2)cc(OC)c1OC 50382649COc1cc(Nc2nccc(n2)N2CCC[C@@H](C2)C(=O)NCc2cccc(Oc3ccccc3)c2)cc(OC)c1OC 50382651COc1cc(Nc2nccc(n2)N2CCC[C@@H](C2)C(=O)NCc2cccc(c2)-c2ccccc2)cc(OC)c1OC 50382653COC(=O)c1cccc(CNC(=O)[C@H]2CCCN(C2)c2ccnc(Nc3cc(OC)c(OC)c(OC)c3)n2)c1 50382655COc1cc(Nc2nccc(n2)N2CCC[C@@H](C2)C(=O)NCc2cccc(c2)[N+]([O-])=O)cc(OC)c1OC 50382656COc1cc(Nc2nccc(n2)N2CCC[C@@H](C2)C(=O)NCc2ccc(Cl)cc2)cc(OC)c1OC 50382657COc1cc(Nc2nccc(n2)N2CCC[C@@H](C2)C(=O)NCc2cccc(Cl)c2)cc(OC)c1OC 50382658COc1cc(Nc2nccc(n2)N2CCC[C@@H](C2)C(=O)NCc2ccccc2Cl)cc(OC)c1OC 50382659COc1cc(Nc2nccc(n2)N2CCC[C@@H](C2)C(=O)NCc2ccc(OC(F)(F)F)cc2)cc(OC)c1OC 50382660COc1cc(Nc2nccc(n2)N2CCC[C@@H](C2)C(=O)NCc2cccc(OC(F)(F)F)c2)cc(OC)c1OC 50382661COc1cc(Nc2nccc(n2)N2CCC[C@@H](C2)C(=O)NCc2cccc(C)c2)cc(OC)c1OC 50382662COc1cc(Nc2nccc(n2)N2CCC[C@@H](C2)C(=O)NCc2ccccc2C)cc(OC)c1OC 50382665COc1cc(Nc2nccc(n2)N2CCC[C@@H](C2)C(=O)NCC(=O)c2ccccc2)cc(OC)c1OC 50382666COc1cc(Nc2nccc(n2)N2CCC[C@@H](C2)C(=O)NCCCc2ccccc2)cc(OC)c1OC 50382668COc1cc(Nc2nccc(n2)N2CCC[C@@H](C2)C(=O)NCc2ccccc2)cc(OC)c1OC 50382669COc1cc(Nc2nccc(n2)N2CCC[C@@H](C2)C(=O)Nc2ccccc2)cc(OC)c1OC 50382670COc1cc(Nc2nccc(n2)N2CCC[C@@H](C2)C(=O)NCc2ccc(C)cc2)cc(OC)c1 50383168COc1ccc2c(Oc3ccc(NC(=O)c4c(-c5ccccn5)n(C)n(-c5ccccc5)c4=O)nc3)ccnc2c1 50383169COc1ccc2c(Oc3ccc(NC(=O)c4c(-c5ccncc5)n(C)n(-c5ccccc5)c4=O)nc3)ccnc2c1 50383170COc1ccc2c(Oc3ccc(NC(=O)c4c(C5CCOCC5)n(C)n(-c5ccccc5)c4=O)nc3)ccnc2c1 50383171COc1ccc2c(Oc3ccc(NC(=O)c4c(C5CCOCC5)n(C)n(-c5ccccc5)c4=O)cc3F)ccnc2c1 50383172COc1ccc2c(Oc3ccc(NC(=O)c4c(C5CCOC5)n(C)n(-c5ccccc5)c4=O)cc3F)ccnc2c1 50383173COc1ccc2c(Oc3ccc(NC(=O)c4c(C5CCCO5)n(C)n(-c5ccccc5)c4=O)cc3F)ccnc2c1 50383174COc1ccc2c(Oc3ccc(NC(=O)c4c([C@@H]5CCCN5)n(C)n(-c5ccccc5)c4=O)nc3)ccnc2c1 50383175COc1ccc2c(Oc3ccc(NC(=O)c4c([C@@H]5CCCN5)n(C)n(-c5ccccc5)c4=O)cc3F)ccnc2c1 50383176COc1ccc2c(Oc3ccc(NC(=O)c4c(n(C)n(-c5ccccc5)c4=O)C(C)(C)N)cc3F)ccnc2c1 50383177COc1ccc2c(Oc3ccc(NC(=O)c4c(CN5CCCC5)n(C)n(-c5ccccc5)c4=O)nc3)ccnc2c1 50383178COc1ccc2c(Oc3ccc(NC(=O)c4c(CN5CCCC5)n(C)n(-c5ccccc5)c4=O)cc3F)ccnc2c1 50383179CCN(C)Cc1c(C(=O)Nc2ccc(Oc3ccnc4cc(OC)ccc34)c(F)c2)c(=O)n(-c2ccccc2)n1C 50383181COc1ccc2c(Oc3ccc(NC(=O)c4c(CN)n(C)n(-c5ccccc5)c4=O)cc3F)ccnc2c1 50383182COc1ccc2c(Oc3cnc(NC(=O)c4c(C)n(C)n(-c5ccccc5)c4=O)nc3)ccnc2c1 50383183COc1ccc2c(Oc3ccc(NC(=O)c4c(C)n(C)n(-c5ccccc5)c4=O)nc3)ccnc2c1 50383184COc1cc2nccc(Oc3ccc(NC(=O)c4c(C)n(C)n(-c5ccccc5)c4=O)nc3)c2cc1OC 50383185COc1ccc2c(Oc3ccc(NC(=O)c4c(C)n(C)n(-c5ccccc5)c4=O)c(OC)c3)ccnc2c1 50383186COc1cc2nccc(Oc3ccc(NC(=O)c4c(C)n(C)n(-c5ccccc5)c4=O)c(Cl)c3)c2cc1OC 50383187COc1cc2nccc(Oc3ccc(NC(=O)c4c(C)n(C)n(-c5ccccc5)c4=O)cn3)c2cc1OC 50383188CCc1cc2c(Oc3ccc(NC(=O)c4c(C)n(C)n(-c5ccccc5)c4=O)cc3F)ccnc2cc1OC 50383189COc1cc2nccc(Oc3ccc(NC(=O)c4c(C)n(C)n(-c5ccccc5)c4=O)cc3F)c2cc1C 50383190COc1cc2nccc(Oc3ccc(NC(=O)c4c(C)n(C)n(-c5ccccc5)c4=O)cc3F)c2cc1Br 50383191COc1cc2nccc(Oc3ccc(NC(=O)c4c(C)n(C)n(-c5ccccc5)c4=O)cc3F)c2cc1OC 50383192COc1ccc2c(Oc3ccc(NC(=O)c4c(C)n(CC5CNC(=O)O5)n(-c5ccccc5)c4=O)cc3F)ccnc2c1 50383193COc1ccc2c(Oc3ccc(NC(=O)c4c(C)n(CCN)n(-c5ccccc5)c4=O)cc3F)ccnc2c1 50383194COc1ccc2c(Oc3ccc(NC(=O)c4c(-c5cc(C)on5)n(C)n(-c5ccccc5)c4=O)nc3)ccnc2c1 50383195COc1ccc2c(Oc3ccc(NC(=O)c4c(C)n(CC(O)CN)n(-c5ccccc5)c4=O)cc3F)ccnc2c1 50383196COc1ccc2c(Oc3ccc(NC(=O)c4c(C)n(CC(O)C(C)C)n(-c5ccccc5)c4=O)cc3F)ccnc2c1 50383197CC[C@H](O)Cn1c(C)c(C(=O)Nc2ccc(Oc3ccnc4cc(OC)ccc34)c(F)c2)c(=O)n1-c1ccccc1 50383198COc1ccc2c(Oc3ccc(NC(=O)c4c(C)n(CC(C)O)n(-c5ccccc5)c4=O)nc3)ccnc2c1 50383199COCCn1c(C)c(C(=O)Nc2ccc(Oc3ccnc4cc(OC)ccc34)cn2)c(=O)n1-c1ccccc1 50383200COc1ccc2c(Oc3ccc(NC(=O)c4c(C)n(CCO)n(-c5ccccc5)c4=O)nc3)ccnc2c1 50383201COc1ccc2c(Oc3ccc(NC(=O)c4c(C)n(CCO)n(-c5ccccc5)c4=O)cc3F)ccnc2c1 50383202COc1ccc2c(Oc3ccc(NC(=O)c4c(C)n(CC(C)=C)n(-c5ccccc5)c4=O)cc3F)ccnc2c1 50383203CCCn1c(C)c(C(=O)Nc2ccc(Oc3ccnc4cc(OC)ccc34)cn2)c(=O)n1-c1ccccc1 50383204CCn1c(C)c(C(=O)Nc2ccc(Oc3ccnc4cc(OC)ccc34)cn2)c(=O)n1-c1ccccc1 50383205CCn1c(C)c(C(=O)Nc2ccc(Oc3ccnc4cc(OC)ccc34)c(F)c2)c(=O)n1-c1ccccc1 50383206COc1ccc2c(Oc3ccc(NC(=O)c4c(-c5csc(C)n5)n(C)n(-c5ccccc5)c4=O)nc3)ccnc2c1 50383207COc1ccc2c(Oc3ccc(NC(=O)c4c(-c5cnccn5)n(C)n(-c5ccccc5)c4=O)nc3)ccnc2c1 50383208COc1ccc2c(Oc3ccc(NC(=O)c4c(-c5cccnc5)n(C)n(-c5ccccc5)c4=O)nc3)ccnc2c1 50391732CNC(=O)[C@@H](Cc1c[nH]c2cc(Cl)ccc12)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccc(cc1)C(=O)P(O)(O)O)NC(=O)[C@H]1CCCC[C@@H]1C(O)=O 50409194COc1cc(\C=C(/C#N)c2ccccn2)ccc1O 50420941Cc1cc(Nc2nc(NCCCc3cn[nH]c3C)ncc2Br)[nH]n1 50420942Cc1cc(Nc2nc(NCCc3ccco3)ncc2Br)[nH]n1 50420947Cc1cc(Nc2ccnc(NCc3cc(no3)C(N)=O)n2)[nH]n1 50420948CCc1cc(Nc2nc(NCc3ccccn3)ncc2Br)[nH]n1 50420949CCc1cc(Nc2nc(NCc3cc(no3)-c3ccccn3)ncc2Br)[nH]n1 50420950CCCc1cc(Nc2nc(NCc3cccnc3)ncc2Br)[nH]n1 50420954Cc1cc(Nc2nc(NCCc3cccnc3)ncc2Br)[nH]n1 50420955Cc1cc(Nc2nc(NCC=C)ncc2Br)[nH]n1 50420956Cc1cc(Nc2nc(NCc3cc(C)no3)ncc2Br)[nH]n1 50420958CCCc1cc(Nc2nc(NCc3cc(C)no3)ncc2Br)[nH]n1 50420959Cc1cc(CNc2ncc(Br)c(Nc3cc(CCc4ccccc4)n[nH]3)n2)on1 50420960Cc1cc(Nc2nc(NCc3cc(no3)C(C)(C)C)ncc2Br)[nH]n1 50420961COc1cc(CCc2cc(Nc3ccnc(NCc4cc(C)no4)n3)[nH]n2)cc(OC)c1 50420963Cc1cc(Nc2nc(NCc3cc(C)no3)ncc2Cl)[nH]n1 50420967CC(C)c1cc(Nc2nc(NCc3cccnc3)ncc2Br)[nH]n1 50420996CCN1CCC(CC1)Nc1ccc2NC(=O)C(=C(c3ncc[nH]3)c3ccc(Cl)cc3)c2c1 50423773C[C@]12O[C@@H](C[C@@]1(O)CO)n1c3ccccc3c3c4C(=O)NCc4c4c5ccccc5n2c4c13 50428737Oc1ccc(CCNC(=O)C(Cc2cc(Br)c(O)c(c2)-c2cc(CC(N=O)C(=O)NCCc3ccc(O)c(Br)c3)cc(Br)c2O)N=O)cc1Br 50428738Oc1ccc(CCNC(=O)C(Cc2cc(Br)c(O)c(Oc3ccc(CCNC(=O)C(Cc4cc(Br)c(O)c(c4)-c4cc(CC(N=O)C(=O)NCCc5ccc(O)c(Br)c5)cc(Br)c4O)N=O)cc3Br)c2)N=O)cc1Br 50436850CC(C)Oc1cc(C2CCNCC2)c(C)cc1Nc1ncc(Cl)c(Nc2ccccc2S(=O)(=O)C(C)C)n1 50437357CCOc1cc(nc2cc(ccc12)-c1nc([C@H]2C[C@@](C)(O)C2)n2ccnc(N)c12)-c1ccccc1 50437358COc1cc(nc2cc(ccc12)-c1nc([C@H]2C[C@@](C)(O)C2)n2ccnc(N)c12)-c1ccccc1 50437359CN1CCN(CC1)[C@H]1C[C@H](C1)c1nc(-c2ccc3c(Oc4ccccc4)cc(nc3c2F)-c2ccccc2)c2c(N)nccn12 50437360CC(C)Oc1cc(nc2c(F)c(ccc12)-c1nc([C@@H]2C[C@@H](C2)N2CCN(C)CC2)n2ccnc(N)c12)-c1ccccc1 50437361CCOc1cc(nc2c(F)c(ccc12)-c1nc([C@@H]2C[C@@H](C2)N2CCN(C)CC2)n2ccnc(N)c12)-c1ccccc1 50437362COc1cc(nc2c(F)c(ccc12)-c1nc([C@@H]2C[C@@H](C2)N2CCN(C)CC2)n2ccnc(N)c12)-c1ccccc1 50437363CN1CCN(CC1)[C@H]1C[C@H](C1)c1nc(-c2ccc3c(Oc4ccccc4)cc(nc3c2)-c2ccccc2)c2c(N)nccn12 50437364CC(C)Oc1cc(nc2cc(ccc12)-c1nc([C@@H]2C[C@@H](C2)N2CCN(C)CC2)n2ccnc(N)c12)-c1ccccc1 50437365CCOc1cc(nc2cc(ccc12)-c1nc([C@@H]2C[C@@H](C2)N2CCN(C)CC2)n2ccnc(N)c12)-c1ccccc1 50437366COc1cc(nc2cc(ccc12)-c1nc([C@@H]2C[C@@H](C2)N2CCN(C)CC2)n2ccnc(N)c12)-c1ccccc1 50437367C[C@@]1(O)C[C@@H](C1)c1nc(-c2ccc3c(Oc4ccccc4)cc(nc3c2F)-c2ccccc2)c2c(N)nccn12 50437368CC(C)Oc1cc(nc2c(F)c(ccc12)-c1nc([C@H]2C[C@@](C)(O)C2)n2ccnc(N)c12)-c1ccccc1 50437369CCOc1cc(nc2c(F)c(ccc12)-c1nc([C@H]2C[C@@](C)(O)C2)n2ccnc(N)c12)-c1ccccc1 50437370COc1cc(nc2c(F)c(ccc12)-c1nc([C@H]2C[C@@](C)(O)C2)n2ccnc(N)c12)-c1ccccc1 50437371C[C@@]1(O)C[C@@H](C1)c1nc(-c2ccc3c(Oc4ccccc4)cc(nc3c2)-c2ccccc2)c2c(N)nccn12 50437372CC(C)Oc1cc(nc2cc(ccc12)-c1nc([C@H]2C[C@@](C)(O)C2)n2ccnc(N)c12)-c1ccccc1 50441567CN1CCN(Cc2ccc(cc2)-c2cnc3[nH]cc(-c4ccc5[nH]ccc5c4)c3c2)CC1 50445471COCc1c(C)c(O)c(O)c(O)c1C=O 50445472COC1OC(=O)c2c1c(C)c(O)c(O)c2O 50445473Cc1c(O)c(O)c2O[C@H]3O[C@H](C(=O)c4c(O)c(O)c(O)c(C)c34)c2c1C=O 50445474Cc1c(O)c(O)c2oc(cc2c1C=O)-c1c(C)c(O)c(O)c(O)c1C=O 50445475Cc1c2COC(=O)c2c(O)c(O)c1O 50446565COc1cc2nc(C)oc2c(C[C@]2(C)[C@@H](C)CC[C@]3(C)[C@H]2CCC=C3C)c1O 50446566CC(C)CC=Nc1cc(O)c(O)c(C[C@]2(C)[C@@H](C)CC[C@]3(C)[C@H]2CCC=C3C)c1O