520CC(C)[C@H](NC(=O)N(C)Cc1csc(n1)C(C)C)C(=O)N[C@H](C[C@H](O)[C@H](Cc1ccccc1)NC(=O)OCc1cncs1)Cc1ccccc1 19188CNCc1cc(=O)oc2cc(OCc3cccc(Cl)c3)ccc12 22416Fc1ccc(cc1)[C@@H]1CCNC[C@H]1COc1ccc2OCOc2c1 25761CC(C)NCC(O)COc1cccc2ccccc12 26467CN(c1ccc2c(C)n[nH]c2c1)c1ccnc(Nc2cccc(c2)S(N)(=O)=O)n1 26468CN(c1ccc2c(C)nn(C)c2c1)c1ccnc(Nc2cccc(c2)S(N)(=O)=O)n1 36108CC(C)[NH2+]C[C@@H](O)COc1cccc2ccccc12 48320CCN(CC)CCNC(=O)c1cc(Cl)c(N)cc1OC 84745CNCC[C@H](Oc1cccc2ccccc12)c1cccs1 87123Fc1cccc(c1)N1CNC(=O)C11CCN(CCNC(=O)c2ccc(F)c(F)c2)CC1 87351COc1cc(NS(C)(=O)=O)ccc1Nc1c2ccccc2nc2ccccc12 93132CC(C)(O)CCCC1(C)CC(=O)c2cc(O)c(Br)cc2O1 93133CC(CCCC(C)(C)O)=CC(=O)c1cc(O)c(Br)cc1O 112777[#6]-[#7]-[#6]-[#6]\[#6]=[#6]-1/c2ccccc2-[#6]-[#6]-c2ccccc-12 126700Oc1cc(CC2CCN(CCc3ccc4OCCC(=O)c4c3)CC2)ccc1Br 50001888CN(C)CCCN1c2ccccc2Sc2ccc(Cl)cc12 50007344CN([C@H](CN1CCCC1)c1ccccc1)C(=O)Cc1ccc(Cl)c(Cl)c1 50013515COC(=O)[C@H]1[C@@H](O)CC[C@H]2CN3CCc4c([nH]c5ccccc45)[C@@H]3C[C@H]12 50014779Clc1ccc(cc1)C(N1CCNCC1)c1ccc(Cl)cc1 50015547[H][C@]12COCC[C@]1([H])[C@]1(COC(N)=N1)c1cc(ccc1O2)-c1cncc(Cl)c1 50015550[H][C@]12COCC[C@]1([H])[C@@]1(COC(N)=N1)c1cc(ccc1O2)-c1cncc(Cl)c1 50015560[H][C@@]12COCC[C@@]1([H])[C@@]1(COC(N)=N1)c1cc(ccc1O2)-c1cncc(Cl)c1 50017297Cc1cccc2nc(cn12)C(=O)N[C@H]1CC[C@H](CC1)NC(=O)c1cc(F)cnc1Oc1cccc(c1)-c1ccc(CN2CCC(CC2)N2CCCC2)cc1 50017299C[C@H]1CN(Cc2ccc(cc2)-c2cccc(Oc3ncc(F)cc3C(=O)N[C@@H]3CC[C@@H](CC3)NC(=O)c3cn4c(C)cccc4n3)c2)C[C@@H](C)N1 50017338C[C@H]1CN(CCCc2ccc(cc2)-c2cccc(Oc3ncc(F)cc3C(=O)N[C@@H]3CC[C@@H](CC3)NC(=O)c3cc(C)n(C)n3)c2)C[C@@H](C)N1 50017339Cc1cc(nn1C)C(=O)N[C@H]1CC[C@H](CC1)NC(=O)c1cc(F)cnc1Oc1cccc(c1)-c1ccc(CCN2CCC(CC2)N2CCCC2)cc1 50017681COc1ccc2nccc([C@H](O)C3CC4CCN3CC4C=C)c2c1 50021822COc1cc2ccnc(Oc3ccc(F)cc3)c2cc1OC 50022784CNCCC(Oc1ccccc1C)c1ccccc1 50027058COC(=O)[C@@H]1[C@@H](O)CC[C@H]2CN3CCc4c([nH]c5ccccc45)[C@@H]3C[C@H]12 50028094CN[C@H]1CC[C@@H](c2ccc(Cl)c(Cl)c2)c2ccccc12 50029559CC(C)(C)Sc1c(CC(C)(C)C(O)=O)n(Cc2ccc(Cl)cc2)c2ccc(OCc3ccc4ccccc4n3)cc12 50030612COC(=O)C1=CO[C@@H](C)[C@H]2CN3CCc4c([nH]c5ccccc45)[C@@H]3C[C@H]12 50032651C[C@@H]([C@@H](O)c1ccc(O)cc1)N1CCC(O)(CC1)c1ccccc1 50039966CN([C@H](CN1CCCC1)c1ccccc1)C(=O)Cc1ccccc1 50041457CCN(CC)Cc1cc(Nc2ccnc3cc(Cl)ccc23)ccc1O 50047001CCC1CN2CCC1CC2C(O)c1ccnc2ccccc12 50047003COC(=O)C1=CO[C@@H](C)[C@H]2C[n+]3ccc-4c([NH2+]c5ccccc-45)c3C[C@H]12 50047004C1CCC2C[n+]3ccc4c([n-]c5ccccc45)c3CC2C1 50047006CC1OC=C(CO)[C@H]2C[C@@H]3N(CCc4c3[nH]c3ccccc43)CC12 50047010COC(=O)C1=CO[C@@H](C)[C@H]2C=[N+]3CCc4c([nH]c5ccccc45)[C@@H]3C[C@H]12 50047011OC1CCC2CN3CCc4c([nH]c5ccccc45)[C@@H]3C[C@@H]2C1C(O)=O 50047016OC1(CCN(CCCC(=O)c2ccc(F)cc2)CC1)c1cccc(c1)C(F)(F)F 50047017COc1ccc2nccc(C(=O)C3CC4CCN3CC4C=C)c2c1 50047018COC(=O)C1C=NC(C)C2CN3CCc4c([nH]c5ccccc45)[C@@H]3C[C@H]12 50047020CC(C)N1CCC(CC1)(c1ccccc1)c1ccccc1 50056190CCNCc1cc(Nc2ccnc3cc(Cl)ccc23)ccc1O 50060418CSc1cc2CCN(C(=O)Nc3cccnc3)c2cc1C(F)(F)F 50066721CCN(CC)CCNc1ccc(CO)c2sc3ccccc3c(=O)c12 50067935COc1ccc(OC(F)(F)F)cc1CN[C@H]1CCCN[C@H]1c1ccccc1 50111469Cc1cc(CCCOc2c(C)cc(cc2C)-c2noc(n2)C(F)(F)F)on1 50116806Fc1ccc(cc1)C(OCCN1CCC(CCCc2ccccc2)CC1)c1ccc(F)cc1 50116913CC(C)(C)NC(=O)[C@@H]1CN(CCN1C[C@@H](O)C[C@@H](Cc1ccccc1)C(=O)N[C@@H]1[C@H](O)COc2ccccc12)C(C)(C)c1cc2cnccc2o1 50117922COCC(=O)O[C@]1(CCN(C)CCCc2nc3ccccc3[nH]2)CCc2cc(F)ccc2[C@@H]1C(C)C 50121975COc1ccc2nccc([C@H](O)[C@H]3C[C@@H]4CCN3C[C@@H]4C=C)c2c1 50125266CCN(CC)CCN(Cc1ccc(cc1)-c1ccc(cc1)C(F)(F)F)C(=O)Cn1c(SCc2ccc(F)cc2)nc(=O)c2CCCCc12 50125267CCN(CC)CCN(Cc1ccc(cc1)-c1ccc(Cl)cc1)C(=O)Cn1c(SCc2ccc(F)cc2)nc(=O)c2CCCCc12 50133282COc1ccnc2[nH]cc(C(=O)C(=O)N3CCN(C[C@H]3C)C(=O)c3ccccc3)c12 50134931CCN(CC)Cc1ccc(Nc2ccnc3cc(Cl)ccc23)cc1O 50134934CCNCc1ccc(Nc2ccnc3cc(Cl)ccc23)cc1O 50134936CC(C)(C)NCc1ccc(Nc2ccnc3cc(Cl)ccc23)cc1O 50136034CCCCOc1ccc(cc1)-c1ccncc1 50136037CCCCOc1ccc(cc1)-n1ccnc1 50136038CCCCOc1ccc(cc1)-n1cncn1 50136041CCCCOc1ccc(cc1)-c1ncc[nH]1 50136043CCCCOc1ccc(cc1)-c1ccncn1 50136047CCCCOc1ccc(cc1)-c1cnccn1 50136052CCCCOc1ccc(cc1)-c1cnco1 50136056CCCCOc1ccc(cc1)-n1cncc1C 50136059CCCCOc1ccc(cc1)-c1c[nH]cn1 50136061CCCCOc1ccc(cc1)-n1cnc(C)c1 50138231C(CN1CCOCC1)Oc1ccc(cc1)-n1ccnc1 50138232C(Oc1ccc(cc1)-n1ccnc1)c1ccccn1 50138233C(COc1ccc(cc1)-n1ccnc1)Cc1ccccn1 50138234CN(C)CCCOc1ccc(cc1)-n1ccnc1 50138235CN(C)CCCCCCOc1ccc(cc1)-n1ccnc1 50138236CCCCCCOc1ccc(cn1)-n1ccnc1 50138237C(COc1ccc(cc1)-n1ccnc1)Cc1cccnc1 50138238C(COc1ccc(cc1)-n1ccnc1)Cc1ccncc1 50138239CCOC(=O)N1CCN(CCOc2ccc(cc2)-n2ccnc2)CC1 50138240CN(C)CCOc1ccc(cc1)-n1ccnc1 50142448CC(=O)c1cccc(NC(=O)NCCCN2CCC[C@@H](Cc3ccc(F)cc3)C2)c1 50142453Cn1nnnc1-c1cccc(NC(=O)NCCCN2CCC[C@@H](Cc3ccc(F)cc3)C2)c1 50142468CC(=O)c1cc(NC(=O)NCCCN2CCC[C@@H](Cc3ccc(F)cc3)C2)cc(c1)C(C)=O 50143945COc1ccc(OCC(O)CN2CCC(CC2)N(C(=O)c2ccc(Cl)cc2)c2ccccc2)cc1 50143946COc1ccc(OCC(O)CN2CCN(CC2)C(CNC(=O)c2ccccc2)c2ccccc2)cc1 50143947OC(COc1ccccc1)CN1CCN(CC1)C(CNC(=O)c1ccc(F)cc1)c1ccccc1 50143948OC(COc1ccccc1)CN1CCN(CC1)C(c1ccccc1)c1ccc(cc1)C(F)(F)F 50143949Cc1cccc(C)c1OCC(O)CN1CCN(CC1)C(C(=O)NCc1ccccc1)c1ccc(cc1)C(F)(F)F 50143950Cc1cccc(C)c1OCC(O)CN1CCN(CC1)C(C(=O)NCc1ccccc1)c1ccc(F)cc1 50143951OC(COCC=C)CN1CCN(CC1)C(c1ccccc1)c1ccc(Cl)cc1 50143952COc1ccc(OCC(O)CN2CCC(CC2)N(C(=O)c2ccc(OC)cc2)c2ccccc2)cc1 50143953COc1ccc(OCC(O)CN2CCN(CC2)C(CNC(=O)c2ccc(OC)cc2)c2ccccc2)cc1 50143954COc1ccc(OCC(O)CN2CCC(CC2)N(C(=O)c2ccc(OC)cc2)c2ccc(F)cc2)cc1 50143955COc1ccc(CNC(=O)C(N2CCN(CC(O)COc3ccc(OC)cc3)CC2)c2ccc(cc2)C(F)(F)F)cc1 50143956COc1ccc(CNC(=O)C(N2CCN(CC(O)COc3c(C)cccc3C)CC2)c2ccc(C)cc2)cc1 50143957COc1ccc(OCC(O)CN2CCN(CC2)C(C(=O)NCc2ccccc2)c2ccc(F)cc2)cc1 50143958COc1ccc(OCC(O)CN2CCC(CC2)N(C(=O)c2ccccc2)c2ccc(F)cc2)cc1 50143959COc1ccc(cc1)C(=O)NCC(N1CCN(CC(O)COc2ccc(Cl)cc2)CC1)c1ccccc1 50143960COc1ccc(OCC(O)CN2CCN(CC2)C(CNC(=O)c2ccccc2OC)c2ccccc2)cc1 50143961COc1ccc(OCC(O)CN2CCC(CC2)N(C(=O)c2ccccc2)c2ccccc2)cc1 50143962OC(COc1ccc(Cl)cc1)CN1CCN(CC1)C(CNC(=O)c1ccc(cc1)C(F)(F)F)c1ccccc1 50143964COc1ccc(OCC(O)CN2CCC(CC2)N(C(=O)c2ccc(Cl)cc2)c2ccc(F)cc2)cc1 50143965COc1ccccc1C(=O)NCC(N1CCN(CC(O)COc2ccc(Cl)cc2)CC1)c1ccccc1 50143967Cc1ccc(cc1)C(N1CCN(CC(O)COc2c(C)cccc2C)CC1)C(=O)NCc1ccccc1 50143968COc1ccc(OCC(O)CN2CCN(CC2)C(CNC(=O)c2ccc(F)cc2)c2ccccc2)cc1 50143970COc1ccc(OCC(O)CN2CCN(CC2)C(CNC(=O)c2ccc(cc2)C(F)(F)F)c2ccccc2)cc1 50143971COc1ccc(OCC(O)CN2CCN(CC2)C(C(=O)NCc2ccccc2)c2ccc(cc2)C(F)(F)F)cc1 50143972COc1ccc(CNC(=O)C(N2CCN(CC(O)COc3c(C)cccc3C)CC2)c2ccc(OC)cc2)cc1 50143973COc1ccc(OCC(O)CN2CCN(CC2)C(C(=O)NCc2ccccc2)c2ccc(C)cc2)cc1 50143974COc1ccc(CNC(=O)C(N2CCN(CC(O)COc3c(C)cccc3C)CC2)c2ccc(cc2)C(F)(F)F)cc1 50143975COc1ccc(CNC(=O)C(N2CCN(CC(O)COc3ccc(OC)cc3)CC2)c2ccc(F)cc2)cc1 50143976COc1ccc(CNC(=O)C(N2CCN(CC(O)COc3c(C)cccc3C)CC2)c2ccc(F)cc2)cc1 50154452NCC(O)CSCc1ccc(Cl)cc1 50154453OC(C1CCN(CCCC(=O)c2ccc(F)cc2)CC1)c1ccc(F)cc1 50154454CCCCNc1c(CN)cnc2cc(Cl)ccc12 50154459CN(C)CCOc1ccc(cc1)C(=C\c1ccccc1)\c1ccccc1 50154460COc1ccc2n(CCCN)c3c(C)c4ccncc4c(C)c3c2c1 50154461CSc1ccc2n(Cc3ccccc3Cl)c(C)c(CCN)c2c1 50154467Clc1ccc(Cl)c(SCCCN2CCNCC2)c1 50154468NCCN1C(=O)c2ccccc2C1(O)c1ccc(Cl)cc1 50154469CCN(CC)CCOC(=O)Cc1cccc2c1oc(cc2=O)-c1ccccc1 50158528Oc1ccc2[nH]cc(C[C@H](NC(=O)c3ccc4n(C5CCCCC5)c(nc4c3)-c3ccoc3)c3cscn3)c2c1 50161093CC(C)(Cc1ccc2ccccc2c1)NC[C@@H](O)COc1cccc(Cl)c1C#N 50163634Cn1nnnc1-c1cccc(NC(=O)N[C@@H]2CCCC[C@H]2CN2CCC[C@@H](Cc3ccc(F)cc3)C2)c1 50163636CC(=O)c1sc(NC(=O)N[C@@H]2CCCC[C@H]2CN2CCC[C@@H](Cc3ccc(F)cc3)C2)nc1C 50164618Clc1ccc(s1)N1C[C@@]2(CN3CCC2CC3)OC1=O 50166613CCCCS(=O)(=O)NCc1ccc(CC(=O)N(C)[C@H](CN2CC[C@H](O)C2)c2ccccc2)cc1 50166614CN([C@H](CN1CC[C@H](O)C1)c1ccccc1)C(=O)Cc1ccc(CNS(=O)(=O)Cc2ccccc2)cc1 50166616CN([C@H](CN1CCCC1)c1ccccc1)C(=O)Cc1ccccc1CNS(C)(=O)=O 50166617CN([C@H](CN1CC[C@H](O)C1)c1ccccc1)C(=O)Cc1ccc(CNS(=O)(=O)c2ccc(F)cc2)cc1 50166621CN([C@H](CN1CC[C@H](O)C1)c1ccccc1)C(=O)Cc1ccc(NS(C)(=O)=O)cc1 50166622CN([C@H](CN1CCCC1)c1ccccc1)C(=O)Cc1cccc(CNS(C)(=O)=O)c1 50166623CN([C@H](CN1CC[C@H](O)C1)c1ccccc1)C(=O)Cc1ccc(CNS(=O)(=O)c2ccc(C)cc2)cc1 50166625CN([C@H](CN1CCCC1)c1ccccc1)C(=O)Cc1cccc(CNC(C)=O)c1 50166627CN([C@H](CN1CCCC1)c1ccccc1)C(=O)Cc1ccccc1CN 50166629CN([C@H](CN1CCCC1)c1ccccc1)C(=O)Cc1ccc(CNC(C)=O)cc1 50166630CN([C@H](CN1CC[C@H](O)C1)c1ccccc1)C(=O)Cc1ccc(CNS(=O)(=O)c2ccccc2)cc1 50166631CN([C@H](CN1CCCC1)c1ccccc1)C(=O)Cc1ccc2CN(Cc2c1)S(C)(=O)=O 50166632CNC(=O)NCc1ccc(CC(=O)N(C)[C@H](CN2CCCC2)c2ccccc2)cc1 50166633CN([C@H](CN1CCCC1)c1ccccc1)C(=O)Cc1ccccc1CNC(C)=O 50166634CN([C@H](CN1CCCC1)c1ccccc1)C(=O)Cc1cccc(CN)c1 50166635CN([C@H](CN1CCCC1)c1ccccc1)C(=O)Cc1ccc(CN)cc1 50166636CN([C@H](CN1CC[C@H](O)C1)c1ccccc1)C(=O)Cc1ccc(CNS(=O)(=O)Cc2cccs2)cc1 50169786COc1ccc2c(CC(C)(C)NCC(O)COc3ccccc3C#N)c[nH]c2c1 50169788CC(C)(Cc1c[nH]c2ccccc12)NCC(O)COc1ccccc1 50169790CCc1ncnc2cc(OC)c(OCC(O)CNC(C)(C)Cc3cc4ccccc4[nH]3)cc12 50169791CC(C)N[C@@H](C)C(O)COc1cccc2ccccc12 50169792CCc1cccc2cc(CC(O)CNC(C)(C)C)oc12 50169793CC(C)(Cc1c[nH]c2ccc(O)cc12)NCC(O)COc1ccccc1C#N 50169794CC(C)(Cc1cc2ccccc2[nH]1)N(CC#C)CC(O)COc1ccccc1C#N 50169795CC(C)(Cc1csc2ccccc12)NCC(O)COc1ccccc1C#N 50169796CC(C)(Cc1c[nH]c2ccccc12)NCC(O)COc1cccc2ccccc12 50169798CC(C)(Cc1cc2ccccc2[nH]1)NCC(O)COc1ccccc1S(C)(=O)=O 50169799CC(C)(Cc1cc2ccccc2[nH]1)N(CC=C)CC(O)COc1ccccc1C#N 50169800CC(C)(Cc1cc2ccccc2[nH]1)NCC(O)COc1ccc(cc1)S(C)(=O)=O 50169801CN(CC(O)COc1ccccc1C#N)C(C)(C)Cc1cc2ccccc2[nH]1 50169802CC(C)(Cc1c[nH]c2ccccc12)NCC(O)COc1ccc(F)cc1C#N 50169803COc1ccc2[nH]cc(CC(C)(C)NCC(O)COc3ccccc3C#N)c2c1 50169804Cc1cc(OCC(O)CNC(C)(C)Cc2cc3ccccc3[nH]2)ccc1S(C)(=O)=O 50169805COc1ccc2c(OCC(O)CNC(C)C)cccc2c1 50169806CCc1ccccc1OCC(O)CNC(C)(C)Cc1cc2ccccc2[nH]1 50169807COCCc1ccc(OCC(O)CNC(C)(C)CSc2ccccc2C)cc1 50169808CC(C)(Cc1c[nH]c2ccccc12)NCC(O)COc1ccccc1C#N 50169809CCOC(=O)CCc1ccc(OCC(O)CNC(C)(C)Cc2c[nH]c3ccccc23)c(c1)C#N 50169810Cc1ccccc1OCC(O)CNC(C)(C)Cc1cc2ccccc2n1C 50169811CC(C)(Cc1c[nH]c2ccccc12)NCC(O)COc1ccc(O)cc1C#N 50169812CC(C)(Cc1cc2ccccc2[nH]1)NCC(O)COc1ccc(cc1)C#N 50169813CCc1ncnc2cc(OCC(O)CNC(C)(C)Cc3cc4ccccc4[nH]3)c(OC)cc12 50169815CC(C)(Cc1c[nH]c2ccccc12)NCC(O)COc1c(ccc2ccccc12)C#N 50172467CC1(C)CCC(CC1)c1ccc(cc1)-c1ccc(cc1F)C1(CC1)C(O)=O 50174943CN([C@H](CN1CC[C@H](O)C1)c1ccccc1)C(=O)C1CCc2cc(NC(C)=O)ccc2O1 50174944CCCS(=O)(=O)NCc1ccc2O[C@@H](Cc2c1)C(=O)N(C)[C@H](CN1CC[C@H](O)C1)c1ccccc1 50174945CCCS(=O)(=O)NCc1ccc2O[C@H](Cc2c1)C(=O)N(C)[C@H](CN1CC[C@H](O)C1)c1ccccc1 50174946COC(=O)Nc1ccc2OC(CCc2c1)C(=O)N(C)[C@H](CN1CC[C@H](O)C1)c1ccccc1 50174947COC(=O)Nc1ccc2O[C@H](Cc2c1)C(=O)N(C)[C@H](CN1CC[C@H](O)C1)c1ccccc1 50174948CN([C@H](CN1CC[C@H](O)C1)c1ccccc1)C(=O)[C@H]1Cc2cccc(NS(C)(=O)=O)c2O1 50174949CN([C@H](CN1CC[C@H](O)C1)c1ccccc1)C(=O)C1CCc2cc(NS(C)(=O)=O)ccc2O1 50174950CN([C@H](CN1CC[C@H](O)C1)c1ccccc1)C(=O)C1CCc2cc(ccc2O1)S(N)(=O)=O 50174952CCCS(=O)(=O)Nc1ccc2O[C@@H](CCc2c1)C(=O)N(C)[C@H](CN1CC[C@H](O)C1)c1ccccc1 50174953CN([C@H](CN1CC[C@H](O)C1)c1ccccc1)C(=O)C1Cc2cc(NC(C)=O)ccc2O1 50174955CN([C@H](CN1CC[C@H](O)C1)c1ccccc1)C(=O)[C@@H]1Cc2ccccc2O1 50174956CN([C@H](CN1CC[C@H](O)C1)c1ccccc1)C(=O)[C@H]1CCc2ccccc2O1 50174957CN([C@H](CN1CC[C@H](O)C1)c1ccccc1)C(=O)[C@@H]1Cc2cccc(NS(C)(=O)=O)c2O1 50174958CN([C@H](CN1CC[C@H](O)C1)c1ccccc1)C(=O)[C@@H]1CCc2ccccc2O1 50174960COC(=O)NCc1ccc2O[C@H](CCc2c1)C(=O)N(C)[C@H](CN1CC[C@H](O)C1)c1ccccc1 50174961CN([C@H](CN1CC[C@H](O)C1)c1ccccc1)C(=O)[C@H]1Cc2ccccc2O1 50174962COC(=O)Nc1ccc2O[C@@H](Cc2c1)C(=O)N(C)[C@H](CN1CC[C@H](O)C1)c1ccccc1 50174963CN([C@H](CN1CC[C@H](O)C1)c1ccccc1)C(=O)[C@@H]1Cc2cc(NS(C)(=O)=O)ccc2O1 50174964CCCS(=O)(=O)Nc1ccc2O[C@H](CCc2c1)C(=O)N(C)[C@H](CN1CC[C@H](O)C1)c1ccccc1 50174965CNS(=O)(=O)c1ccc2OC(Cc2c1)C(=O)N(C)[C@H](CN1CC[C@H](O)C1)c1ccccc1 50174966CNS(=O)(=O)c1ccc2OC(CCc2c1)C(=O)N(C)[C@H](CN1CC[C@H](O)C1)c1ccccc1 50174967CN([C@H](CN1CC[C@H](O)C1)c1ccccc1)C(=O)[C@H]1Cc2cc(NS(C)(=O)=O)ccc2O1 50174968CN([C@H](CN1CC[C@H](O)C1)c1ccccc1)C(=O)[C@H]1CCc2cc(CNS(C)(=O)=O)ccc2O1 50175387CC(C)(Cc1ccc2ccccc2c1)NC[C@@H](O)COc1ccccc1C#N 50175828Fc1cccc(NC(=O)CCN2CCC(Cc3cnc[nH]3)CC2)c1 50175833Clc1ccc(NC(=O)CCN2CCC(Cc3cnc[nH]3)CC2)cc1 50175839C(COc1ccccc1)CN1CCC(Cc2cnc[nH]2)CC1 50176362CN(CC(=O)N(C)[C@H](CN1CC[C@H](O)C1)c1ccccc1)c1ccc(cc1)C#N 50176364CN([C@H](CN1CC[C@H](O)C1)c1ccccc1)C(=O)CN(C(C)=O)c1ccccc1 50176365CN([C@H](CN1CC[C@H](O)C1)c1ccccc1)C(=O)CNc1ccc(cc1)C(F)(F)F 50176366CN([C@H](CN1CC[C@H](O)C1)c1ccccc1)C(=O)CNc1cccc(CNS(C)(=O)=O)c1 50176367CN([C@H](CN1CC[C@H](O)C1)c1ccccc1)C(=O)CNc1cccc(c1)C#N 50176368CN([C@H](CN1CC[C@H](O)C1)c1ccccc1)C(=O)CNc1ccc(CNS(C)(=O)=O)cc1 50176369CN([C@H](CN1CC[C@H](O)C1)c1ccccc1)C(=O)CNc1ccccc1 50176370CN([C@H](CN1CC[C@H](O)C1)c1ccccc1)C(=O)CNc1ccc(cc1)[N+]([O-])=O 50176371CCCS(=O)(=O)Nc1ccc(NCC(=O)N(C)[C@H](CN2CC[C@H](O)C2)c2ccccc2)cc1 50176372CN([C@H](CN1CC[C@H](O)C1)c1ccccc1)C(=O)CNc1ccccc1CNS(C)(=O)=O 50176373CN([C@H](CN1CC[C@H](O)C1)c1ccccc1)C(=O)CNc1ccccc1C#N 50176374CN(CC(=O)N(C)[C@H](CN1CC[C@H](O)C1)c1ccccc1)c1ccccc1 50176375CN([C@H](CN1CC[C@H](O)C1)c1ccccc1)C(=O)CNc1ccc(Cl)c(Cl)c1 50176376CN([C@H](CN1CC[C@H](O)C1)c1ccccc1)C(=O)CNc1ccc(cc1)C#N 50177524C(COc1ccc(cc1)-c1ncccn1)CN1CCC(Cc2cnc[nH]2)CC1 50177525O=C(CCOc1ccc(CN2CCCCC2)cc1)N1CCC(Cc2cnc[nH]2)CC1 50177527C(COc1ccc(NC2CCCCC2)cc1)CN1CCC(Cc2cnc[nH]2)CC1 50177530C(COc1cccc(OC2CCCCC2)c1)CN1CCC(Cc2cnc[nH]2)CC1 50177531C(COc1ccc(CCN2CCCCC2)cc1)CN1CCC(Cc2cnc[nH]2)CC1 50177532C(COc1ccc(OC2CCCCC2)cc1)CN1CCC(Cc2cnc[nH]2)CC1 50177533O=C(N1CCCCC1)c1ccc(OCCCN2CCC(Cc3cnc[nH]3)CC2)nc1 50177535CCN(CC)Cc1ccc(OCCCN2CCC(Cc3cnc[nH]3)CC2)cc1 50177537C(COc1ccc2ncccc2c1)CN1CCC(Cc2cnc[nH]2)CC1 50177539O=C1CCCCN1Cc1ccc(OCCCN2CCC(Cc3cnc[nH]3)CC2)cc1 50177540O=C(CCN1CCC(Cc2cnc[nH]2)CC1)Nc1ccc(CN2CCCCC2)cc1 50177541C(COc1ccc(CN2CCCCC2)nc1)CN1CCC(Cc2cnc[nH]2)CC1 50177542FC1(F)CCN(Cc2ccc(OCCCN3CCC(Cc4cnc[nH]4)CC3)cc2)CC1 50177543C(COc1cccc(CN2CCCCC2)c1)CN1CCC(Cc2cnc[nH]2)CC1 50177544C(CN1CCC(Cc2cnc[nH]2)CC1)Oc1ccc(CN2CCCCC2)cc1 50177545O=C(N1CCCCC1)c1ccc(OCCCN2CCC(Cc3cnc[nH]3)CC2)cc1 50177546O=C(Nc1ncccn1)N1CCC(Cc2cnc[nH]2)CC1 50177548C(COc1ccc(cc1)-c1cccnc1)CN1CCC(Cc2cnc[nH]2)CC1 50177551O=C(Nc1nccs1)N1CCC(Cc2cnc[nH]2)CC1 50177554O=C(CCc1ccc(CN2CCCCC2)cc1)N1CCC(Cc2cnc[nH]2)CC1 50177555C(COc1ccc(cc1)N1CCCCC1)CN1CCC(Cc2cnc[nH]2)CC1 50177556C(COc1ccc(cc1)-c1cncnc1)CN1CCC(Cc2cnc[nH]2)CC1 50185248[#6]-[#6]-1-[#6]-2-[#6]-[#6]-[#6]-1-[#6]=[#6](-[#6]-2)\[#6]=[#6]-1/c2ccccc2-[#6]-[#6]-c2ccccc-12 50185249CN(C)CCC1(O)c2ccccc2CCc2ccc3ccccc3c12 50185250CCCCCCCCCCCc1cccn1C1c2ccccc2CCc2ccccc12 50185254CC(Cc1ccccc1)NC1CC2c3c1cccc3CCc1ccccc21 50185257C(CC1c2ccccc2Sc2ccccc12)NCCc1ccccc1 50185666CCN(C1CCN(CC[C@H](c2ccc(cc2)S(C)(=O)=O)c2cc(F)cc(F)c2)CC1)C(=O)Cc1ccc(cc1)S(C)(=O)=O 50188049Clc1ccccc1CC(N1CCNCC1)c1ccccc1 50188062FC(F)(F)Oc1ccccc1CC(N1CCNCC1)c1ccccc1 50190261CC1CCC(CC1)N[C@@H]1CCN(C1)C(=O)N1CC[C@@H](C1)N(C)C(=O)c1ccc(cc1)-c1ccc(cc1)C(F)(F)F 50190290CN([C@H]1CCN(C1)C(=O)N1CC[C@H](C1)NCCC(C)(C)c1ccc(Cl)cc1)C(=O)c1ccc(cc1)-c1ccc(cc1)C(F)(F)F 50190296CN([C@H]1CCN(C1)C(=O)N1CC[C@H](C1)NCCCc1ccccc1)C(=O)c1ccc(cc1)-c1ccc(cc1)C(F)(F)F 50190516CCCCN1C(=O)C(CC2CCCCC2)NC(=O)C11CCN(Cc2ccc(Oc3ccccc3)cc2)CC1 50190520CCCCN1C(=O)C(CC(C)C)NC(=O)C11CCN(Cc2ccc(Oc3ccccc3)cc2)CC1 50190696Brc1ccc(s1)N1C[C@]2(CN3CCC2CC3)OC1=O 50190788O=C(N[C@H]1CN2CCC1CC2)c1ccc2occc2c1 50190918CN([C@H]1CCN(C1)C(=O)N1CC[C@H](C1)NC1CCC(C)(C)CC1)C(=O)c1ccc(s1)-c1ccc(cc1)C(F)(F)F 50190919COc1ccc(cc1)-c1ccc(s1)C(=O)N(C)[C@H]1CCN(C1)C(=O)N1CC[C@H](C1)NC1CCC(C)(C)CC1 50190920CCc1ccc(cc1)-c1ccc(cc1)C(=O)N(C)[C@H]1CCN(C1)C(=O)N1CC[C@H](C1)N[C@@H](C)C(C)C 50190922CCc1ccc(cc1)-c1ccc(s1)C(=O)N(C)[C@H]1CCN(C1)C(=O)N1CC[C@H](C1)NC1CCOCC1 50190927CCc1ccc(cc1)-c1ccc(s1)C(=O)N(C)[C@H]1CCN(C1)C(=O)N1CC[C@H](C1)NC1CCC(C)(C)CC1 50190931CCc1ccc(cc1)-c1ccc(s1)C(=O)N(C)[C@H]1CCN(C1)C(=O)N1CC[C@H](C1)NC1CCCC1 50190933CCc1ccc(cc1)-c1ccc(s1)C(=O)N(C)[C@H]1CCN(C1)C(=O)N1CC[C@H](C1)NCC1CCOCC1 50190938CCc1ccc(cc1)-c1ccc(s1)C(=O)N(C)[C@H]1CCN(C1)C(=O)N1CC[C@H](C1)NC(C)C 50190940COc1ccc(-c2ccc(s2)C(=O)N(C)[C@H]2CCN(C2)C(=O)N2CC[C@H](C2)NC2CCC(C)(C)CC2)c(C)c1 50190942CN([C@H]1CCN(C1)C(=O)N1CC[C@H](C1)NC1CCC(C)(C)CC1)C(=O)c1ccc(s1)-c1ccccc1 50190943CN([C@H]1CCN(C1)C(=O)N1CC[C@H](C1)NC1CCC(C)(C)CC1)C(=O)c1ccc(s1)-c1ccc2OCCOc2c1 50190948CN([C@H]1CCN(C1)C(=O)N1CC[C@H](C1)NC1CCC(C)(C)CC1)C(=O)c1ccc(s1)-c1ccc(C)cc1 50193172CC(C)N1CCN(CC1)C(=O)N1CCC(CC1)C(C)(C)C 50196930NCC1CCC(CNc2nc(NCc3ccccc3Cl)ncc2[N+]([O-])=O)CC1 50196931CN(C)CC1CCC(CNc2nc(NCc3ccccc3Cl)ncc2[N+]([O-])=O)CC1 50196932CSc1ccccc1CNc1ncc(c(NCC2CCC(CN)CC2)n1)[N+]([O-])=O 50197858CN1CCc2ccc(NS(=O)(=O)c3ccc(cc3)-c3ccc(Cl)cc3)cc2CC1 50197859CCCCc1ccc(cc1)S(=O)(=O)Nc1ccc2CCN(C)CCc2c1 50198075COc1cc(OC)c2c(C)[n+](c(C)cc2c1)-c1cccc2ccccc12 50198392CC1(C)[C@@H]2C[C@H]1C(CN1CCC(CC1)NC(=O)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F)=CC2 50198394O=C(NC1CCN(C\C2=C\CCCCCC2)CC1)Nc1ccc2ccccc2c1 50198936CCCCN1C(=O)[C@H](NC(=O)C11CCN(Cc2ccc(Oc3ccccc3)cc2)CC1)[C@H](O)C1CCCCC1 50200841C[C@H](NC(=O)C(C)(C)Oc1ccc(cn1)C(F)(F)F)[C@@H](Cc1ccc(Cl)cc1)c1cccc(c1)C#N 50203300O=C(OCc1ccccc1)N1CCC(CNc2cnccn2)CC1 50203302O=C(OCc1ccccc1)N1CCC(CNc2ccncn2)CC1 50203303O=C(OCc1ccccc1)N1CCC(CNc2cccnc2)CC1 50203931Cc1c(CN([C@H]2CCNC2)C2CCOCC2)cccc1C(F)(F)F 50203934Fc1ccc(CN([C@H]2CCNC2)C2CCOCC2)c(F)c1F 50203935Cc1cccc(CN([C@@H]2CCNC2)C2CCOCC2)c1C 50203936COc1cccc(CN([C@H]2CCNC2)C2CCOCC2)c1C 50203937Clc1cccc(CN(CC2CC2)[C@H]2CCNC2)c1Cl 50203938Clc1cccc(CN([C@H]2CCNC2)C2CCOCC2)c1Cl 50203939Clc1cccc(CN(Cc2ccccn2)[C@H]2CCNC2)c1Cl 50203943C(N([C@H]1CCNC1)C1CCOCC1)c1ccccc1-c1ccccc1 50203944Clc1cccc(CN(Cc2ccccn2)[C@@H]2CCNC2)c1Cl 50203945Cc1cccc(CN([C@H]2CCNC2)C2CCOCC2)c1C 50205678CN([C@H](CN1CC[C@H](O)C1)c1ccccc1)C(=O)CCC(=O)Nc1nccs1 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50246491CNC[C@]1(O)Cc2ccccc2[C@@H]1Oc1ccccc1-c1cccc2ccccc12 50246492CNC[C@@H]1Cc2ccccc2[C@@H]1Oc1ccccc1C 50246493CNCC1(O)Cc2ccccc2C1Oc1ccccc1C 50246494CNC[C@]1(O)Cc2ccccc2[C@@H]1Oc1ccccc1C 50246547CNC[C@@]1(O)Cc2ccccc2[C@H]1Oc1ccccc1C 50246548CNCC1(O)Cc2ccccc2C1Sc1ccccc1C 50246549CNCC1(O)Cc2ccccc2C1Cc1ccccc1C 50246550CNC[C@@]1(Cc2ccccc2[C@@H]1Oc1ccccc1C)OC 50246551CCNCC1(O)Cc2ccccc2C1Oc1ccccc1C 50246936CC(C)NC[C@H](O)COc1cccc2ccccc12 50246956C(S\C(NC1CCCCC1)=N/C1CCCCC1)C1=CSC2=NCCN12 50247128CC1(C)CN2C(CS\C(NC3CCCCC3)=N/C3CCCCC3)=CSC2=N1 50247629CC(C)(C)NCc1cc(Nc2ccnc3cc(Cl)ccc23)ccc1F 50248347CN(CCC1c2ccccc2-c2ccccc12)CCC(=O)N1CCN(CC1)c1ccc(F)c(F)c1 50250187CCC(=O)c1cc(-c2ccc(Cl)cc2)n(c1C)-c1ccc(cc1)S(N)(=O)=O 50252659Clc1ccc(cc1Cl)C(=O)N[C@H]1CCN(Cc2ccc(OC3CCNCC3)c(Br)c2)C1 50252876CCN(CC)C(=O)c1ccc(cc1)C1=CC2(CCNCC2)Oc2ccccc12 50254448CCN(CCCc1ccc(F)cc1)CC1OC(=O)N(C)CC1(C)NC(=O)Nc1cccc(c1)-c1nnnn1C 50255006CN1C[C@@H](NC(=O)Nc2cccc(c2)-c2nnnn2C)[C@H](CN2CCC[C@@H](Cc3ccc(F)cc3)C2)OC1=O 50255042CN1CC(C)(NC(=O)Nc2nc(C)cs2)C(CN2CCC[C@@H](Cc3ccc(F)cc3)C2)OC1=O 50255702COc1cc(OC)c2c(C)[n+](c(C)cc2c1)-c1ccc(C)cc1 50255812COc1cc(OC)c2c(C)[n+](c(C)cc2c1)-c1ccc(cc1)C(C)C 50256563COCc1c2CC[C@@H](c3ncc[nH]3)c2ccc1Cl 50259063CC(C)(C)OC(=O)NCc1noc(n1)-c1nn(Cc2ccc3OCOc3c2)c2ccccc12 50259240NCc1noc(n1)-c1nn(Cc2ccccc2)c2ccccc12 50259243Cc1cccc(Cn2nc(-c3nc(CN)no3)c3ccccc23)c1 50259287Cc1cc(C)cc(Cn2nc(-c3nc(CN)no3)c3ccccc23)c1 50259356NCc1noc(n1)-c1nn(Cc2ccc(cc2)C(N)=O)c2ccccc12 50259376C[C@@H](Nc1c(Nc2ccncc2)c(=O)c1=O)c1ccccc1 50259554NCc1noc(n1)-c1nn(CCc2ccccc2)c2ccccc12 50259555NCc1noc(n1)-c1n(CCc2ccccc2)nc2ccccc12 50259557NCc1noc(n1)-c1n[nH]c2ccccc12 50259585COc1ccc(cc1OC)S(=O)(=O)n1nc(-c2nc(CN)no2)c2ccccc12 50262279COc1cc2COC(C)(c2cc1CN[C@H]1CCCN[C@H]1c1ccccc1)C(F)(F)F 50262280COc1ccc(cc1CN[C@H]1CCCN[C@H]1c1ccccc1)C(C)C(F)(F)F 50262281COc1ccc(CC(F)(F)F)cc1CN[C@H]1CCCN[C@H]1c1ccccc1 50262337COc1ccc(cc1CN[C@H]1CCCN[C@H]1c1ccccc1)C(C(F)(F)F)C(F)(F)F 50262395COc1cc2CCC(c2cc1CN[C@H]1CCCN[C@H]1c1ccccc1)C(F)(F)F 50262415CC(C)C(=O)N(Cc1ccccc1-c1ccccc1)[C@H]1CCNC1 50262510COc1cc2CCCC(C)(c2cc1CN[C@H]1CCCN[C@H]1c1ccccc1)C(F)(F)F 50262567COc1ccc(cc1CN[C@H]1C2CCN(CC2)[C@H]1C(c1ccccc1)c1ccccc1)C(C)C 50262625CS(=O)(=O)N(Cc1ccccc1-c1ccccc1)[C@H]1CCNC1 50262626CCS(=O)(=O)N(Cc1ccccc1-c1ccccc1)[C@H]1CCNC1 50262627CCCS(=O)(=O)N(Cc1ccccc1-c1ccccc1)[C@H]1CCNC1 50262630CCOC(=O)N(Cc1ccccc1-c1ccccc1)[C@@H]1CCNC1 50262631CS(=O)(=O)N(Cc1ccccc1-c1ccccc1)[C@@H]1CCNC1 50262678CCOC(=O)N(Cc1ccccc1-c1ccccc1)[C@H]1CCNC1 50262679CC(C)S(=O)(=O)N(Cc1ccccc1-c1ccccc1)[C@H]1CCNC1 50262684CN(C)S(=O)(=O)N(Cc1ccccc1-c1ccccc1)[C@H]1CCNC1 50262733CCOC(=O)N(Cc1ccccc1Oc1ccccc1)[C@H]1CCNC1 50263399Clc1ccc(cc1)C(NC(=O)CNC(=O)c1ccc(cc1)C#N)c1ccccc1 50264142Fc1ccc2cc(CN3C4CCC3CC(C4)NC(=O)c3ccccc3-c3ccccc3)ccc2c1 50264144Fc1ccc2cc(CN3[C@@H]4CC[C@@H]3CC(C4)NC(=O)c3ccccc3-c3cccnc3)ccc2c1 50264155Fc1ccc2cc(CN3[C@@H]4CC[C@@H]3CC(C4)NC(=O)c3ccccc3-c3nccs3)ccc2c1 50264157Fc1ccc2cc(CN3[C@@H]4CC[C@@H]3CC(C4)NC(=O)c3ccccc3C(=O)N3CCCCC3)ccc2c1 50264158CN1CCN(CC1)C(=O)c1ccccc1C(=O)NC1C[C@H]2CC[C@H](C1)N2Cc1ccc2cc(F)ccc2c1 50264159Fc1ccc2cc(CN3[C@@H]4CC[C@@H]3CC(C4)NC(=O)c3ccccc3C(=O)N3CCOCC3)ccc2c1 50264161Fc1ccc2cc(CN3[C@@H]4CC[C@@H]3CC(C4)NC(=O)c3ccncc3C(=O)N3CCCCC3)ccc2c1 50264191Fc1ccc2cc(CN3[C@@H]4CC[C@@H]3CC(C4)NC(=O)c3ccccc3-c3ccccn3)ccc2c1 50264206Fc1ccc2cc(CN3[C@@H]4CC[C@@H]3CC(C4)NC(=O)c3ccccc3OC3CCCCC3)ccc2c1 50264208CN(C1CCCCC1)C(=O)c1ccccc1C(=O)NC1C[C@H]2CC[C@H](C1)N2Cc1ccc2cc(F)ccc2c1 50264209Fc1ccc2cc(CN3[C@@H]4CC[C@@H]3CC(C4)NC(=O)c3ccccc3C(=O)N3CCCC3)ccc2c1 50264210Fc1ccc2cc(CN3[C@@H]4CC[C@@H]3CC(C4)NC(=O)c3ccccc3C(=O)N3CCCCCC3)ccc2c1 50267987COc1ccc(CC(C)(C)NCC(O)COc2ccccc2C#N)cc1 50267988COc1ccc(CC(C)(C)NCC(O)COc2cccc(Cl)c2C#N)cc1 50268077COc1ccc(CC(C)(C)NC[C@H](O)COc2cccc3[nH]c(=O)[nH]c23)cc1 50268484Cc1cc(C[C@@H](NC(=O)N2CCC(CC2)N2Cc3cccc(F)c3NC2=O)C(=O)N2CCC(CC2)N2CCCCC2)cc2cn[nH]c12 50268742CCc1cccc(C)c1CNc1cccn2c(C)c(C)nc12 50268782Cc1nc2c(NCc3c(C)cccc3C)cc(cn2c1C)-c1ccccn1 50268887Cc1nc2c(NCc3c(C)cccc3C)cc(cn2c1C)-c1ccco1 50269055CC(C)N1CCC(CC1)Oc1ccc2n(C(C)C)c(cc2c1)C(=O)N1CCC(F)(F)CC1 50269061C[C@@H](N[C@@H]1CCCc2c1[nH]c1ccc(Br)cc21)c1ccccc1 50272643CNC[C@@H]1COc2ccccc2[C@@H]1Oc1ccccc1Cl 50272645CNC[C@@H]1COc2ccccc2[C@@H]1Oc1ccccc1C 50272646CNC[C@@H]1CCc2ccccc2[C@@H]1Oc1ccccc1C 50272647CNC[C@H]1COc2ccccc2[C@@H]1Oc1ccccc1C 50272654CNC[C@@H]1OCc2ccccc2[C@@H]1Oc1ccccc1C(F)(F)F 50272655CNC[C@@H]1OCc2ccccc2[C@@H]1Oc1cccc(F)c1C 50272686CNC[C@H]1OCc2ccccc2[C@H]1Oc1ccccc1C 50272687Cc1ccccc1O[C@H]1[C@@H](CN)COc2ccccc12 50272688Cc1ccccc1O[C@@H]1[C@H](CN)OCc2ccccc12 50272690CNC[C@@H]1COc2ccccc2[C@H]1Oc1ccccc1C 50272691CNC[C@@H]1OCc2ccccc2[C@@H]1Oc1ccccc1Cl 50272692CNC[C@H]1OCc2ccccc2[C@H]1Oc1ccccc1Cl 50272693CNC[C@H]1OCc2ccccc2[C@H]1Oc1ccccc1C(F)(F)F 50272694CNC[C@H]1OCc2ccccc2[C@H]1Oc1cccc(C)c1C 50272715Cc1ccccc1O[C@@H]1[C@H](CN)COc2ccccc12 50272717CNC[C@@H]1OCc2ccccc2[C@@H]1Oc1ccccc1C 50272719CNC[C@H]1OCc2ccccc2[C@@H]1Oc1ccccc1C 50272728CNC[C@@H]1OCc2ccccc2[C@@H]1Oc1c(C)cccc1F 50272730CNC[C@@H]1OCc2ccccc2[C@@H]1Oc1c(F)cccc1C(F)(F)F 50272742CNC[C@H]1CCc2ccccc2[C@H]1Oc1ccccc1C 50272743CNC[C@H]1COc2ccccc2[C@H]1Oc1ccccc1C 50272744CNC[C@@H]1OCc2ccccc2[C@H]1Oc1ccccc1C 50272745CCc1ccccc1O[C@@H]1[C@H](CNC)COc2ccccc12 50272746CCc1ccccc1O[C@H]1[C@@H](CNC)COc2ccccc12 50272747CNC[C@H]1COc2ccccc2[C@H]1Oc1ccccc1Cl 50272748CNC[C@@H]1OCc2ccccc2[C@@H]1Oc1cccc(C)c1C 50272749CNC[C@@H]1OCc2ccccc2[C@@H]1Oc1ccc(O)cc1C 50272853CCn1cc(c(n1)-c1cccc(NC(=O)Nc2ccc(cc2)C(F)(F)F)c1)-c1ccnc2[nH]ccc12 50272893CCn1cc(c(n1)-c1cccc(NC(=O)Nc2cccc(OC)c2)c1)-c1ccnc2[nH]ccc12 50274918C(c1ccccc1)C1(CCNC1)c1ccc2cc[nH]c2c1 50274919C(c1ccccc1)C1(CCNC1)c1c[nH]c2ccccc12 50274920C(c1ccccn1)C1(CCNC1)c1ccc2[nH]ccc2c1 50274921Fc1ccc(CC2(CCNC2)c2ccc3[nH]ccc3c2)cc1 50274949COc1cccc(CC2(CCNC2)c2ccc3[nH]ccc3c2)c1 50274950C(CC1(CCNC1)c1ccc2[nH]ccc2c1)c1ccccc1 50274951Cn1ccc2cc(ccc12)C1(Cc2ccccc2)CCNC1 50274952CCOC(=O)c1cc2cc(ccc2[nH]1)C1(Cc2ccccc2)CCNC1 50274953N#Cc1cc2cc(ccc2[nH]1)C1(Cc2ccccc2)CCNC1 50274954NC(=O)c1cc2cc(ccc2[nH]1)C1(Cc2ccccc2)CCNC1 50274974CNC(=O)c1cc2cc(ccc2[nH]1)C1(Cc2ccccc2)CCNC1 50274975CN(C)C(=O)c1cc2cc(ccc2[nH]1)C1(Cc2ccccc2)CCNC1 50274976N#Cc1c[nH]c2ccc(cc12)C1(Cc2ccccc2)CCNC1 50274977CC1(CCNC1)c1ccc2[nH]ccc2c1 50274978CCCC1(CCNC1)c1ccc2[nH]ccc2c1 50274979CCCCC1(CCNC1)c1ccc2[nH]ccc2c1 50275378CNCCC(c1c[nH]c2ccccc12)c1ccccc1 50275438C(c1ccccc1)C1(CCNC1)c1ccc2[nH]ccc2c1 50275439C(c1ccccc1)C1(CCNC1)c1ccc2[nH]ncc2c1 50275735COc1ccc2nc(SCc3cc(OC)cc(OC)c3)[nH]c2c1 50275736COc1ccc2nc(SCc3ccc4ccccc4c3)[nH]c2c1 50275773CCN(CC(F)=C)C(=O)[C@]1(C[C@H]1CN)c1cccs1 50275774NC[C@@H]1C[C@@]1(C(=O)N(CC=C)CC=C)c1cccs1 50293132CC(C)(C#N)c1ccc(CCC2(CC(=O)C(Cc3cn4ccccc4n3)C(=O)O2)C2CCCC2)cc1F 50293133COc1cccc(CC2C(=O)CC(CCc3ccc(c(F)c3)C(C)(C)C#N)(OC2=O)C2CCCC2)c1 50293851CC[C@@H](Oc1cccc(Cn2c(C)c(C(=O)c3ccc(Cl)cc3)c3ccc(OC(F)(F)F)cc23)c1)C(O)=O 50294257Clc1cccc(OC([C@H]2CCNC2)c2ccccn2)c1Cl 50294270Clc1cccc(OC(C2CCNCC2)c2cccnc2)c1Cl 50294271Cc1ccc(cn1)C(Oc1cccc(Cl)c1Cl)C1CCNCC1 50294286Clc1cccc(OC([C@@H]2CCCNC2)c2cccnc2)c1Cl 50296487[NH3+][C@H]1C[n+]2c(C[C@@H]1c1cc(F)c(F)cc1F)[nH]c1ncccc21 50296488CS(=O)(=O)c1ccc2n3C[C@H]([NH3+])[C@H](Cc3nc2c1)c1cc(F)c(F)cc1F 50296754N[C@@H](CC(=O)N1CCC[C@H]1CN(C1CC1)S(=O)(=O)C(F)(F)F)Cc1cc(F)c(F)cc1F 50296755CN(C[C@@H]1CCCN1C(=O)C[C@H](N)Cc1cc(F)c(F)cc1F)S(=O)(=O)C(F)(F)F 50296759CN(C[C@@H]1CCCN1C(=O)C[C@H](N)Cc1cc(F)c(F)cc1F)C(=O)C(C)(F)F 50296760CN(C[C@@H]1CCCN1C(=O)C[C@H](N)Cc1cc(F)c(F)cc1F)C(=O)C(C)(C)C 50296761CN(C[C@@H]1CCCN1C(=O)C[C@H](N)Cc1cc(F)c(F)cc1F)C(=O)C1CC1 50296763CC(F)(F)C(=O)NC[C@@H]1CCCN1C(=O)C[C@H](N)Cc1cc(F)c(F)cc1F 50296769N[C@@H](CC(=O)N1CCC[C@H]1CNC(=O)C1(CC1)C(F)(F)F)Cc1cc(F)c(F)cc1F 50296770N[C@@H](CC(=O)N1CCC[C@H]1COCC1CC1)Cc1cc(F)c(F)cc1F 50296771N[C@@H](CC(=O)N1CCC[C@H]1COc1ccnc(n1)C(F)(F)F)Cc1cc(F)c(F)cc1F 50296772N[C@@H](CC(=O)N1CCC[C@H]1COc1cc(ccn1)C#N)Cc1cc(F)c(F)cc1F 50296773N[C@@H](CC(=O)N1CCC[C@H]1COc1ccc(cn1)C#N)Cc1cc(F)c(F)cc1F 50296774N[C@@H](CC(=O)N1CCC[C@H]1CNc1nccc(n1)C(F)(F)F)Cc1cc(F)c(F)cc1F 50296775N[C@@H](CC(=O)N1CCC[C@H]1CNc1ncc(F)cn1)Cc1cc(F)c(F)cc1F 50296776N[C@@H](CC(=O)N1CCC[C@H]1CNc1ncccn1)Cc1cc(F)c(F)cc1F 50296777N[C@@H](CC(=O)N1CCC[C@H]1CNc1ccc(nc1)C(F)(F)F)Cc1cc(F)c(F)cc1F 50296778N[C@@H](CC(=O)N1CCC[C@H]1CNc1ccc(F)cn1)Cc1cc(F)c(F)cc1F 50296779N[C@@H](CC(=O)N1CCC[C@H]1CNc1ncccc1C#N)Cc1cc(F)c(F)cc1F 50296780CN(C[C@@H]1CCCN1C(=O)C[C@H](N)Cc1cc(F)c(F)cc1F)c1ccc(cn1)C#N 50296781N[C@@H](CC(=O)N1CCC[C@H]1CNc1ccc(cn1)C#N)Cc1cc(F)c(F)cc1F 50297078CCSc1ccccc1C(=O)N(CC1CCC1)[C@H]1CCNC1 50297079CC(C)c1ccccc1C(=O)N(CC1CCC1)[C@H]1CCNC1 50297080O=C(N(CC1CCC1)[C@H]1CCNC1)c1ccccc1C1CCCC1 50297081O=C(N(CC1CCC1)[C@H]1CCNC1)c1ccccc1Oc1ccccc1 50297086O=C(N(C1CCC1)[C@H]1CCNC1)c1ccccc1Oc1ccccc1 50297087CC(C)CN([C@H]1CCNC1)C(=O)c1ccccc1Oc1ccccc1 50297088O=C(N([C@H]1CCNC1)c1ccccc1)c1ccccc1Oc1ccccc1 50297304CN(C)CCC1=C(Cc2ccc(F)cc2)c2ccccc2C1 50297305CN(C)CCC1=C(Cc2cnccn2)c2ccccc2C1 50297306CN(C)CCc1sc2ccccc2c1Cc1ccc(F)cc1 50297309C[C@H](c1c(CCN(C)C)sc2ccccc12)c1ccccn1 50297310C[C@H](c1c(CCN(C)C)oc2ccccc12)c1ccccn1 50297312CCNC(=O)c1ccc(cc1)C1=CC2(CCNCC2)Oc2ccccc12 50297313NC(=O)c1ccc(cc1)C1=CC2(CCNCC2)Oc2ccccc12 50297314CNC(=O)c1ccc(cc1)C1=CC2(CCNCC2)Oc2ccccc12 50297315CC(C)CNC(=O)c1ccc(cc1)C1=CC2(CCNCC2)Oc2ccccc12 50297316CC(C)N(C(C)C)C(=O)c1ccc(cc1)C1=CC2(CCNCC2)Oc2ccccc12 50297317CN(C)C(=O)c1ccc(cc1)C1=CC2(CCNCC2)Oc2ccccc12 50297318O=C(N1CCCC1)c1ccc(cc1)C1=CC2(CCNCC2)Oc2ccccc12 50297319O=C(N1CCCCC1)c1ccc(cc1)C1=CC2(CCNCC2)Oc2ccccc12 50297320O=C(N1CCOCC1)c1ccc(cc1)C1=CC2(CCNCC2)Oc2ccccc12 50297321O=C(N1Cc2ccccc2C1)c1ccc(cc1)C1=CC2(CCNCC2)Oc2ccccc12 50297322CN(Cc1ccccc1)C(=O)c1ccc(cc1)C1=CC2(CCNCC2)Oc2ccccc12 50297323CCN1CCc2cc(ccc2C1=O)C1=CC2(CCNCC2)Oc2ccccc12 50297324CCN(CC)C(=O)c1ccc(cc1)C1=CC2(CCCNCC2)Oc2ccccc12 50297325CCN(CC)C(=O)c1ccc(cc1)C1=CC2(CCNC2)Oc2ccccc12 50297326CCN(CC)C(=O)c1ccc(cc1)C1=CC2(CCCNC2)Oc2ccccc12 50297328CCN(CC)C(=O)c1ccc(cc1)C1CC2(CCNCC2)Oc2ccccc12 50297329CCN(CC)C(=O)c1ccc(cc1)[C@H]1CC2(CCNCC2)Oc2ccccc12 50297330CCN(CC)C(=O)c1ccc(cc1)[C@@H]1CC2(CCNCC2)Oc2ccccc12 50297331CCN(CC)C(=O)c1ccc(s1)C1=CC2(CCNCC2)Oc2ccccc12 50297332CCN(CC)C(=O)c1ccc(o1)C1=CC2(CCNCC2)Oc2ccccc12 50297333CCN(CC)C(=O)c1cc(cs1)C1=CC2(CCNCC2)Oc2ccccc12 50297337CCN(CC)C(=O)c1ccc(cc1C)C1=CC2(CCNCC2)Oc2ccccc12 50297338CCN(CC)C(=O)c1ccc(cc1F)C1=CC2(CCNCC2)Oc2ccccc12 50297339CCN(CC)C(=O)c1ccc(cc1O)C1=CC2(CCNCC2)Oc2ccccc12 50297340CCN(CC)C(=O)c1ccc(C2=CC3(CCNCC3)Oc3ccccc23)c(C)c1 50297341CCN(CC)C(=O)c1ccc(C2=CC3(CCNCC3)Oc3ccccc23)c(F)c1 50297370CC(C)(C)Sc1c(CC(C)(C)C(O)=O)n(Cc2ccc(cc2)-c2nccs2)c2ccc(OCc3ccccn3)cc12 50297374CC(C)(C)Sc1c(CC(C)(C)C(O)=O)n(Cc2ccc(cc2)-c2cccnc2)c2ccc(OCc3ccccn3)cc12 50297849COc1ccc(Cn2c(nc3ccccc23)N2CCC(CC2)n2cc(C)cn2)cc1 50297850Cc1cnn(c1)C1CCN(CC1)c1nc2ccccc2n1Cc1ccc(F)cc1 50297851Fc1ccc(Cn2c(nc3ccccc23)N2CCC(CC2)n2cccn2)cc1 50297852Fc1ccc(Cn2c(nc3ccccc23)N2CCC(CC2)n2ccnc2)cc1 50297853Fc1ccc(Cn2c(nc3ccccc23)N2CCC(CC2)n2cccc2)cc1 50297854Fc1ccc(Cn2c(nc3ccccc23)N2CCC(CC2)N2CCCCC2=O)cc1 50297855CN(C)CCN(C)C1CCN(CC1)c1nc2ccccc2n1Cc1ccc(F)cc1 50297859COCCN(C)C1CCN(CC1)c1nc2ccccc2n1Cc1ccc(F)cc1 50297860COc1ccc(Cn2c(nc3ccccc23)N2CCC(CC2)N(C)CC2CCOCC2)cc1 50297862COc1ccc(Cn2c(nc3ccccc23)N2CCC(CC2)N(C)C)cc1 50297863CN(C)C1CCN(CC1)c1nc2ccccc2n1Cc1ccc(C)cc1 50297865CN(C1CCOCC1)C1CCN(CC1)c1nc2ccccc2n1Cc1ccc(F)cc1 50297866CNC1CCN(CC1)c1nc2ccccc2n1Cc1ccc(F)cc1 50297867CN(C1CCCCC1)C1CCN(CC1)c1nc2ccccc2n1Cc1ccc(F)cc1 50297868CN(CC1CCCCC1)C1CCN(CC1)c1nc2ccccc2n1Cc1ccc(F)cc1 50297869CN(CCc1ccccc1)C1CCN(CC1)c1nc2ccccc2n1Cc1ccc(F)cc1 50297870CN(Cc1ccccc1)C1CCN(CC1)c1nc2ccccc2n1Cc1ccc(F)cc1 50297872CN(C1CCN(CC1)c1nc2ccccc2n1Cc1ccc(F)cc1)c1ncccn1 50298028CN1CC[C@@H](C1)N(Cc1ccccc1C(F)(F)F)c1ccc(C#N)c(Cl)c1 50299545CC(C)(Cc1ccc2ccccc2c1)NC[C@@H](O)COc1ccc(CCC(O)=O)cc1 50299633Cc1cc(ccc1O)-c1ccc(s1)-c1cccc(O)c1 50299643Oc1cccc(c1)-c1ccc(s1)-c1ccc(O)c(F)c1 50299645Cc1cc(ccc1O)-c1csc(c1)-c1cccc(O)c1 50302545C[C@@H]1CN(CCN1C(=O)C(=O)c1c[nH]c2ccccc12)C(=O)c1ccccc1 50304834Cc1cc(NC2CCCCC2)nc(NCc2ccccc2)n1 50304967CCCS(=O)(=O)N1CC[C@@H](C1)N(Cc1ccccc1C(F)(F)F)c1ccc(C#N)c(Cl)c1 50304975COC(=O)N1CC[C@@H](C1)N(Cc1ccccc1C(F)(F)F)c1ccc(C#N)c(Cl)c1 50304976COC(=O)N1CC[C@@H](C1)N(Cc1ccccc1F)c1ccc(C#N)c(Cl)c1 50304979COC(=O)N1CC[C@@H](C1)N(Cc1cccc(F)c1F)c1ccc(C#N)c(Cl)c1 50304985CC(C)C(=O)N1CC[C@@H](C1)N(Cc1ccccc1C(F)(F)F)c1ccc(C#N)c(Cl)c1 50304987CCC(=O)N1CC[C@@H](C1)N(Cc1ccccc1Br)c1ccc(C#N)c(Cl)c1 50304988COC(=O)N1CC[C@@H](C1)N(Cc1ccccc1)c1ccc(C#N)c(Cl)c1 50305760FC(F)(F)c1ccccc1OC1CCN(CC1)c1ccc(nn1)-n1ccnc1 50305878Cc1n[nH]c2ccc(cc12)-c1cc(OC[C@@H](N)Cc2c[nH]c3ccccc23)cnc1-c1ccoc1 50308246Clc1ccc(cc1Cl)[C@]1(COCC2CC2)[C@H]2CNC[C@@H]12 50308251CCOC[C@H]1[C@@H]2CNC[C@]12c1ccc(Cl)c(Cl)c1 50308253Clc1ccc(cc1Cl)[C@@]12CNC[C@@H]1[C@H]2COCC1CC1 50308254FC(F)(F)COC[C@]1([C@H]2CNC[C@@H]12)c1ccc(Cl)c(Cl)c1 50309954CN1C[C@@H]2C[C@@H](C[C@@H]2C1)N(Cc1cccc(OC(F)(F)F)c1)C(=O)c1cn(C)cn1 50309963CCN1C[C@@H]2C[C@@H](C[C@@H]2C1)N(Cc1ccc(F)c(c1)C(F)(F)F)C(=O)c1cn(C)cn1 50309965Cn1cnc(c1)C(=O)N(Cc1cccc(OC(F)(F)F)c1)[C@H]1C[C@H]2CN(CC(C)(C)O)C[C@H]2C1 50309966Cn1cnc(c1)C(=O)N(Cc1cccc(OC(F)(F)F)c1)[C@H]1C[C@H]2CN(CC(O)c3ccccc3)C[C@H]2C1 50309967Cn1cnc(c1)C(=O)N(Cc1cccc(OC(F)(F)F)c1)[C@H]1C[C@H]2CN(CCC(F)(F)F)C[C@H]2C1 50309968CC(F)CN1C[C@@H]2C[C@@H](C[C@@H]2C1)N(Cc1cccc(OC(F)(F)F)c1)C(=O)c1cn(C)cn1 50309969CCN1C[C@@H]2C[C@@H](C[C@@H]2C1)N(Cc1cccc(OC(F)(F)F)c1)C(=O)c1cn(C)cn1 50311414O=S(=O)(Nc1ccc2CCN(Cc3ccn[nH]3)CCc2c1)c1ccc(s1)-c1ccccn1 50311415CC1(C)CCc2cc(ccc2O1)S(=O)(=O)Nc1ccc2CCN(Cc3ccn[nH]3)CCc2c1 50311416CC(C)Oc1ccc(cc1)S(=O)(=O)Nc1ccc2CCN(Cc3ccn[nH]3)CCc2c1 50311417O=S(=O)(Nc1ccc2CCN(Cc3ccn[nH]3)CCc2c1)c1ccc(cc1)C#N 50311419Fc1ccc(Nc2ccc(cn2)S(=O)(=O)Cc2ccc3CCNCCc3c2)cc1 50311420O=S(=O)(Cc1ccc2CCNCCc2c1)c1ccc(nc1)N1CCCCC1 50311421CC(C)Oc1ccc(cn1)S(=O)(=O)Cc1ccc2CCNCCc2c1 50311422Fc1ccc(Oc2ccc(cn2)S(=O)(=O)Cc2ccc3CCNCCc3c2)cc1 50311423Fc1ccc(cc1)-c1ccc(cn1)S(=O)(=O)Cc1ccc2CCNCCc2c1 50311424Fc1ccc(cc1F)-c1ccc(cc1)S(=O)(=O)Cc1ccc2CCNCCc2c1 50311425Fc1ccc(cc1)-c1ccc(cc1)S(=O)(=O)Cc1ccc2CCNCCc2c1 50311746C[C@H]1C[C@@H]1Cn1c(C)c(C)c2cnnc(OCc3ccc(F)cc3)c12 50311748Cc1[nH]c2c(NCc3c(C)cccc3C)ncnc2c1C 50311754Cc1nc2c(OCc3c(C)cccc3C)cccn2c1C 50311756Cc1[nH]c2c(NCc3c(C)cccc3C)nc(cc2c1C)N1CCNC1=O 50311759Cc1[nH]c2c(NCc3c(C)cccc3C)nc(cc2c1C)N1CCCC1=O 50311760Cc1[nH]c2c(NCc3c(C)cccc3C)nc(cc2c1C)-c1ccccc1 50312665OP([O-])(=O)OC1CC(=Nc2cc3OCOc3cc12)c1ccccc1F 50312945COc1ccc(C[C@H](C)CN2C[C@@H]3CCCC[C@@H]3[C@@H](C2)C(=O)N2CCN(CC2)c2ccc(F)c(F)c2)cn1 50313618Clc1cccc(c1)N1CCN(CC2CCCCN2)C1=O 50314261C[C@@H](c1c(CCN(C)C)sc2ccccc12)c1ccccn1 50314262CNCCc1sc2ccccc2c1[C@@H](C)c1ccccn1 50314263C[C@H](c1c(CCN2CCCC2)sc2ccccc12)c1ccccn1 50314265CC(c1c(CCN(C)C)sc2ccccc12)c1cccnc1 50314266C[C@@H](c1c(CCN(C)C)sc2ccccc12)c1cccnc1 50314267C[C@H](c1c(CCN(C)C)sc2ccccc12)c1cccnc1 50314268CC(c1c(CCN(C)C)sc2ccccc12)c1ccncc1 50314269C[C@H](c1c(CCN(C)C)sc2ccccc12)c1ncccc1Cl 50314274COc1ncccc1[C@@H](C)c1c(CCN(C)C)sc2ccccc12 50314275C[C@@H](c1c(CCN(C)C)sc2ccccc12)c1cccnc1F 50314276C[C@@H](c1c(CCN(C)C)sc2ccccc12)c1cccnc1Cl 50314280C[C@H](c1c(CCN(C)C)sc2ccccc12)c1ncccc1C 50314281COc1cccnc1[C@H](C)c1c(CCN(C)C)sc2ccccc12 50314282C[C@H](c1c(CCN(C)C)sc2ccccc12)c1ncccc1F 50315184CN(C)CCC1=C(Cc2cncc(C)n2)c2ccccc2C1 50315186CN(C)CCC1=C(Cc2cnc(C)cn2)c2ccccc2C1 50315187COc1nccnc1CC1=C(CCN(C)C)Cc2ccccc12 50315191C[C@H](C1=C(CCN(C)C)Cc2ccccc12)c1nccs1 50315193CN(C)CCC1=C(Cc2cnccn2)c2ccc(C)cc2C1 50315194COc1ccc2C(Cc3cnccn3)=C(CCN(C)C)Cc2c1 50315197COc1nccnc1CC1=C(CCN(C)C)Cc2cc(Cl)ccc12 50315198COc1nccnc1CC1=C(CCN(C)C)Cc2cc(F)ccc12 50315204COc1ccc2C([C@@H](C)c3nccnc3OC)=C(CCN(C)C)Cc2c1 50315205COc1nccnc1[C@H](C)C1=C(CCN(C)C)Cc2cc(F)ccc12 50315206C[C@H](C1=C(CCN(C)C)Cc2cc(F)ccc12)c1nccs1 50315207C[C@H](C1=C(CCN(C)C)Cc2cc(C)ccc12)c1nccs1 50315208COc1ccc2C([C@@H](C)c3nccs3)=C(CCN(C)C)Cc2c1 50316513Cc1cc([nH]n1)C(=O)N[C@@H]1CC(C)(C)Oc2nc(-c3ccc(Cl)cc3Cl)c(cc12)-c1ccc(Cl)cc1 50316938CN1CCCC(C1)c1nc2ccccc2n1Cc1ccc(F)cc1 50316940CN1CCC[C@H](C1)c1nc2ccccc2n1Cc1ccc(F)cc1 50317865CC(C)(C)c1ccc(SCCc2cnc[nH]2)cc1 50319818FC(F)Oc1ccccc1CC(N1CCNCC1)c1ccccc1 50319828Fc1ccccc1C(Cc1ccccc1OC(F)(F)F)N1CCNCC1 50319830Fc1ccc(cc1)C(Cc1ccccc1OC(F)(F)F)N1CCNCC1 50320009Cc1ccccc1[C@H](OC[C@H](O)CNC(C)(C)Cc1ccc2ccccc2c1)C1CC1 50320377OCc1ccccc1S(=O)(=O)c1ccc(\C=C\c2ccc(F)cc2)cc1 50321337C(C1CCOCC1)C1CNCCN1c1ccc2[nH]ncc2c1 50321338COCCC1CNCCN1c1ccc2[nH]ncc2c1 50321339CCOCC1CNCCN1c1ccc2[nH]ncc2c1 50321340COCC1CNCCN1c1ccc2[nH]ncc2c1 50321341C(C1CCCCC1)C1CNCCN1c1ccc2[nH]ncc2c1 50321342CC(C)CC1CNCCN1c1ccc2[nH]ncc2c1 50321343CCCCC1CNCCN1c1ccc2[nH]ncc2c1 50321344CCC[C@@H]1CNCCN1c1ccc2[nH]ncc2c1 50321345CCC[C@H]1CNCCN1c1ccc2[nH]ncc2c1 50321346C(Cc1ccccc1)C1CNCCN1c1ccc2[nH]ncc2c1 50321347C1CN(C(CN1)c1ccccc1)c1ccc2[nH]ncc2c1 50321348C(C1CNCCN1c1ccc2[nH]ncc2c1)c1ccccc1 50321349C(C1CCOCC1)[C@H]1CNCCN1c1ccc2[nH]ncc2c1 50321350C(C1CCOCC1)[C@@H]1CNCCN1c1ccc2[nH]ncc2c1 50322696COC(CC=C)[C@@]12C[C@]1(CCNC2)c1ccc(Cl)c(Cl)c1 50322697COC[C@]12C[C@]1(CCNC2)c1ccc2ccccc2c1 50322698COC[C@]12C[C@]1(CCNC2)c1ccc(Cl)c(Cl)c1 50322852Cc1ncoc1-c1nnc(SCCCN2CC3CC3(C2)c2ccc(cc2)S(F)(F)(F)(F)F)n1C 50322854Cc1ncoc1-c1nnc(SCCCN2CC3CC3(C2)c2cccc(c2)S(F)(F)(F)(F)F)n1C 50322916CS(=O)(=O)N(c1ccccc1)c1cc(cc(c1)C(=O)N[C@@H](Cc1ccccc1)[C@H](O)CNCc1cccc(c1)C(F)(F)F)C1CCCC1 50325063CNC(=O)c1ccc(cc1)C(N1CCCN(CC1)C1CCC1)c1nnnn1Cc1ccccc1 50325065CN1CCN(Cc2ccc(cc2)C(N2CCCN(CC2)C2CCC2)c2nnnn2Cc2ccccc2)CC1 50325066C(c1ccccc1)n1nnnc1C(N1CCCN(CC1)C1CCC1)c1ccc(cc1)-n1cncn1 50325067C(c1ccc(cc1)C(N1CCCN(CC1)C1CCC1)c1nnnn1Cc1ccccc1)n1cncn1 50325068C(c1ccccc1)n1nnnc1C(N1CCCN(CC1)C1CCC1)c1ccc2occc2c1 50325449O=C(C1CCN(Cc2ccncc2)CC1)N1CCC(CC1)n1c2ccccc2n(CCN2CCCCC2)c1=O 50325461COc1cccc(Cn2c3ccccc3n(C3CCN(CC3)C(=O)C3CCN(Cc4ccncc4)CC3)c2=O)c1 50325462Clc1ccc(Cn2c3ccccc3n(C3CCN(CC3)C(=O)C3CCN(Cc4ccncc4)CC3)c2=O)cc1 50325463Clc1cccc(Cn2c3ccccc3n(C3CCN(CC3)C(=O)C3CCN(Cc4ccncc4)CC3)c2=O)c1 50325464Clc1ccccc1Cn1c2ccccc2n(C2CCN(CC2)C(=O)C2CCN(Cc3ccncc3)CC2)c1=O 50325465O=C(C1CCN(Cc2ccncc2)CC1)N1CCC(CC1)n1c2ccccc2n(Cc2ccccc2)c1=O 50325466CN(C)CCCn1c2ccccc2n(C2CCN(CC2)C(=O)C2CCN(Cc3ccncc3)CC2)c1=O 50325473CC(C)Cn1c2ccccc2n(C2CCN(CC2)C(=O)C2CCN(Cc3ccncc3)CC2)c1=O 50325614Fc1cc(cc2cc[nH]c12)C(=O)C1(Cc2ccccc2)CCNC1 50325615CCCC1(CCNC1)C(=O)c1cc(F)c2[nH]ccc2c1 50325616CC(C)CC1(CCNC1)C(=O)c1cc(F)c2[nH]ccc2c1 50325617CCOCC1(CCNC1)C(=O)c1cc(F)c2[nH]ccc2c1 50325618CCCCC1(CCNC1)C(=O)c1cc(F)c2[nH]ccc2c1 50325619CC(C)CCC1(CCNC1)C(=O)c1cc(F)c2[nH]ccc2c1 50325620CC(C)(C)CCC1(CCNC1)C(=O)c1cc(F)c2[nH]ccc2c1 50325622CC(C)(C)CCC1(CCNC1)C(=O)c1ccc(Cl)c(Cl)c1 50325625CC(C)(C)CCC1(CCNC1)C(=O)c1ccc(Cl)c(Cl)n1 50325626CC(C)(C)CCC1(CCNC1)C(=O)c1ccc(N)c(Cl)c1 50325631CCCC1(CCCN1)C(=O)c1ccc2[nH]ccc2c1 50325632CCCC1(CCCN1)C(=O)c1cc(F)c2[nH]ccc2c1 50325633CCCC1(CCCN1)C(=O)c1ccc(Cl)c(Cl)c1 50325634CCCC1(CCCN1)C(=O)c1ccc(N)c(Cl)c1 50325637CC(C)CC1(CCCN1)C(=O)c1ccc2[nH]ncc2c1 50325638CC(C)(C)CCC1(CCCN1)C(=O)c1ccc2[nH]ncc2c1 50325639CC(C)(C)CCC1(CCNC1)C(=O)c1ccc2ccccc2n1 50325640Cc1cccc2nc(ccc12)C(=O)C1(CCC(C)(C)C)CCNC1 50325933CNCC[C@@H](c1ccc(Cl)c(Cl)c1)n1nnc(C)n1 50326286FC(F)(F)c1ccc(SC[C@H](C2CCNCC2)c2cnc[nH]2)cc1 50326287CC(C)(C)c1ccc(SCC(c2cnc[nH]2)c2ccccn2)cc1 50326289FC(F)(F)c1ccc(SCC(c2cnc[nH]2)c2ccncc2)cc1 50326292CC(C)(C)c1ccc(SCC(C2CCNCC2)c2cnc[nH]2)cc1 50327481CC(C)N1CCC(CC1)Oc1ccc2n3CCNC(=O)c3cc2c1 50327484CC(C)N1CCC(CC1)Oc1ccc2n3CCN(CCO)C(=O)c3cc2c1 50329265Cc1cc(N[C@H](CCCCNCc2ccc(F)cc2)C(=O)NO)cc(C)c1F 50329312NC(=O)[C@@]12CC3CC(C1)[C@H](OC(=O)N1CC[C@H](C1)Nc1cccc(n1)C(F)(F)F)C(C3)C2 50332231Cn1c2cc(N3CCC[C@@](C)(N)C3)n(Cc3cc(F)ccc3Cl)c2c(=O)n(C)c1=O 50332233CCn1c2cc(N3CCC[C@@](C)(N)C3)n(Cc3cc(F)ccc3C#N)c2c(=O)n(C)c1=O 50332235Cn1c(=O)n(CCCO)c2cc(N3CCC[C@@](C)(N)C3)n(Cc3cc(F)ccc3Cl)c2c1=O 50334764CN[C@@H]1C[C@@H](c2ccc(Cl)c(Cl)c2)c2ccccc2C1 50334765CN[C@H]1C[C@H](c2ccc(Cl)c(Cl)c2)c2ccccc2C1 50334766CN[C@H]1C[C@@H](c2ccc(Cl)c(Cl)c2)c2ccccc2C1 50334767CN[C@@H]1C[C@H](c2ccc(Cl)c(Cl)c2)c2ccccc2C1 50334775CNC[C@@H]1C[C@@H](c2ccc(Cl)c(Cl)c2)c2ccccc2C1 50334776CNC[C@H]1C[C@H](c2ccc(Cl)c(Cl)c2)c2ccccc2C1 50334777CNC[C@H]1C[C@@H](c2ccc(Cl)c(Cl)c2)c2ccccc2C1 50334781NCC[C@H]1C[C@@H](c2ccc(Cl)c(Cl)c2)c2ccccc2C1 50334783CN[C@H]1CCc2ccccc2[C@@H]1c1ccc(Cl)c(Cl)c1 50334784CN[C@@H]1CCc2ccccc2[C@@H]1c1ccc(Cl)c(Cl)c1 50334785CN[C@@H]1CCc2ccccc2[C@H]1c1ccc(Cl)c(Cl)c1 50334786CN[C@H]1CCc2ccccc2[C@H]1c1ccc(Cl)c(Cl)c1 50334917CNC1CCN(c2ccc(Cl)c(Cl)c2)c2ccccc12 50334918N[C@@H]1CCN(c2ccc(Cl)c(Cl)c2)c2ccccc12 50334919CN[C@@H]1CCN(c2ccc(Cl)c(Cl)c2)c2ccccc12 50334920CN(C)[C@@H]1CCN(c2ccc(Cl)c(Cl)c2)c2ccccc12 50334925CN[C@@H]1CN(c2ccc(Cl)c(Cl)c2)c2ccccc2C1 50334932CCCCN(C)C(=O)c1ccc(cc1)-n1nc(c2CCCCc12)C(F)(F)F 50334936FC(F)(F)c1nn(c2CCCCc12)-c1ccc(CC(=O)NC2CCCC2)cc1 50334941CS(=O)(=O)c1ccc(cc1)-n1nc(c2CCCCc12)C(F)(F)F 50334943FC(F)(F)c1nn(c2CCCCc12)-c1ccc(cc1)C(=O)N1CCCC1 50334950CN(C)C(=O)c1ccc(cc1)-n1nc(c2CCCCc12)C(F)(F)F 50335379[#6]-c1ccc(-[#7]-[#6](=O)-[#7]-2-[#6]-[#6]\[#6](-[#6]-[#6]-2)=[#6]\c2cccc(-[#8]-c3ccc(cn3)C(F)(F)F)c2)cn1 50335380FC(F)(F)c1ccc(-[#8]-c2cccc(\[#6]=[#6]-3\[#6]-[#6]-[#7](-[#6]-[#6]-3)-[#6](=O)-[#7]-c3cccnc3)c2)nc1 50336066CCN(C)CCC1=C(Cc2cnccn2)c2ccccc2C1 50336067CCCN(C)CCC1=C(Cc2cnccn2)c2ccccc2C1 50336068CN(CCF)CCC1=C(Cc2cnccn2)c2ccccc2C1 50336069C[C@H](C1=C(CCN(C)CCF)Cc2ccccc12)c1cnccn1 50336072C[C@H](C1=C(CCN(C)CCC(F)(F)F)Cc2ccccc12)c1cnccn1 50336073C(CC1=C(Cc2cnccn2)c2ccccc2C1)N1CCC1 50336074C(CC1=C(Cc2cnccn2)c2ccccc2C1)N1CCCC1 50336075FC1CN(CCC2=C(Cc3cnccn3)c3ccccc3C2)C1 50336077FC1(F)CCN(CCC2=C(Cc3cnccn3)c3ccccc3C2)C1 50336078FC1CCN(CCC2=C(Cc3cnccn3)c3ccccc3C2)C1 50336079C[C@H](C1=C(CCN(C)Cc2ccco2)Cc2ccccc12)c1cnccn1 50336080C[C@H](C1=C(CCN(C)Cc2cccs2)Cc2ccccc12)c1cnccn1 50336083C[C@H](C1=C(CCN(C)Cc2ncc[nH]2)Cc2ccccc12)c1cnccn1 50336084C[C@H](C1=C(CCN(C)Cc2nccn2C)Cc2ccccc12)c1cnccn1 50336085C[C@H](C1=C(CCN(C)Cc2ccccn2)Cc2ccccc12)c1cnccn1 50336086C[C@H](C1=C(CCN(C)Cc2ccncc2)Cc2ccccc12)c1cnccn1 50336088C[C@H](C1=C(CCN(C)CC2CCOCC2)Cc2ccccc12)c1cnccn1 50336974O=C(Nc1cnc(-c2ccncc2)c(n1)-c1ccco1)C1CC1 50336976O=C(Nc1cnc(-c2ccncc2)c(n1)-c1ccncc1)C1CC1 50337104C[C@@H](OC[C@H](O)CNC(C)(C)Cc1ccc2ccccc2c1)c1ccccc1CCC(O)=O 50337105CC(C)(Cc1ccc2ccccc2c1)NC[C@@H](O)CO[C@H](C1CC1)c1ccccc1CO 50337910CNC(C)C1(CCCCC1)c1ccc(Cl)c(Cl)c1 50338821Nc1nc(CC(=O)Nc2ccc(C[C@@H]3CC[C@@H](N3)[C@H](O)c3ccccc3)cc2)cs1 50339996CNCC[C@@H](Oc1cc(Cl)ccc1C#N)c1ccccc1 50339997NCC[C@@H](Oc1cc(Cl)ccc1C#N)c1ccccc1 50339998NCC[C@@H](Sc1cc(Cl)ccc1C#N)c1ccccc1 50339999CNCC[C@@H](Oc1cc(ccc1C#N)C(F)(F)F)c1ccccc1 50340000CNCC[C@@H](Oc1cc(OC)ccc1C#N)c1ccccc1 50340001CCC(CCNC)Oc1cc(Cl)ccc1C#N 50340002NCC[C@@H](Oc1cc(Cl)c(F)cc1C#N)c1ccccc1 50340003Cc1ccc(C#N)c(S[C@H](CCN)c2ccccc2)n1 50340754Cc1cc(C[C@H](CCCCNCc2ccc(F)cc2)C(=O)NO)cc(C)c1F 50340758CO[C@H](C[C@H](CCCCNCc1ccc(F)cc1)C(=O)NO)c1ccc(F)cc1 50340768Cc1cc(O[C@H](CCCCNCc2ccc(F)cc2)C(=O)NO)cc(C)c1F 50341075COc1ccccc1N1CCN(CC1)C(=O)c1cc(n[nH]1)-c1ccc(Cl)cc1 50341447Clc1ccc(Cc2nn(C[C@H]3CCCN3CCCCc3ccc(OCCCN4CCCCCC4)cc3)c(=O)c3ccccc23)cc1 50341448CN1CCCC(CC1)n1nc(Cc2ccc(Cl)cc2)c2ccccc2c1=O 50342128COC(=O)C(C)(C)C(c1ccc(Nc2ccc3ccccc3c2)cc1)n1ccnc1 50342133C[C@H]([C@@H](c1ccc(Nc2nc3ccccc3s2)cc1)n1ccnc1)N(C)C 50344232COc1cc(F)ccc1-c1cncc(CNCC2CC2)n1 50344250COc1cc(F)ccc1-c1cncc(CNC2CCCC2)c1 50344584Cn1c(-c2ccoc2)c(C2CCCCC2)c2ccc(cc12)C(=O)NC(C)(C)C(=O)Nc1ccc(\C=C\C(O)=O)cc1 50350378CN1C[C@H]2CCCC[C@]2(C1)c1ccc(Cl)c(Cl)c1 50350379CN1C[C@@H]2CCCC[C@@]2(C1)c1ccc(Cl)c(Cl)c1 50350380Clc1ccc(cc1Cl)[C@@]12CNC[C@@H]1CCCC2 50350381Clc1ccc(cc1Cl)[C@]12CNC[C@H]1CCCC2 50350382CCN1C[C@H]2CCCC[C@]2(C1)c1ccc(Cl)c(Cl)c1 50350383CCN1C[C@@H]2CCCC[C@@]2(C1)c1ccc(Cl)c(Cl)c1 50350384CN1C[C@@H]2CCCC[C@@]2(C1)c1ccc2ccccc2c1 50350386CN1C[C@@H]2CCC[C@@]2(C1)c1ccc(Cl)c(Cl)c1 50350387CN1C[C@H]2CCC[C@]2(C1)c1ccc(Cl)c(Cl)c1 50350388Clc1ccc(cc1Cl)[C@]12CCC[C@H]1CNC2 50350389Clc1ccc(cc1Cl)[C@@]12CCC[C@@H]1CNC2 50350390C1C[C@H]2CNC[C@]2(C1)c1ccc2ccccc2c1 50350392CN1C[C@@H]2CCC[C@@]2(C1)c1ccc2ccccc2c1 50351399Cn1c2cc(N3CCC[C@@H](N)C3)n(Cc3cc(F)ccc3C#N)c2c(=O)n(C)c1=O 50352702Cc1c(Cl)cccc1N1CCN(CCCNC(=O)c2nc(-c3ccccc3)n(c2Cn2cncn2)-c2ccccc2)CC1 50352707Cc1c(nc(-c2ccccc2)n1-c1ccccc1)C(=O)NCCCN1CCN(CC1)c1cccc(Cl)c1C 50353232CCCCCCc1nc2cc(\C=C\C(=O)NO)ccc2n1CCN(C)C 50353578COC(=O)C(C)(C)C(c1ccc(Nc2ccc3ccccc3c2)cc1)n1cncn1 50355852CN(C)S(=O)(=O)NCCCCCNc1nc(cs1)-c1ccccn1 50356019Cc1c(O)c2ccccc2nc1COc1cccc(OCCCC(F)(F)F)c1 50356020COC(C)(C)CCOc1cccc(OCc2nc3ccccc3c(O)c2C)c1 50356024Cc1c(COc2cccc(OCC3CCOCC3)n2)nc2ccccc2c1O 50356025CCCCOc1cccc(OCc2nc3ccccc3c(O)c2C)c1 50356029CCCCCCC=CCc1nc2ccccc2c(O)c1C 50356030Cc1c(COc2cccc(OCC3CCOCC3)c2)nc2ccccc2c1O 50356031Cc1c(COc2cccc(OCC3CCOCC3)c2)nc2ccc(cc2c1O)-c1cccnc1 50357427CC(C)(C)c1cc(C(=O)Nc2nc(CN)cs2)n(Cc2ccccc2)n1 50360603Clc1ccc2[nH]c(cc2c1)C(=O)N1C[C@]2(CCN(C2)C2CCNC2)c2ccccc12 50360611Fc1ccc2cc([nH]c2c1)C(=O)N1C[C@]2(CCN(C2)C2CCNC2)c2ccccc12 50360973O=S1(=O)CCC(CC1)Oc1ccc2OC3(CCN(CC3)C3CCC3)CCc2c1 50360994CN(C)C(=O)CN1CCCC(C1)c1nc2ccccc2n1Cc1ccc(F)cc1 50360995CCN(CC)C(=O)CN1CCCC(C1)c1nc2ccccc2n1Cc1ccc(F)cc1 50360996Fc1ccc(Cn2c(nc3ccccc23)C2CCCN(CC(=O)N3CCCCC3)C2)cc1 50360999OCCN1CCCC(C1)c1nc2ccccc2n1Cc1ccc(F)cc1 50361003CN(C)C(=O)CN1CCCC(C1)c1nc2ccccc2n1CCOc1ccccc1 50361006Cc1ccc(Cn2c(nc3ccccc23)C2CNCCO2)cc1C 50361007Cc1ccc(Cn2c(nc3ccccc23)C2CNCCS2)cc1 50361008Fc1ccc(Cn2c(nc3ccccc23)[C@H]2CNCCS2)cc1 50361009COc1ccc(Cn2c(nc3ccccc23)[C@H]2CNCCS2)cc1 50363196CN1C\C=C\CCOc2cccc(c2)-c2ccnc(Nc3cccc(C1)c3)n2 50364664CCCOc1sc(C(=O)N2CCC(CC2)c2cccc(CN)c2)c(C)c1Br 50364665CCCOc1sc(C(=O)N2[C@H]3CC[C@H]2CC(C3)c2cc(CN)ccc2F)c(C)c1Br 50364777COc1cc(NCC2CCNCC2)nc2n(nnc12)-c1cccc(OC(F)(F)F)c1 50366567CNCC[C@@H](Oc1ccccc1C)c1ccccc1 50366613COc1ccc2C[C@H]3[C@H]4CCCC[C@@]4(CCN3C)c2c1 50367247COc1ccc2nccc([C@@H](O)[C@@H]3C[C@@H]4CCN3C[C@@H]4C=C)c2c1 50370411O[C@H]([C@H]1C[C@@H]2CC[N@]1C[C@@H]2C=C)c1ccnc2ccccc12 50371684CC(C)(N)C(=O)N[C@H](COCc1ccccc1)c1nnnn1[C@@H](COc1ccccc1O)CC#N 50372824CCC[C@H](C[C@@H](O)N1CCC[C@@H](Cc2ccc(F)cc2)C1)NC(=O)Nc1cccc(c1)-c1nnnn1C 50372825C[C@H](C[C@@H](O)N1CCC[C@@H](Cc2ccc(F)cc2)C1)NC(=O)Nc1cc(cc(c1)-n1ccnn1)-n1ccnn1 50372826C[C@H](C[C@@H](O)N1CCC[C@@H](Cc2ccc(F)cc2)C1)NC(=O)Nc1cc(cc(c1)-n1cccn1)-n1cccn1 50372827C[C@H](C[C@@H](O)N1CCC[C@@H](Cc2ccc(F)cc2)C1)NC(=O)Nc1cc(C)cc(c1)-c1nnnn1C 50372829C[C@H](CC(=O)N1CCC[C@@H](Cc2ccc(F)cc2)C1)NC(=O)Nc1cccc(c1)-c1nnnn1C 50372830C[C@H](CCN1CCC[C@@H](Cc2ccc(F)cc2)C1)NC(=O)Nc1cc(cc(c1)-n1cccn1)-n1cccn1 50372831C[C@@H](CCN1CCC[C@@H](Cc2ccc(F)cc2)C1)NC(=O)Nc1cc(cc(c1)C(C)=O)C(C)=O 50372833CCc1cc(NC(=O)N[C@H](C)CCN2CCC[C@@H](Cc3ccc(F)cc3)C2)cc(c1)-c1nnnn1C 50372834C[C@H](CCN1CCC[C@@H](Cc2ccc(F)cc2)C1)NC(=O)Nc1cccc(c1)-c1nnnn1C 50372835C[C@H](C[C@@H](C)N1CCC[C@@H](Cc2ccc(F)cc2)C1)NC(=O)Nc1cccc(c1)-c1nnnn1C 50372836CNC(=O)O[C@H](C[C@@H](C)NC(=O)Nc1cccc(c1)-c1nnnn1C)N1CCC[C@@H](Cc2ccc(F)cc2)C1 50372837C[C@H](C[C@@H](O)N1CCC[C@@H](Cc2ccc(F)cc2)C1)NC(=O)Nc1cc(cc(c1)-c1ccon1)-c1ccon1 50372838C[C@H](C[C@@H](O)N1CCC[C@@H](Cc2ccc(F)cc2)C1)NC(=O)Nc1cccc(c1)-c1nccn1C 50372839CCc1cc(NC(=O)N[C@H](C)C[C@@H](O)N2CCC[C@@H](Cc3ccc(F)cc3)C2)cc(c1)-c1nnnn1C 50372840Fc1ccc(C[C@@H]2CCCN(CCCNC(=O)Nc3cc(cc(c3)-n3cccn3)-n3cccn3)C2)cc1 50372841CC(C)c1cc(NC(=O)NCCCN2CCC[C@@H](Cc3ccc(F)cc3)C2)cc(c1)-c1nnnn1C 50372842C[C@H](CCN1CCC[C@@H](Cc2ccc(F)cc2)C1)NC(=O)Nc1cc(cc(c1)-c1nnnn1C)C(C)C 50372843CCc1cc(NC(=O)NCCCN2CCC[C@@H](Cc3ccc(F)cc3)C2)cc(c1)-c1nnnn1C 50372844C[C@H](CCN1CCC[C@@H](Cc2ccc(F)cc2)C1)NC(=O)Nc1cc(C)cc(c1)-c1nnnn1C 50372845CCc1cc(NC(=O)N[C@H](C)C[C@@H](N(C)C)N2CCC[C@@H](Cc3ccc(F)cc3)C2)cc(c1)-c1nnnn1C 50372846C[C@H](C[C@@H](NC(C)=O)N1CCC[C@@H](Cc2ccc(F)cc2)C1)NC(=O)Nc1cccc(c1)-c1nnnn1C 50372847C[C@H](C[C@@H](N)N1CCC[C@@H](Cc2ccc(F)cc2)C1)NC(=O)Nc1cccc(c1)-c1nnnn1C 50372848CC(C)C[C@H](C[C@@H](O)N1CCC[C@@H](Cc2ccc(F)cc2)C1)NC(=O)Nc1cccc(c1)-c1nnnn1C 50372849CC(C)[C@H](C[C@@H](O)N1CCC[C@@H](Cc2ccc(F)cc2)C1)NC(=O)Nc1cccc(c1)-c1nnnn1C 50372850CC[C@H](C[C@@H](O)N1CCC[C@@H](Cc2ccc(F)cc2)C1)NC(=O)Nc1cccc(c1)-c1nnnn1C 50372851C[C@H](C[C@@H](O)N1CCC[C@@H](Cc2ccc(F)cc2)C1)NC(=O)Nc1cc(cc(c1)-c1ncco1)-c1ncco1 50372852C[C@H](CCN1CCC[C@@H](Cc2ccc(F)cc2)C1)NC(=O)Nc1cc(cc(c1)-n1ccnn1)-n1ccnn1 50372853C[C@H](C[C@@H](O)N1CCC[C@@H](Cc2ccc(F)cc2)C1)NC(=O)Nc1cc(cc(c1)-c1nccs1)-c1nccs1 50372854C[C@H](C[C@@H](O)N1CCC[C@@H](Cc2ccc(F)cc2)C1)NC(=O)Nc1cc(cc(c1)-c1nnnn1C)C(C)C 50372855C[C@H](C[C@@H](O)N1CCC[C@@H](Cc2ccc(F)cc2)C1)NC(=O)Nc1cc(Br)cc(c1)-c1nnnn1C 50372856C[C@H](CCN1CCC[C@@H](Cc2ccc(F)cc2)C1)NC(=O)Nc1cc(Br)cc(c1)-c1nnnn1C 50372857C[C@H](C[C@@H](O)N1CCC[C@@H](Cc2ccc(F)cc2)C1)NC(=O)Nc1cc(cc(c1)C(C)=O)C(C)=O 50372858C[C@@H](CCN1CCC[C@@H](Cc2ccc(F)cc2)C1)NC(=O)Nc1cccc(c1)-c1nnnn1C 50372859CCC[C@H](CCN1CCC[C@@H](Cc2ccc(F)cc2)C1)NC(=O)Nc1cc(cc(c1)C(C)(C)O)-c1nnnn1C 50372860CC[C@H](CCN1CCC[C@@H](Cc2ccc(F)cc2)C1)NC(=O)Nc1cc(cc(c1)C(C)(C)O)-c1nnnn1C 50372861C[C@H](CCN1CCC[C@@H](Cc2ccc(F)cc2)C1)NC(=O)Nc1cc(cc(c1)-c1nnnn1C)C(C)=O 50372862C[C@H](CCN1CCC[C@@H](Cc2ccc(F)cc2)C1)NC(=O)Nc1cc(cc(c1)C(C)=O)C(C)=O 50375697CN(C)Cc1cnc(C)cc1Oc1ccccc1Oc1ccccc1 50376027COc1cc2nccc(Oc3ccc4c(cccc4c3)C(=O)Nc3ccncc3)c2cc1OC 50377214Cc1cc2ncc(=O)n(CC(=O)N3CCCC(C3CN3CCOCC3)c3ccccc3)c2cc1C 50377215Cc1cc2ncc(=O)n(CC(=O)N3CCCC(C3CN3CCCC3)c3ccccc3)c2cc1C 50377217Clc1cc2ncc(=O)n(CC(=O)N3CCCC(C3CN3CCCC3)c3ccccc3)c2cc1Cl 50377218Cc1cc2OCC(=O)N(CC(=O)N3CCCC(C3CN3CCCC3)c3ccccc3)c2cc1C 50377219Clc1cc2OCC(=O)N(CC(=O)N3CCCC(C3CN3CCOCC3)c3ccccc3)c2cc1Cl 50377220Clc1cc2OCC(=O)N(CC(=O)N3CCCC(C3CN3CCCC3)c3ccccc3)c2cc1Cl 50377221COCCN(CC(=O)N1CCCC(C1CN1CCOCC1)c1ccccc1)c1ccc(Cl)c(Cl)c1 50377222COCCN(CC(=O)N1CCCC(C1CN1CCCC1)c1ccccc1)c1ccc(Cl)c(Cl)c1 50377223Clc1ccc(cc1Cl)N(CC#N)CC(=O)N1CCCC(C1CN1CCOCC1)c1ccccc1 50377224Clc1ccc(cc1Cl)N(CC#N)CC(=O)N1CCCC(C1CN1CCCC1)c1ccccc1 50377225CN(CC(=O)N1CCCC(C1CN1CCOCC1)c1ccccc1)c1ccc(Cl)c(Cl)c1 50377226Clc1ccc2sc(=O)n(CC(=O)N3CCCC(C3CN3CCOCC3)c3ccccc3)c2c1 50377227Clc1ccc2sc(=O)n(CC(=O)N3CCCC(C3CN3CCCC3)c3ccccc3)c2c1 50377228Clc1ccc2oc(=O)n(CC(=O)N3CCCC(C3CN3CCOCC3)c3ccccc3)c2c1 50377229Clc1ccc2oc(=O)n(CC(=O)N3CCCC(C3CN3CCCC3)c3ccccc3)c2c1 50377956Fc1ccc2cc(CN3[C@@H]4CC[C@@H]3CC(C4)NC(=O)c3ccccc3-c3cncnc3)ccc2c1 50378146CCOC(=O)CCc1ccc(OC[C@H](O)CNC(C)(C)Cc2ccc3ccccc3c2)c(c1)C#N 50379157Cc1nc2cc(OC(F)(F)F)ccc2n1-c1ccc(s1)C(=O)NC1CC1 50379533CCC(NCCCC[C@@H](C[C@@H](OC)c1ccc(F)cc1)C(=O)NO)c1ccc(F)cc1 50379534CCC(NCCCC[C@@H](Oc1cc(C)c(F)c(C)c1)C(=O)NO)c1ccc(F)cc1 50379535CCC(NCCCC[C@@H](Cc1cc(C)c(F)c(C)c1)C(=O)NO)c1ccc(F)cc1 50379536CCC(NCCCC[C@@H](Nc1cc(C)c(F)c(C)c1)C(=O)NO)c1ccc(F)cc1 50379670Oc1ccc2nc([nH]c2c1CN1CCCCC1)-c1ccccc1 50379681C(N1CCCCC1)c1cccc2nc([nH]c12)-c1ccccc1 50379684Fc1ccc2nc([nH]c2c1CN1CCCC1)-c1ccccc1 50380410Fc1ccc(Oc2ccc(NC(=O)[C@@H]3C[C@@H](Cc4ccccc4)CN3C(=O)Cn3cncn3)cc2)cc1 50380412Fc1ccc(C[C@H]2C[C@H](N(C2)C(=O)Cn2cncn2)C(=O)Nc2ccc(Oc3ccc(F)cc3)cc2)cc1 50380415Fc1ccc(Oc2ccc(NC(=O)[C@@H]3C[C@@H](Cc4ccccc4)CN3C(=O)Cc3cnc[nH]3)cc2)cc1 50380416Fc1ccc(Oc2ccc(NC(=O)[C@@H]3C[C@H](CN3C(=O)Cc3cnc[nH]3)c3ccccc3)cc2)cc1 50380417Fc1ccc(C[C@@H]2C[C@H](N(C2)C(=O)Cn2cncn2)C(=O)Nc2ccc(Oc3ccc(F)cc3)cc2)cc1 50380505COc1ccc2nc(SCc3ccc(Cl)cc3)[nH]c2c1 50380506COc1ccc2nc(SCc3ccc(Br)cc3)[nH]c2c1 50380507COc1ccc2nc(SCc3ccc(I)cc3)[nH]c2c1 50380508COc1ccc2nc(SCc3cccc(c3)-c3ccccc3)[nH]c2c1 50380510COc1ccc2nc(SCc3cccc(Oc4ccccc4)c3)[nH]c2c1 50380511COc1ccc2nc(SCc3ccc(OCc4ccccc4)cc3)[nH]c2c1 50380514C(Sc1nc2ccccc2[nH]1)c1ccccn1 50380517Nc1ccc2nc(SCc3ccccn3)[nH]c2c1 50380518CCSc1nc2ccc(OC)cc2[nH]1 50380519CCCSc1nc2ccc(OC)cc2[nH]1 50380520CCCCSc1nc2ccc(OC)cc2[nH]1 50380522CCCCCCSc1nc2ccc(OC)cc2[nH]1 50380527COc1ccc2nc(SCCCO)[nH]c2c1 50380529COc1ccc2nc(SCc3ccccc3)[nH]c2c1 50380530COc1ccc2nc(SCc3ccc(C)cc3)[nH]c2c1 50380531COc1ccc2nc(SCc3ccc(cc3)C(C)C)[nH]c2c1 50380532COc1ccc2nc(SCc3ccc(cc3)C(C)(C)C)[nH]c2c1 50380534CCCCCCCSc1nc2ccc(OC)cc2[nH]1 50380592COc1ccc(cc1)-n1c(SCc2nc(no2)-c2ccc(C)cc2)nnc1-c1ccncc1 50382558Cc1cccc(c1)C(CCCN)(c1ccccc1)c1ccccc1 50384896CN[C@H]1CC[C@H](CC1)c1c[nH]c2ccc(cc12)N=C(N)c1cccs1 50384898CCN[C@H]1CC[C@H](CC1)c1c[nH]c2ccc(cc12)N=C(N)c1cccs1 50384899CN[C@H]1CCC[C@H](C1)c1c[nH]c2ccc(cc12)N=C(N)c1cccs1 50384930CCOC(=O)N1CCN(CC(=O)c2ccc(OCCCN3CCC[C@H]3C)cc2)CC1 50385469Clc1ccc(NC(=O)N2CCN(C[C@@H]3CCCN(C3)C3CC3)CC2)cc1Cl 50385791CNC(=O)c1ccc(cc1)-c1ccc(cc1)N1C(=O)N(c2cc(OC)ncn2)C2(CCN(Cc3ncccc3C)CC2)C1=O 50387877CCN1CCN(CC1)c1nc(C)nc2sc(cc12)-c1ccccc1 50388470CCc1c(CCCC(O)=O)cccc1-c1cnc(nc1)-c1ccc(OC(C)C)c(c1)C#N 50389658O=C(NCc1ccncc1)c1nnc(CS(=O)(=O)c2ccccc2)o1 50389659O=C(NCc1ccncc1)c1nc(CS(=O)(=O)c2ccccc2)no1 50390396CS(=O)(=O)c1ccc2nc(sc2c1)N1CCN(CC1)C(=O)[C@@H]1CCCC[C@H]1C(=O)NC1(CC1)C#N 50392994C1CCN(CC1)[C@H]([C@@H](N1CCCCC1)c1ccccc1)c1ccccc1 50392995C1CCN(CC1)[C@@H]([C@H](N1CCCCC1)c1ccccc1)c1ccccc1 50392996C1CCN(C1)[C@H]([C@@H](N1CCCC1)c1ccccc1)c1ccccc1 50392997C1CCN(C1)[C@@H]([C@H](N1CCCC1)c1ccccc1)c1ccccc1 50397830COc1nc(Nc2cccc3n(C)c(nc23)-c2ccc(F)cc2)ccc1-n1cnc(C)c1 50398687CN1C(N)=N[C@]2(CN(C[C@H]2C1=O)c1ccc(F)cn1)c1cc(cs1)-c1cccc(c1)C#N 50399004CN1C[C@@H]([C@H](C1)c1ccc(\C=C\C(=O)Nc2ccccc2N)cc1F)C(=O)Nc1ccc(Cl)cc1 50399006CN1C[C@@H]([C@H](C1)c1ccc(\C=C\C(=O)Nc2ccccc2N)cc1)C(=O)Nc1ccc(Cl)cc1 50399007Nc1ccccc1NC(=O)\C=C\c1ccc(cc1)[C@H]1CN(CCO)C[C@@H]1C(=O)Nc1ccc(Cl)cc1 50399008CC(C)(O)CN1C[C@@H]([C@H](C1)c1ccc(\C=C\C(=O)Nc2ccccc2N)cc1)C(=O)Nc1ccc(Cl)cc1 50400880Cc1ccc(Sc2ccccc2N2CCNCC2)cc1 50400882Clc1ccc(Sc2ccccc2N2CCNCC2)cc1 50400889Cc1cccc(Sc2ccccc2N2CCNCC2)c1C 50400890Clc1cccc(Sc2ccccc2N2CCNCC2)c1Cl 50400892Cc1ccc(Sc2ccccc2N2CCNCC2)cc1C 50400899Cc1ccc(Sc2ccccc2N2CCNCC2)c(Cl)c1 50400902Cc1ccc(Sc2ccccc2N2CCNCC2)c(C)c1 50400903Clc1ccc(Sc2ccccc2N2CCNCC2)c(Cl)c1 50401154COC(=O)C(C)(C)C(c1ccc(Nc2ccccc2)cc1)n1cncn1 50401271NC(=Nc1ccc2N(CCc2c1)C1CCNCC1)c1cccs1 50401730CN1C[C@@H](c2ccc(F)cc2)c2ccc(C)cc2C1 50407151COC(=O)C1=CO[C@H](C)[C@H]2CN3CCc4c([nH]c5ccccc45)[C@@H]3C[C@H]12 50407152COC(=O)[C@H]1[C@H](O)CC[C@H]2CN3CCc4c([nH]c5ccccc45)[C@@H]3C[C@H]12 50407153CCC1CN2CCC1CC2[C@H](O)c1ccnc2ccccc12 50407154CCC1CN2CCC1CC2[C@H](O)c1ccnc2ccc(OC)cc12 50407155O[C@@H]([C@@H]1CC2CCN1CC2C=C)c1ccnc2ccc(Cl)cc12 50407156COC(=O)C1=CO[C@@H](C)[C@@H]2CN3CCc4c([nH]c5ccccc45)[C@@H]3C[C@H]12 50407157CCC1CN2CCC1CC2[C@@H](O)c1ccnc2ccc(OC)cc12 50407158O[C@H]([C@H]1CC2CCN1CC2C=C)c1ccnc2ccc(Cl)cc12 50409213O=C(N[C@H]1CC[C@H](CCN2CCc3ccc(cc3C2)C#N)CC1)c1cc2ccccc2[nH]1 50410855COc1ccc2nccc([C@H](O)[C@H]3CC4CCN3C[C@@H]4C=C)c2c1 50412340CC(C)OC(=O)c1ccc(NC(=O)N[C@@H](Cc2ccc(O)cc2)C(=O)N[C@H]2CCC[N+](C)(Cc3cccc(O)c3)C2)cc1 50413014CCCCNc1nccc2[nH]c3ccccc3c12 50415478CCOC[C@H]1[C@@H]2CNC[C@]12C 50418098CCN(CC1CCN(CC1)S(C)(=O)=O)[C@@H](C)Cc1ccc2OCCc2c1 50418099CCc1nc(C)c(CN2CCN(CC2)c2cc(ccn2)C(F)(F)F)[nH]1 50418100Fc1cnc(nc1)N1CCN(Cc2cnc([nH]2)-c2ccccc2)CC1 50418123CCCCN(c1cccc(-c2ccc(OC(F)(F)F)cc2)c1Cl)S(=O)(=O)c1ccc(OC(C)C(O)=O)c(C)c1C 50418124CCCCN(c1cccc(-c2ccc(cc2)C(F)(F)F)c1Cl)S(=O)(=O)c1ccc(OC(C)C(O)=O)c(C)c1C 50422013CN1[C@@H](C[C@H](O)c2ccccc2)CCC[C@H]1CC(=O)c1ccccc1 50426342CN1CC=CCC(C1)c1cc2ccccc2o1 50426345Fc1ccc(cc1Cl)C1CNCC=CC1 50426348Cc1ccc(cc1Cl)C1CNCC=CC1 50426349C1NCC(CC=C1)c1ccc2ccccc2c1 50426350Clc1ccc(cc1Cl)[C@H]1CNCC=CC1 50426351Clc1ccc(cc1Cl)[C@@H]1CNCC=CC1 50426352CN1CC=CC[C@@H](C1)c1ccc(Cl)c(Cl)c1 50426358COCCN1CC=CC[C@@H](C1)c1ccc(Cl)c(Cl)c1 50426360Clc1ccc(cc1Cl)C1CCCCNC1 50426362C1NCC(CC=C1)c1cc2ccccc2o1 50427800C[C@@H](CN1CCC2(CC1)N(CNC2=O)c1cccc(C)c1)NC(=O)c1ccc(Br)cc1 50428596CC(C)(C)NC(=O)NCCN1CCCC(C1)NC(=O)c1cc(Cl)cc(Cl)c1 50428597CC(C)(C)NC(=O)NCCN1CCC(C1)NC(=O)c1cc(Cl)cc(Cl)c1 50428598CC(C)(C)NC(=O)NCCN1CC(C1)NC(=O)c1cc(Cl)cc(Cl)c1 50428599CC(C)(C)NC(=O)NCCN1CCC(CNC(=O)c2cc(Cl)cc(Cl)c2)C1 50428601CC(C)(C)NC(=O)NCCN1CCCC(CNC(=O)c2cc(Cl)cc(Cl)c2)C1 50428602CC(C)(C)NC(=O)NCCN1CCC(CNC(=O)c2cc(Cl)cc(Cl)c2)CC1 50428603CC(C)(C)NC(=O)NCCN1CCN(CC(=O)Nc2cc(Cl)cc(Cl)c2)CC1 50429069COc1cc2CCN3CC[C@@](O)(C[C@@H]3c2cc1O)c1ccc(OC(F)(F)F)cc1 50431134COc1cccc(CN(CCN(C)C)C(=O)Nc2ccc(cc2)-c2cn[nH]c2)c1 50431380CC(C)(C)NC(=O)c1c[nH]c2ncc(nc12)-c1n[nH]c2c(cccc12)C(C)(C)O 50431398Cc1ccc2c(nn(C)c2c1)-c1cnc2[nH]cc(C(=O)NC3(C)CCNC3)c2n1 50434673Cc1cccc(c1)-c1ccc2c3nc([nH]c3c(=O)[nH]c2c1)-c1c(F)cccc1Cl 50436481Cc1nc(NC(=O)CN(Cc2ccccc2)C(=O)c2ccncc2)sc1-c1ccc(N)nc1 50436482Nc1ccc(cn1)-c1cnc(NC(=O)CN(Cc2ccccc2)C(=O)c2ccncc2)s1 50436849C[C@]1(CCOC(N)=N1)c1cc(NC(=O)c2ncc(Cl)cc2Cl)ccc1F 50437809Nc1ccccc1NC(=O)c1ccc(CN=C2N[C@H](CS2)c2ccccc2)cc1 50437837CN(C)Cc1ccc(\C=C\c2n[nH]c3cc(\C=C4\C(=O)Nc5ccccc45)ccc23)cc1 50438845CC(C)(C)n1nnnc1C(N1CCCC1)c1cccc(Nc2ccnc3cc(Cl)ccc23)c1 50438846CCN(CC)C(c1nnnn1C(C)(C)C)c1cccc(Nc2ccnc3cc(Cl)ccc23)c1 50439304O=C(NCc1ccc(cc1)S(=O)(=O)c1ccccc1)N1Cc2ccncc2C1 50440366Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(cc1)-c1n[nH]c(=S)n1C)C(C)(C)C 50440367Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(cc1)-n1cnnc1)C(C)(C)C 50440368Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(cc1)-n1ccnc1)C(C)(C)C 50441514Nc1cc(CN2CCC(F)(CC2)C(=O)N2CCC(CC2)N2Cc3ccccc3-c3ccccc3C2)ccn1 50441569Nc1ccc(cn1)-c1cnc2[nH]cc(-c3ccc4[nH]ccc4c3)c2c1 50443195C[C@H](C(=O)Nc1ccc(cc1)-c1ccnc(C)c1)c1cc(cc(c1)C(F)(F)F)C(F)(F)F 50443196C[C@@H](C(=O)Nc1ccc(cc1)-c1ccnc(C)c1)c1cc(cc(c1)C(F)(F)F)C(F)(F)F 50443200CCCc1cc(ccn1)-c1ccc(NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)cc1 50443201CCc1cc(ccn1)-c1ccc(NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)cc1 50443202FC(F)(F)c1cc(cc(c1)S(=O)(=O)Nc1ccc(cc1)-c1ccnc(C=C)c1)C(F)(F)F 50443203COc1cc(ccc1NS(=O)(=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)-c1ccnc(C)c1 50443204Cc1cc(ccn1)-c1ccc(NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)cc1 50443205Cc1cc(ccn1)-c1ccc(NS(=O)(=O)c2cc(Cl)cc(Cl)c2)cc1 50443206Clc1cc(Cl)cc(c1)S(=O)(=O)Nc1ccc(cc1)-c1cncnc1 50443208Clc1cc(Cl)cc(c1)S(=O)(=O)Nc1ccc(cc1)-c1ccncc1 50443210Clc1cc(Cl)cc(c1)S(=O)(=O)Nc1ccc(cc1)-n1ccnc1 50443215Clc1cc(Cl)cc(c1)S(=O)(=O)Nc1ccc(cc1)-c1cnco1 50443780Cn1c2ccc(COc3ccc4CCN(CCc4c3)C3CCC3)cc2ccc1=O 50443781C(Oc1ccc2CCN(CCc2c1)C1CCCC1)c1ccccc1 50443782C(Oc1ccc2CCN(CCc2c1)C1CCC1)c1ccccc1 50443783C(Oc1ccc2CCN(CC3CC3)CCc2c1)c1ccccc1 50443879COc1ccc(cc1)[C@H]1CN(CCO1)c1nc(cc(=O)n1C)-c1ccncn1 50443880Cn1c(nc(cc1=O)-c1ccncn1)N1CCO[C@H](C1)c1ccc(cc1)C#N 50444546CC(C)(C)n1nnnc1C(NCCNc1ccnc2cc(Cl)ccc12)c1ccc(Cl)cc1 50444547Cc1ccc(cc1)C(NCCNc1ccnc2cc(Cl)ccc12)c1nnnn1C(C)(C)C 50446305COCCOc1ccn2c(cnc2c1)-c1ccc2cccc(O[C@@H]3CCNC[C@@H]3F)c2n1 50446472ONC(=O)[C@@H]1[C@@H]([C@H]1c1ccc(cc1)-c1cnco1)c1ccccc1 50447388CC(C)[C@H](NC(=O)N(C)Cc1csc(n1)C(C)C)C(=O)N[C@@H](Cc1ccccc1)[C@H](Cc1ccccc1)NC(=O)OCc1cncs1 50447389CC(C)CN(CC[C@H](Cc1ccccc1)NC(=O)OCc1cncs1)C(=O)[C@H](CCN1CCOCC1)NC(=O)N(C)Cc1csc(n1)C(C)C 50447390CC(C)c1nc(CN(C)C(=O)N[C@@H](CCN2CCOCC2)C(=O)N[C@H](CCN(Cc2ccccc2)C(=O)OCc2cncs2)Cc2ccccc2)cs1 50447391CC(C)[C@H](NC(=O)N(C)Cc1csc(n1)C(C)C)C(=O)N[C@H](CCN(Cc1ccccc1)C(=O)OCc1cncs1)Cc1ccccc1 50447392CC(C)[C@H](NC(=O)N(C)Cc1csc(n1)C(C)C)C(=O)N(CCCCN(Cc1ccccc1)C(=O)OCc1cncs1)Cc1ccccc1 50447393CC(C)[C@H](NC(=O)N(C)Cc1csc(n1)C(C)C)C(=O)N[C@@H](CC[C@@H](Cc1ccccc1)NC(=O)OCc1cncs1)Cc1ccccc1 50447394CC[C@@H](CC[C@H](CC)NC(=O)[C@@H](NC(=O)N(C)Cc1csc(n1)C(C)C)C(C)C)NC(=O)OCc1cncs1 50447395CC(C)[C@H](NC(=O)N(C)Cc1csc(n1)C(C)C)C(=O)N[C@H](CC[C@H](Cc1ccccc1)NC(=O)OCc1cncs1)Cc1ccccc1 50447466CC(C)c1nc(CN(C)C(=O)N[C@@H](Cc2cnc[nH]2)C(=O)N[C@@H](CC[C@@H](Cc2ccccc2)NC(=O)OCc2cncs2)Cc2ccccc2)cs1 50447467CC(C)c1nc(CN(C)C(=O)N[C@@H](CCNC(C)=O)C(=O)N[C@@H](CC[C@@H](Cc2ccccc2)NC(=O)OCc2cncs2)Cc2ccccc2)cs1 50447468CC(C)c1nc(CN(C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC[C@@H](Cc2ccccc2)NC(=O)OCc2cncs2)Cc2ccccc2)cs1 50447469CC(C)c1nc(CN(C)C(=O)N[C@@H](Cc2cn(C)cn2)C(=O)N[C@H](CC[C@H](Cc2ccccc2)NC(=O)OCc2cncs2)Cc2ccccc2)cs1 50447470CC(C)c1nc(CN(C)C(=O)N[C@H](CCN2CCOCC2)C(=O)N[C@H](CC[C@H](Cc2ccccc2)NC(=O)OCc2cncs2)Cc2ccccc2)cs1 50447471CC(C)c1nc(CN(C)C(=O)N[C@@H](CCN2CCOCC2)C(=O)N[C@H](CC[C@H](Cc2ccccc2)NC(=O)OCc2cncs2)Cc2ccccc2)cs1 50447472CC(C)c1nc(CN(C)C(=O)N[C@@H](CCN)C(=O)N[C@H](CC[C@H](Cc2ccccc2)NC(=O)OCc2cncs2)Cc2ccccc2)cs1 50447694NC[C@@]1(CC[C@@H](CC1)N1CCn2c(nnc2C(F)(F)F)C1=O)c1cccc(Cl)c1 50448471OCc1cc(ccc1O)[C@@H](O)CNCCCCCCOCCCCc1cccc(c1)S(=O)(=O)C1CCCC1 50448616FC(F)(F)Oc1cccc(c1)S(=O)(=O)c1ccc(NC(=O)[C@@H]2C[C@H]2c2cccnc2)cc1 50448622O=C(Nc1ccc(cc1)S(=O)(=O)c1ccccc1)[C@@H]1C[C@H]1c1cccnc1