73956Cn1c2ccccc2n(CC(=O)c2ccc(Cl)c(Cl)c2)c1=N 84297Cn1c2ccccc2n(CC(=O)c2ccc(Br)cc2)c1=N 94647Cn1c2ccccc2n(CC(=O)c2ccc(Cl)cc2)c1=N 94737CCCn1c2ccccc2n(CC(=O)c2ccc(Cl)cc2)c1=N 50018551Fc1ccc(CN2CCC(CC2)C2(CCC(=O)NC2=O)c2ccccc2)cc1 50018553Brc1ccc(CN2CCC(CC2)C2(CCC(=O)NC2=O)c2ccccc2)cc1 50018560Clc1ccc(CN2CCC(CC2)C2(CCC(=O)NC2=O)c2ccccc2)cc1 50167778CCCCCCCCCC(=O)N(CCN(C)C)C(C)c1nc2ccccc2c(=O)n1-c1ccc(F)cc1 50167781CCCCCCCCCC(=O)N(CCN(C)C)C(C)c1nc2ccccc2c(=O)n1-c1ccc(C)cc1 50167782CCCCCCCCCC(=O)N(CCN(C)C)C(C)c1nc2ccccc2c(=O)n1-c1ccc(OC)cc1 50167783CCCCCCCCCC(=O)N(CCN(C)C)C(C)c1nc2ccccc2c(=O)n1-c1ccc(cc1)C#N 50167784CCCCCCCCCC(=O)N(CCN(C)C)C(C)c1nc2ccccc2c(=O)n1-c1cccc(c1)C#N 50175160CCNC(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1cccc(Cl)c1)C(=O)NC(C)C 50175161CCNC(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)cc1)C(=O)NCCc1ccc(Cl)cc1Cl 50175162CCNC(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1cccc(Cl)c1)C(=O)NCC1CC1 50175163CCNC(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1cccc(Cl)c1)C(=O)NCCc1ccc(OC)c(OC)c1 50175164CCNC(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1cccc(Cl)c1)C(=O)NCCc1ccccc1Cl 50175165CCNC(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1ccncc1)C(=O)NCCc1ccc(Cl)cc1Cl 50175166CCNC(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1cccc(Cl)c1)C(=O)NCCc1ccc(F)cc1 50175167COC(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1cccc(Cl)c1)C(=O)NCCc1ccc(Cl)cc1Cl 50175168CC(C)NC(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1cccc(Cl)c1)C(=O)NCCc1ccc(Cl)cc1Cl 50175169CCNC(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1cccs1)C(=O)NCCc1ccc(Cl)cc1Cl 50175170CCNC(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1cccc(c1)C#N)C(=O)NCCc1ccc(Cl)cc1Cl 50175171CCNC(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1cccc(Cl)c1)C(=O)NCCc1ccccc1 50175172CCNC(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1ccco1)C(=O)NCCc1ccc(Cl)cc1Cl 50175173CCNC(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1cccc(Cl)c1)C(=O)NCCc1ccc(Cl)cc1Cl 50175174CCNC(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1ccsc1)C(=O)NCCc1ccc(Cl)cc1Cl 50175175CCNC(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1ccccc1F)C(=O)NCCc1ccc(Cl)cc1Cl 50175176CCNC(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1cccc(F)c1)C(=O)NCCc1ccc(Cl)cc1Cl 50175177CCNC(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1cccc(Cl)c1)C(=O)NCc1ccc(Cl)cc1 50175178CCNC(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1cccc(Cl)c1)C(=O)NCCc1ccc(Cl)cc1 50175179CN(C)C(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1cccc(Cl)c1)C(=O)NCCc1ccc(Cl)cc1Cl 50175180CCNC(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1cccnc1)C(=O)NCCc1ccc(Cl)cc1Cl 50175181CNC(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1cccc(Cl)c1)C(=O)NCCc1ccc(Cl)cc1Cl 50175182CCNC(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1ccc(F)c(F)c1)C(=O)NCCc1ccc(Cl)cc1Cl 50175183CCCNC(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1cccc(Cl)c1)C(=O)NCCc1ccc(Cl)cc1Cl 50175184CCNC(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1ccccc1Cl)C(=O)NCCc1ccc(Cl)cc1Cl 50175185CCNC(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1cccc(OC)c1)C(=O)NCCc1ccc(Cl)cc1Cl 50175187CCNC(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1ccccc1)C(=O)NCCc1ccc(Cl)cc1Cl 50175188CCNC(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1cccc(Cl)c1)C(=O)NCCc1cccc(F)c1 50175189CCNC(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1cccc(Cl)c1)C(=O)NCc1ccccc1 50175190CCNC(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1cc(F)cc(F)c1)C(=O)NCCc1ccc(Cl)cc1Cl 50175191CCNC(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1cccc(Cl)c1)C(=O)NCCc1ccccc1F 50175192CCNC(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1cccc(Cl)c1)C(=O)NCCc1cccc(Cl)c1 50175193CCCCNC(=O)N1CCCN(CC1)c1ccc(cc1NC(=O)c1cccc(Cl)c1)C(=O)NCCc1ccc(Cl)cc1Cl 50198385CC1(C)[C@@H]2C[C@H]1C(CN1CCC(CC1)NC(=O)Nc1ccccc1)=CC2 50198386CC1(C)[C@@H]2C[C@H]1C(CN1CCC(CC1)NC(=O)Nc1cc(F)cc(OC3CCOC3)c1)=CC2 50198387CC(=O)c1cccc(NC(=O)NC2CCN(CC3=CC[C@H]4C[C@@H]3C4(C)C)CC2)c1 50198388CC1(C)[C@@H]2C[C@H]1C(CN1CCC(CC1)NC(=O)Nc1cc(F)cc(F)c1)=CC2 50198389CC1(C)[C@@H]2C[C@H]1C(CN1CCC(CC1)NC(=O)Nc1ccc(s1)-c1ccc(cc1)C(F)(F)F)=CC2 50198390CC1(C)[C@@H]2C[C@H]1C(CN1CCC(CC1)NC(=O)Nc1cccc(OC(F)(F)F)c1)=CC2 50198391Fc1cc(NC(=O)NC2CCN(C\C3=C\CCCCCC3)CC2)cc(c1)C(F)(F)F 50198392CC1(C)[C@@H]2C[C@H]1C(CN1CCC(CC1)NC(=O)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F)=CC2 50198393CC1(C)[C@@H]2C[C@H]1C(CN1CCC(CC1)NC(=O)Nc1cc(ccc1F)C(F)(F)F)=CC2 50198394O=C(NC1CCN(C\C2=C\CCCCCC2)CC1)Nc1ccc2ccccc2c1 50198395NA 50198396CC1(C)C2CC1C(CCN1CCC(CC1)NC(=O)Nc1ccc3ccccc3c1)=CC2 50198397Clc1cncc(Cl)c1NC(=O)NC1CCN(C\C2=C\CCCCCC2)CC1 50198398Clc1cccc(NC(=O)NC2CCN(C\C3=C\CCCCCC3)CC2)c1 50198399CC1(C)[C@@H]2C[C@H]1C(CN1CCC(CC1)NC(=O)Nc1cccc(OC3CCOCC3)c1)=CC2 50198400CC1(C)[C@@H]2C[C@H]1C(CN1CCC(CC1)NC(=O)Nc1cccc(OC3CCOC3)c1)=CC2 50198401CC1(C)[C@@H]2C[C@H]1C(CN1CCC(CC1)NC(=O)Nc1cncc(Br)c1)=CC2 50198402CC(=O)c1cccc(NC(=O)NC2CCN(C\C3=C\CCCCCC3)CC2)c1 50198403COC(=O)c1cccc(NC(=O)NC2CCN(C\C3=C\CCCCCC3)CC2)c1 50198404FC(F)(F)c1cccc(NC(=O)NC2CCN(C\C3=C\CCCCCC3)CC2)c1 50198405COc1cccc(c1)-c1ccc(NC(=O)NC2CCN(CC3=CC[C@H]4C[C@@H]3C4(C)C)CC2)s1 50198406CC1(C)[C@@H]2C[C@H]1C(CN1CCC(CC1)NC(=O)Nc1cncc(c1)-c1ccsc1)=CC2 50198407O=C(NC1CCN(C\C2=C\CCCCCC2)CC1)Nc1ccc(s1)-c1ccccc1 50198408CC1(C)[C@@H]2C[C@H]1C(CN1CCC(CC1)NC(=O)Nc1ccc(s1)-c1ccccc1Cl)=CC2 50198409COC(=O)c1cccc(NC(=O)NC2CCN(CC3=CC[C@H]4C[C@@H]3C4(C)C)CC2)c1 50198410CC1(C)[C@@H]2C[C@H]1C(CN1CCC(CC1)NC(=O)Nc1cncc(c1)-c1cccs1)=CC2 50198411CC1(C)[C@@H]2C[C@H]1C(CN1CCC(CC1)NC(=O)Nc1ccc(OC(F)(F)F)cc1)=CC2 50198412FC(F)(F)Oc1cccc(NC(=O)NC2CCN(C\C3=C\CCCCCC3)CC2)c1 50198413O=C(NC1CCN(CCCc2ccccc2)CC1)Nc1ccc2ccccc2c1 50198414CC1(C)[C@@H]2C[C@H]1C(CN1CCC(CC1)NC(=O)Nc1ccc(F)c(c1)C(F)(F)F)=CC2 50198415FC(F)(F)c1cc(NC(=O)NC2CCN(C\C3=C\CCCCCC3)CC2)cc(c1)C(F)(F)F 50198416O=C(NC1CCN(CCc2ccccc2)CC1)Nc1ccc2ccccc2c1 50198417CC1(C)[C@@H]2C[C@H]1C(CN1CCC(CC1)NC(=O)Nc1ccc(s1)-c1ccccc1)=CC2 50198418Clc1cc(Cl)cc(NC(=O)NC2CCN(C\C3=C\CCCCCC3)CC2)c1 50198419CC1(C)[C@@H]2C[C@H]1C(CN1CCC(CC1)NC(=O)Nc1cc(F)cc(c1)C(F)(F)F)=CC2 50198420O=C(NC1CCN(C\C2=C\CCCCCC2)CC1)Nc1ccc(Oc2ccccc2)cc1 50198421CC(C)(C)c1ccc(NC(=O)NC2CCN(C\C3=C\CCCCCC3)CC2)cc1 50198422COc1cccc(NC(=O)NC2CCN(CC3=CC[C@H]4C[C@@H]3C4(C)C)CC2)c1 50211114CCOc1ccc(cc1)-n1c(nc2ncccc2c1=O)[C@@H](C)N(Cc1cccnc1)C(=O)Cc1ccc(OC(F)(F)F)cc1 50211115C[C@@H](N(Cc1cccnc1)C(=O)Cc1ccc(cc1)C(F)(F)F)c1nc2ccccc2c(=O)n1-c1ccc(C)cc1 50211117C[C@@H](N(CCN(C)C)C(=O)Cc1ccc(cc1)C(F)(F)F)c1nc2ccccc2c(=O)n1-c1ccc(F)cc1 50211118C[C@@H](N(Cc1ccccn1)C(=O)Cc1ccc(cc1)C(F)(F)F)c1nc2ccccc2c(=O)n1-c1ccc(F)cc1 50211119CCOCCN([C@H](C)c1nc2ccccc2c(=O)n1-c1ccc(F)cc1)C(=O)Cc1ccc(cc1)C(F)(F)F 50211120CCCCCCCCCCS(=O)(=O)N(CCN(C)C)[C@H](C)c1nc2ccccc2c(=O)n1-c1ccc(F)cc1 50211121C[C@@H](N(Cc1cccnc1)C(=O)Cc1ccc(cc1)C(F)(F)F)c1nc2ccccc2c(=O)n1-c1ccc(cc1)C#N 50211122C[C@@H](N(Cc1cccnc1)C(=O)Cc1ccc(cc1)C(F)(F)F)c1nc2ccccc2c(=O)n1-c1ccc(Cl)cc1 50211123C[C@@H](N(Cc1cccnc1)C(=O)Cc1ccc(cc1)C(F)(F)F)c1nc2ccccc2c(=O)n1-c1ccc(F)cc1 50211125CCCCCCCCN(CCN(C)C)[C@H](C)c1nc2ccccc2c(=O)n1-c1ccc(F)cc1 50211128CCOCCN([C@H](CC)c1nc2ccccc2c(=O)n1-c1ccc(OCC)cc1)C(=O)Cc1ccc(cc1)-c1ccccc1 50211129C[C@@H](N(Cc1nccs1)C(=O)Cc1ccc(cc1)C(F)(F)F)c1nc2ccccc2c(=O)n1-c1ccc(F)cc1 50211130CCOc1ccc(cc1)-n1c(nc2ccccc2c1=O)[C@@H](C)N(Cc1cccnc1)C(=O)Cc1ccc(OC(F)(F)F)cc1 50211132CCOCCN([C@H](C)c1nc2ccccc2c(=O)n1-c1ccc(OCC)cc1)C(=O)Cc1ccc(cc1)-c1ccccc1 50211134CCCCCCCCCN(CCN(C)C)[C@H](C)c1nc2ccccc2c(=O)n1-c1ccc(F)cc1 50211135CCOCCN(Cc1nc2ccccc2c(=O)n1-c1ccc(OCC)cc1)C(=O)Cc1ccc(cc1)-c1ccccc1 50211136CCOc1ccc(cc1)-n1c(nc2cccnc2c1=O)[C@@H](C)N(Cc1cccnc1)C(=O)Cc1ccc(OC(F)(F)F)cc1 50211137C[C@@H](N(Cc1cccnc1)C(=O)Cc1ccc(cc1)C(F)(F)F)c1nc2ccccc2c(=O)n1-c1ccc(cc1)[N+]([O-])=O 50211138CCOc1ccc(cc1)-n1c(nc2ccccc2c1=O)[C@@H](C)N(Cc1cccnc1)C(=O)Cc1ccc(cc1)C(F)(F)F 50211140CCCCCCCCCC(=O)N(CCN(C)C)[C@H](C)c1nc2ccccc2c(=O)n1-c1ccc(F)cc1 50211142C[C@@H](N(Cc1cccnc1)C(=O)Cc1ccc(cc1)C(F)(F)F)c1nc2ccccc2c(=O)n1-c1ccccc1 50211143COc1ccc(cc1)-n1c(nc2ccccc2c1=O)[C@@H](C)N(Cc1cccnc1)C(=O)Cc1ccc(cc1)C(F)(F)F 50211144C[C@@H](N(CC(=O)c1cn(C)cn1)C(=O)Cc1ccc(cc1)C(F)(F)F)c1nc2ccccc2c(=O)n1-c1ccc(F)cc1 50211145C[C@@H](N(CC(=O)c1ncc[nH]1)C(=O)Cc1ccc(cc1)C(F)(F)F)c1nc2ccccc2c(=O)n1-c1ccc(F)cc1 50211146CCOCCN([C@H](c1ccccc1)c1nc2ccccc2c(=O)n1-c1ccc(OCC)cc1)C(=O)Cc1ccc(cc1)-c1ccccc1 50211147CCOc1ccc(cc1)-n1c(nc2nccnc2c1=O)[C@@H](C)N(Cc1cccnc1)C(=O)Cc1ccc(OC(F)(F)F)cc1 50211148CC#Cc1ccc(cc1)-n1c(nc2ccccc2c1=O)[C@@H](C)N(Cc1cccnc1)C(=O)Cc1ccc(cc1)C(F)(F)F 50211149CCCCCCCCS(=O)(=O)N(CCN(C)C)[C@H](C)c1nc2ccccc2c(=O)n1-c1ccc(F)cc1 50211150C[C@@H](N(CCN(C)C)C(=O)Cc1ccc(OC(F)(F)F)cc1)c1nc2ccccc2c(=O)n1-c1ccc(F)cc1 50211151CCCCCCCCCCCC(=O)N(CCN(C)C)[C@H](C)c1nc2ccccc2c(=O)n1-c1ccc(F)cc1 50211152CCOc1ccc(cc1)-n1c(nc2cnccc2c1=O)[C@@H](C)N(Cc1cccnc1)C(=O)Cc1ccc(OC(F)(F)F)cc1 50211153C[C@@H](N(CC(=O)c1cnc[nH]1)C(=O)Cc1ccc(cc1)C(F)(F)F)c1nc2ccccc2c(=O)n1-c1ccc(F)cc1 50211154C[C@@H](N(Cc1cccnc1)C(=O)Cc1ccc(cc1)C(F)(F)F)c1nc2ccccc2c(=O)n1-c1ccc(cc1)C(O)=O 50211155CCCCCCCC(=O)N(CCN(C)C)[C@H](C)c1nc2ccccc2c(=O)n1-c1ccc(F)cc1 50211156C[C@@H](N(CCN(C)C)C(=O)Cc1ccc(cc1)-c1ccccc1)c1nc2ccccc2c(=O)n1-c1ccc(F)cc1 50211157COCCN([C@H](C)c1nc2ccccc2c(=O)n1-c1ccc(F)cc1)C(=O)Cc1ccc(cc1)C(F)(F)F 50225709CC1(C)[C@@H]2C[C@H]1C(CN1CCC(CC1)Nc1nc3ccccc3o1)=CC2 50225710CC1(C)[C@@H]2C[C@H]1C(CN1CCC(CC1)n1cc(O)n(-c3cccc(c3)C(F)(F)F)c1=O)=CC2 50225711CN(C1CCN(CC2=CC[C@H]3C[C@@H]2C3(C)C)CC1)c1nc2ccccc2s1 50225712CN(C1CCN(CC2=CC[C@H]3C[C@@H]2C3(C)C)CC1)c1nc2c(Cl)cccc2s1 50225713CCN(C1CCN(CC2=CC[C@H]3C[C@@H]2C3(C)C)CC1)C(=O)Nc1cccc(c1)C(F)(F)F 50225714CC1(C)[C@@H]2C[C@H]1C(CN1CCC(CC1)N1CCN(C1=O)c1cc(F)cc(c1)C(F)(F)F)=CC2 50225715CC1(C)[C@@H]2C[C@H]1C(CN1CCC(CC1)n1cc(O)n(-c3cc(cc(c3)C(F)(F)F)C(F)(F)F)c1=O)=CC2 50225716CCc1cccc(c1)-n1c(O)cn(C2CCN(CC3=CC[C@H]4C[C@@H]3C4(C)C)CC2)c1=O 50225717CC1(C)[C@@H]2C[C@H]1C(CN1CCC(CC1)Nc1nc3ccccc3s1)=CC2 50225718CC1(C)[C@@H]2C[C@H]1C(CN1CCC(CC1)n1cc(O)n(-c3cc(F)cc(c3)C(F)(F)F)c1=O)=CC2 50225719CSc1cccc(c1)-n1c(O)cn(C2CCN(CC3=CC[C@H]4C[C@@H]3C4(C)C)CC2)c1=O 50225720CC1(C)[C@@H]2C[C@H]1C(CN1CCC(CC1)Nc1nc(cs1)-c1ccc(Cl)c(Cl)c1)=CC2 50225721CN(C1CCN(CC2=CC[C@H]3C[C@@H]2C3(C)C)CC1)c1nc2cccc(Cl)c2s1 50225722CN(C1CCN(CC2=CC[C@H]3C[C@@H]2C3(C)C)CC1)c1nc2cc(Cl)ccc2s1 50225723CN(C1CCN(CC2=CC[C@H]3C[C@@H]2C3(C)C)CC1)c1nc2ccccc2o1 50225724CC1(C)[C@@H]2C[C@H]1C(CN1CCC(CC1)Nc1nc(cs1)-c1cc(cc(c1)C(F)(F)F)C(F)(F)F)=CC2 50225725CC1(C)[C@@H]2C[C@H]1C(CN1CCC(CC1)Nc1nc3ccc(Br)cc3s1)=CC2 50225726CC1(C)[C@@H]2C[C@H]1C(CN1CCC(CC1)Nc1nc3c(Br)cccc3s1)=CC2 50225727CN(C1CCN(CC2=CC[C@H]3C[C@@H]2C3(C)C)CC1)c1nc2ccccc2[nH]1 50225728CC1(C)[C@@H]2C[C@H]1C(CN1CCC(CC1)Nc1nc(ns1)-c1cc(cc(c1)C(F)(F)F)C(F)(F)F)=CC2 50225729CC1(C)[C@@H]2C[C@H]1C(CN1CCC(CC1)n1cc(O)n(-c3ccc(Cl)c(c3)C(F)(F)F)c1=O)=CC2 50225730CCc1cccc(c1)N(C)C(=O)NC1CCN(CC2=CC[C@H]3C[C@@H]2C3(C)C)CC1 50225731CC1(C)[C@@H]2C[C@H]1C(CN1CCC(CC1)N1CCN(C1=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)=CC2 50225732CN(C1CCN(CC2=CC[C@H]3C[C@@H]2C3(C)C)CC1)C(=O)Nc1cccc(c1)C(F)(F)F 50225733CN(C1CCN(CC2=CC[C@H]3C[C@@H]2C3(C)C)CC1)c1nc2ccc(Cl)cc2s1 50225734CC1(C)[C@@H]2C[C@H]1C(CN1CCC(CC1)Nc1nc(cs1)-c1ccccc1)=CC2 50227861CC(C)(C)C(=O)N1C2CCCC1C=C(CN1CCC(CC1)NC(=O)Nc1cc(F)cc(c1)C(F)(F)F)C2 50227862Fc1cc(NC(=O)NC2CCN(CC3=CC4CCC(C3)N4C(=O)C3CC3)CC2)cc(c1)C(F)(F)F 50227863CC(=O)N1C2CCCC1C=C(CN1CCC(CC1)NC(=O)Nc1cc(F)cc(c1)C(F)(F)F)C2 50227864CC(C)Oc1cc(F)cc(NC(=O)NC2CCN(CC3=CC4CCCC(C3)N4C(C)=O)CC2)c1 50227865CC(C)(C)C(=O)N1C2CCC1C=C(CN1CCC(CC1)NC(=O)Nc1cc(F)cc(c1)C(F)(F)F)C2 50227866CC(=O)N1C2CCCC1C=C(CN1C3CCC1CC(C3)NC(=O)Nc1cc(F)cc(c1)C(F)(F)F)C2 50227867CC(C)Oc1cccc(NC(=O)NC2CCN(CC3=CC4CCCC(C3)N4C(C)=O)CC2)c1 50227868CC(C)(C)C(=O)N1CCC(CN2CCC(CC2)NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)CC1 50227869CC(=O)N1C2CCC1C=C(CN1CCC(CC1)NC(=O)Nc1cc(F)cc(c1)C(F)(F)F)C2 50227870CC(=O)N1C2CCCC1C=C(CN1CCC(CC1)NC(=O)Nc1cccc(c1)C(C)=O)C2 50227871CC(=O)N1C2CCC1CC(CN1CCC(CC1)NC(=O)Nc1cc(F)cc(c1)C(F)(F)F)C2 50227872FC(F)(F)c1cc(NC(=O)NC2CCN(CCC3CCS(=O)(=O)C3)CC2)cc(c1)C(F)(F)F 50227873CC(C)C(=O)N1C2CCC1C=C(CN1CCC(CC1)NC(=O)Nc1cc(F)cc(c1)C(F)(F)F)C2 50227874CCOC(=O)N1C2CCC1C=C(CN1CCC(CC1)NC(=O)Nc1cc(F)cc(c1)C(F)(F)F)C2 50227875CC(=O)N1CCC(CN2CCC(CC2)NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)CC1 50229376CCS(=O)(=O)CCN([C@H](C)c1nc2ncccc2c(=O)n1-c1ccc(cc1)C#N)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50229377CCS(=O)(=O)CCN([C@H](C)c1nc2ccccn2c(=O)c1-c1ccc(cc1)C#N)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50229378CCS(=O)(=O)CCN([C@H](C)c1nc2ccccn2c1-c1ccc(cc1)C#N)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50229379CCS(=O)(=O)CCN([C@H](C)c1nc2ccccc2n1-c1ccc(cc1)C#N)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50229380CCS(=O)(=O)CCN([C@H](C)c1nc2N(C)CCCc2c(=O)n1-c1ccc(cc1)C#N)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50229381CCS(=O)(=O)CCN([C@H](C)c1nc2ccccc2cc1-c1ccc(cc1)C#N)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50229382CCS(=O)(=O)CCN([C@H](C)c1nc2ncccn2c1-c1ccc(cc1)C#N)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50229383CCS(=O)(=O)CCN([C@H](C)c1nc2ncccc2cc1-c1ccc(cc1)C#N)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50229384CCS(=O)(=O)CCN([C@H](C)c1cc2ccccc2nc1-c1ccc(cc1)C#N)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50229385CCS(=O)(=O)CCN([C@H](C)c1nc2ccccc2nc1-c1ccc(cc1)C#N)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50229386CCS(=O)(=O)CCN([C@H](C)c1nn2ccccc2c1-c1ccc(cc1)C#N)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50229439CCS(=O)(=O)CCN([C@H](C)c1nc(cn1-c1ccc(cc1)C#N)-c1ccccc1)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50229462CCOc1ccc(cc1)-n1c(nc2ccccc2c1=O)[C@@H](C)N(Cc1cccnc1)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50254678C[C@H]1CN(CCN1c1ncc(cc1F)C(F)(F)F)S(=O)(=O)C[C@]12CC[C@H](CC1=O)C2(C)C 50254758C[C@H]1CN(CCN1c1ncc(cc1F)C(F)(F)F)S(=O)(=O)C[C@]12CC[C@H](C[C@@H]1O)C2(C)C 50292637Fc1ccc(c(F)c1)C1(CCC(=O)NC1=O)C1CCN(Cc2ccc(Br)cc2)CC1 50292638Brc1ccc(CN2CCC(CC2)C2(CCCN(C2)C(=O)Nc2ccccc2)c2ccccc2)cc1 50292639Clc1ccc(CN2CCC(CC2)C2(CCC(=O)NC2=O)c2ccccc2)cc1Cl 50292640Fc1cc(CN2CCC(CC2)C2(CCC(=O)NC2=O)c2ccccc2)ccc1Cl 50292641FC(F)(F)c1cc(CN2CCC(CC2)C2(CCC(=O)NC2=O)c2ccccc2)ccc1Cl 50292642Brc1ccc(CN2CCC(CC2)C2(CCC(=O)NC2=O)c2ccccn2)cc1 50292643Brc1ccc(CN2CCC(CC2)C2(CCC(=O)NC2=O)c2cccnc2)cc1 50292644Brc1ccc(CN2CCC(CC2)C2(CCC(=O)NC2=O)c2ccncc2)cc1 50292645Fc1ccc(cc1)C1(CCC(=O)NC1=O)C1CCN(Cc2ccc(Br)cc2)CC1 50292646COc1ccc(cc1)C1(CCC(=O)NC1=O)C1CCN(Cc2ccc(Br)cc2)CC1 50292647COc1cccc(c1)C1(CCC(=O)NC1=O)C1CCN(Cc2ccc(Br)cc2)CC1 50292648COc1ccc(cc1C1(CCC(=O)NC1=O)C1CCN(Cc2ccc(Br)cc2)CC1)S(O)(=O)=O 50292649Clc1cccc(c1)C1(CCC(=O)NC1=O)C1CCN(Cc2ccc(Br)cc2)CC1 50292650OC(=O)c1ccc(cc1)C1(CCC(=O)NC1=O)C1CCN(Cc2ccc(Br)cc2)CC1 50292651OC(=O)c1cccc(c1)C1(CCC(=O)NC1=O)C1CCN(Cc2ccc(Br)cc2)CC1 50292652NC(=O)c1cccc(c1)C1(CCC(=O)NC1=O)C1CCN(Cc2ccc(Br)cc2)CC1 50292653CNC(=O)c1cccc(c1)C1(CCC(=O)NC1=O)C1CCN(Cc2ccc(Br)cc2)CC1 50292654OCCCNC(=O)c1cccc(c1)C1(CCC(=O)NC1=O)C1CCN(Cc2ccc(Br)cc2)CC1 50292655Brc1ccc(CN2CCC(CC2)C2(CCC(=O)NC2=O)c2cccc(c2)C(=O)N2CCOCC2)cc1 50292656CN(N1CCNCC1)C(=O)c1cccc(c1)C1(CCC(=O)NC1=O)C1CCN(Cc2ccc(Br)cc2)CC1 50292657Nc1cccc(c1)C1(CCC(=O)NC1=O)C1CCN(Cc2ccc(Br)cc2)CC1 50292658Oc1cccc(c1)C1(CCC(=O)NC1=O)C1CCN(Cc2ccc(Br)cc2)CC1 50292659CN1C(=O)CCC(C2CCN(Cc3ccc(Br)cc3)CC2)(C1=O)c1ccccc1 50292660CCN1C(=O)CCC(C2CCN(Cc3ccc(Br)cc3)CC2)(C1=O)c1ccccc1 50292661CCCN1C(=O)CCC(C2CCN(Cc3ccc(Br)cc3)CC2)(C1=O)c1ccccc1 50292662CC(C)N1C(=O)CCC(C2CCN(Cc3ccc(Br)cc3)CC2)(C1=O)c1ccccc1 50292663COCCN1C(=O)CCC(C2CCN(Cc3ccc(Br)cc3)CC2)(C1=O)c1ccccc1 50292664CSCN1C(=O)CCC(C2CCN(Cc3ccc(Br)cc3)CC2)(C1=O)c1ccccc1 50292665CC(=O)N1CCCC(C1)(C1CCN(Cc2ccc(Br)cc2)CC1)c1ccccc1 50292666CCOC(=O)N1CCCC(C1)(C1CCN(Cc2ccc(Br)cc2)CC1)c1ccccc1 50292667Brc1ccc(CN2CCC(CC2)C2(CCCN(C2)C=O)c2ccccc2)cc1 50292668FC(F)(F)C(=O)N1CCCC(C1)(C1CCN(Cc2ccc(Br)cc2)CC1)c1ccccc1 50292669CCC(=O)N1CCCC(C1)(C1CCN(Cc2ccc(Br)cc2)CC1)c1ccccc1 50292670Brc1ccc(CN2CCC(CC2)C2(CCCN(C2)C2CC2=O)c2ccccc2)cc1 50292671NC(=O)CN1CCCC(C1)(C1CCN(Cc2ccc(Br)cc2)CC1)c1ccccc1 50292672NC(=O)N1CCCC(C1)(C1CCN(Cc2ccc(Br)cc2)CC1)c1ccccc1 50292673NS(=O)(=O)N1CCCC(C1)(C1CCN(Cc2ccc(Br)cc2)CC1)c1ccccc1 50292674Brc1ccc(CN2CCC(CC2)C2(CCC(=O)NC2)c2ccccc2)cc1 50292676Brc1ccc(CN2CCC(CC2)C2(CCCNC2=O)c2ccccc2)cc1 50292677Cc1ccc(CN2CCC(CC2)C2(CCC(=O)NC2=O)c2ccccc2)cc1 50292678COc1ccc(CN2CCC(CC2)C2(CCC(=O)NC2=O)c2ccccc2)cc1 50292679Clc1ccc(CN2CCC(CC2)C2(CCC(=O)NC2=O)c2ccccc2)c(Cl)c1 50299165CCN(CC)C(=O)[C@H]1CN([C@@H]2Cc3c[nH]c4cccc(C2=C1)c34)C(=O)Nc1ccccc1 50299168CCN(CC)C(=O)[C@H]1CN([C@@H]2Cc3c[nH]c4cccc(C2=C1)c34)C(=O)Oc1ccccc1 50299170CCN(CC)C(=O)[C@@H]1CC2[C@@H](Cc3c[nH]c4cccc2c34)N(C1)C(=O)Nc1ccccc1 50299171CCN(CC)C(=O)[C@H]1CN([C@@H]2Cc3cn(C)c4cccc(C2=C1)c34)C(=O)Nc1ccccc1 50299172CCN(CC)C(=O)[C@H]1CN([C@@H]2Cc3cn(Cc4ccccc4)c4cccc(C2=C1)c34)C(=O)Nc1ccccc1 50299173CCN(CC)C(=O)[C@H]1CN([C@@H]2Cc3c[nH]c4cccc(C2=C1)c34)C(=O)Nc1ccccc1C 50299174CCN(CC)C(=O)[C@H]1CN([C@@H]2Cc3c[nH]c4cccc(C2=C1)c34)C(=O)Nc1cccc(C)c1 50299175CCN(CC)C(=O)[C@H]1CN([C@@H]2Cc3c[nH]c4cccc(C2=C1)c34)C(=O)Nc1ccc(C)cc1 50299176CCN(CC)C(=O)[C@H]1CN([C@@H]2Cc3c[nH]c4cccc(C2=C1)c34)C(=O)Nc1ccccn1 50299177CCN(CC)C(=O)[C@H]1CN([C@@H]2Cc3c[nH]c4cccc(C2=C1)c34)C(=O)Nc1cccnc1 50299178CCN(CC)C(=O)[C@H]1CN([C@@H]2Cc3c[nH]c4cccc(C2=C1)c34)C(=O)Nc1ccncc1 50299179CCN(CC)C(=O)[C@H]1CN([C@@H]2Cc3c[nH]c4cccc(C2=C1)c34)C(=O)Nc1cc(OC)c(OC)c(OC)c1 50299180CCN(CC)C(=O)[C@H]1CN([C@@H]2Cc3c[nH]c4cccc(C2=C1)c34)C(=O)NC1CCCCC1 50300898C[C@@H](N(CC1CCS(=O)(=O)CC1)C(=O)Cc1ccc(cc1)C(F)(F)F)c1nc2c(nccn2c1-c1ccc(cc1)C#N)C1CC1 50300899CCS(=O)(=O)CCN([C@H](C)c1nc2c(nccn2c1-c1ccc(cc1)C#N)C1CC1)C(=O)Cc1ccc(c(F)c1)C(F)(F)F 50300900CCS(=O)(=O)CCN([C@H](C)c1nc2c(OC)nccn2c1-c1ccc(cc1)C#N)C(=O)Cc1ccc(c(F)c1)C(F)(F)F 50300901CCS(=O)(=O)CCN([C@H](C)c1nc2c(C)nccn2c1-c1ccc(cc1)C#N)C(=O)Cc1ccc(c(F)c1)C(F)(F)F 50300902CCc1nccn2c(c(nc12)[C@@H](C)N(CCS(=O)(=O)CC)C(=O)Cc1ccc(c(F)c1)C(F)(F)F)-c1ccc(cc1)C#N 50300903CCS(=O)(=O)CCN(C(C)c1nc2c(nccn2c1-c1ccc(cc1)C#N)N(C)C)C(=O)Cc1ccc(c(F)c1)C(F)(F)F 50300904CCS(=O)(=O)CCN(C(C)c1nc2n(cc[nH]c2=O)c1-c1ccc(cc1)C#N)C(=O)Cc1ccc(c(F)c1)C(F)(F)F 50300905C[C@@H](N(CC1CCS(=O)(=O)CC1)C(=O)Cc1ccc(c(F)c1)C(F)(F)F)c1nc2c(nccn2c1-c1ccc(cc1)C#N)C1CC1 50300906C[C@@H](N(CC1CCS(=O)(=O)CC1)C(=O)Cc1ccc(OC(F)(F)F)cc1)c1nc2c(nccn2c1-c1ccc(cc1)C#N)C1CC1 50300907C[C@@H](N(CC1CCS(=O)(=O)CC1)C(=O)Cc1ccc(F)c(c1)C(F)(F)F)c1nc2c(nccn2c1-c1ccc(cc1)C#N)C1CC1 50300908C[C@@H](N(CC1CCS(=O)(=O)CC1)C(=O)Cc1cccc(c1)C(F)(F)F)c1nc2c(nccn2c1-c1ccc(cc1)C#N)C1CC1 50300909C[C@@H](N(CC1CCS(=O)(=O)CC1)C(=O)Cc1cccc(OC(F)(F)F)c1)c1nc2c(nccn2c1-c1ccc(cc1)C#N)C1CC1 50300910CCS(=O)(=O)CCN([C@H](C)c1nc2nc(C)ccc2c(=O)n1-c1ccc(cc1)C#N)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50300911CCS(=O)(=O)CCN([C@H](C)c1nc2nc(OC)ccc2c(=O)n1-c1ccc(cc1)C#N)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50300912CCS(=O)(=O)CCN([C@H](C)c1nc2ncccc2c(=O)n1-c1ccc(cc1)C#N)C(=O)Cc1ccc(c(F)c1)C(F)(F)F 50300913CCS(=O)(=O)CCN([C@H](C)c1nc2nc(OC)ccc2c(=O)n1-c1ccc(cc1)C#N)C(=O)Cc1ccc(c(F)c1)C(F)(F)F 50300914CCS(=O)(=O)CCN([C@H](C)c1nc2nc(C)ccn2c1-c1ccc(cc1)C#N)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50300915CCS(=O)(=O)CCN(C(C)c1nc2c(Cl)nccn2c1-c1ccc(cc1)C#N)C(=O)Cc1ccc(c(F)c1)C(F)(F)F 50300916CCOc1ccc2c(n1)nc(C(C)N(CCS(=O)(=O)CC)C(=O)Cc1ccc(F)c(c1)C(F)(F)F)n(-c1ccc(cc1)C#N)c2=O 50300918CCS(=O)(=O)CCN(C(C)c1nc2nc(ccc2c(=O)n1-c1ccc(cc1)C#N)C(F)(F)F)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50300919CCS(=O)(=O)CCN([C@H](C)c1nc2cnccn2c1-c1ccc(cc1)C#N)C(=O)Cc1ccc(c(F)c1)C(F)(F)F 50301324Clc1ccc(CN2CCC(CC2)N2CCN(CC2)c2ncc(CNC(=O)c3ccc(Cl)c(Cl)c3)cc2Cl)cc1 50301325Clc1ccc(CN2CCC(CC2)N2CCN(CC2)c2ccc(cc2Cl)C(=O)NCc2ccc(Cl)c(Cl)c2)cc1 50301326Fc1ccc(CNC(=O)c2cnc(N3CCN(CC3)C3CCN(Cc4ccc(cc4)C#N)CC3)c(Cl)c2)cc1 50301327Fc1ccc(CNC(=O)c2ccc(nc2)N2CCN(CC2)C2CCN(Cc3ccc(cc3)C#N)CC2)cc1 50301328C[C@@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2)CC1)c1ncc(cc1Cl)C(=O)NCc1ccc(Cl)c(Cl)c1 50301329C[C@H]1CC(CCN1Cc1ccc(Cl)cc1)N1CCN(CC1)c1ncc(cc1Cl)C(=O)NCc1ccc(Cl)c(Cl)c1 50301330CNC(=O)c1cnc(N2CCN(CC2)C2CCN(Cc3ccc(Cl)cc3)[C@@H](C)C2)c(Cl)c1 50301331Clc1ccc(CN2CCC(CC2)C2CCN(CC2)c2ncc(cc2Cl)C(=O)NCc2ccc(Cl)c(Cl)c2)cc1 50301332Clc1ccc(CN2CCN(CC2)C2CCN(CC2)c2ncc(cc2Cl)C(=O)NCc2ccc(Cl)c(Cl)c2)cc1 50301334CN(CCCN1CCN(CC1)c1ncc(cc1Cl)C(=O)NCCOc1ccccc1)c1ccc(Cl)cc1 50301335Clc1cc(cnc1N1CCN(CC1)C1CCN(Cc2ccc(cc2)C#N)CC1)C(=O)NCCOc1ccccc1 50301336Clc1cc(cnc1N1CCN(CC1)C1CCN(Cc2ccccc2)CC1)C(=O)NCCOc1ccccc1 50301337Clc1cc(cnc1N1CCN(CC1)C1CCN(Cc2cccc(c2)C#N)CC1)C(=O)NCCOc1ccccc1 50301338Clc1cc(cnc1N1CCN(CC1)C1CCN(Cc2ccccc2C#N)CC1)C(=O)NCCOc1ccccc1 50301339Clc1cc(cnc1N1CCN(CC1)C1CCN(CC1)C(=O)c1ccc(cc1)C#N)C(=O)NCCOc1ccccc1 50301340Clc1ccc(CN2CCC(CC2)N2CCN(CC2)c2ncc(cc2Cl)C(=O)NCCOc2ccccc2)cc1 50301341Clc1cc(cnc1N1CCN(CC1)C1CCN(Cc2ccc(Br)cc2)CC1)C(=O)NCCOc1ccccc1 50301342Fc1ccc(CN2CCC(CC2)N2CCN(CC2)c2ncc(cc2Cl)C(=O)NCCOc2ccccc2)cc1 50301343FC(F)(F)c1ccc(CN2CCC(CC2)N2CCN(CC2)c2ncc(cc2Cl)C(=O)NCCOc2ccccc2)cc1 50301344COc1ccc(CN2CCC(CC2)N2CCN(CC2)c2ncc(cc2Cl)C(=O)NCCOc2ccccc2)cc1 50301345CN(C)c1ccc(CN2CCC(CC2)N2CCN(CC2)c2ncc(cc2Cl)C(=O)NCCOc2ccccc2)cc1 50301346CNC(=O)c1cnc(N2CCN(CC2)C2CCN(Cc3ccc(Cl)cc3)CC2)c(Cl)c1 50301347CCCCNC(=O)c1cnc(N2CCN(CC2)C2CCN(Cc3ccc(Cl)cc3)CC2)c(Cl)c1 50301348Clc1ccc(CN2CCC(CC2)N2CCN(CC2)c2ncc(cc2Cl)C(=O)NCc2ccccc2)cc1 50301349Clc1ccc(CN2CCC(CC2)N2CCN(CC2)c2ncc(cc2Cl)C(=O)NCCc2ccccc2)cc1 50301350COc1cccc(CNC(=O)c2cnc(N3CCN(CC3)C3CCN(Cc4ccc(Cl)cc4)CC3)c(Cl)c2)c1 50301351Clc1ccc(CN2CCC(CC2)N2CCN(CC2)c2ncc(cc2Cl)C(=O)NCc2ccc(Cl)c(Cl)c2)cc1 50301352Clc1ccc(CN2CCC(CC2)N2CCN(CC2)c2ncc(NC(=O)Cc3ccc(Cl)c(Cl)c3)cc2Cl)cc1 50301354Clc1ccc(CN2CCC(CC2)N2CCN(CC2)c2ncc(CNCc3ccc(Cl)c(Cl)c3)cc2Cl)cc1 50301355CN(Cc1ccc(Cl)c(Cl)c1)Cc1cnc(N2CCN(CC2)C2CCN(Cc3ccc(Cl)cc3)CC2)c(Cl)c1 50310479CCOc1ccc(cc1)-n1c(nc2ncccc2c1=O)[C@@H](C)N(C[C@H]1CCCN1C(C)C)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50310480CCOc1ccc(cc1)-n1c(nc2ncccc2c1=O)[C@@H](C)N(C[C@@H]1CCCN1C(C)C)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50310481CCOc1ccc(cc1)-n1c(nc2ncccc2c1=O)[C@@H](C)N(C[C@H]1CCCN1)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50310482CCOc1ccc(cc1)-n1c(nc2ncccc2c1=O)[C@@H](C)N(CC1CCN(C)CC1)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50310483CCOc1ccc(cc1)-n1c(nc2ncccc2c1=O)[C@@H](C)N(C1CCN(CC1)C(C)C)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50310484CCOc1ccc(cc1)-n1c(nc2ncccc2c1=O)[C@@H](C)N(C1CCN(CC1)C(C)=O)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50310485CCOc1ccc(cc1)-n1c(nc2ncccc2c1=O)[C@@H](C)N(C1CCOCC1)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50310486CCOc1ccc(cc1)-n1c(nc2ncccc2c1=O)[C@@H](C)N(CCS(=O)(=O)CC)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50310487CCS(=O)(=O)CCN([C@H](C)c1nc2ncccc2c(=O)n1-c1ccc(OCC(F)(F)F)cc1)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50310488CCOc1ccc(cc1)-n1c(nc2ncccc2c1=O)[C@@H](C)N(Cc1ccc[n+]([O-])c1)C(=O)Cc1ccc(OC(F)(F)F)cc1 50310489CCOc1ccc(cc1)-n1c(nc2ccccc2c1=O)[C@@H](C)N(Cc1cccnc1)C(=O)CN1CCN(CCC(F)(F)F)CC1 50310490CCOc1ccc(cc1)-n1c(nc2ccccc2c1=O)[C@@H](C)N(Cc1cccnc1)C(=O)Cc1nc2ccc(cc2[nH]1)C(F)(F)F 50310491CCOc1ccc(cc1)-n1c(nc2ccccc2c1=O)[C@@H](C)N(Cc1cccnc1)C(=O)Cn1cnc(c1)C(F)(F)F 50310492CCOc1ccc(cc1)-n1c(nc2ccccc2c1=O)[C@@H](C)N(Cc1cccnc1)C(=O)Cc1ccc(cn1)C(F)(F)F 50310493CCOc1ccc(cc1)-n1c(nc2ccccc2c1=O)[C@@H](C)N(Cc1cccnc1)C(=O)CCc1ccc(cc1)C(F)(F)F 50310494CCOc1ccc(cc1)-n1c(nc2ccccc2c1=O)[C@@H](C)N(Cc1cccnc1)C(=O)Cc1cccc(c1)C(F)(F)F 50310495CCOc1ccc(cc1)-n1c(nc2ccccc2c1=O)[C@@H](C)N(Cc1cccnc1)C(=O)Cc1ccc(cc1)C#N 50310496CCOc1ccc(cc1)-n1c(nc2ccccc2c1=O)[C@@H](C)N(Cc1cccnc1)C(=O)Cc1ccc(cc1)S(C)(=O)=O 50310497CCOc1ccc(cc1)-n1c(nc2ccccc2c1=O)[C@@H](C)N(Cc1cccnc1)C(=O)Cc1ccc(F)c(F)c1 50310498CCOc1ccc(cc1)-n1c(nc2ccccc2c1=O)[C@@H](C)N(Cc1cccnc1)C(=O)Cc1cc(F)c(F)c(F)c1 50310499CCOc1ccc(cc1)-n1c(nc2ccccc2c1=O)[C@@H](C)N(Cc1cccnc1)C(=O)Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F 50310500CCOc1ccc(cc1)-n1c(nc2ccccc2c1=O)[C@@H](C)N(Cc1cccnc1)C(=O)Cc1ccc(OC(F)(F)F)c(F)c1 50310501CCOc1ccc(cc1)-n1c(nc2ccccc2c1=O)[C@@H](C)N(Cc1cccnc1)C(=O)Cc1ccc(c(F)c1)C(F)(F)F 50310502CCOc1ccc(cc1)-n1c(nc2ncccc2c1=O)[C@@H](C)N(Cc1cccnc1)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50310503CCOc1ccc(cc1)-n1c(nc2cnccc2c1=O)[C@@H](C)N(Cc1cccnc1)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50310504CCOc1ccc(cc1)-n1c(nc2cccnc2c1=O)[C@@H](C)N(Cc1cccnc1)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50310505CCOc1ccc(cc1)-n1c(nc2nccnc2c1=O)[C@@H](C)N(Cc1cccnc1)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50310506CCOc1ccc(cc1)-n1c(nc2ncccc2c1=O)[C@@H](C)N(Cc1cc(C)no1)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50320127CC(=O)Nc1cccc(c1)C(C)=NNC(=O)c1ccc(CN(Cc2ccccc2)S(=O)(=O)c2ccc(Cl)cc2)cc1 50320128Clc1ccc(cc1)S(=O)(=O)N(Cc1ccccc1)Cc1ccc(cc1)C(=O)NC[C@@H]1CCCO1 50320129Clc1ccc(cc1)S(=O)(=O)N(Cc1ccccc1)Cc1ccc(cc1)C(=O)NCC1CC1 50320130Clc1ccc(cc1)S(=O)(=O)N(Cc1ccccc1)Cc1ccc(cc1)C(=O)NCc1cccc(Cl)c1 50320131Clc1ccc(cc1)S(=O)(=O)N(Cc1ccccc1)Cc1ccc(cc1)C(=O)NCc1cccs1 50320132Clc1ccc(cc1)S(=O)(=O)N(Cc1ccccc1)Cc1ccc(cc1)C(=O)NC1(CC1)c1ccccc1 50320133[O-][N+](=O)c1cccc(CCNC(=O)c2ccc(CN(Cc3ccccc3)S(=O)(=O)c3ccc(Cl)cc3)cc2)c1 50320134COc1ccc(cc1)S(=O)(=O)N(Cc1ccccc1)Cc1ccc(cc1)C(=O)NCC1CC1 50320135COc1ccc(cc1)S(=O)(=O)N(Cc1ccccc1)Cc1ccc(cc1)C(=O)NCc1ccccc1 50320136CCOc1ccc(cc1)S(=O)(=O)N(Cc1ccccc1)Cc1ccc(cc1)C(=O)NCC1CC1 50320137FC(F)(F)Oc1ccc(cc1)S(=O)(=O)N(Cc1ccccc1)Cc1ccc(cc1)C(=O)NCC1CC1 50320138Clc1ccc(cc1)S(=O)(=O)N(Cc1ccc(cc1)C(=O)NCC1CC1)Cc1ccccn1 50320139Clc1ccc(cc1)S(=O)(=O)N(Cc1ccc(cc1)C(=O)NCc1cccc(Cl)c1)Cc1ccccn1 50320140COc1ccc(cc1)S(=O)(=O)N(Cc1ccc(cc1)C(=O)NCC1CC1)Cc1cccnc1 50320141O=C(NCC1CC1)c1ccc(CN(Cc2ccccn2)S(=O)(=O)c2ccc(cc2)C#N)cc1 50320142Fc1ccccc1CN(Cc1ccc(cc1)C(=O)NCC1CC1)S(=O)(=O)c1ccc(Cl)cc1 50320143Clc1ccc(cc1)S(=O)(=O)N(Cc1ccc(cc1)C(=O)NCC1CC1)Cc1cccc(Cl)c1 50320144Clc1ccc(cc1)S(=O)(=O)N(Cc1ccc(cc1)C(=O)NC1(CC1)c1ccccc1)Cc1ccccn1 50320145O=C(NC1(CC1)c1ccccc1)c1ccc(CN(Cc2ccccn2)S(=O)(=O)c2ccc(cc2)C#N)cc1 50320146OC(=O)c1ccc(CN(Cc2ccccc2)S(=O)(=O)c2ccc(Cl)cc2)cc1 50320147COc1ccc(cc1)S(=O)(=O)N(Cc1ccccc1)Cc1ccc(cc1)C(O)=O 50320148OC(=O)c1ccc(CN(Cc2ccccn2)S(=O)(=O)c2ccc(Cl)cc2)cc1F 50320149OC(=O)c1ccc(CN(Cc2ccccc2F)S(=O)(=O)c2ccc(Cl)cc2)cc1F 50320150OC(=O)c1ccc(CN(Cc2ccccn2)S(=O)(=O)c2ccc(cc2)C#N)cc1F 50320151Clc1ccc(cc1)S(=O)(=O)N(Cc1ccc(cc1)-c1n[nH]c(=O)o1)Cc1ccccn1 50320152Clc1ccc(cc1)S(=O)(=O)N(Cc1ccc(cc1)-c1nnn[nH]1)Cc1ccccn1 50320153Fc1ccccc1CN(Cc1ccc(cc1)-c1nnn[nH]1)S(=O)(=O)c1ccc(Cl)cc1 50320154Clc1ccc(cc1)S(=O)(=O)N(Cc1ccc(cc1)-c1nnn[nH]1)Cc1cccc(Cl)c1 50320155Clc1ccc(CN(Cc2ccc(cc2)-c2nnn[nH]2)S(=O)(=O)c2ccc(Cl)cc2)cc1 50320156O=S(=O)(N(Cc1ccc(cc1)-c1nnn[nH]1)Cc1ccccn1)c1ccc(cc1)C#N 50320157CCOc1ccc(cc1)S(=O)(=O)N(Cc1ccc(cc1)-c1nnn[nH]1)Cc1ccccn1 50320158COc1ccc(CN(Cc2ccc(cc2)-c2nnn[nH]2)S(=O)(=O)c2ccc(Cl)cc2)cc1 50320159COc1cccc(CN(Cc2ccc(cc2)-c2nnn[nH]2)S(=O)(=O)c2ccc(Cl)cc2)c1 50320160Fc1ccc(CN(Cc2ccc(cc2)-c2nnn[nH]2)S(=O)(=O)c2ccc(Cl)cc2)cc1 50320161Clc1ccc(cc1)S(=O)(=O)N(CCc1cc2ccccc2cn1)Cc1ccc(cc1)-c1nnn[nH]1 50320162CC(C)(C)c1nc(CCN(Cc2ccc(cc2)-c2nnn[nH]2)S(=O)(=O)c2ccc(Cl)cc2)no1 50320163Fc1cc(CN(Cc2ccccn2)S(=O)(=O)c2ccc(Cl)cc2)ccc1-c1nnn[nH]1 50320164COc1ccc(cc1)S(=O)(=O)N(Cc1ccc(-c2nnn[nH]2)c(F)c1)Cc1ccccn1 50320165Fc1ccccc1CN(Cc1ccc(-c2nnn[nH]2)c(F)c1)S(=O)(=O)c1ccc(cc1)C#N 50320166Fc1ccccc1CN(Cc1ccc(-c2nnn[nH]2)c(F)c1)S(=O)(=O)c1ccc(Cl)cc1 50320167Fc1ccccc1CN(Cc1ccc(cc1)-c1nnn[nH]1)S(=O)(=O)c1ccc(cc1)C#N 50320168Clc1ccc(cc1)S(=O)(=O)N(Cc1ccc(cc1)-c1cccc(Cl)c1)Cc1ccccn1 50320169Fc1cccc(c1)-c1ccc(CN(Cc2ccccn2)S(=O)(=O)c2ccc(Cl)cc2)cc1 50320170Clc1ccc(cc1)S(=O)(=O)N(Cc1ccc(Cc2ccccc2)cc1)Cc1ccccn1 50320171[O-][N+](=O)c1cccc(Cc2ccc(CN(Cc3ccccn3)S(=O)(=O)c3ccc(Cl)cc3)cc2)c1 50337210CNC(=O)c1cnc(N2CCN([C@@H](C)C2)C2CCN(Cc3ccc(Cl)cc3Cl)CC2)c(Cl)c1 50337211CNC(=O)c1cnc(N2CCN([C@@H](C)C2)C2CCN(Cc3ccc(F)cc3Cl)CC2)c(Cl)c1 50337212CNC(=O)c1cnc(N2CCN([C@@H](C)C2)C2CCN(CC2)C(C)c2ccc(Cl)cc2)c(Cl)c1 50337213CNC(=O)c1cnc(N2CCN([C@@H](C)C2)C2CCN(CC2)C2CCc3cc(Cl)ccc23)c(Cl)c1 50337214CNC(=O)c1cnc(N2CCN([C@@H](C)C2)C2CCN(CC2)C(=O)c2ccc(Cl)cc2)c(Cl)c1 50337217Fc1ccc(CNC(=O)c2cnc(N3CCN(CC3)C3CCN(Cc4ccc(Cl)cc4)CC3)c(Cl)c2)cc1F 50337218C[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2)CC1)c1ncc(cc1Cl)C(=O)NCc1ccc(F)c(F)c1 50337219C[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2)CC1)c1ncc(cc1Cl)C(=O)NCc1ccc(Cl)c(Cl)c1 50337220C[C@H]1CN(CCN1c1ncc(cc1Cl)C(=O)NCc1ccc(Cl)c(Cl)c1)C1CCN(Cc2ccc(Cl)cc2)CC1 50337221C[C@@H]1CN(CCN1c1ncc(cc1Cl)C(=O)NCc1ccc(Cl)c(Cl)c1)C1CCN(Cc2ccc(Cl)cc2)CC1 50337222CC1CN(CCN1c1ccc(cn1)C(=O)NCc1ccc(F)c(F)c1)C1CCN(Cc2ccc(Cl)cc2)CC1 50337223CNC(=O)c1cnc(N2CCN(CC2)C2CCN(Cc3ccc(Cl)cc3)CC2C)c(Cl)c1 50337224CC1(CCN(Cc2ccc(Cl)cc2)CC1)N1CCN(CC1)c1ncc(cc1Cl)C(=O)NCc1ccc(Cl)c(Cl)c1 50337225Fc1ccc(CNC(=O)c2cnc(N3CCN(C4CCN(Cc5ccc(Cl)cc5)CC4)C(=O)C3)c(Cl)c2)cc1F 50337226CNC(=O)c1cnc(N2CCN([C@@H](C)C2)C2CCN(Cc3ccc(Cl)cc3)C(=O)C2)c(Cl)c1 50337228CNC(=O)c1cnc(N2CCC(CC2)N2CCN(Cc3ccc(Cl)cc3)C[C@H]2C)c(Cl)c1 50337229CNC(=O)c1cnc(N2CCC(C(C)C2)N2CCN(Cc3ccc(Cl)cc3)CC2)c(Cl)c1 50337230C[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2)CC1)c1ncc(cc1Cl)C(C)=O 50337231C[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2)CC1)c1ncc(cc1Cl)C(N)=N 50337232CCNC(=N)c1cnc(N2CCN([C@@H](C)C2)C2CCN(Cc3ccc(Cl)cc3)CC2)c(Cl)c1 50337233C[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2)CC1)c1ncc(NC(C)=O)cc1Cl 50337234C[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2)CC1)c1ncc(NC(=O)C2CC2)cc1Cl 50337235C[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2)CC1)c1ncc(cc1Cl)C(N)=O 50337236CCNC(=O)c1cnc(N2CCN([C@@H](C)C2)C2CCN(Cc3ccc(Cl)cc3)CC2)c(Cl)c1 50337237CC(C)NC(=O)c1cnc(N2CCN([C@@H](C)C2)C2CCN(Cc3ccc(Cl)cc3)CC2)c(Cl)c1 50337238C[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2)CC1)c1ncc(cc1Cl)C(=O)NCC1CCCCC1 50337239C[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2)CC1)c1ncc(cc1Cl)C(=O)Nc1ccc(F)c(F)c1 50337240C[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2)CC1)c1ncc(cc1Cl)C(=O)N1CCCCC1 50337241C[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2)CC1)c1ncc(cc1Cl)C(=O)N1CCC1 50337242CC[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2)CC1)c1ncc(cc1Cl)C(=O)NC 50337243CNC(=O)c1cnc(N2CCN([C@@H](CC(C)C)C2)C2CCN(Cc3ccc(Cl)cc3)CC2)c(Cl)c1 50337244CNC(=O)c1cnc(N2CCN(C3CCN(Cc4ccc(Cl)cc4)CC3)[C@H](C2)c2ccccc2)c(Cl)c1 50337245CNC(=O)c1cnc(N2CCN(C3CCN(Cc4ccc(Cl)cc4)CC3)C(C2)C(=O)OC)c(Cl)c1 50337246CNC(=O)c1cnc(N2CCN(C(CO)C2)C2CCN(Cc3ccc(Cl)cc3)CC2)c(Cl)c1 50337247CNC(=O)c1cnc(N2CCN(C(COC)C2)C2CCN(Cc3ccc(Cl)cc3)CC2)c(Cl)c1 50337249CNOC(=O)C1CN(CCN1C1CCN(Cc2ccc(Cl)cc2)CC1)c1ncc(cc1Cl)C(=O)NC 50337250CCNC(=O)c1cnc(N2CCN([C@@H](CC)C2)C2CCN(Cc3ccc(Cl)cc3)CC2)c(Cl)c1 50337251CCNC(=O)c1cnc(N2CCN([C@@H](CC)C2)C2CCN(Cc3ccc(Cl)cc3F)CC2)c(Cl)c1 50337252CCNC(=O)c1cnc(N2CCN(C3CCN(Cc4ccc(Cl)cc4)CC3)[C@H](C2)C(C)C)c(Cl)c1 50337253CCNC(=O)c1cnc(N2CCN(C3CCN(Cc4ccc(Cl)cc4F)CC3)C(C2)C2CC2)c(Cl)c1 50337254CNC(=O)c1cnc(N2CCN([C@@H](C)C2)C2CCN(Cc3ccc(Cl)cc3)CC2)c(Cl)c1 50337255CNC(=O)c1cnc(N2CCN([C@@H](C)C2)C2CCN(Cc3ccco3)CC2)c(Cl)c1 50337256CNC(=O)c1cnc(N2CCN([C@@H](C)C2)C2CCN(Cc3cccs3)CC2)c(Cl)c1 50337257CNC(=O)c1cnc(N2CCN([C@@H](C)C2)C2CCN(Cc3ccc[nH]3)CC2)c(Cl)c1 50337258CNC(=O)c1cnc(N2CCN([C@@H](C)C2)C2CCN(Cc3ccccn3)CC2)c(Cl)c1 50337260CNC(=O)c1cnc(N2CCN([C@@H](C)C2)C2CCN(Cc3ccc(C)cc3)CC2)c(Cl)c1 50337261CNC(=O)c1cnc(N2CCN([C@@H](C)C2)C2CCN(CC2)C(F)(F)F)c(Cl)c1 50337262CNC(=O)c1cnc(N2CCN([C@@H](C)C2)C2CCN(Cc3ccc(Cl)cc3F)CC2)c(Cl)c1 50349637CCNC(=O)[C@H]1CN([C@@H]2Cc3c[nH]c4cccc(C2=C1)c34)C(=O)Nc1ccccc1 50349638CN(C)C(=O)[C@H]1CN([C@@H]2Cc3c[nH]c4cccc(C2=C1)c34)C(=O)Nc1ccccc1 50349639COCCN(CCOC)C(=O)[C@H]1CN([C@@H]2Cc3c[nH]c4cccc(C2=C1)c34)C(=O)Nc1ccccc1 50349640CN(CCO)C(=O)[C@H]1CN([C@@H]2Cc3c[nH]c4cccc(C2=C1)c34)C(=O)Nc1ccccc1 50349641O=C(Nc1ccccc1)N1C[C@@H](C=C2[C@H]1Cc1c[nH]c3cccc2c13)C(=O)N1CCC1 50349642O=C(Nc1ccccc1)N1C[C@@H](C=C2[C@H]1Cc1c[nH]c3cccc2c13)C(=O)N1CCCCCC1 50349643O=C(Nc1ccccc1)N1C[C@@H](C=C2[C@H]1Cc1c[nH]c3cccc2c13)C(=O)N1CC=CC1 50349644O=C(Nc1ccccc1)N1C[C@@H](C=C2[C@H]1Cc1c[nH]c3cccc2c13)C(=O)N1CCCC=C1 50349645O=C(Nc1ccccc1)N1C[C@@H](C=C2[C@H]1Cc1c[nH]c3cccc2c13)C(=O)N1CCNCC1 50349646O=C(Nc1ccccc1)N1C[C@@H](C=C2[C@H]1Cc1c[nH]c3cccc2c13)C(=O)N1CCNC(=O)C1 50349647CN1CCN(CC1)C(=O)[C@H]1CN([C@@H]2Cc3c[nH]c4cccc(C2=C1)c34)C(=O)Nc1ccccc1 50349648CC(=O)N1CCN(CC1)C(=O)[C@H]1CN([C@@H]2Cc3c[nH]c4cccc(C2=C1)c34)C(=O)Nc1ccccc1 50349649O=C(Nc1ccccc1)N1C[C@@H](C=C2[C@H]1Cc1c[nH]c3cccc2c13)C(=O)N1CCOCC1 50349650CC1CN(CC(C)O1)C(=O)[C@H]1CN([C@@H]2Cc3c[nH]c4cccc(C2=C1)c34)C(=O)Nc1ccccc1 50349651O=C(Nc1ccccc1)N1C[C@@H](C=C2[C@H]1Cc1c[nH]c3cccc2c13)C(=O)N1CCS(=O)(=O)CC1 50349652OC1CCN(CC1)C(=O)[C@H]1CN([C@@H]2Cc3c[nH]c4cccc(C2=C1)c34)C(=O)Nc1ccccc1 50349653O[C@@H]1CCN(C[C@@H]1O)C(=O)[C@H]1CN([C@@H]2Cc3c[nH]c4cccc(C2=C1)c34)C(=O)Nc1ccccc1 50349654O[C@H]1CCN(C1)C(=O)[C@H]1CN([C@@H]2Cc3c[nH]c4cccc(C2=C1)c34)C(=O)Nc1ccccc1 50349655Fc1ccccc1NC(=O)N1C[C@@H](C=C2[C@H]1Cc1c[nH]c3cccc2c13)C(=O)N1CCCC1 50349656Fc1cccc(NC(=O)N2C[C@@H](C=C3[C@H]2Cc2c[nH]c4cccc3c24)C(=O)N2CCCC2)c1 50349657Fc1ccc(NC(=O)N2C[C@@H](C=C3[C@H]2Cc2c[nH]c4cccc3c24)C(=O)N2CCCC2)cc1 50349658COc1ccccc1NC(=O)N1C[C@@H](C=C2[C@H]1Cc1c[nH]c3cccc2c13)C(=O)N1CCCC1 50349659COc1ccc(NC(=O)N2C[C@@H](C=C3[C@H]2Cc2c[nH]c4cccc3c24)C(=O)N2CCCC2)cc1 50349660O=C(Nc1ccsc1)N1C[C@@H](C=C2[C@H]1Cc1c[nH]c3cccc2c13)C(=O)N1CCCC1 50349661O=C(Nc1cccs1)N1C[C@@H](C=C2[C@H]1Cc1c[nH]c3cccc2c13)C(=O)N1CCCC1 50349663O=C(NC1CCCCC1)N1C[C@@H](C=C2[C@H]1Cc1c[nH]c3cccc2c13)C(=O)N1CCCC1 50349664O=C(NC1CCCCCC1)N1C[C@@H](C=C2[C@H]1Cc1c[nH]c3cccc2c13)C(=O)N1CCCC1 50349665OC1CCC(CC1)NC(=O)N1C[C@@H](C=C2[C@H]1Cc1c[nH]c3cccc2c13)C(=O)N1CCCC1 50349667O=C(NCc1ccccc1)N1C[C@@H](C=C2[C@H]1Cc1c[nH]c3cccc2c13)C(=O)N1CCCC1 50349668O=C(NCc1ccco1)N1C[C@@H](C=C2[C@H]1Cc1c[nH]c3cccc2c13)C(=O)N1CCCC1 50349669O=C([C@H]1CN([C@@H]2Cc3c[nH]c4cccc(C2=C1)c34)C(=O)c1ccccc1)N1CCCC1 50349670O=C(Cc1ccccc1)N1C[C@@H](C=C2[C@H]1Cc1c[nH]c3cccc2c13)C(=O)N1CCCC1 50349671CC(C)OC(=O)Cn1cc2C[C@H]3N(C[C@@H](C=C3c3cccc1c23)C(=O)N1CCCC1)C(=O)Nc1ccccc1 50349672OCCn1cc2C[C@H]3N(C[C@@H](C=C3c3cccc1c23)C(=O)N1CCCC1)C(=O)Nc1ccccc1 50349673CN(C)CCn1cc2C[C@H]3N(C[C@@H](C=C3c3cccc1c23)C(=O)N1CCCC1)C(=O)Nc1ccccc1 50349674O=C(Nc1ccccc1)N1C[C@@H](C=C2[C@H]1Cc1cn(CCN3CCCC3)c3cccc2c13)C(=O)N1CCCC1 50349675O=C(Nc1ccccc1)N1C[C@@H](C=C2[C@H]1Cc1cn(CCN3CCCCC3)c3cccc2c13)C(=O)N1CCCC1 50349676CN1CCN(CCn2cc3C[C@H]4N(C[C@@H](C=C4c4cccc2c34)C(=O)N2CCCC2)C(=O)Nc2ccccc2)CC1 50349677O=C(Nc1ccccc1)N1C[C@@H](C=C2[C@H]1Cc1cn(CCN3CCOCC3)c3cccc2c13)C(=O)N1CCCC1 50349678O=C(Nc1ccccc1)N1C[C@@H](C=C2[C@H]1Cc1c[nH]c3cccc2c13)C(=O)N1CCCC1 50349679O=C(Nc1ccccc1)N1C[C@@H](C=C2[C@H]1Cc1c[nH]c3cccc2c13)C(=O)N1CCCCC1 50349680O[C@@H]1CCN(C1)C(=O)[C@H]1CN([C@@H]2Cc3c[nH]c4cccc(C2=C1)c34)C(=O)Nc1ccccc1 50349681COc1cccc(NC(=O)N2C[C@@H](C=C3[C@H]2Cc2c[nH]c4cccc3c24)C(=O)N2CCCC2)c1 50349683CN(C)Cc1ccc(NC(=O)N2C[C@@H](C=C3[C@H]2Cc2c[nH]c4cccc3c24)C(=O)N2CCCC2)cc1 50349684O=C(NC1CCCC1)N1C[C@@H](C=C2[C@H]1Cc1c[nH]c3cccc2c13)C(=O)N1CCCC1 50349686CN(C)Cc1cccc(NC(=O)N2C[C@@H](C=C3[C@H]2Cc2c[nH]c4cccc3c24)C(=O)N2CCCC2)c1 50358605CC[C@H]1CN([C@H](CC)CN1C1CCN(CC1)C(=O)c1ccc(Cl)cc1)c1ncc(nc1C)C(N)=O 50358607CC[C@H]1CN([C@H](C)CN1C1CCN(CC1)C(=O)c1ccc(Cl)cc1)c1ncc(nc1C)C(=O)NC 50358608CC[C@H]1CN([C@H](C)CN1C1CCN(CC1)C(=O)c1ccc(Cl)cc1)c1ncc(nc1C)C(=O)NC1CC1 50358609CC[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2)CC1)c1nc(N)c(nc1Cl)C(N)=O 50358610CC[C@H]1CN(CCN1C1CCN(Cc2ccc(OC(F)(F)F)cc2)CC1)c1nc(N)c(nc1Cl)C(N)=O 50358611CC[C@H]1CN(CCN1C1CCN(Cc2ccc(cc2)C#N)CC1)c1nc(N)c(nc1Cl)C(N)=O 50358612CC[C@H]1CN(CCN1C1CCN(CC1)C(CO)c1ccc(Cl)cc1)c1nc(N)c(nc1Cl)C(N)=O 50358613CC[C@H]1CN(CCN1C1CCN(CC1)C(=O)c1ccc(Cl)cc1)c1nc(N)c(nc1Cl)C(N)=O 50358614CC[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2)CC1)c1nc(N)c(nc1Cl)C(=O)NC 50358615CC[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2)CC1)c1nc(N)c(nc1Cl)C(=O)NCC(F)(F)F 50358616CC[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2)CC1)c1nc(N)c(nc1Cl)C(=O)NCCO 50358617CC[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2)CC1)c1nc(N)c(nc1Cl)C(=O)NCC(C)O 50358618CC[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2)CC1)c1nc(N)c(nc1Cl)C(=O)NCC(C)(C)O 50358619CC[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2)CC1)c1nc(N)c(nc1Cl)C(=O)NCCNS(=O)(=O)C(F)(F)F 50358620CC[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2)CC1)c1nc(N)c(nc1Cl)C(=O)NCCNS(N)(=O)=O 50358621CC[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2)CC1)c1nc(N)c(nc1Cl)C(=O)NCCS(C)(=O)=O 50358622CC[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2)CC1)c1nc(N)c(nc1Cl)C(=O)N[C@@H]1CCOC1=O 50358623CC[C@H]1CN(CCN1C1CCN(Cc2ccc(F)c(F)c2)CC1)c1nc(N)c(nc1Cl)C(=O)NCCNS(N)(=O)=O 50358624CC[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2)CC1)c1nc(N)c(nc1Cl)C(=O)NCCNS(C)(=O)=O 50358625CC[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2[C@H](O)C(N)=O)CC1)c1nc(N)c(nc1Cl)C(N)=O 50358626CC[C@H]1CN(CCN1C1CCN(CC1)C(=O)c1ccc(Cl)nc1N)c1nc(N)c(nc1Cl)C(=O)NCCO 50358627CC[C@H]1CN(CCN1C1CCN(CC1)C(=O)c1ccc(Cl)nc1N)c1ncc(nc1Cl)C(N)=O 50358628CC[C@H]1CN(CCN1C1CCN(CC1)C(=O)c1ccc(Cl)nc1N)c1ncc(nc1Cl)C(=O)NC(C)(C)C 50358629CC[C@H]1CN(CCN1C1CCN(CC1)C(=O)c1ccc(Cl)nc1N)c1ncc(nc1Cl)C(=O)NC1CC1 50358630CC[C@H]1CN(CCN1C1CCN(CC1)C(=O)c1ccc(Cl)nc1N)c1ncc(nc1Cl)C(=O)NC(C)C 50358631CC[C@H]1CN(CCN1C1CCN(CC1)C(=O)c1ccc(Cl)nc1N)c1ncc(nc1Cl)C(=O)NCCO 50358632CC[C@H]1CN(CCN1C1CCN(CC1)C(=O)c1ccc(Cl)nc1N)c1ncc(nc1Cl)C(=O)NC[C@@H](C)O 50358633CC[C@H]1CN(CCN1C1CCN(CC1)C(=O)c1ccc(Cl)nc1N)c1ncc(nc1C(F)(F)F)C(N)=O 50358634CC[C@H]1CN(CCN1C1CCN(CC1)C(=O)c1ccc(Cl)nc1N)c1ncc(nc1C(F)(F)F)C(=O)NC 50358635CC[C@H]1CN(CCN1C1CCN(CC1)C(=O)c1ccc(Cl)nc1N)c1ncc(nc1C(F)(F)F)C(=O)NC1CC1 50358636CC[C@H]1CN(CCN1C1CCN(CC1)C(=O)c1ccc(Cl)nc1N)c1ncc(nc1C)C(N)=O 50358637CC[C@H]1CN(CCN1C1CCN(CC1)C(=O)c1ccc(Cl)nc1N)c1ncc(nc1C)C(=O)NC 50358638CC[C@H]1CN(CCN1C1CCN(CC1)C(=O)c1ccc(Cl)nc1N)c1ncc(nc1C)C(=O)NC1CC1 50358639CC[C@H]1CN(CCN1C1CCN(CC1)C(=O)c1ccc(Cl)cc1)c1ncc(nc1C)C(N)=O 50358640CC[C@H]1CN(CCN1C1CCN(CC1)C(=O)c1ccc(Cl)cc1)c1ncc(nc1C)C(=O)NC 50358641CCNC(=O)c1cnc(N2CCN([C@@H](CC)C2)C2CCN(CC2)C(=O)c2ccc(Cl)cc2)c(C)n1 50358642CC[C@H]1CN(CCN1C1CCN(CC1)C(=O)c1ccc(Cl)cc1)c1ncc(nc1C)C(=O)NC1CC1 50358643CC[C@H]1CN([C@H](C)CN1C1CCN(CC1)C(=O)c1ccc(Cl)cc1)c1ncc(nc1C)C(N)=O 50361979CCS(=O)(=O)CCN([C@H](C)c1nc2ncccc2c(=O)n1-c1ccc(F)cc1)C(=O)Cc1ccc(c(F)c1)C(F)(F)F 50361980C[C@@H](N(CC1CCS(=O)(=O)CC1)C(=O)Cc1ccc(OC(F)(F)F)cc1)c1nc2ccccn2c(=O)c1-c1ccc(cc1)C#N 50361981C[C@@H](N(CC1CCS(=O)(=O)CC1)C(=O)Cc1ccc(F)c(c1)C(F)(F)F)c1nc2ncccc2c(=O)n1-c1ccc(cc1)C#N 50361982C[C@@H](N(CC1CCS(=O)(=O)CC1)C(=O)Cc1ccc(c(F)c1)C(F)(F)F)c1nc2ncccc2c(=O)n1-c1ccc(cc1)C#N 50361983C[C@@H](N(Cc1cccnc1)C(=O)Cc1ccc(OC(F)(F)F)cc1)c1nc2ncccc2c(=O)n1-c1ccc(O)cc1 50361984C[C@@H](N(CC1CCS(=O)(=O)CC1)C(=O)Cc1ccc(c(F)c1)C(F)(F)F)c1nc2ncccc2c(=O)n1-c1ccc(F)cc1 50361985C[C@@H](N(CC1CCS(=O)(=O)CC1)C(=O)Cc1ccc(F)c(c1)C(F)(F)F)c1nc2ncccc2c(=O)n1-c1ccc(F)cc1 50361986CCS(=O)(=O)CCN([C@H](C)c1nc2ncccc2c(=O)n1-c1ccc(F)cc1)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50361987C[C@@H](N(CC1CCS(=O)(=O)CC1)C(=O)Cc1ccc(c(F)c1)C(F)(F)F)c1nc2ncccc2c(=O)n1-c1ccc(Cl)cc1 50361988C[C@@H](N(CC1CCS(=O)(=O)CC1)C(=O)Cc1ccc(F)c(c1)C(F)(F)F)c1nc2ncccc2c(=O)n1-c1ccc(Cl)cc1 50361989CCS(=O)(=O)CCN([C@H](C)c1nc2ncccc2c(=O)n1-c1ccc(Cl)cc1)C(=O)Cc1ccc(c(F)c1)C(F)(F)F 50361990CCS(=O)(=O)CCN([C@H](C)c1nc2ncccc2c(=O)n1-c1ccc(Cl)cc1)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50361991C[C@@H](N(CCS(C)(=O)=O)C(=O)Cc1ccc(F)c(c1)C(F)(F)F)c1nc2ncccc2c(=O)n1-c1ccc(cc1)C#N 50371483CCOc1ccc(cc1)-n1cc(nc1[C@@H](C)N(Cc1cccnc1)C(=O)Cc1ccc(F)c(c1)C(F)(F)F)-c1ccccc1 50371484CCS(=O)(=O)CCN([C@H](C)c1nc(C2CC2)c(Cl)n1-c1ccc(cc1)C#N)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50371485CCS(=O)(=O)CCN([C@H](C)c1nc(C2CC2)c(CF)n1-c1ccc(cc1)C#N)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50371486CCS(=O)(=O)CCN([C@H](C)c1nc(C2CC2)c(C=C)n1-c1ccc(cc1)C#N)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50371487CCS(=O)(=O)CCN([C@H](C)c1nc(cn1-c1ccc(cc1)C#N)-c1ccccn1)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50371488CCOc1ccc(cc1)-n1cc(nc1[C@@H](C)N(CCS(=O)(=O)CC)C(=O)Cn1nnc(n1)C1CC1)-c1ccccc1 50371489CCOc1ccc(cc1)-n1cc(nc1[C@@H](C)N(CCS(=O)(=O)CC)C(=O)Cn1nnc(n1)-c1ccccc1)-c1ccccc1 50371490CCOc1ccc(cc1)-n1ccnc1[C@@H](C)N(Cc1cccnc1)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50371491CCOc1ccc(cc1)-n1cc(nc1[C@@H](C)N(CCS(=O)(=O)CC)C(=O)Cn1cnc(c1)-c1ccccc1)-c1ccccc1 50371492CCOc1ccc(cc1)-n1cc(nc1[C@@H](C)N(CCS(=O)(=O)CC)C(=O)Cc1ccc(OC(F)(F)F)cc1)-c1ccccc1 50371493CCOc1ccc(cc1)-n1cc(nc1[C@@H](C)N(CCCS(=O)(=O)CC)C(=O)Cc1ccc(F)c(c1)C(F)(F)F)-c1ccccc1 50371494CCOc1ccc(cc1)-n1cc(nc1[C@@H](C)N(CCS(=O)(=O)CC)C(=O)Cc1ccc(F)c(c1)C(F)(F)F)-c1ccccc1 50371495CCOCCN([C@H](C)c1nc(cn1-c1ccc(OCC)cc1)-c1ccccc1)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50371496CCOc1ccc(cc1)-n1cc(nc1[C@@H](C)N(C[C@@H]1CCCN1C)C(=O)Cc1ccc(F)c(c1)C(F)(F)F)-c1ccccc1 50371497CCOc1ccc(cc1)-n1cc(nc1[C@@H](C)N(C[C@H]1CCCN1C)C(=O)Cc1ccc(F)c(c1)C(F)(F)F)-c1ccccc1 50371498CCOc1ccc(cc1)-n1cc(nc1[C@@H](C)N(C[C@@H]1CCCN1)C(=O)Cc1ccc(F)c(c1)C(F)(F)F)-c1ccccc1 50371499CCOc1ccc(cc1)-n1cc(nc1[C@@H](C)N(C[C@H]1CCCN1)C(=O)Cc1ccc(F)c(c1)C(F)(F)F)-c1ccccc1 50371500CCOc1ccc(cc1)-n1cc(nc1[C@@H](C)N(Cc1ccccn1)C(=O)Cc1ccc(F)c(c1)C(F)(F)F)-c1ccccc1 50371501CCOc1ccc(cc1)-n1cc(nc1[C@@H](C)N(Cc1ccncc1)C(=O)Cc1ccc(F)c(c1)C(F)(F)F)-c1ccccc1 50371502CCS(=O)(=O)CCN([C@H](C)c1nc(C2CC2)c(-c2ccccc2)n1-c1ccc(cc1)C#N)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50371503CCS(=O)(=O)CCN([C@H](C)c1nc(C2CC2)c(C#N)n1-c1ccc(cc1)C#N)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50371504CCS(=O)(=O)CCN([C@H](C)c1nc(C2CC2)c(n1-c1ccc(cc1)C#N)C(F)(F)F)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50371505CCS(=O)(=O)CCN([C@H](C)c1nc(C2CC2)c(C(F)F)n1-c1ccc(cc1)C#N)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50371506CCS(=O)(=O)CCN([C@H](C)c1nc(C2CC2)c(CO)n1-c1ccc(cc1)C#N)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50371507CCc1c(nc([C@@H](C)N(CCS(=O)(=O)CC)C(=O)Cc2ccc(F)c(c2)C(F)(F)F)n1-c1ccc(cc1)C#N)C1CC1 50371508CCS(=O)(=O)CCN([C@H](C)c1nc(cn1-c1ccc(cc1)C#N)C(C)(C)C)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50371509CCS(=O)(=O)CCN([C@H](C)c1nc(cn1-c1ccc(cc1)C#N)C(C)C)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50371510CCS(=O)(=O)CCN([C@H](C)c1nc(cn1-c1ccc(cc1)C#N)C1CC1)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50371511CCS(=O)(=O)CCN([C@H](C)c1nc(cn1-c1ccc(cc1)C#N)-c1cccnc1)C(=O)Cc1ccc(F)c(c1)C(F)(F)F 50371512CCOc1ccc(cc1)-n1cc(nc1[C@@H](C)N(CCS(=O)(=O)CC)C(=O)Cn1ccc(n1)C(F)(F)F)-c1ccccc1 50371513CCOc1ccc(cc1)-n1cc(nc1[C@@H](C)N(CCS(=O)(=O)CC)C(=O)Cn1nnc(n1)-c1ccc(cc1)C(F)(F)F)-c1ccccc1 50371514CCOc1ccc(cc1)-n1cc(nc1[C@@H](C)N(CCS(=O)(=O)CC)C(=O)Cn1nnc(n1)-c1ccc(F)cc1)-c1ccccc1 50371515CCOc1ccc(cc1)-n1cc(nc1[C@@H](C)N(CCS(=O)(=O)CC)C(=O)Cn1cc(nn1)-c1ccccc1)-c1ccccc1 50371834CC(=O)c1nc2ccccc2n1CC(=O)c1ccc(cc1)[N+]([O-])=O 50371835Cn1c2c(cccc2n(CC(=O)c2ccc(Cl)cc2)c1=N)C(F)(F)F 50371836Cn1c2c(Cl)cccc2n(CC(=O)c2ccc(Cl)cc2)c1=N 50371837CCc1cccc2n(CC(=O)c3ccc(Cl)cc3)c(=N)n(C)c12 50371838Cc1cccc2n(CC(=O)c3ccc(Cl)cc3)c(=N)n(C)c12 50371839Cc1ccc2n(CC(=O)c3ccc(Cl)cc3)c(=N)n(C)c2c1 50371841Cn1c2ccccc2n(CCCC(=O)c2ccc(Br)cc2)c1=N 50371842Cn1c2ccccc2n(CS(=O)c2ccc(Cl)cc2)c1=N 50371847CN=c1n(C)c2ccccc2n1CC(=O)c1ccc(Cl)cc1 50371853COc1cccc2n(CC(=O)c3ccc(Br)cc3)c(nc12)C(C)=O 50371855CC(=O)c1nc2ccccc2n1CC(=O)c1ccc(Br)cc1 50371857COc1cccc2n(CC(=O)c3ccc(Br)cc3)c(=N)n(C)c12 50371858CCCc1cccc2n(CC(=O)c3ccc(Cl)cc3)c(=N)n(C)c12 50371859Cc1ccc2n(C)c(=N)n(CC(=O)c3ccc(Cl)cc3)c2c1 50371862COCCN=c1n(C)c2ccccc2n1CC(=O)c1ccc(Br)cc1 50371865CC(=O)c1nc2ccccc2n1CC(=O)c1ccc(Cl)cc1 50372000CC(=O)N1C2CCCC1C=C(CN1[C@H]3CC[C@@H]1C[C@H](C3)Nc1ccc3ccc(cc3n1)C(F)(F)F)C2 50372001CC(C)Oc1cc(F)c2ccc(NC3CCN(CC4=CC5CCCC(C4)N5C(C)=O)CC3)nc2c1 50372002CC(=O)N1C2CCCC1C=C(CN1CCC(CC1)Nc1ccc3cc(ccc3n1)C(F)(F)F)C2 50372003CC(=O)N1C2CCCC1C=C(CN1CCC(CC1)Nc1ccc3cccc(Cl)c3n1)C2 50372004CN(C1CCN(CC2=CC3CCCC(C2)N3C(C)=O)CC1)c1nc2ccccc2s1 50372005CC(C)Oc1cc(F)c2ccc(N[C@H]3C[C@@H]4CC[C@H](C3)N4CC3=CC4CCCC(C3)N4C(C)=O)nc2c1 50372006CC(C)Oc1ccc2ccc(N[C@H]3C[C@@H]4CC[C@H](C3)N4CC3=CC4CCCC(C3)N4C(C)=O)nc2c1 50372007CC(=O)N1C2CCCC1C=C(CN1[C@H]3CC[C@@H]1C[C@H](C3)Nc1ccc3cc(ccc3n1)C(F)(F)F)C2 50372008CC(=O)N1C2CCCC1C=C(CN1[C@H]3CC[C@@H]1C[C@H](C3)Nc1ccc3cc(OC(F)(F)F)ccc3n1)C2 50372009COc1cc(F)c2ccc(NC3CCN(CC4=CC5CCCC(C4)N5C(C)=O)CC3)nc2c1 50372010CC(C)Oc1ccc2ccc(NC3CCN(CC4=CC5CCCC(C4)N5C(C)=O)CC3)nc2c1 50372011CC(=O)N1C2CCCC1C=C(CN1CCC(CC1)Nc1ccc3ccc(cc3n1)C(F)(F)F)C2 50372012CC(=O)N1C2CCCC1C=C(CN1CCC(CC1)Nc1ccc3cc(OC(F)(F)F)ccc3n1)C2 50372013CC(=O)N1C2CCCC1C=C(CN1CCC(CC1)Nc1ccc3cc(Cl)ccc3n1)C2 50372014CC(=O)N1C2CCCC1C=C(CN1CCC(CC1)Nc1cnc3ccccc3n1)C2 50372015CC(=O)N1C2CCCC1C=C(CN1CCC(CC1)Nc1ccc3c(cc(nc3n1)C(F)(F)F)C(F)(F)F)C2 50372016CC(=O)N1C2CCCC1C=C(CN1CCC(CC1)Nc1ccc3ccccc3n1)C2 50375111CN(CCCn1c2c(Cl)cccc2n(CC(=O)c2ccc(Cl)cc2)c1=N)C(=O)c1ccccc1 50375112CN(CCCCn1c2c(Cl)cccc2n(CC(=O)c2ccc(Cl)cc2)c1=N)C(=O)Cc1ccccc1 50375113CN(CCn1c2ccccc2n(CC(=O)c2ccc(Cl)cc2)c1=N)C(=O)Cc1ccccc1 50375114CN(Cc1ccccc1)C(=O)CCn1c2ccccc2n(CC(=O)c2ccc(Cl)cc2)c1=N 50375116Clc1ccc(cc1)C(=O)Cn1c2cccc(Cl)c2n(C[C@H]2CCCN(C2)C(=O)c2cccc3cccnc23)c1=N 50375117CN(CCCn1c2c(Cl)cccc2n(CC(=O)c2ccc(Cl)cc2)c1=N)C(=O)c1ccccn1 50375118CN(CCCn1c2c(Cl)cccc2n(CC(=O)c2ccc(Cl)cc2)c1=N)C(=O)C(C)(C)C 50375119Clc1ccc(cc1)C(=O)Cn1c2cccc(Cl)c2n(CCCN(C2CC2)C(=O)c2cccc3cccnc23)c1=N 50375120Clc1ccc(cc1)C(=O)Cn1c2cccc(Cl)c2n(CC[C@@H]2CCCN2C(=O)c2cccc3cccnc23)c1=N 50375121Clc1ccc(cc1)C(=O)Cn1c2cccc(Cl)c2n(C[C@@H]2CCCN(C2)C(=O)c2cccc3cccnc23)c1=N 50375122CN(CCCn1c2c(Cl)cccc2n(CC(=O)c2ccc(Cl)cc2)c1=N)C(=O)c1cccc2cccnc12 50375123COc1ccccc1C(=O)N(C)CCCn1c2c(Cl)cccc2n(CC(=O)c2ccc(Cl)cc2)c1=N 50375124CN(CCCn1c2c(Cl)cccc2n(CC(=O)c2ccc(Cl)cc2)c1=N)C(=O)c1ccc2ccccc2c1 50375125CCc1cccc2n(CC(=O)c3ccc(Cl)cc3)c(=N)n(CCCN(C)C(=O)Cc3ccccc3)c12 50375126CN(CCCn1c2c(Cl)cccc2n(CC(=O)c2ccc(Cl)cc2)c1=N)C(=O)Cc1ccccc1 50375127CN(CCn1c2c(Cl)cccc2n(CC(=O)c2ccc(Cl)cc2)c1=N)C(=O)Cc1ccccc1 50375128CN(CCn1c2ccccc2n(CC(=O)c2ccc(Cl)cc2)c1=N)C(=O)c1ccccc1 50375129CN(CCn1c2ccccc2n(CC(=O)c2ccc(Cl)cc2)c1=N)C(=O)C1CCCCC1 50375130CN(CCn1c2ccccc2n(CC(=O)c2ccc(Cl)cc2)c1=N)C(C)=O 50375131CN(Cc1ccccc1)C(=O)Cn1c2ccccc2n(CC(=O)c2ccc(Cl)cc2)c1=N 50375132CCOC(=O)CCn1c2ccccc2n(CC(=O)c2ccc(Cl)cc2)c1=N 50375133CCn1c2ccccc2n(CC(=O)c2ccc(Cl)cc2)c1=N 50399980NCCCC[C@H](NC(=O)[C@@H]1Cc2ccccc2CN1C(=O)CCC(=O)c1ccccc1)C(=O)NCC(c1ccccc1)c1ccccc1 50399981CC1(C)[C@H]2C[C@@H]1C(C[N+](C)(C)Cc1ccc(cc1)-c1ccccc1I)=CC2 50399982CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccc(cc1)-c1ccccc1I)=CC2 50399983CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccc(cc1)-c1ccccc1Br)=CC2 50399984CC1(C)[C@@H]2C[C@H]1[C@H](C[N+](C)(C)Cc1ccc(cc1)-c1ccccc1I)CC2 50399985CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccc(cc1)-c1ccccc1Cl)=CC2 50399986COc1ccccc1-c1ccc(C[N+](C)(C)CC2=CC[C@H]3C[C@@H]2C3(C)C)cc1 50399987Cc1ccccc1-c1ccc(C[N+](C)(C)CC2=CC[C@H]3C[C@@H]2C3(C)C)cc1 50399988CC1(C)[C@@H]2C[C@H]1C=C(C[N+](C)(C)Cc1ccc(cc1)-c1ccccc1I)C2 50399989CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccc(cc1)-c1cccc(Br)c1)=CC2 50399990CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccc(c(Cl)c1)-c1ccccc1Cl)=CC2 50399991CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccc(Cl)cc1)=CC2 50399992CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccc(cc1)-c1cc(Cl)ccc1Cl)=CC2 50399993CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccc(cc1)-c1cccc(Cl)c1)=CC2 50399994CC1(C)[C@H]2C[C@@H]1C(C[N+](C)(C)Cc1ccc(cc1)-c1cccc(Cl)c1)=CC2 50399995CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccc(cc1)-c1c(Cl)cccc1Cl)=CC2 50399996CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccc(cc1)-c1cccc(Cl)c1Cl)=CC2 50399997CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccc-3c(Cc4ccccc-34)c1)=CC2 50399998CC1(C)[C@@H]2C[C@H]1C=C(C[N+](C)(C)Cc1ccc(cc1)-c1cccc(Cl)c1)C2 50399999CC1(C)[C@@H]2C[C@H]1[C@H](C[N+](C)(C)Cc1ccc(cc1)-c1cccc(Cl)c1)CC2 50400000CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccc(c(Cl)c1)-c1cccc(Cl)c1)=CC2 50400001CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccc(cc1)-c1ccccc1F)=CC2 50400002CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccc(c(Cl)c1)-c1ccccc1)=CC2 50400003CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccc(cc1)-c1ccccc1)=CC2 50400004Cc1cccc(C)c1-c1ccc(C[N+](C)(C)CC2=CC[C@H]3C[C@@H]2C3(C)C)cc1 50400005CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccc(cc1)-c1ccccc1O)=CC2 50400006CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccccc1)=CC2 50400912CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccc(cc1)-c1ccsc1)=CC2 50400913CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccc(I)cc1)=CC2 50400914NC(Nc1ccc(I)cc1)=NC1C2CC3CC(C2)CC1C3 50400915CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccc(cc1)-c1ccoc1)=CC2 50400916CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccc(cc1)-c1cc(Cl)cc(Cl)c1)=CC2 50400917CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccc(cc1)-c1ccc(Cl)cc1)=CC2 50400918CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccc(cc1)-c1cccc(N)c1)=CC2 50400919CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccc(cc1)-c1cccc(O)c1)=CC2 50400920CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccc(cc1)-c1cccc(c1)[N+]([O-])=O)=CC2 50400921Cc1cccc(c1)-c1ccc(C[N+](C)(C)CC2=CC[C@H]3C[C@@H]2C3(C)C)cc1 50400922COc1ccc(cc1OC)-c1ccc(C[N+](C)(C)CC2=CC[C@H]3C[C@@H]2C3(C)C)cc1 50400923CC(=O)c1cccc(c1)-c1ccc(C[N+](C)(C)CC2=CC[C@H]3C[C@@H]2C3(C)C)cc1 50400924COC(=O)c1cccc(c1)-c1ccc(C[N+](C)(C)CC2=CC[C@H]3C[C@@H]2C3(C)C)cc1 50400925CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccc(cc1)-c1ccc(cc1)C(F)(F)F)=CC2 50400926CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccc(cc1)-c1cccc(c1)C(F)(F)F)=CC2 50400927CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccc(cc1)-c1cccc(F)c1)=CC2 50400928CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccc3oc4ccccc4c3c1)=CC2 50400929Cn1c2ccccc2c2ccc(C[N+](C)(C)CC3=CC[C@H]4C[C@@H]3C4(C)C)cc12 50400930CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccc(Oc3ccccc3)cc1)=CC2 50400931CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1cccc(c1)-c1ccccc1)=CC2 50400932CN(CC1=CC[C@H]2C[C@@H]1C2(C)C)Cc1ccc(cc1)-c1ccsc1 50400933CN(CC1=CC[C@H]2C[C@@H]1C2(C)C)Cc1ccc(cc1)-c1ccoc1 50400936CN(CC1=CC[C@H]2C[C@@H]1C2(C)C)Cc1ccc(cc1)-c1cccc(Cl)c1 50400937CN(CC1=CC[C@H]2C[C@@H]1C2(C)C)Cc1ccc(cc1)-c1cccc(N)c1 50400939CN(CC1=CC[C@H]2C[C@@H]1C2(C)C)Cc1ccc(cc1)-c1cccc(c1)[N+]([O-])=O 50400947CN(CC1=CC[C@H]2C[C@@H]1C2(C)C)Cc1ccc(cc1)-c1cccc(F)c1 50400953CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)CCc1ccc(Cl)cc1)=CC2 50400954CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccc(Cl)c(Cl)c1)=CC2 50400955CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccc(Br)cc1)=CC2 50400956CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccc(F)cc1)=CC2 50400957CC1(C)[C@@H]2C[C@H]1C(C[N+]1(C)CCc3ccccc3C1)=CC2 50400958CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1ccccc1I)=CC2 50400959CC1(C)[C@@H]2C[C@H]1C(C[N+](C)(C)Cc1cccc(I)c1)=CC2 50400960CN(CC1=CC[C@H]2C[C@@H]1C2(C)C)Cc1ccc(cc1)-c1ccccc1 50400961CN(CCc1ccc(Cl)cc1)CC1=CC[C@H]2C[C@@H]1C2(C)C 50400962CN(CC1=CC[C@H]2C[C@@H]1C2(C)C)Cc1ccc(Cl)c(Cl)c1 50400963CN(CC1=CC[C@H]2C[C@@H]1C2(C)C)Cc1ccc(Br)cc1 50400964CN(CC1=CC[C@H]2C[C@@H]1C2(C)C)Cc1ccc(Cl)cc1 50400965CN(CC1=CC[C@H]2C[C@@H]1C2(C)C)Cc1ccc(F)cc1 50400968CN(CC1=CC[C@H]2C[C@@H]1C2(C)C)Cc1ccccc1I 50400969CN(CC1=CC[C@H]2C[C@@H]1C2(C)C)Cc1cccc(I)c1 50400970CC[N+](C)(CC1=CC[C@H]2C[C@@H]1C2(C)C)Cc1ccc(I)cc1 50400971CC1(C)[C@@H]2CC[C@@]1(C)C(C[N+](C)(C)Cc1ccc(I)cc1)C2 50400972C[N+](C)(Cc1ccc(I)cc1)C\C1=C\CCCCCC1 50400973C[N+](C)(CCC12CC3CC(CC(C3)C1)C2)Cc1ccc(I)cc1 50400974C[N+](C)(Cc1ccc(I)cc1)CC12CC3CC(CC(C3)C1)C2 50400975C[N+](C)(CC1C2CC3CC(C2)CC1C3)Cc1ccc(I)cc1 50400976CCN(CC1=CC[C@H]2C[C@@H]1C2(C)C)Cc1ccc(I)cc1 50400977CN(CC1=CC[C@H]2C[C@@H]1C2(C)C)Cc1ccc(I)cc1 50400978CN(CC1C[C@H]2CC[C@]1(C)C2(C)C)Cc1ccc(I)cc1 50400979CN(Cc1ccc(I)cc1)C\C1=C\CCCCCC1 50400980CN(CCC12CC3CC(CC(C3)C1)C2)Cc1ccc(I)cc1 50400981CN(CC1C2CC3CC(C2)CC1C3)Cc1ccc(I)cc1 50400982Ic1ccc(CNCC2C3CC4CC(C3)CC2C4)cc1 50412551CC1(C)[C@@H]2CC[C@@]1(CS(=O)(=O)N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(N)C2 50412552CC1(C)[C@@H]2CC[C@@]1(CS(=O)(=O)N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(C2)NS(C)(=O)=O 50412553CCNC(=O)NC1C[C@H]2CC[C@]1(CS(=O)(=O)N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C2(C)C 50412554C[C@@H]1CN(CCN1c1ncc(cc1F)C(F)(F)F)S(=O)(=O)C[C@]12CC[C@H](CC1=O)C2(C)C 50412555C[C@H]1CN(CCN1c1ccc(cn1)C(F)(F)F)S(=O)(=O)C[C@]12CC[C@H](CC1O)C2(C)C 50412556C[C@H]1CN(CCN1c1ccc(cn1)C(F)(F)F)S(=O)(=O)C[C@]12CC[C@H](C[C@@H]1O)C2(C)C 50412557C[C@H]1CN(CCN1c1ncc(cc1F)C(F)(F)F)S(=O)(=O)C[C@]12CC[C@H](CC11OCCO1)C2(C)C 50412558CC1(C)[C@@H]2CC[C@@]1(CS(=O)(=O)N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(=O)C2 50412559C[C@H]1CN(CCN1c1ncc(cn1)C(F)(F)F)S(=O)(=O)C[C@]12CC[C@H](CC1=O)C2(C)C 50412560C[C@H]1CN(CCN1c1ncc(cc1F)C(F)(F)F)S(=O)(=O)C[C@]12CC[C@H](C[C@H]1O)C2(C)C 50412561C[C@H]1CN(CCN1c1ccc(cn1)C(F)(F)F)S(=O)(=O)C[C@]12CC[C@H](C[C@H]1O)C2(C)C 50412562CC1(C)[C@@H]2CC[C@@]1(CS(=O)(=O)N1CCN([C@H](CO)C1)c1ncc(cc1F)C(F)(F)F)C(=O)C2 50412563C[C@H]1CN(CCN1c1ccc(cn1)C(F)(F)F)S(=O)(=O)C[C@]12CC[C@H](CC1=O)C2(C)C 50412564CC1(C)[C@@H]2CC[C@@]1(CS(=O)(=O)N1CCN(CC1)c1ncc(cc1F)C(F)(F)F)C(=O)C2 50412573CC1(C)[C@@H]2CC[C@@]1(CS(=O)(=O)N1CCN(CC1)c1ncc(cc1[N+]([O-])=O)C(F)(F)F)C(=O)C2 50412574CC1(C)[C@@H]2CC[C@@]1(CS(=O)(=O)N1CCN(CC1)c1ncc(cc1Cl)C(F)(F)F)C(=O)C2 50412575CC1(C)[C@@H]2CC[C@@]1(CS(=O)(=O)N1CCN(CC1)c1ccc(c(Cl)n1)C(F)(F)F)C(=O)C2 50412576CC1(C)[C@@H]2CC[C@@]1(CS(=O)(=O)N1CCN(CC1)c1nc(Cl)c(cc1Cl)C(F)(F)F)C(=O)C2 50412578CC1(C)[C@@H]2CC[C@@]1(CS(=O)(=O)N1CCN(CC1)c1ccc(cc1F)C(F)(F)F)C(=O)C2 50412579CC1(C)[C@@H]2CC[C@@]1(CS(=O)(=O)N1CCN(CC1)c1ncc(cn1)C(F)(F)F)C(=O)C2 50412580CC1(C)[C@@H]2CC[C@@]1(CS(=O)(=O)N1CCN(CC1)c1ncc(Br)cn1)C(=O)C2 50412581CC1(C)[C@@H]2CC[C@@]1(CS(=O)(=O)N1CCN(CC1)c1ccc(nn1)C(F)(F)F)C(=O)C2 50412584CC1CN(CCN1S(=O)(=O)C[C@]12CC[C@H](CC1=O)C2(C)C)c1ccc(cn1)C(F)(F)F 50412585C[C@H]1CN([C@H](C)CN1c1ccc(cn1)C(F)(F)F)S(=O)(=O)C[C@]12CC[C@H](CC1=O)C2(C)C 50412587C[C@@H]1CN(CCN1c1ccc(cn1)C(F)(F)F)S(=O)(=O)C[C@]12CC[C@H](CC1=O)C2(C)C 50412588CCC1CN(CCN1c1ccc(cn1)C(F)(F)F)S(=O)(=O)C[C@]12CC[C@H](CC1=O)C2(C)C 50412589CC1(C)[C@@H]2CC[C@@]1(CS(=O)(=O)N1CCN(C(CO)C1)c1ccc(cn1)C(F)(F)F)C(=O)C2 50412592CC1(C)[C@@H]2CC[C@@]1(CS(=O)(=O)N1CCCN(CC1)c1ccc(cn1)C(F)(F)F)C(=O)C2 50412595CC1(C)[C@@H]2CC[C@]1(CS(=O)(=O)N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(=O)C2 50412596CC1(C)[C@@H]2CC[C@@]1(CS(=O)(=O)N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(F)C2 50412597CC1(O)C[C@H]2CC[C@]1(CS(=O)(=O)N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C2(C)C 50412598CC1(C)[C@H]2CC[C@]1(CS(=O)(=O)N1CCN(CC1)c1ccc(cn1)C(F)(F)F)CC2 50412599CC1(C)[C@@H]2CC[C@@]1(CS(=O)(=O)N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(O)C2 50412600CC1(C)[C@@H]2CC[C@@]1(CS(=O)(=O)N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C1(C2)OCCO1 50412601CC(=O)NC1C[C@H]2CC[C@]1(CS(=O)(=O)N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C2(C)C 50412602CCNC1C[C@H]2CC[C@]1(CS(=O)(=O)N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C2(C)C 50412603CC1(C)[C@@H]2CC[C@@]1(CS(=O)(=O)N1CCN(CC1)c1ccc(Br)cn1)C(=O)C2 50413567CC1(C)[C@@H]2CC[C@@]1(C)[C@@H](C2)NC1CCN(Cc2c(F)c(F)c(F)c(F)c2F)CC1 50413568Clc1ccc(CN2CCC(CC2)NC23CC4CC(CC(C4)C2)C3)cc1 50413569Fc1cc(Cl)ccc1CN1CCC(CC1)NCC1C2CC3CC(C2)CC1C3 50413570Fc1cc(Cl)ccc1CN1CCC(CC1)NCC12CC3CC(CC(C3)C1)C2 50413571CN(C1CCN(Cc2ccc(Cl)cc2F)CC1)C1C2CC3CC(C2)CC1C3 50413572CN(CC1C2CC3CC(C2)CC1C3)C1CCN(Cc2ccc(Cl)cc2F)CC1 50413573CC12CC3CC(C)(CC(C1)C3NC1CCN(Cc3ccc(Cl)cc3F)CC1)C2 50413574Fc1cc(Cl)ccc1CN1CCC(CC1)NC1C2CC3CC1CN(C3)C2 50413575CC(N1CCC(CC1)NC1C2CC3CC(C2)CC1C3)c1ccc(Cl)cc1F 50413576Fc1cc(Cl)ccc1CN1CCC(CNC2C3CC4CC(C3)CC2C4)CC1 50413577CCOC(=O)C1=C(CCN(Cc2ccc(Cl)cc2F)C1)NC1C2CC3CC(C2)CC1C3 50413578CCOC(=O)C1CN(Cc2ccc(Cl)cc2F)CCC1NC1C2CC3CC(C2)CC1C3 50413579Fc1cc(Cl)ccc1CNC1CCN(CC1)C1C2CC3CC(C2)CC1C3 50413580Fc1cc(Cl)ccc1CN1CCCC(C1)NC1C2CC3CC(C2)CC1C3 50413581Fc1cc(Cl)ccc1CN1CCCN(CC1)C1C2CC3CC(C2)CC1C3 50413583CC1(C)[C@@H]2CC[C@@]1(C)[C@@H](C2)NC1CCN(Cc2ccc(Cl)cc2F)CC1 50413584CC1(C)[C@@H]2CC[C@@]1(C)[C@@H](C2)NC1CCN(Cc2ccccc2)CC1 50413585CC1(C)[C@@H]2CC[C@@]1(C)[C@@H](C2)NC1CCN(Cc2ccccn2)CC1 50413587CC1(C)[C@@H]2CC[C@@]1(C)[C@@H](C2)NC1CCN(Cc2ccc(F)c(c2)C(F)(F)F)CC1 50413588CC1(C)[C@@H]2CC[C@@]1(C)[C@@H](C2)NC1CCN(Cc2cc(F)cc(c2)C(F)(F)F)CC1 50413589CC1(C)[C@@H]2CC[C@@]1(C)[C@@H](C2)NC1CCN(Cc2ccc(Cl)cc2)CC1 50413590COc1ccc(CN2CCC(CC2)N[C@@H]2C[C@H]3CC[C@]2(C)C3(C)C)c(F)c1 50413591COc1ccc(CN2CCC(CC2)N[C@@H]2C[C@H]3CC[C@]2(C)C3(C)C)cc1 50413593CC1(C)[C@@H]2CC[C@@]1(C)[C@@H](C2)NC1CCN(Cc2cccc(OC(F)(F)F)c2)CC1 50413595CC1(C)[C@@H]2CC[C@@]1(C)[C@@H](C2)NC1CCN(Cc2ccc(N)cc2)CC1 50413596CN(C)c1ccc(CN2CCC(CC2)N[C@@H]2C[C@H]3CC[C@]2(C)C3(C)C)cc1 50413597CC1(C)[C@@H]2CC[C@@]1(C)[C@H](C2)NC1CCN(Cc2ccc(Cl)cc2F)CC1 50413598CN([C@H]1C[C@H]2CC[C@]1(C)C2(C)C)C1CCN(Cc2ccc(Cl)cc2F)CC1 50413599CC1(C)C2CC[C@@]1(C)C(CNC1CCN(Cc3ccc(Cl)cc3F)CC1)C2 50413601Fc1cc(Cl)ccc1CN1CCC(CC1)N1CCc2ccccc2C1 50413603Fc1cc(Cl)ccc1CN1CCC(CC1)NC\C1=C\CCCCCC1 50413604Fc1cc(Cl)ccc1CN1CCC(CC1)NC1CCCCC1 50413605Fc1cc(Cl)ccc1CN1CCC(CC1)NCC1CCCCC1 50413606CC1(C)C2CC1C(CNC1CCN(Cc3ccc(Cl)cc3F)CC1)=CC2 50413608Fc1cc(Cl)ccc1CN1CCC(CC1)NC1C2CC3CC(C2)CC1C3 50413609Clc1ccc(CN2CCC(CC2)NC2C3CC4CC(C3)CC2C4)cc1 50413610C(N1CCC(CC1)NC1C2CC3CC(C2)CC1C3)c1ccccc1 50413611CC1(C)[C@@H]2CC[C@@]1(C)[C@@H](C2)NC1CCN(Cc2ccco2)CC1 50413612CC1(C)[C@@H]2CC[C@@]1(C)[C@@H](C2)NC1CCN(Cc2ccc(F)cc2F)CC1 50413613CC1(C)[C@@H]2CC[C@@]1(C)[C@@H](C2)NC1CCN(Cc2ccccc2F)CC1 50413614COc1cccc(CN2CCC(CC2)N[C@@H]2C[C@H]3CC[C@]2(C)C3(C)C)c1 50413615COC(=O)c1ccc(CN2CCC(CC2)N[C@@H]2C[C@H]3CC[C@]2(C)C3(C)C)cc1 50413616CC1(C)[C@@H]2CC[C@@]1(C)[C@@H](C2)NC1CCN(Cc2ccc(cc2)N=[N+]=[N-])CC1 50413617CN([C@@H]1C[C@H]2CC[C@]1(C)C2(C)C)C1CCN(Cc2ccc(Cl)cc2F)CC1 50446625CC[C@H]1CN([C@H](C)CN1C1CCN(CC1)C(=O)c1ccc(Cl)cc1)c1ncc(nc1C)-c1nnc[nH]1 50446626CC[C@H]1CN([C@H](C)CN1C1CCN(CC1)C(=O)c1ccc(Cl)cc1)c1ncc(nc1C)-c1ncc[nH]1 50446627CC[C@H]1CN([C@H](C)CN1C1CCN(CC1)C(=O)c1ccc(Cl)cc1)c1ncc(nc1C)-c1nnc(N)o1 50446628CC[C@H]1CN([C@H](C)CN1C1CCN(CC1)C(=O)c1ccc(Cl)cc1)c1ncc(nc1C)-c1nnc(NC)o1 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50446640CCNc1nnc(o1)-c1cnc(N2CCN([C@@H](CC)C2)C2CCN(CC2)C(=O)c2ccc(Cl)nc2N)c(Cl)n1 50446641CCNc1nnc(o1)-c1nc(Cl)c(nc1N)N1CCN([C@@H](CC)C1)C1CCN(CC1)C(=O)c1ccc(Cl)nc1N 50446642CC[C@H]1CN(CCN1C1CCN(CC1)C(=O)c1ccc(Cl)nc1N)c1nc(N)c(nc1Cl)-c1nnc(NC)o1 50446643CC[C@H]1CN(CCN1C1CCN(CC1)C(=O)c1ccc(Cl)nc1N)c1nc(N)c(nc1Cl)-c1nnc(NCCO)o1 50446644CC[C@H]1CN(CCN1C1CCN(CC1)C(=O)c1ccc(Cl)nc1N)c1nc(N)c(nc1Cl)-c1nnc(o1)N(C)C 50446645CC[C@H]1CN(CCN1C1CCN(CC1)C(=O)c1ccc(Cl)nc1N)c1nc(N)c(nc1Cl)-c1nnc(NS(C)(=O)=O)o1 50446646CC[C@H]1CN(CCN1C1CCN(CC1)C(=O)c1ccc(Cl)nc1N)c1nc(N)c(nc1Cl)-c1nnc(N)o1 50446647CC[C@H]1CN(CCN1C1CCN(CC1)C(=O)c1ccc(Cl)nc1N)c1nc(N)c(nc1Cl)-c1nnc(CO)o1 50446648CC[C@H]1CN(CCN1C1CCN(CC1)C(=O)c1ccc(Cl)nc1N)c1nc(N)c(nc1Cl)-c1nnc(o1)C1CC1 50446649CC[C@H]1CN(CCN1C1CCN(CC1)C(=O)c1ccc(Cl)nc1N)c1nc(N)c(nc1Cl)-c1nnc(C)o1 50446650CC[C@H]1CN(CCN1C1CCN(CC1)C(=O)c1ccc(Cl)cc1)c1nc(N)c(nc1Cl)-c1nnc(C)o1 50446651CC[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2)CC1)c1nc(N)c(nc1Cl)-c1nnc(C)o1 50446652CC[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2)CC1)c1nc(N)c(nc1Cl)-c1nnco1 50446653CC[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2F)CC1)c1ncc(cc1Cl)-c1nnco1 50446654CC[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2F)CC1)c1ncc(cc1Cl)-c1ncon1 50446655CC[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2F)CC1)c1ncc(cc1Cl)-c1nc(=O)o[nH]1 50446656CC[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2F)CC1)c1ncc(cc1Cl)-c1nnn[nH]1 50446657CC[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2F)CC1)c1ncc(cc1Cl)-c1nnc[nH]1 50446658CC[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2F)CC1)c1ncc(cc1Cl)C1=NCCN1 50446659CC[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2F)CC1)c1ncc(cc1Cl)-c1ncc[nH]1 50446660CC[C@H]1CN(CCN1C1CCN(Cc2ccc(Cl)cc2F)CC1)c1ncc(cc1Cl)C#N