4814CCN(CC)CCNC(=O)c1c(C)[nH]c(\C=C2/C(=O)Nc3ccc(F)cc23)c1C 5655CN1CC[C@@H]([C@H](O)C1)c1c(O)cc(O)c2c1oc(cc2=O)-c1ccccc1Cl 5718Cn1cnc2c(NCc3ccccc3)nc(NCCO)nc12 5931CC(C)(C)c1cnc(CSc2cnc(NC(=O)C3CCNCC3)s2)o1 6866Nc1nc(Nc2ccc(cc2)S(N)(=O)=O)nn1C(=O)c1c(F)cccc1F 6939COc1ccc(cc1)-c1n[nH]c2-c3cccc(NC(=O)NNC(=O)c4ccc(O)cc4)c3C(=O)c12 7108O=C(Cc1ccc2ccccc2c1)Nc1cc(n[nH]1)C1CC1 7238COc1ccc2NC(=O)C(=Cc3cnc[nH]3)c2c1 7262[O-][N+](=O)c1ccc2[nH]c-3c(CC(=O)Nc4ccccc-34)c2c1 7263O=C1Cc2c([nH]c3ccc(cc23)C#N)-c2ccccc2N1 7264COc1cc2NC(=O)Cc3c([nH]c4ccc(cc34)[N+]([O-])=O)-c2cc1OC 7265COc1cc2NC(=O)Cc3c([nH]c4ccc(cc34)C#N)-c2cc1OC 7266Brc1ccc2[nH]c-3c(CC(=O)Nc4ccccc-34)c2c1 7267Clc1ccc2[nH]c-3c(CC(=O)Nc4ccccc-34)c2c1 7268FC(F)(F)c1ccc2[nH]c-3c(CC(=O)Nc4ccccc-34)c2c1 7269FC(F)(F)c1ccc2[nH]c-3c(CC(=O)Nc4ccc(CCC#N)cc-34)c2c1 7270COc1cc2NC(=O)Cc3c([nH]c4ccc(cc34)C(F)(F)F)-c2cc1OC 7272Fc1ccc2[nH]c-3c(CC(=O)Nc4ccccc-34)c2c1 7273COc1cc2NC(=O)Cc3c([nH]c4ccc(Br)cc34)-c2cc1OC 7274Oc1cc2NC(=O)Cc3c([nH]c4ccc(Br)cc34)-c2cc1O 7275Cc1ccc2[nH]c-3c(CC(=O)Nc4ccccc-34)c2c1 7276Brc1ccc2c3CC(=O)Nc4ccccc4-c3[nH]c2c1 7277Brc1ccc2NC(=O)Cc3c([nH]c4ccccc34)-c2c1 7278Clc1cccc2c3CC(=O)Nc4ccccc4-c3[nH]c12 7279OCC#Cc1ccc2NC(=O)Cc3c([nH]c4ccc(cc34)C(F)(F)F)-c2c1 7280[O-][N+](=O)c1ccc2[nH]c-3c(CC(=O)Nc4ccc(Br)cc-34)c2c1 7281Ic1ccc2NC(=O)Cc3c([nH]c4ccccc34)-c2c1 7284FC(F)(F)c1ccc2[nH]c-3c(CC(=O)Nc4ccc(\C=C\C#N)cc-34)c2c1 7285COC(=O)CN1c2ccccc2-c2[nH]c3ccc(Br)cc3c2CC1=O 7286Cc1cccc2c3CC(=O)Nc4ccccc4-c3[nH]c12 7287O=C1Cc2c([nH]c3ccccc23)-c2ccccc2N1 7289ONC1=Nc2ccccc2-c2[nH]c3ccc(Br)cc3c2C1 7291Brc1cccc2c3CC(=O)Nc4ccccc4-c3[nH]c12 7292COc1cc2NC(=O)Cc3c([nH]c4ccccc34)-c2cc1OC 7297Brc1ccc2[nH]c-3c(CC(=S)Nc4ccccc-34)c2c1 7298FC(F)(F)c1ccc2[nH]c-3c(CC(=O)Nc4ccc(Br)cc-34)c2c1 7299OC1(CCCCC1)C#Cc1ccc2NC(=O)Cc3c([nH]c4ccc(cc34)C(F)(F)F)-c2c1 7301COc1ccc2[nH]c-3c(CC(=O)Nc4ccccc-34)c2c1 7302FC(F)(F)c1ccc2[nH]c-3c(CC(=O)Nc4ccc(I)cc-34)c2c1 7320COc1ccc2-c3[nH]c4ccc(cc4c3CC(=O)Nc2c1)C(F)(F)F 7322Oc1ccc2-c3[nH]c4ccc(Br)cc4c3CC(=O)Nc2c1 7323CC(=O)Nc1ccc2[nH]c-3c(CC(=O)Nc4ccccc-34)c2c1 7325CC(=O)Cc1ccc2NC(=O)Cc3c([nH]c4ccc(cc34)C(F)(F)F)-c2c1 7328COc1ccc2-c3[nH]c4ccc(cc4c3CC(=O)Nc2c1)C#N 7329COc1ccc2-c3[nH]c4ccc(cc4c3CC(=O)Nc2c1)[N+]([O-])=O 7330COc1ccc2NC(=O)Cc3c([nH]c4ccc(cc34)[N+]([O-])=O)-c2c1 7332O=C1Cc2c([nH]c3ncccc23)-c2ccccc2N1 7333[O-][N+](=O)c1ccc2[nH]c-3c(CC(=S)Nc4ccccc-34)c2c1 7336Brc1ccc2[nH]c-3c(CC(=O)Nc4ccsc-34)c2c1 7338Clc1ccc2[nH]c-3c(CC(=O)Nc4ccsc-34)c2c1 7339O=C1Cc2c([nH]c3ccc(cc23)C#N)-c2sccc2N1 7340[O-][N+](=O)c1ccc2[nH]c-3c(CC(=O)Nc4ccsc-34)c2c1 7341c1c([nH]c2nccnc12)-c1ccccc1 7343Oc1ccccc1-c1cc2nccnc2[nH]1 7346COc1ccc(cc1)-c1cc2nccnc2[nH]1 7347Oc1ccc(cc1)-c1cc2nccnc2[nH]1 7350Fc1ccc(cc1)-c1cc2nccnc2[nH]1 7358COc1ccc(cc1)-c1[nH]c2nccnc2c1C 7359COc1ccc(cc1OC)-c1[nH]c2nccnc2c1C 7360CCCc1c([nH]c2nccnc12)-c1ccc(OC)cc1 7361COc1ccc(cc1)-c1[nH]c2nccnc2c1CCCCl 7362COc1ccc(cc1)-c1[nH]c2nccnc2c1C(C)C 7363COc1ccc(cc1)-c1[nH]c2nccnc2c1CC=C 7364CCCCc1c([nH]c2nccnc12)-c1ccc(OC)cc1 7368CN(C)S(=O)(=O)Oc1ccc(cc1)-c1[nH]c2nccnc2c1C 7369Cc1c([nH]c2nccnc12)-c1ccc(Cl)cc1 7375Cc1c([nH]c2nccnc12)-c1ccc(O)cc1 7376CCCc1c([nH]c2nccnc12)-c1ccc(O)cc1 7377CCCCc1c([nH]c2nccnc12)-c1ccc(O)cc1 7379c1coc(c1)-c1cc2nccnc2[nH]1 7380c1csc(c1)-c1cc2nccnc2[nH]1 7381c1cc(cs1)-c1cc2nccnc2[nH]1 7389Cn1c(cc2nccnc12)-c1ccccc1 7393O=Nc1c([nH]c2ccccc12)C1C(=O)Nc2ccccc12 7394CC(=O)ON=C1C(Nc2ccccc12)=C1C(=O)Nc2ccccc12 7395CO\N=C1\C(\Nc2ccccc\12)=C1\C(=O)Nc2ccccc12 7397Brc1ccc2C(C(=O)Nc2c1)c1[nH]c2cc(Br)ccc2c1N=O 7399Brc1ccc2c(N=O)c([nH]c2c1)C1C(=O)Nc2ccccc12 7401Brc1ccc2C(C(=O)Nc2c1)c1[nH]c2ccccc2c1N=O 7402CC(=O)ON=C1C(Nc2ccccc12)=C1C(=O)Nc2cc(Br)ccc12 7403CO\N=C1\C(\Nc2ccccc\12)=C1\C(=O)Nc2cc(Br)ccc12 7407Clc1ccc2C(C(=O)Nc2c1)c1[nH]c2ccccc2c1N=O 7408CC(=O)ON=C1C(Nc2ccccc12)=C1C(=O)Nc2cc(Cl)ccc12 7409Ic1ccc2\C(C(=O)Nc2c1)=C1\Nc2ccccc2C1=O 7410Ic1ccc2C(C(=O)Nc2c1)c1[nH]c2ccccc2c1N=O 7411CC(=O)ON=C1C(Nc2ccccc12)=C1C(=O)Nc2cc(I)ccc12 7412C=Cc1ccc2\C(C(=O)Nc2c1)=C1\Nc2ccccc2C1=O 7413C=Cc1ccc2C(C(=O)Nc2c1)c1[nH]c2ccccc2c1N=O 7414CC(=O)ON=C1C(Nc2ccccc12)=C1C(=O)Nc2cc(C=C)ccc12 7415Fc1ccc2\C(C(=O)Nc2c1)=C1\Nc2ccccc2C1=O 7416Fc1ccc2C(C(=O)Nc2c1)c1[nH]c2ccccc2c1N=O 7417CC(=O)ON=C1C(Nc2ccccc12)=C1C(=O)Nc2cc(F)ccc12 7421Cc1cc2C(C(=O)Nc2cc1Br)c1[nH]c2ccccc2c1N=O 7424Clc1cc2NC(=O)C(c2cc1Cl)c1[nH]c2ccccc2c1N=O 7425CC(=O)ON=C1C(Nc2ccccc12)=C1C(=O)Nc2cc(Cl)c(Cl)cc12 7427[O-][N+](=O)c1cc2[c-](-c3[nH]c4ccccc4c3N=[OH+])c(=O)[nH]c2cc1Br 7454CCOc1cnc2oc3ccc(O)cc3c2c1-c1ccccc1 7457Oc1ccc2c(c1)oc(-c1ccc(O)c(O)c1)c(O)c2=O 7458Oc1ccc(cc1)-c1cc(=O)c2c(O)cc(O)cc2o1 7459Oc1cc(O)c2c(c1)oc(cc2=O)-c1ccc(O)c(O)c1 7461Oc1cc(O)c2c(c1)oc(cc2=O)-c1ccccc1 7478CC(C)[C@H](CO)Nc1nc(Nc2ccc(C(O)=O)c(Cl)c2)c2ncn(C(C)C)c2n1 7491NC1=NC(=O)C(N1)=C1CCNC(=O)c2[nH]c(Br)cc12 7492Ic1ccc2NC(=O)C(c2c1)c1[nH]c2ccccc2c1N=O 7497Brc1ccc2[nH]c-3c(CC(=O)Nc4cccnc-34)c2c1 7514CC(C)n1cnc2c(NCc3ccccc3)nc(nc12)N1CCC[C@H]1CO 7515CC(C)n1cnc2c(NCc3ccccc3)nc(nc12)N1CCC[C@@H]1CO 7516CC(C)n1cnc2c(NCc3ccccc3)nc(nc12)N(CCO)Cc1ccccc1 7517CC(C)n1cnc2c(NCc3ccccc3)nc(NCC(O)c3ccccc3)nc12 7518CCCCC(CO)Nc1nc(NCc2ccccc2)c2ncn(C(C)C)c2n1 7519CC(C)n1cnc2c(NCc3ccccc3)nc(N[C@H](CO)c3ccccc3)nc12 7520CC(C)n1cnc2c(NCc3ccccc3)nc(N[C@@H](CO)c3ccccc3)nc12 7521CC(C)n1cnc2c(NCc3ccccc3)nc(N[C@H](CO)Cc3ccccc3)nc12 7522CC(C)n1cnc2c(NCc3ccccc3)nc(N[C@@H](CO)Cc3ccccc3)nc12 7523CCCC(CO)Nc1nc(NCc2ccccc2)c2ncn(C(C)C)c2n1 7524C[C@H](CO)Nc1nc(NCc2ccccc2)c2ncn(C(C)C)c2n1 7526CC(C)n1cnc2c(NCc3cccc(I)c3)nc(nc12)N1CCC[C@@H]1CO 7527CC(C)n1cnc2c(NCc3ccccc3)nc(nc12)N1CCC(O)C1 7529OC[C@H]1CCCN1c1nc(NCc2ccccc2)c2ncn(C3CCCC3)c2n1 7533CC[C@H](CO)Nc1nc(NCc2ccccc2)c2ncn(C(C)C)c2n1 7555CCC(C)(O)C#Cc1nc(NCc2ccccc2)c2ncn(C(C)C)c2n1 7573CCC(C)(O)C#Cc1nc(NCc2ccc(OC)cc2)c2ncn(C(C)C)c2n1 7575CCC(C)(O)C#Cc1nc(NCc2ccc(Cl)c(Cl)c2)c2ncn(C(C)C)c2n1 7576CCC(C)(O)C#Cc1nc(NCc2ccc(Cl)cc2)c2ncn(C(C)C)c2n1 7577CCC(C)(O)C#Cc1nc(NCc2ccc3OCOc3c2)c2ncn(C(C)C)c2n1 7578CCC(C)(O)C#Cc1nc(NCc2ccc(OC)c(OC)c2)c2ncn(C(C)C)c2n1 7579CCC(C)(O)C#Cc1nc(NCc2ccc(cc2)N(C)C)c2ncn(C(C)C)c2n1 7580CCC(C)(O)C#Cc1nc(Nc2ccccc2)c2ncn(C(C)C)c2n1 7581CCC(C)(O)C#Cc1nc(Nc2ccc(OC)cc2)c2ncn(C(C)C)c2n1 7582CCOc1ccc(Nc2nc(nc3n(cnc23)C(C)C)C#CC(C)(O)CC)cc1 7583CCC(C)(O)C#Cc1nc(Nc2ccc(Cl)c(Cl)c2)c2ncn(C(C)C)c2n1 7584CCC(C)(O)C#Cc1nc(Nc2cccc(Cl)c2)c2ncn(C(C)C)c2n1 7585CCC(CO)Nc1nc(NCc2ccccc2)c2ncn(C(C)C)c2n1 10643COCCNc1nc(nc2n(cnc12)C(C)C)-c1ccc(C=O)cc1 10644COCCNc1nc(nc2n(cnc12)C(C)C)-c1ccc(cc1)C(C)=O 10645COCCNc1nc(nc2n(cnc12)C(C)C)-c1ccc(NS(C)(=O)=O)cc1 10646CNC(=O)c1ccc(cc1)-c1nc(NCCOC)c2ncn(C(C)C)c2n1 10647COCCNc1nc(nc2n(cnc12)C(C)C)-c1ccc(cc1)C(=O)NCCC#N 10648COCCNc1nc(nc2n(cnc12)C(C)C)-c1ccc(NC(=O)OC)cc1 10649COCCNc1nc(nc2n(cnc12)C(C)C)-c1ccc(s1)C(C)=O 10650COCCNc1nc(nc2n(cnc12)C(C)C)-c1ccc(s1)C#N 10651COc1ccc(CNc2nc(nc3n(cnc23)C(C)C)-c2ccc(C=O)cc2)cc1 10838Nc1nccc(n1)-c1c[nH]c2cccc(O)c12 10839Nc1nccc(n1)-c1c[nH]c2cc(Br)cc(O)c12 10840Nc1nccc(n1)-c1c[nH]c2ccc(Br)cc12 10841Nc1nccc(n1)-c1c[nH]c2cc(Br)ccc12 10842Nc1nccc(n1)-c1c[nH]c2c(Br)ccc(O)c12 10844Nc1nccc(n1)-c1c[nH]c2ccccc12 12097CCCCNC(=O)N1Cc2n[nH]c(NC(=O)Cc3ccc(cc3)N3CCCC3)c2C1 12100CCCCNC(=O)N1Cc2n[nH]c(NC(=O)[C@@H](C)c3ccc4ccccc4c3)c2C1 12621COc1ccc(F)c(F)c1C(=O)c1cnc(NC2CCN(CC2)S(C)(=O)=O)nc1N 16673CNC(=O)c1cc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(c3)C(F)(F)F)cc2)ccn1 20816O=C(Nc1csc(n1)-c1ccncc1)Nc1ccccc1 20818O=c1[nH]c2ccccc2n1-c1csc(n1)-c1ccncc1 20819O=C1Nc2ccccc2CN1c1csc(n1)-c1ccncc1 20820O=C1Nc2ccccc2CN1c1nc(cs1)-c1ccncc1 20822O=C1Nc2ccccc2CN1c1nc(ns1)-c1ccncc1 20825Fc1cccc2NC(=O)N(Cc12)c1csc(n1)-c1ccncc1 20826Clc1cccc2NC(=O)N(Cc12)c1csc(n1)-c1ccncc1 20827Brc1cccc2NC(=O)N(Cc12)c1csc(n1)-c1ccncc1 20828Cc1cccc2NC(=O)N(Cc12)c1csc(n1)-c1ccncc1 20829COc1cccc2NC(=O)N(Cc12)c1csc(n1)-c1ccncc1 20830Fc1ccc2NC(=O)N(Cc2c1)c1csc(n1)-c1ccncc1 20831Cc1ccc2NC(=O)N(Cc2c1)c1csc(n1)-c1ccncc1 20832Fc1ccc2CN(c3csc(n3)-c3ccncc3)C(=O)Nc2c1 20833Brc1ccc2CN(c3csc(n3)-c3ccncc3)C(=O)Nc2c1 20834O=C1Nc2cc(ccc2CN1c1csc(n1)-c1ccncc1)-c1ccccc1 20835CN1CCN(CC1)c1cccc2NC(=O)N(Cc12)c1csc(n1)-c1ccncc1 20836CN1CCN(CC1)c1ccc2NC(=O)N(Cc2c1)c1csc(n1)-c1ccncc1 20837O=C1Nc2cccc(CN3CCOCC3)c2CN1c1csc(n1)-c1ccncc1 20838O=C1Nc2cc(CN3CCOCC3)ccc2CN1c1csc(n1)-c1ccncc1 20839O=C1Nc2ccccc2CN1c1nc(cs1)-c1cccnc1 20840O=C1Nc2ccccc2CN1c1nc(cs1)-c1ccccn1 20841CCc1cc(ccn1)-c1nc(cs1)N1Cc2ccccc2NC1=O 20842O=c1[nH]c2ccccc2cc1-c1csc(n1)-c1ccncc1 20843COC(=O)c1cccc2[nH]c(=O)c(cc12)-c1csc(n1)-c1ccncc1 20845CCN(CC)C(=O)c1cccc2[nH]c(=O)c(cc12)-c1csc(n1)-c1ccncc1 20846Fc1ccc2[nH]c(=O)c(cc2c1)-c1csc(n1)-c1ccncc1 20847Clc1ccc2[nH]c(=O)c(cc2c1)-c1csc(n1)-c1ccncc1 20848FC(F)(F)c1ccc2cc(-c3csc(n3)-c3ccncc3)c(=O)[nH]c2c1 20849CCN(CCN(C)C)C(=O)c1ccc2cc(-c3csc(n3)-c3ccncc3)c(=O)[nH]c2c1 20850CN1CCN(CC1)C(=O)c1ccc2cc(-c3csc(n3)-c3ccncc3)c(=O)[nH]c2c1 20851O=C(N1CCCCC1)c1ccc2cc(-c3csc(n3)-c3ccncc3)c(=O)[nH]c2c1 20852Oc1c(-c2csc(n2)-c2ccncc2)c(=O)[nH]c2ccccc12 20853O=c1[nH]c2ccccc2c(-c2ccccc2)c1-c1csc(n1)-c1ccncc1 20854Cc1c(-c2csc(n2)-c2ccncc2)c(=O)[nH]c2ccccc12 20855Nc1c(-c2csc(n2)-c2ccncc2)c(=O)[nH]c2ccccc12 20856Nc1c(-c2csc(n2)-c2ccncc2)c(=O)[nH]c2ccc(Cl)cc12 20857Nc1c(-c2csc(n2)-c2ccncc2)c(=O)[nH]c2ccc(cc12)N1CCCCC1 20858CN1CCN(CC1)c1ccc2[nH]c(=O)c(-c3csc(n3)-c3ccncc3)c(N)c2c1 20859O=c1[nH]c2ccccc2cc1-c1csc(n1)-c1ccccc1 20860O=c1[nH]c2ccccc2cc1-c1csc(n1)-c1ccsc1 20861O=c1[nH]c2ccccc2cc1-c1csc(n1)-c1cccnc1 20865Nc1ccc(cc1)-c1nc(cs1)-c1cc2ccccc2[nH]c1=O 20866Oc1ccc(cc1)-c1nc(cs1)-c1cc2ccccc2[nH]c1=O 20868O=c1[nH]c2ccccc2cc1-c1csc(CS(=O)(=O)c2ccccc2)n1 20869O=c1[nH]c2ccccc2cc1-c1csc(CS(=O)(=O)c2ccccn2)n1 20870O=c1[nH]c2ccccc2cc1-c1csc(CS(=O)(=O)c2cccs2)n1 20871Clc1ccc(cc1)S(=O)(=O)Cc1nc(cs1)-c1cc2ccccc2[nH]c1=O 20872CS(=O)(=O)Cc1nc(cs1)-c1cc2ccccc2[nH]c1=O 20873CC(C)(C)S(=O)(=O)Cc1nc(cs1)-c1cc2ccccc2[nH]c1=O 20874O=S(Cc1nc(cs1)-c1cc2ccccc2[nH]c1=O)c1ccccc1 24654Clc1cccc(Cl)c1C(=O)Nc1cn[nH]c1C(=O)NC1CCNCC1 27216CC(C)[C@H](CO)Nc1nc(Nc2cccc(Cl)c2)c2ncn(C(C)C)c2n1 27217CC[C@H](CO)Nc1nc(NCc2ccccc2)n2ncc(C(C)C)c2n1 27218CC(C)[C@H](CO)Nc1nc(Nc2cccc(Cl)c2)n2ncc(C(C)C)c2n1 27219CC[C@H](CO)Nc1nc(NCc2ccccc2)c2ncc(C(C)C)n2n1 27220CC[C@@H](CO)Nc1nc(NCc2ccccc2)n2ncc(C(C)C)c2n1 27344O=C1NCCc2[nH]c(cc12)-c1ccncc1 31085CCN1CCN(Cc2ccc(NC(=O)Nc3ccc(Oc4cc(NC)ncn4)cc3)cc2C(F)(F)F)CC1 31545CNC(=O)c1nn(C)c-2c1C(C)(C)Cc1cnc(Nc3ccc(cc3)N3CCN(C)CC3)nc-21 41575COc1ccc(cc1Nc1ncc2CCc3c(nn(C)c3-c2n1)C(N)=O)N1CCN(C)CC1 59194Nc1nc(Nc2ccc(Cl)cc2)sc1C(=O)c1cccc(c1)N(=O)=O 59195Nc1nc(Nc2ccc(Cl)cc2)sc1C(=O)c1ccc(Cl)cc1Cl 59200CC(=O)Nc1ccc(CN2CCC(CC2)N2Cc3cc(Cl)c4cccnc4c3O2)cc1 59201Clc1cc2CN(Oc2c2ncccc12)C1CCN(Cc2ccc(cc2)-c2ccccc2)CC1 59227CC(C)c1nn(-c2c(Cl)cccc2Cl)c2nc(Cc3ccc(OCCO)cc3)[nH]c(=O)c12 84528O=C1Cc2c([nH]c3ccc(cc23)N(=O)=O)-c2ccccc2N1 84529NCCCCc1ccc2NC(=O)Cc3c([nH]c4ccc(cc34)N(=O)=O)-c2c1 84530NCCCc1ccc2NC(=O)Cc3c([nH]c4ccc(cc34)N(=O)=O)-c2c1 84531OC(=O)CCc1ccc2NC(=O)Cc3c([nH]c4ccc(cc34)N(=O)=O)-c2c1 84532COC(=O)CCc1ccc2NC(=O)Cc3c([nH]c4ccc(cc34)N(=O)=O)-c2c1 84533O=C1Cc2c([nH]c3ccc(cc23)N(=O)=O)-c2cc(CCC#N)ccc2N1 100152COc1ccc2c(c1)[nH]c1c(C)nccc21 124970Cc1nc(Nc2nc3ccc(nc3s2)-c2cccc(c2)C(=O)Nc2cccc(c2)C(F)(F)F)cc(n1)N1CCNCC1 50012188O\N=C1\C(\Nc2ccccc\12)=C1\C(=O)Nc2cc(Br)ccc12 50021604OC1CNC(=O)c2c(I)c3ccccc3n2C1 50021605COc1cccc2n3CC(O)CNC(=O)c3c(I)c12 50021607COc1ccc2c(I)c3C(=O)NCC(O)Cn3c2c1 50021609OC1CNC(=O)c2c(Br)c3ccccc3n2C1 50021611COc1ccc2c(Br)c3C(=O)NCC(O)Cn3c2c1 50021612OC1CNC(=O)c2c(I)c3ccc(O)cc3n2C1 50021616COc1c(O)ccc2c1[nH]c1c3C=CC(C)(C)Oc3cc(O)c1c2=O 50059889CN[C@@H]1CC2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13 50077360COc1ccc(cc1O)-c1c2c(n3ccc4cc(O)c(OC)cc4c13)c(=O)oc1cc(O)c(OC)cc21 50093389CCCCNc1nc(nc2n(cnc12)C(C)C)C#CC(C)(O)Cc1ccccc1 50093390CC(C)n1cnc2c(NCc3cccc(I)c3)nc(nc12)N1CCCC1CO 50093411OCC1CCCN1c1nc(NCc2ccccc2)c2ncn(C3CCCC3)c2n1 50111434Cc1[nH]cnc1-c1[nH]ccc2c3ccccc3nc12 50132003Oc1[nH]c2ccccc2c1-c1[nH]c2ccccc2c1N=O 50133549CONC(=O)Nc1csc(Cc2c(Cl)cccc2Cl)n1 50133551CN(C)NC(=O)Nc1csc(Cc2c(Cl)cccc2Cl)n1 50133555Clc1cccc(Cl)c1Cc1nc(NC(=O)NN2CCCCC2)cs1 50133556O=C(NN1CCOCC1)Nc1csc(n1)-c1ccccc1 50133557Clc1cccc(Cl)c1Cc1nc(NC(=O)NN2CCOCC2)cs1 50133564Clc1cccc(Cl)c1Cc1nc(NC(=O)NN2CCCC2)cs1 50133566CS(=O)(=O)Cc1nc(NC(=O)NOc2ccccc2)cs1 50133567Clc1cccc(Cl)c1Cc1nc(NC(=O)NOCC=C)cs1 50133573Clc1cccc(Cl)c1Cc1nc(NC(=O)NOc2ccccc2)cs1 50133575Clc1cccc(Cl)c1Cc1nc(NC(=O)NOC2CCCCO2)cs1 50133576O=C(NOc1ccccc1)Nc1csc(n1)-c1ccccc1 50133579CC(C)(C)ONC(=O)Nc1csc(Cc2c(Cl)cccc2Cl)n1 50133580CCONC(=O)Nc1csc(Cc2c(Cl)cccc2Cl)n1 50134580O=C1NC(=O)c2c1c1c3ccccc3[nH]c1c1ccccc21 50148063COc1ccc2N=C(C(=O)c2c1)c1c(O)[nH]c2ccccc12 50148066Cc1ccc2N=C(C(=O)c2c1)c1c(O)[nH]c2ccccc12 50148067COc1ccc2[nH]c(O)c(C3=Nc4ccccc4C3=O)c2c1 50148068COc1ccc2N=C(C(=O)c2c1)c1c(O)[nH]c2ccc(OC)cc12 50148069Cc1ccc2[nH]c(O)c(C3=Nc4ccccc4C3=O)c2c1 50155206O=C(Cc1ccccc1)Nc1ncc(s1)C1CCCC1 50155207O=C(Nc1ncc(s1)C1CCC1)Nc1cccc2ncccc12 50155208CC(C)c1cnc(NC(=O)Oc2ccccc2)s1 50155209O=C(Nc1ncc(s1)C1CCC1)Nc1cccc2cnccc12 50155210CC(C)c1cnc(NC(=O)Cc2ccccc2)s1 50155211O=C(Nc1ncc(s1)C1CCC1)Nc1ccccc1 50155212CC(C)C(=O)Nc1ncc(s1)C(C)C 50155213O=C(Nc1ncc(s1)C1CCC1)Nc1cccc2ccncc12 50155214O=C(Cc1c[nH]c2ccccc12)Nc1ncc(s1)C1CCC1 50155215CCCCCc1cnc(NC(=O)Cc2ccccc2)s1 50155216CSc1cnc(NC(=O)Cc2ccccc2)s1 50155217O=C(Cc1ccccc1)Nc1ncc(s1)-c1ccccc1 50155218CN(C)c1cnc(NC(=O)Cc2ccccc2)s1 50155219CC(C)c1cnc(NC(=O)C(=O)c2ccccc2)s1 50155220O=C(Cn1ccc2ccccc12)Nc1ncc(s1)C1CCC1 50155221O=C(Nc1ncc(s1)C1CCC1)Nc1ccc2ncccc2c1 50155222O=C(Nc1ncc(s1)C1CCC1)Nc1ccc2cnccc2c1 50155223O=C(Nc1ncc(s1)C1CCC1)Nc1cccc2c[nH]nc12 50155224CC(=O)c1cnc(NC(=O)Cc2ccccc2)s1 50155225O=C(Cc1ccccc1)Nc1ncc(s1)C1CCC1 50155226CCc1cnc(NC(=O)Cc2ccccc2)s1 50155227Brc1cnc(NC(=O)Cc2ccccc2)s1 50155228O=C(Cc1ccccc1)Nc1ncc(s1)C1CCCCC1 50155229O=C(Cc1ccccc1)Nc1ncc(s1)C1=CCCC1 50155230Cc1cc2ncn(CC(=O)Nc3ncc(s3)C3CCC3)c2cc1C 50155231O=C(Cc1ccc2nc[nH]c2c1)Nc1ncc(s1)C1CCC1 50155232O=C(Nc1ncc(s1)C1CCC1)Nc1cccc2nn[nH]c12 50155233CC(C)c1cnc(NC(=O)c2ccccc2)s1 50155234CC(C)c1cnc(NC(=O)Nc2ccccc2)s1 50155235Cc1nc2ccc(CC(=O)Nc3ncc(s3)C3CCC3)cc2s1 50155236O=C(Cc1ccc2ncccc2c1)Nc1ncc(s1)C1CCC1 50155237O=C(Cc1cccc2cnccc12)Nc1ncc(s1)C1CCC1 50155420COc1cc(O)c2c(c1)oc1c(O)ccc(O)c1c2=O 50155426Oc1cc(O)c2c(c1)oc1c(O)ccc(O)c1c2=O 50169892OCCCNc1cc(ccn1)-c1ncnc(Nc2cccc(Cl)c2)n1 50180964Oc1ccc2[nH]c3c(c4C(=O)NC(=O)c4c4ccccc34)c2c1 50186073CC(C)n1cnc2ccc3nc(sc3c2c1=O)C(=N)NCCN(C)C 50186373C1CCC(CC1)Oc1nccc(n1)-c1cnc(Nc2ccccn2)s1 50186375CN1CCN(Cc2cnc(Nc3ncc(s3)-c3cc(C)nc(OC4CCCCC4)n3)cn2)CC1 50191394CC(=O)ON=C1C(=Nc2ccccc12)c1c(O)[nH]c2ccccc12 50191418Oc1[nH]c2c(Cl)cccc2c1-c1[nH]c2ccccc2c1N=O 50191421CO\N=C1/C(=Nc2ccccc12)c1c(O)[nH]c2ccccc12 50191431Oc1[nH]c2ccc(Br)cc2c1-c1[nH]c2ccccc2c1N=O 50191448Oc1[nH]c2c(F)cccc2c1-c1[nH]c2ccccc2c1N=O 50197305CC(C)C(=O)Nc1nc(NCc2ccc(Cl)cc2)c2ncn(C(C)C)c2n1 50197307COc1ccc(CNc2nc(nc3n(cnc23)C(C)C)C(=O)NCC(C)C)cc1 50197308CC(C)NC(=O)c1nc(NCc2ccc(Cl)cc2)c2ncn(C(C)C)c2n1 50197310CCCC(=O)Nc1nc(NCc2ccc(OC)cc2)c2ncn(C(C)C)c2n1 50197311COCCNc1nc(NC(=O)C(C)C)nc2n(cnc12)C(C)C 50197312CC(C)CC(=O)Nc1nc(NCc2ccc(Cl)cc2)c2ncn(C(C)C)c2n1 50197314COCCNc1nc(NC(=O)CC(C)C)nc2n(cnc12)C(C)C 50197316COc1ccc(CNc2nc(NC(=O)CC(C)=O)nc3n(cnc23)C(C)C)cc1 50197317COc1ccc(CNc2nc(NC(=O)C(C)C)nc3n(cnc23)C(C)C)cc1 50197318COc1ccc(CNc2nc(nc3n(cnc23)C(C)C)C(=O)NC(C)C)cc1 50197319COc1ccc(CNc2nc(NC(=O)CC(C)C)nc3n(cnc23)C(C)C)cc1 50197321COc1ccc(CNc2nc(NC(=O)c3ccc(OC)cc3)nc3n(cnc23)C(C)C)cc1 50197322CCCC(=O)Nc1nc(NCc2ccc(Cl)cc2)c2ncn(C(C)C)c2n1 50204948CC(=O)NNC(=O)CSc1nnc(Cc2csc(NC(=O)CCl)n2)n1NC(=O)c1ccccc1 50204949CC(=O)Nn1c(Cc2csc(NC(=O)CCl)n2)nnc1SCC(=O)NN=Cc1ccccc1 50204950CC(=O)Nc1nc(Cc2nnc(SCC(=O)NN=Cc3ccccc3)n2NC(=O)c2ccccc2)cs1 50204951ClCC(=O)Nc1nc(Cc2nnc(SCSc3nnc(Cc4csc(NC(=O)CCl)n4)n3NC(=O)c3ccccc3)n2NC(=O)c2ccccc2)cs1 50204952CC(=O)NNC(=O)CSc1nnc(Cc2csc(NC(=O)c3ccccc3)n2)n1NC(C)=O 50204953CC(=O)Nc1nc(Cc2nnc(SCC#N)n2NC(C)=O)cs1 50204954CC(=O)Nn1c(Cc2csc(NCCC(O)=O)n2)n[nH]c1=S 50204955COC(=O)CSc1nnc(Cc2csc(NC(=O)c3ccccc3)n2)n1NC(=O)c1ccccc1 50204956O=C(CSc1nnc(Cc2csc(NC(=O)c3ccccc3)n2)n1NC(=O)c1ccccc1)NN=Cc1ccccc1 50204957CC(=O)Nc1nc(Cc2nnc(SCC(=O)NN)n2NC(=O)c2ccc(Cl)cc2)cs1 50204958CC(=O)Nn1c(Cc2csc(NC(=O)CCl)n2)nnc1SCC(=O)NNC(=O)c1ccccc1 50204959CC(=O)Nc1nc(Cc2n[nH]c(=S)n2N)cs1 50204960CC(=O)Nn1c(Cc2csc(NCCC(O)=O)n2)nnc1SCC(=O)NN=Cc1ccccc1 50204961OC(=O)CCNc1nc(Cc2n[nH]c(=S)n2NC(=O)c2ccccc2)cs1 50204962CC(=O)Nn1c(Cc2csc(NCCC(O)=O)n2)nnc1SCC(=O)NNC(=O)c1ccccc1 50204963CC(=O)Nc1nc(Cc2nnc(SCC(=O)NNC(=O)c3ccccc3)n2NC(=O)c2ccc(Cl)cc2)cs1 50204964CC(=O)Nc1nc(Cc2nnc(SCC(=O)NNC(=O)c3ccccc3)n2NC(C)=O)cs1 50204965COC(=O)CSc1nnc(Cc2csc(NC(C)=O)n2)n1NC(C)=O 50204966CC(=O)Nc1nc(Cc2nnc(SCC(=O)NNC(=O)CCl)n2NC(C)=O)cs1 50204967CC(=O)Nc1nc(Cc2nnc(SCc3n[nH]c(=S)n3N)n2NC(=O)c2ccccc2)cs1 50204968ClCC(=O)NNC(=O)CSc1nnc(Cc2csc(NC(=O)c3ccccc3)n2)n1NC(=O)c1ccc(Cl)cc1 50204969NNC(=O)CSc1nnc(Cc2csc(NC(=O)c3ccccc3)n2)n1NC(=O)c1ccc(Cl)cc1 50204970CC(=O)Nn1c(Cc2csc(NC(=O)c3ccccc3)n2)nnc1SCC#N 50204971CC(=O)Nn1c(Cc2csc(NC(=O)CCl)n2)nnc1SCC#N 50204972NNC(=O)CSc1nnc(Cc2csc(NC(=O)c3ccccc3)n2)n1NC(=O)c1ccccc1 50204973NNC(=O)CSc1nnc(Cc2csc(NC(=O)CCl)n2)n1NC(=O)c1ccc(Cl)cc1 50204974OC(=O)CCNc1nc(Cc2nnc(SCC(=O)NNC(=O)c3ccccc3)n2NC(=O)c2ccc(Cl)cc2)cs1 50204975Nn1c(CSc2nnc(Cc3csc(NC(=O)c4ccccc4)n3)n2NC(=O)c2ccccc2)n[nH]c1=S 50204976Nn1c(CSc2nnc(Cc3csc(NC(=O)CCl)n3)n2NC(=O)c2ccc(Cl)cc2)n[nH]c1=S 50204977CC(=O)Nc1nc(Cc2nnc(SCC(=O)NNC(=O)c3ccccc3)n2NC(=O)c2ccccc2)cs1 50204978CC(=O)NNC(=O)CSc1nnc(Cc2csc(NC(C)=O)n2)n1NC(=O)c1ccccc1 50204979COC(=O)CSc1nnc(Cc2csc(NC(C)=O)n2)n1NC(=O)c1ccccc1 50204980CC(=O)Nc1nc(Cc2nnc(SCC(=O)NN=Cc3ccccc3)n2NC(=O)c2ccc(Cl)cc2)cs1 50204981OC(=O)CCNc1nc(Cc2nnc(SCC#N)n2NC(=O)c2ccc(Cl)cc2)cs1 50204982CC(=O)Nn1c(Cc2csc(NC(=O)c3ccccc3)n2)n[nH]c1=S 50204983NNC(=O)CSc1nnc(Cc2csc(NCCC(O)=O)n2)n1NC(=O)c1ccccc1 50204984CC(=O)NNC(=O)CSc1nnc(Cc2csc(NCCC(O)=O)n2)n1NC(=O)c1ccccc1 50204985CC(=O)Nc1nc(Cc2nnc(SCc3n[nH]c(=S)n3N)n2NC(=O)c2ccc(Cl)cc2)cs1 50204986COC(=O)CSc1nnc(Cc2csc(NCCC(O)=O)n2)n1NC(=O)c1ccc(Cl)cc1 50204987ClCC(=O)NNC(=O)CSc1nnc(Cc2csc(NC(=O)CCl)n2)n1NC(=O)c1ccccc1 50204988COC(=O)CSc1nnc(Cc2csc(NC(=O)CCl)n2)n1NC(C)=O 50204989CC(=O)Nn1c(Cc2csc(NC(=O)c3ccccc3)n2)nnc1SCC(=O)NN=Cc1ccccc1 50204990CC(=O)Nn1c(Cc2csc(NC(=O)CCl)n2)n[nH]c1=S 50204991ClCC(=O)Nc1nc(Cc2nnc(SCC(=O)NNC(=O)c3ccccc3)n2NC(=O)c2ccccc2)cs1 50204992ClCC(=O)Nc1nc(Cc2nnc(SCC#N)n2NC(=O)c2ccc(Cl)cc2)cs1 50204993Nn1c(Cc2csc(NC(=O)c3ccccc3)n2)n[nH]c1=S 50204994ClCC(=O)Nc1nc(Cc2nnc(SCC(=O)NNC(=O)c3ccccc3)n2NC(=O)c2ccc(Cl)cc2)cs1 50204995NNC(=O)CSc1nnc(Cc2csc(NC(=O)CCl)n2)n1NC(=O)c1ccccc1 50204996CC(=O)Nn1c(Cc2csc(NCCC(O)=O)n2)nnc1SCC(=O)NNC(=O)CCl 50204997CC(=O)Nc1nc(Cc2n[nH]c(=S)n2NC(C)=O)cs1 50204998CC(=O)Nc1nc(Cc2nnc(SCC(=O)NNC(=O)CCl)n2NC(=O)c2ccc(Cl)cc2)cs1 50204999ClCC(=O)NNC(=O)CSc1nnc(Cc2csc(NC(=O)CCl)n2)n1NC(=O)c1ccc(Cl)cc1 50205000CC(=O)Nn1c(Cc2csc(NCCC(O)=O)n2)nnc1SCc1n[nH]c(=S)n1N 50205001ClCC(=O)Nc1nc(Cc2nnc(SCC(=O)NN=Cc3ccccc3)n2NC(=O)c2ccccc2)cs1 50205002CC(=O)Nc1nc(Cc2nnc(SCC#N)n2NC(=O)c2ccc(Cl)cc2)cs1 50205003CC(=O)Nc1nc(Cc2nnc(SCC#N)n2NC(=O)c2ccccc2)cs1 50205004OC(=O)CCNc1nc(Cc2nnc(SCC(=O)NNC(=O)c3ccccc3)n2NC(=O)c2ccccc2)cs1 50205005O=C(CSc1nnc(Cc2csc(NC(=O)c3ccccc3)n2)n1NC(=O)c1ccccc1)NNC(=O)c1ccccc1 50205006CC(=O)Nn1c(Cc2csc(NC(=O)c3ccccc3)n2)nnc1SCC(=O)NNC(=O)CCl 50205007CC(=O)NNC(=O)CSc1nnc(Cc2csc(NC(C)=O)n2)n1NC(C)=O 50205008CC(=O)Nc1nc(Cc2nnc(SCSc3nnc(Cc4csc(NC(C)=O)n4)n3NC(=O)c3ccc(Cl)cc3)n2NC(=O)c2ccc(Cl)cc2)cs1 50205009Clc1ccc(cc1)C(=O)Nn1c(Cc2csc(NC(=O)c3ccccc3)n2)n[nH]c1=S 50205010CC(=O)NNC(=O)CSc1nnc(Cc2csc(NC(=O)c3ccccc3)n2)n1NC(=O)c1ccccc1 50205011Nn1c(CSc2nnc(Cc3csc(NCCC(O)=O)n3)n2NC(=O)c2ccccc2)n[nH]c1=S 50205012ClCC(=O)Nc1nc(Cc2nnc(SCC(=O)NN=Cc3ccccc3)n2NC(=O)c2ccc(Cl)cc2)cs1 50205013CC(=O)Nn1c(Cc2csc(NC(=O)c3ccccc3)n2)nnc1SCC(=O)NNC(=O)c1ccccc1 50205014OC(=O)CCNc1nc(Cc2nnc(SCC(=O)NN=Cc3ccccc3)n2NC(=O)c2ccccc2)cs1 50205015O=C(Nc1nc(Cc2n[nH]c(=S)n2NC(=O)c2ccccc2)cs1)c1ccccc1 50205016CC(=O)Nn1c(Cc2csc(NC(=O)c3ccccc3)n2)nnc1SCC(=O)NN 50205017ClCC(=O)Nc1nc(Cc2nnc(SCSc3nnc(Cc4csc(NC(=O)CCl)n4)n3NC(=O)c3ccc(Cl)cc3)n2NC(=O)c2ccc(Cl)cc2)cs1 50205018CC(=O)NNC(=O)CSc1nnc(Cc2csc(NC(=O)c3ccccc3)n2)n1NC(=O)c1ccc(Cl)cc1 50205019CC(=O)Nc1nc(Cc2nnc(SCc3n[nH]c(=S)n3N)n2NC(C)=O)cs1 50205020CC(=O)Nn1c(Cc2csc(NC(=O)CCl)n2)nnc1SCSc1nnc(Cc2csc(NC(=O)CCl)n2)n1NC(C)=O 50205021Clc1ccc(cc1)C(=O)Nn1c(Cc2csc(NC(=O)c3ccccc3)n2)nnc1SCC#N 50205022OC(=O)CCNc1nc(Cc2nnc(SCSc3nnc(Cc4csc(NC(=O)CCC(O)=O)n4)n3NC(=O)c3ccccc3)n2NC(=O)c2ccccc2)cs1 50205023OC(=O)CCNc1nc(Cc2nnc(SCSc3nnc(Cc4csc(NCCC(O)=O)n4)n3NC(=O)c3ccc(Cl)cc3)n2NC(=O)c2ccc(Cl)cc2)cs1 50205024ClCC(=O)Nc1nc(Cc2n[nH]c(=S)n2NC(=O)c2ccc(Cl)cc2)cs1 50205025Nn1c(CSc2nnc(Cc3csc(NC(=O)c4ccccc4)n3)n2NC(=O)c2ccc(Cl)cc2)n[nH]c1=S 50205026CC(=O)Nc1nc(Cc2nnc(SCC(=O)NN=Cc3ccccc3)n2NC(C)=O)cs1 50205027CC(=O)NNC(=O)CSc1nnc(Cc2csc(NC(=O)CCl)n2)n1NC(C)=O 50205028CC(=O)Nn1c(Cc2csc(NC(=O)c3ccccc3)n2)nnc1SCSc1nnc(Cc2csc(NC(=O)c3ccccc3)n2)n1NC(C)=O 50205029OC(=O)CCNc1nc(Cc2nnc(SCC#N)n2NC(=O)c2ccccc2)cs1 50205030CC(=O)Nc1nc(Cc2n[nH]c(=S)n2NC(=O)c2ccccc2)cs1 50205031COC(=O)CSc1nnc(Cc2csc(NCCC(O)=O)n2)n1NC(C)=O 50205032ClCC(=O)Nc1nc(Cc2nnc(SCC#N)n2NC(=O)c2ccccc2)cs1 50205033CC(=O)Nc1nc(Cc2nnc(SCC(=O)NN)n2NC(C)=O)cs1 50205034CC(=O)Nc1nc(Cc2nnc(SCSc3nnc(Cc4csc(NC(C)=O)n4)n3NC(=O)c3ccccc3)n2NC(=O)c2ccccc2)cs1 50205035CC(=O)Nn1c(Cc2csc(NC(=O)CCl)n2)nnc1SCC(=O)NN 50205036CC(=O)Nn1c(Cc2csc(NCCC(O)=O)n2)nnc1SCSc1nnc(Cc2csc(NCCC(O)=O)n2)n1NC(C)=O 50205037Clc1ccc(cc1)C(=O)Nn1c(Cc2csc(NC(=O)c3ccccc3)n2)nnc1SCSc1nnc(Cc2csc(NC(=O)c3ccccc3)n2)n1NC(=O)c1ccc(Cl)cc1 50205038ClCC(=O)Nc1nc(Cc2n[nH]c(=S)n2NC(=O)c2ccccc2)cs1 50205039COC(=O)CSc1nnc(Cc2csc(NC(=O)c3ccccc3)n2)n1NC(=O)c1ccc(Cl)cc1 50205040CC(=O)Nn1c(Cc2csc(NC(=O)CCl)n2)nnc1SCC(=O)NNC(=O)CCl 50205041OC(=O)CCNc1nc(Cc2n[nH]c(=S)n2NC(=O)c2ccc(Cl)cc2)cs1 50205042O=C(Nc1nc(Cc2nnc(SCC#N)n2NC(=O)c2ccccc2)cs1)c1ccccc1 50205043COC(=O)CSc1nnc(Cc2csc(NC(=O)CCl)n2)n1NC(=O)c1ccccc1 50205044Nn1c(Cc2csc(NC(=O)CCl)n2)n[nH]c1=S 50205045ClCC(=O)NNC(=O)CSc1nnc(Cc2csc(NC(=O)c3ccccc3)n2)n1NC(=O)c1ccccc1 50205046CC(=O)NNC(=O)CSc1nnc(Cc2csc(NCCC(O)=O)n2)n1NC(=O)c1ccc(Cl)cc1 50205047CC(=O)Nn1c(Cc2csc(NC(=O)CCl)n2)nnc1SCc1n[nH]c(=S)n1N 50205048Nn1c(CSc2nnc(Cc3csc(NCCC(O)=O)n3)n2NC(=O)c2ccc(Cl)cc2)n[nH]c1=S 50205049OC(=O)CCNc1nc(Cc2nnc(SCC(=O)NN=Cc3ccccc3)n2NC(=O)c2ccc(Cl)cc2)cs1 50205050COC(=O)CSc1nnc(Cc2csc(NC(=O)c3ccccc3)n2)n1NC(C)=O 50205051CC(=O)Nc1nc(Cc2nnc(SCSc3nnc(Cc4csc(NC(C)=O)n4)n3NC(C)=O)n2NC(C)=O)cs1 50205052Nn1c(Cc2csc(NCCC(O)=O)n2)n[nH]c1=S 50205053CC(=O)Nc1nc(Cc2nnc(SCC(=O)NNC(=O)CCl)n2NC(=O)c2ccccc2)cs1 50205054CC(=O)NNC(=O)CSc1nnc(Cc2csc(NC(=O)CCl)n2)n1NC(=O)c1ccc(Cl)cc1 50205055NNC(=O)CSc1nnc(Cc2csc(NCCC(O)=O)n2)n1NC(=O)c1ccc(Cl)cc1 50205056CC(=O)NNC(=O)CSc1nnc(Cc2csc(NCCC(O)=O)n2)n1NC(C)=O 50205057COC(=O)CSc1nnc(Cc2csc(NCCC(O)=O)n2)n1NC(=O)c1ccccc1 50205058CC(=O)Nc1nc(Cc2n[nH]c(=S)n2NC(=O)c2ccc(Cl)cc2)cs1 50205059CC(=O)Nc1nc(Cc2nnc(SCC(=O)NN)n2NC(=O)c2ccccc2)cs1 50205060CC(=O)Nn1c(Cc2csc(NC(=O)c3ccccc3)n2)nnc1SCc1n[nH]c(=S)n1N 50205061Clc1ccc(cc1)C(=O)Nn1c(Cc2csc(NC(=O)c3ccccc3)n2)nnc1SCC(=O)NN=Cc1ccccc1 50205062Clc1ccc(cc1)C(=O)Nn1c(Cc2csc(NC(=O)c3ccccc3)n2)nnc1SCC(=O)NNC(=O)c1ccccc1 50205063CC(=O)Nn1c(Cc2csc(NCCC(O)=O)n2)nnc1SCC#N 50205064CC(=O)Nn1c(Cc2csc(NCCC(O)=O)n2)nnc1SCC(=O)NN 50205065Nn1c(CSc2nnc(Cc3csc(NC(=O)CCl)n3)n2NC(=O)c2ccccc2)n[nH]c1=S 50205066O=C(Nc1nc(Cc2nnc(SCSc3nnc(Cc4csc(NC(=O)c5ccccc5)n4)n3NC(=O)c3ccccc3)n2NC(=O)c2ccccc2)cs1)c1ccccc1 50205067OC(=O)CCNc1nc(Cc2nnc(SCC(=O)NNC(=O)CCl)n2NC(=O)c2ccc(Cl)cc2)cs1 50205068CC(=O)NNC(=O)CSc1nnc(Cc2csc(NC(C)=O)n2)n1NC(=O)c1ccc(Cl)cc1 50205069OC(=O)CCNc1nc(Cc2nnc(SCC(=O)NNC(=O)CCl)n2NC(=O)c2ccccc2)cs1 50205070COC(=O)CSc1nnc(Cc2csc(NC(C)=O)n2)n1NC(=O)c1ccc(Cl)cc1 50205071COC(=O)CSc1nnc(Cc2csc(NC(=O)CCl)n2)n1NC(=O)c1ccc(Cl)cc1 50216159Oc1ccc2[nH]c3c4cccn4c4C(=O)NC(=O)c4c3c2c1 50216171O=C1NC(=O)c2c1c1c3ccccc3[nH]c1c1cccn21 50218333ClCC(=O)Nc1cc(c(s1)-c1nnc2SC(C(=Nn12)c1ccccc1)c1ccccc1)-c1ccccc1 50218334CC(=O)Nc1cc(C)c(s1)-c1nnc2sc(nn12)-c1cccc(c1)[N+]([O-])=O 50218335CC(=O)Nc1cc(C)c(s1)-c1nnc2SCC(C)=Nn12 50218336Cc1cc(NC(=O)CCl)sc1-c1nnc2S\C(=C/c3ccc(Cl)cc3)C(=Nn12)c1cc(F)c(Cl)cc1Cl 50218337Cc1cc(NC(=O)CCl)sc1-c1nnc2sc(nn12)-c1ccccc1 50218338Cc1cc(NC(=O)CCl)sc1-c1nnc2sc(nn12)-c1cccc(c1)[N+]([O-])=O 50218339CC1=Nn2c(SC1)nnc2-c1sc(NC(=O)CCl)cc1-c1ccccc1 50218340CC(=O)Nc1cc(c(s1)-c1nnc2SCC(=O)Nn12)-c1ccccc1 50218341[O-][N+](=O)c1cccc(c1)-c1nn2c(nnc2s1)-c1sc(NC(=O)CCl)cc1-c1ccccc1 50218342CC(=O)Nc1cc(c(s1)-c1nnc2Sc3nc4ccccc4nc3Nn12)-c1ccccc1 50218343CC(=O)Nc1cc(c(s1)-c1nnc2S\C(=C/c3ccc(Cl)cc3)C(=Nn12)c1cc(F)c(Cl)cc1Cl)-c1ccccc1 50218344Cc1cc(NC(=O)CCl)sc1-c1nnc2SCC(=O)Nn12 50218345CC(=O)Nc1cc(C)c(s1)-c1nnc2sc(S)nn12 50218346CC(=O)Nc1cc(C)c(s1)-c1nnc2SC(C(=Nn12)c1ccccc1)c1ccccc1 50218347CC(=O)Nc1cc(C)c(s1)-c1nnc2sc([CH-]c3cccc(c3)[N+]([O-])=O)c(n[n+]12)-c1cc(F)c(Cl)cc1Cl 50218348CC(=O)Nc1cc(c(s1)-c1n[nH]c(=S)n1N)-c1ccccc1 50218350CC(=O)Nc1cc(C)c(s1)-c1n[nH]c(=S)n1N 50218351CC(=O)Nc1cc(c(s1)-c1nnc2sc(nn12)-c1cccc(c1)[N+]([O-])=O)-c1ccccc1 50218352CC(=O)Nc1cc(c(s1)-c1nnc2SCC(C)=Nn12)-c1ccccc1 50218353CC(=O)Nc1cc(C)c(s1)-c1nnc2S\C(=C/c3ccccc3Cl)C(=Nn12)c1cc(F)c(Cl)cc1Cl 50218354CC(=O)Nc1cc(c(s1)-c1nnc2SC(C(=Nn12)c1ccccc1)c1ccccc1)-c1ccccc1 50218355CC(=O)Nc1cc(c(s1)-c1nnc2sc(S)nn12)-c1ccccc1 50218356CC(=O)Nc1cc(C)c(s1)-c1nnc2sc(nn12)-c1ccccc1 50218357ClCC(=O)Nc1cc(c(s1)-c1nnc2Sc3nc4ccccc4nc3Nn12)-c1ccccc1 50218358CC(=O)Nc1cc(C)c(s1)-c1nnc2Sc3nc4ccccc4nc3Nn12 50218359Cc1cc(NC(=O)CCl)sc1-c1nnc2SC(C(=Nn12)c1ccccc1)c1ccccc1 50218360Sc1nn2c(nnc2s1)-c1sc(NC(=O)CCl)cc1-c1ccccc1 50218361Cc1cc(NC(=O)CCl)sc1-c1nnc2Sc3nc4ccccc4nc3Nn12 50218362CC(=O)Nc1cc(C)c(s1)-c1nnc2SCC(=O)Nn12 50218363[O-][N+](=O)c1cccc([CH-]c2sc3nnc(-c4sc(NC(=O)CCl)cc4-c4ccccc4)[n+]3nc2-c2cc(F)c(Cl)cc2Cl)c1 50218364Fc1cc(C2=Nn3c(S\C2=C/c2ccc(Cl)cc2)nnc3-c2sc(NC(=O)CCl)cc2-c2ccccc2)c(Cl)cc1Cl 50218365Cc1cc(NC(=O)CCl)sc1-c1nnc2S\C(=C/c3ccccc3Cl)C(=Nn12)c1cc(F)c(Cl)cc1Cl 50218366CC(=O)Nc1cc(c(s1)-c1nnc2sc([CH-]c3cccc(c3)[N+]([O-])=O)c(n[n+]12)-c1cc(F)c(Cl)cc1Cl)-c1ccccc1 50218367Cc1cc(NC(=O)CCl)sc1-c1nnc2sc(S)nn12 50218368Cc1cc(NC(=O)CCl)sc1-c1nnc2sc([CH-]c3cccc(c3)[N+]([O-])=O)c(n[n+]12)-c1cc(F)c(Cl)cc1Cl 50218369ClCC(=O)Nc1cc(c(s1)-c1nnc2sc(nn12)-c1ccccc1)-c1ccccc1 50218370Cc1cc(NC(=O)CCl)sc1-c1n[nH]c(=S)n1N 50218371Fc1cc(C2=Nn3c(S\C2=C/c2ccccc2Cl)nnc3-c2sc(NC(=O)CCl)cc2-c2ccccc2)c(Cl)cc1Cl 50218373Fc1cc(C2=Nn3c(S\C2=C/c2ccccc2)nnc3-c2sc(NC(=O)CCl)cc2-c2ccccc2)c(Cl)cc1Cl 50218374Cc1cc(NC(=O)CCl)sc1-c1nnc2SCC(C)=Nn12 50218375ClCC(=O)Nc1cc(c(s1)-c1nnc2SCC(=O)Nn12)-c1ccccc1 50218376CC(=O)Nc1cc(C)c(s1)-c1nnc2S\C(=C/c3ccc(Cl)cc3)C(=Nn12)c1cc(F)c(Cl)cc1Cl 50218377Nn1c(n[nH]c1=S)-c1sc(NC(=O)CCl)cc1-c1ccccc1 50218378CC(=O)Nc1cc(c(s1)-c1nnc2S\C(=C/c3ccccc3Cl)C(=Nn12)c1cc(F)c(Cl)cc1Cl)-c1ccccc1 50218379CC(=O)Nc1cc(c(s1)-c1nnc2sc(nn12)-c1ccccc1)-c1ccccc1 50218380CC(=O)Nc1cc(c(s1)-c1nnc2S\C(=C/c3ccccc3)C(=Nn12)c1cc(F)c(Cl)cc1Cl)-c1ccccc1 50232478O[C@@]12CC\C=C/CCCCN3CC[C@@H](C(=C1)c1nccc4c5ccccc5[nH]c14)[C@]1(C[C@@H]4\C=C/CCCCN4[C@@H]21)C3 50242742COc1cc(ccc1Nc1ncc(Cl)c(Nc2ccccc2S(=O)(=O)C(C)C)n1)N1CCC(CC1)N1CCN(C)CC1 50244787CC[C@H](CO)Nc1nc(Nc2cccc(c2)-c2ccccn2)c2ncn(C(C)C)c2n1 50247394CCn1cnc2ccc3nc(sc3c2c1=O)C(=N)OCCc1ccccc1 50267161COc1ccc(cc1O)-c1c[nH]c2C(N=O)c3cccn3-c12 50267607Cn1cc(C2=C(C(=O)NC2=O)c2coc3cc(CO)ccc23)c2cc(Br)ccc12 50295352CCCCc1c([nH]c2nccnc12)-c1ccc(OCCOCCOCCN)cc1 50295872Cn1cc(-c2nc(N)ncc2I)c2ccccc12 50295878Cn1cc(-c2nc(N)ncc2-c2ccncc2)c2ccccc12 50297039Nc1n[nH]c2nc(N)c(C#N)c(-c3ccccc3)c12 50299869CCOC(=O)c1cc(-c2csc(n2)-c2ccncc2)c(=O)[nH]c1C 50304109[O-][N+](=O)c1ccc2NC(=O)C(c2c1)c1[nH]c2ccccc2c1N=O 50304110Nc1ccc2NC(=O)C(=C3Nc4ccccc4C3=O)c2c1 50304111CC(=O)Nc1ccc2NC(=O)\C(=C3/Nc4ccccc4C3=O)c2c1 50304112Nc1ccc2NC(=O)C(c2c1)c1[nH]c2ccccc2c1N=O 50304113CC(=O)Nc1ccc2NC(=O)\C(=C3/Nc4ccc(Br)cc4C3=O)c2c1 50304114CC(=O)Nc1ccc2NC(=O)C(c2c1)c1[nH]c2ccccc2c1N=O 50304119Nc1ccc2NC(=O)C(=C3Nc4ccc(Br)cc4C3=O)c2c1 50304121[O-][N+](=O)c1ccc2NC(=O)C(c2c1)c1[nH]c2ccc(Br)cc2c1N=O 50304123Nc1ccc2NC(=O)C(c2c1)c1[nH]c2ccc(Br)cc2c1N=O 50304124CC(=O)Nc1ccc2NC(=O)C(c2c1)c1[nH]c2ccc(Br)cc2c1N=O 50305006NCCn1cc(-c2cc(-c3cc4ccccc4s3)c3[nH]ncc3c2)c2nc(N)ncc12 50307506Cn1nc(C(N)=O)c2CCc3cnc(NC4CCN(CC4)C(=O)c4ccccc4)nc3-c12 50307507CNC(=O)c1nn(C)c-2c1CCc1cnc(NC3CCN(CC3)C(=O)C3CCN(CC3)S(C)(=O)=O)nc-21 50307535CC(=O)N1CCC(CC1)Nc1ncc2CCc3c(nn(C)c3-c2n1)C(N)=O 50307987CC(C)(C)C(=O)N1Cc2c(NC(=O)c3cc(F)cc(F)c3)[nH]nc2C1(C)C 50312212CN1C(=O)C(=Cc2ccc3OCOc3c2)N=C1NCCN 50312990Cn1cc(C2=C(C(=O)NC2=O)c2cccc(NCC(O)CO)c2)c2cc(F)ccc12 50323213Oc1ccc(cc1)-c1cc(=O)c2c(O)cc(O)c(-c3c(O)cc(O)c4c3oc(cc4=O)-c3ccc(O)cc3)c2o1 50331277COc1ccc2cc([nH]c2c1)-c1n[nH]c2cccnc12 50340882COc1ccc(cc1)C(=O)c1sc(Nc2ccncc2)nc1N 50340883Nc1nc(Nc2cccnc2)sc1C(=O)c1ccccn1 50340884Nc1nc(Nc2cccnc2)sc1C(=O)c1cccnc1 50340885Nc1nc(Nc2cccnc2)sc1C(=O)c1ccncc1 50340887Nc1nc(Nc2ccc(nc2)C(F)(F)F)sc1C(=O)c1ccccc1F 50340888Nc1nc(Nc2ccc(Cl)cc2)sc1C(=O)c1cccc(c1)[N+]([O-])=O 50340889Nc1nc(Nc2ccc(Cl)cc2)sc1C(=O)c1cccc(F)c1 50340890COc1cccc(c1)C(=O)c1sc(Nc2ccc(Cl)cc2)nc1N 50340891Nc1nc(NC2CCCNC2)sc1C(=O)c1cccc(F)c1 50340892Nc1nc(NC2CCNCC2)sc1C(=O)c1cccc(F)c1 50340893Nc1nc(Nc2cccc(N)c2)sc1C(=O)c1cccc(F)c1 50340894CNc1cccc(Nc2nc(N)c(s2)C(=O)c2cccc(F)c2)c1 50340895CN(C)c1ccc(Nc2nc(N)c(s2)C(=O)c2cccc(F)c2)cc1 50340896Nc1nc(Nc2ccccn2)sc1C(=O)c1cccc(F)c1 50340897Nc1nc(Nc2ccccn2)sc1C(=O)c1ccccc1F 50340898Nc1nc(Nc2ccccn2)sc1C(=O)c1ccc(F)cc1 50340899COc1ccccc1C(=O)c1sc(Nc2ccccn2)nc1N 50340900COc1cccc(c1)C(=O)c1sc(Nc2ccccn2)nc1N 50340901COc1ccc(cc1)C(=O)c1sc(Nc2ccccn2)nc1N 50340902Nc1nc(Nc2cccnc2)sc1C(=O)c1ccccc1F 50340903Nc1nc(Nc2cccnc2)sc1C(=O)c1cccc(F)c1 50340904Nc1nc(Nc2cccnc2)sc1C(=O)c1ccc(F)cc1 50340905Nc1nc(Nc2cccnc2)sc1C(=O)c1ccccc1 50340906Nc1nc(Nc2cccnc2)sc1C(=O)c1cccc(c1)[N+]([O-])=O 50340907COc1ccccc1C(=O)c1sc(Nc2cccnc2)nc1N 50340908COc1cccc(c1)C(=O)c1sc(Nc2cccnc2)nc1N 50340909COc1ccc(cc1)C(=O)c1sc(Nc2cccnc2)nc1N 50340910Nc1nc(Nc2ccncc2)sc1C(=O)c1ccccc1F 50340911Nc1nc(Nc2ccncc2)sc1C(=O)c1cccc(F)c1 50340912Nc1nc(Nc2ccncc2)sc1C(=O)c1ccc(F)cc1 50340913COc1ccccc1C(=O)c1sc(Nc2ccncc2)nc1N 50340914COc1cccc(c1)C(=O)c1sc(Nc2ccncc2)nc1N 50341878CC[C@H](CO)Nc1nc(NCc2ccccc2)c2n[nH]c(C(C)C)c2n1 50346235O=C1Cc2c([nH]c3ccncc23)-c2ccccc2N1 50346237[O-][n+]1ccc2[nH]c-3c(CC(=O)Nc4ccccc-34)c2c1 50347740CCCNC1=NC(=Cc2ccc3OCOc3c2)C(=O)N1 50347743CCNC1=NC(=Cc2ccc3OCOc3c2)C(=O)N1 50347744O=C1NC(NCC2CC2)=NC1=Cc1ccc2OCOc2c1 50347746Oc1ccc(NC2=NC(=Cc3ccc4OCOc4c3)C(=O)N2)cc1 50347748O=C1NC(Nc2ccc3OCOc3c2)=NC1=Cc1ccc2OCOc2c1 50347750O=C1NC(Nc2ccccc2)=NC1=Cc1ccc2OCOc2c1 50347756CCCNC1=NC(=Cc2ccc3OCOc3c2)C(=O)N1C 50347757CC(C)NC1=NC(=Cc2ccc3OCOc3c2)C(=O)N1C 50347758CCCCNC1=NC(=Cc2ccc3OCOc3c2)C(=O)N1C 50347759CN1C(=O)C(=Cc2ccc3OCOc3c2)N=C1Nc1ccc(O)cc1 50347760COc1ccc(NC2=NC(=Cc3ccc4OCOc4c3)C(=O)N2C)cc1 50347761CN1C(Nc2ccc3OCOc3c2)=NC(=Cc2ccc3OCOc3c2)C1=O 50347762CN1C(=O)C(=Cc2ccc3OCOc3c2)N=C1Nc1ccc2OCCOc2c1 50347763CC(C)CNC1=NC(=Cc2ccc3OCOc3c2)C(=O)N1C 50347764CC(C)CCNC1=NC(=Cc2ccc3OCOc3c2)C(=O)N1C 50347765CN1C(=O)C(=Cc2ccc3OCOc3c2)N=C1NCC=C 50347766CN1C(=O)C(=Cc2ccc3OCOc3c2)N=C1NCC1CC1 50347767CN1C(NC2CCCC2)=NC(=Cc2ccc3OCOc3c2)C1=O 50347768CN1C(=O)C(=Cc2ccc3OCOc3c2)N=C1NCCO 50347770CN1C(=O)C(=Cc2ccc3OCOc3c2)N=C1NCCCO 50347772CN1C(=O)C(=Cc2ccc3OCOc3c2)N=C1NCCN1CCOCC1 50347778CN1C(Nc2ccccc2)=NC(=Cc2ccc3OCOc3c2)C1=O 50347786CC(=O)Nc1ccc(cc1)-c1cnc(N)nc1-c1c[nH]c2ccc(Br)cc12 50347791CC(=O)c1ccc(cc1)-c1cnc(N)nc1-c1c[nH]c2cccc(Br)c12 50347792Nc1ncc(I)c(n1)-c1c[nH]c2c(Br)cccc12 50347793Nc1ncc(I)c(n1)-c1c[nH]c2cc(Br)ccc12 50347794Nc1ncc(I)c(n1)-c1c[nH]c2ccc(Br)cc12 50347796Nc1nccc(n1)-c1c[nH]c2c(Br)cccc12 50347798Nc1ncc(I)c(n1)-c1c[nH]c2c(N)cccc12 50347799Nc1ccc2c(c[nH]c2c1)-c1nc(N)ncc1I 50347802Nc1ncc(I)c(n1)-c1c[nH]c2ccccc12 50347803Nc1ncc(I)c(n1)-c1c[nH]c2cc(ccc12)[N+]([O-])=O 50347804Nc1ncc(I)c(n1)-c1c[nH]c2ccc(cc12)[N+]([O-])=O 50347806Nc1nccc(n1)-c1c[nH]c2c(cccc12)[N+]([O-])=O 50347810COc1cccc(c1)-c1cnc(N)nc1-c1c[nH]c2cccc(Br)c12 50347814CC(=O)Nc1ccc(cc1)-c1cnc(N)nc1-c1c[nH]c2c(Br)cccc12 50347816COc1cccc(c1)-c1cnc(N)nc1-c1c[nH]c2ccc(Br)cc12 50347817Nc1ncc(-c2ccc(cc2)C(F)(F)F)c(n1)-c1c[nH]c2cccc(Br)c12 50349806O=C1Nc2ccccc2\C1=C1/Nc2ccccc2C1=O 50354392Nc1ncnc2c3ccccc3sc12 50355903Oc1ccc(cc1)-c1cncc(c1)-c1cc2cc(O)ccc2[nH]1 50355904Oc1ccc2[nH]c(cc2c1)-c1cncc(c1)-c1ccc(cc1)C#N 50355905CS(=O)(=O)c1ccc(cc1)-c1cncc(c1)-c1cc2cc(O)ccc2[nH]1 50355906Oc1ccc(cc1)-c1cncc(n1)-c1cc2cc(O)ccc2[nH]1 50355907Oc1ccc2[nH]c(cc2c1)-c1cncc(n1)-c1ccc(cc1)C#N 50355908CS(=O)(=O)c1ccc(cc1)-c1cncc(n1)-c1cc2cc(O)ccc2[nH]1 50355909Oc1ccc(cc1)-c1cncc(c1)-c1cc2ccc(O)cc2[nH]1 50355910Oc1ccc2cc([nH]c2c1)-c1cncc(c1)-c1ccc(cc1)C#N 50355911CS(=O)(=O)c1ccc(cc1)-c1cncc(c1)-c1cc2ccc(O)cc2[nH]1 50355912Oc1ccc(cc1)-c1cncc(n1)-c1cc2ccc(O)cc2[nH]1 50355913Oc1ccc2cc([nH]c2c1)-c1cncc(n1)-c1ccc(cc1)C#N 50355914CS(=O)(=O)c1ccc(cc1)-c1cncc(n1)-c1cc2ccc(O)cc2[nH]1 50355915Oc1ccc(cc1)-c1ccnc(c1)-c1cc2cc(O)ccc2[nH]1 50355916Oc1ccc(cc1)-c1ccnc(c1)-c1cc2ccc(O)cc2[nH]1 50363795Oc1ccc2oc(=O)c3[nH]c4ccc(F)cc4c3c2c1 50363797Oc1ccc2[nH]c3c(c2c1)c1cc(O)ccc1oc3=O 50363802Oc1ccc2oc(=O)c3[nH]c4ccccc4c3c2c1 50363804Oc1ccc2[nH]c3c(c2c1)c1ccc(O)cc1oc3=O 50363805Oc1ccc2c3c4ccccc4[nH]c3c(=O)oc2c1 50366800CC[C@H](CO)Nc1nc(NCc2ccccc2O)c2ncn(C(C)C)c2n1 50371397Cn1cc(-c2ccnc(N)n2)c2c(O)ccnc12 50371399CC(C)Oc1ccnc2[nH]cc(-c3ccnc(N)n3)c12 50371400CCCOc1ccnc2[nH]cc(-c3ccnc(N)n3)c12 50371401CCOc1ccnc2[nH]cc(-c3ccnc(N)n3)c12 50371402COc1ccnc2[nH]cc(-c3ccnc(N)n3)c12 50371403Nc1nccc(n1)-c1c[nH]c2nccc(O)c12 50371404Nc1nccc(n1)-c1c[nH]c2ncccc12 50371405COc1ccnc2c1c(-c1ccnc(N)n1)c1ccnc(N)n21 50371406COc1ccnc2[nH]cc(-c3ccncn3)c12 50371407Oc1ccnc2[nH]cc(-c3ccncn3)c12 50371408COc1ccnc2[nH]cc(-c3ccnc(SC)n3)c12 50371409Nc1nccc(n1)-c1c[nH]c2nccc(Cl)c12 50371411Nc1nccc(n1)-c1c[nH]c2nc(Br)ccc12 50376078O=C1Cc2c([nH]c3ccc(cc23)C#N)-c2cc(ccc2N1)C#N 50376086Cn1c-2c(CC(=O)Nc3cccnc-23)c2ccccc12 50376087COc1ccc2[nH]c-3c(CC(=O)Nc4ccncc-34)c2c1 50376088Clc1ccc2[nH]c-3c(CC(=O)Nc4ccncc-34)c2c1 50376089Fc1ccc2[nH]c-3c(CC(=O)Nc4ccncc-34)c2c1 50376090FC(F)(F)c1ccc2[nH]c-3c(CC(=O)Nc4ccncc-34)c2c1 50376091O=C1Cc2c([nH]c3ccc(cc23)C#N)-c2cnccc2N1 50376092Brc1ccc2[nH]c-3c(CC(=O)Nc4ccncc-34)c2c1 50376094Ic1cc(cc2c3CC(=O)Nc4cccnc4-c3[nH]c12)C#N 50376095Oc1ccc2[nH]c-3c(CC(=O)Nc4cccnc-34)c2c1 50376097COc1ccc2[nH]c-3c(CC(=O)Nc4cccnc-34)c2c1 50376099Ic1ccc2[nH]c-3c(CC(=O)Nc4cccnc-34)c2c1 50376100O=C1Cc2c([nH]c3ccccc23)-c2ncccc2N1 50376104Fc1ccc2[nH]c-3c(CC(=O)Nc4cccnc-34)c2c1 50376106O=C1Cc2c([nH]c3ccc(cc23)C#N)-c2ncccc2N1 50377290CCNC(=O)O[C@@H](C)[C@H]1c2ccccc2-c2c1c1[nH]c3ccccc3c1c1CNC(=O)c21 50378657CC(C)CC(=O)Nc1[nH]nc2c1CN(C(=O)C1CCN(C)CC1)C2(C)C 50378826O=C(Nc1cc(c[nH]1)C1CCC1)Nc1cccc2ccncc12 50379081CC1C\C=C\C(O)C(O)CC\C=C\c2cc(O)cc(O)c2C(=O)O1 50383304CCCCC[C@@H](NC)c1c(O)cc(O)c2c1oc(cc2=O)-c1ccccc1 50383305CN1CCCC[C@H]1c1c(O)cc(O)c2c1oc(cc2=O)-c1ccccc1 50383306CN1CCC[C@@H]1c1c(O)cc(O)c2c1oc(cc2=O)-c1ccccc1 50383307CN1CCCC[C@@H]1c1c(O)cc(O)c2c1oc(cc2=O)-c1ccccc1 50383308Oc1cc(O)c2c(oc(cc2=O)-c2ccccc2)c1C1CCCCN1 50383311CN1CCC[C@H]1c1c(O)cc(O)c2c1oc(cc2=O)-c1ccccc1 50383312Oc1cc(O)c2c(oc(cc2=O)-c2ccccc2)c1C1CCCN1 50383313CCCCC[C@H](NC)c1c(O)cc(O)c2c1oc(cc2=O)-c1ccccc1 50385579Cc1ccc2[nH]c3c4cccn4c4C(=O)NC(=O)c4c3c2c1 50385580O=C1NC(=O)c2c1c1ccnn1c1[nH]c3ccccc3c21 50385583Oc1ccc2[nH]c3c(c4C(=O)NC(=O)c4c4ccnn34)c2c1 50385584O=C1NC(=O)c2c1c1n[nH]cc1c1[nH]c3ccccc3c21 50385585Cc1ccc2[nH]c3c4c[nH]nc4c4C(=O)NC(=O)c4c3c2c1 50390638NS(=O)(=O)c1cc(cs1)-c1nc2ccccc2s1 50390639NS(=O)(=O)c1cc(cs1)-c1nc2ccc(F)cc2s1 50390640NS(=O)(=O)c1cc(cs1)-c1nc2ccc(Cl)cc2s1 50390641Cc1ccc2nc(sc2c1)-c1csc(c1)S(N)(=O)=O 50390642NS(=O)(=O)c1cc(cs1)-c1nc2ccc(cc2s1)[N+]([O-])=O 50390643CC(=O)c1ccc2nc(sc2c1)-c1csc(c1)S(N)(=O)=O 50390645O=S(=O)(Nc1nccs1)c1cc(cs1)-c1nc2ccccc2s1 50390646Cc1nc(NS(=O)(=O)c2cc(cs2)-c2nc3ccccc3s2)sc1C 50390647CCOC(=O)Cc1csc(NS(=O)(=O)c2cc(cs2)-c2nc3ccccc3s2)n1 50390648O=S(=O)(NCc1ccccn1)c1cc(cs1)-c1nc2ccccc2s1 50390649Cc1ccnc(NS(=O)(=O)c2cc(cs2)-c2nc3ccccc3s2)c1 50390650Oc1cccnc1NS(=O)(=O)c1cc(cs1)-c1nc2ccccc2s1 50390651O=S(=O)(Nc1ccc(nc1)N1CCOCC1)c1cc(cs1)-c1nc2ccccc2s1 50390652OC[C@H]1CCCN1S(=O)(=O)c1cc(cs1)-c1nc2ccccc2s1 50390653NS(=O)(=O)c1cc(cs1)-c1nc2ccc(F)c(Cl)c2s1 50390654NS(=O)(=O)c1cc(cs1)-c1nc2cccc(-c3ccc(F)cc3)c2s1 50390655ONS(=O)(=O)c1cc(cs1)-c1nc2ccccc2s1 50393109Nc1nc2c(nccc2[nH]1)-c1ccccn1 50395887Oc1cc2c(oc3ncc(OCc4ccccc4)c(-c4ccccc4)c23)c2ccccc12 50395892Oc1ccc2oc3ncc(O)c(-c4ccccc4)c3c2c1 50395894Oc1cnc2oc3c(cc(O)c4ccccc34)c2c1-c1ccccc1 50399301O=C(Nc1ccccn1)Nc1cccc2C(=O)N3CCCCC3c12 50399302Oc1ccc(NC(=O)Nc2cccc3C(=O)N4CCCCC4c23)nc1 50399303Oc1cccnc1NC(=O)Nc1cccc2C(=O)N3CCCCC3c12 50399304O=C(Nc1ccc(cn1)-c1ccccc1)Nc1cccc2C(=O)N3CCCCC3c12 50399306COc1cccnc1NC(=O)Nc1cccc2C(=O)N3CCCCC3c12 50399308Fc1cnc(NC(=O)Nc2cccc3C(=O)N4CCCCC4c23)c(F)c1 50399309Fc1cccc(NC(=O)Nc2cccc3C(=O)N4CCCCC4c23)n1 50399310Brc1ccnc(NC(=O)Nc2cccc3C(=O)N4CCCCC4c23)c1 50399311Brc1ccc(NC(=O)Nc2cccc3C(=O)N4CCCCC4c23)nc1 50399312Brc1cccc(NC(=O)Nc2cccc3C(=O)N4CCCCC4c23)n1 50399314Oc1cccc2ccc(NC(=O)Nc3cccc4C(=O)N5CCCCC5c34)nc12 50399315O=C(Nc1cc2ccccc2cn1)Nc1cccc2C(=O)N3CCCCC3c12 50399317O=C(Nc1cc(on1)-c1ccccc1)Nc1cccc2C(=O)N3CCCCC3c12 50399318Cc1cc(NC(=O)Nc2cccc3C(=O)N4CCCCC4c23)no1 50399319Cn1ccc(NC(=O)Nc2cccc3C(=O)N4CCCCC4c23)n1 50399320O=C(Nc1ccn[nH]1)Nc1cccc2C(=O)N3CCCCC3c12 50399321O=C(Nc1csc(n1)-c1ccncc1)Nc1cccc2C(=O)N3CCCCC3c12 50399322Cc1nc(NC(=O)Nc2cccc3C(=O)N4CCCCC4c23)cs1 50399323O=C(Nc1cscn1)Nc1cccc2C(=O)N3CCCCC3c12 50399324O=C(Nc1ccncn1)Nc1cccc2C(=O)N3CCCCC3c12 50399326O=C(Nc1cnccn1)Nc1cccc2C(=O)N3CCCCC3c12 50400564CCCn1cnc2c(NCc3ccc(C)s3)nc(N[C@H](CC)CO)nc12 50402020CC(C)(C)Nc1c(Nc2ccnc(Nc3ccc(cc3)-c3ccncc3)n2)c(=O)c1=O 50411426Cc1cc(NC(=O)CCl)sc1-c1nnc2S\C(=C/c3ccccc3)C(=Nn12)c1cc(F)c(Cl)cc1Cl 50411427CC(=O)Nc1cc(C)c(s1)-c1nnc2S\C(=C/c3ccccc3)C(=Nn12)c1cc(F)c(Cl)cc1Cl 50414897CCN(CC)CCCOC(=O)c1cc(-c2csc(n2)-c2ccncc2)c(=O)[nH]c1C(C)C 50414898CCOC(=O)c1cc(-c2csc(n2)-c2ccnc(NCC(C)C)c2)c(=O)[nH]c1C 50414899CCCc1[nH]c(=O)c(cc1C(=O)OCC)-c1csc(n1)-c1ccncc1 50414900CCOC(=O)c1cc(-c2csc(n2)-c2ccnc(NC)c2)c(=O)[nH]c1C(C)C 50414901CCN(CC)CC(C)OC(=O)c1cc(-c2csc(n2)-c2ccncc2)c(=O)[nH]c1C(C)C 50414902CC(C)c1[nH]c(=O)c(cc1C(=O)OCCN1CCCC1)-c1csc(n1)-c1ccncc1 50414903CC(C)c1[nH]c(=O)c(cc1C(=O)OC1CCCN(C)C1)-c1csc(n1)-c1ccncc1 50414904CCN(CC)CCOC(=O)c1cc(-c2csc(n2)-c2ccncc2)c(=O)[nH]c1C(C)C 50414905CCOC(=O)c1cc(-c2csc(n2)-c2ccnc(NCCN(CC)CC)c2)c(=O)[nH]c1C 50414906CCOC(=O)c1cc(-c2csc(n2)-c2ccnc(OC)c2)c(=O)[nH]c1C(C)C 50414907CCOC(=O)c1cc(-c2csc(n2)-c2ccncc2)c(=O)[nH]c1C1CC1 50414908CCOC(=O)c1cc(-c2csc(n2)-c2ccncc2)c(=O)[nH]c1C(C)C 50414909CCOC(=O)c1cc(-c2csc(n2)-c2ccncc2)c(=O)[nH]c1COCc1ccccc1 50414910CC(C)c1[nH]c(=O)c(cc1C(=O)OC1CCN(C)CC1)-c1csc(n1)-c1ccncc1 50414912CCOC(=O)c1cc(-c2csc(n2)-c2ccncc2)c(=O)[nH]c1CC 50414913CCOC(=O)c1cc(-c2csc(n2)-c2ccnc(Cl)c2)c(=O)[nH]c1C 50414914CCOC(=O)c1cc(-c2csc(n2)-c2ccnc(N)c2)c(=O)[nH]c1C 50414915CC(C)c1[nH]c(=O)c(cc1C(=O)OCCc1ccccc1)-c1csc(n1)-c1ccncc1 50414916CCCc1[nH]c(=O)c(cc1C(=O)OCC)-c1csc(CS(=O)(=O)c2ccccc2)n1 50414917CCOC(=O)c1cc(-c2csc(CS(=O)(=O)c3ccccc3)n2)c(=O)[nH]c1C 50414918CCOC(=O)c1cc(-c2csc(CS(=O)(=O)c3ccccc3)n2)c(=O)[nH]c1COCc1ccccc1 50415024O=C(Cc1ccccc1)Nc1cn(cn1)C1CCC1 50415025COc1ccc(CC(=O)Nc2cn(cn2)C2CCC2)cc1 50415026O=C(Cc1cccc2ccccc12)Nc1cn(cn1)C1CCC1 50415028COc1ccc(CC(=O)Nc2cn(cn2)C(C)C)cc1 50415029COc1ccc(CC(=O)Nc2cn(cn2)C2CC2)cc1 50415030COc1ccc(CC(=O)Nc2cn(cn2)C2CCCC2)cc1 50415031COc1ccc(CC(=O)Nc2cn(cn2)C2CCCCC2)cc1 50415032COc1ccc(CC(=O)Nc2cn(Cc3ccccc3)cn2)cc1 50415033COc1ccc(CC(=O)Nc2cn(cn2)[C@@H]2C[C@H](O)C2)cc1 50415034COc1ccc(CC(=O)Nc2cn(cn2)[C@H]2C[C@H](O)C2)cc1 50415035COC(=O)[C@H]1C[C@H](C1)n1cnc(NC(=O)Cc2ccc(OC)cc2)c1 50415036COC(=O)[C@H]1C[C@@H](C1)n1cnc(NC(=O)Cc2ccc(OC)cc2)c1 50415037COc1ccc(CC(=O)Nc2cn(cn2)[C@@H]2C[C@@H](C2)NC(C)=O)cc1 50415038COc1ccc(CC(=O)Nc2cn(cn2)[C@@H]2C[C@@H](C2)NS(C)(=O)=O)cc1 50415039CC(=O)N[C@H]1C[C@H](C1)n1cnc(NC(=O)Cc2cccc3ccccc23)c1 50415040NC(=O)[C@H]1C[C@H](C1)n1cnc(NC(=O)Cc2cccc3ccccc23)c1 50415041CN([C@H]1C[C@H](C1)n1cnc(NC(=O)Cc2cccc3ccccc23)c1)C(C)=O 50415042O=C(Cc1cccc2ccccc12)Nc1cn(cn1)[C@@H]1C[C@@H](C1)NC(=O)c1ccncc1 50415043O=C(Cc1cccc2ccccc12)Nc1cn(cn1)[C@@H]1C[C@@H](C1)NC(=O)c1cccnc1 50415044O=C(Cc1cccc2ccccc12)Nc1cn(cn1)[C@@H]1C[C@@H](C1)NC(=O)c1ccccn1 50415045Clc1cccc(n1)C(=O)N[C@H]1C[C@H](C1)n1cnc(NC(=O)Cc2cccc3ccccc23)c1 50415046Cc1cccc(n1)C(=O)N[C@H]1C[C@H](C1)n1cnc(NC(=O)Cc2cccc3ccccc23)c1 50418617[S-]C(=S)NNC(=O)Cc1c(NC(=O)c2ccccc2)sc2CCCCc12 50418618OC(=O)CCNc1sc2CCCCc2c1CC(=O)NNC([S-])=S 50418619Nn1c(Cc2c3CCCCc3sc2NC(=O)CCl)n[nH]c1=S 50418620CC(=O)Nc1sc2CCCCc2c1Cc1n[nH]c(=S)n1N 50418621Nn1c(Cc2c(NC(=O)c3ccccc3)sc3CCCCc23)n[nH]c1=S 50418622Nn1c(Cc2c3CCCCc3sc2NCCC(O)=O)n[nH]c1=S 50418623ClCC(=O)Nc1sc2CCCCc2c1Cc1n[nH]c(=S)n1NC(=O)c1ccc(Cl)cc1 50418624CC(=O)Nc1sc2CCCCc2c1Cc1n[nH]c(=S)n1NC(=O)c1ccc(Cl)cc1 50418625Clc1ccc(cc1)C(=O)Nn1c(Cc2c(NC(=O)c3ccccc3)sc3CCCCc23)n[nH]c1=S 50418626OC(=O)CCNc1sc2CCCCc2c1Cc1n[nH]c(=S)n1NC(=O)c1ccc(Cl)cc1 50418627ClCC(=O)Nc1sc2CCCCc2c1Cc1n[nH]c(=S)n1NC(=O)c1ccccc1 50418628CC(=O)Nc1sc2CCCCc2c1Cc1n[nH]c(=S)n1NC(=O)c1ccccc1 50418629O=C(Nc1sc2CCCCc2c1Cc1n[nH]c(=S)n1NC(=O)c1ccccc1)c1ccccc1 50418630OC(=O)CCNc1sc2CCCCc2c1Cc1n[nH]c(=S)n1NC(=O)c1ccccc1 50418631CC(=O)Nn1c(Cc2c3CCCCc3sc2NC(=O)CCl)n[nH]c1=S 50418632CC(=O)Nc1sc2CCCCc2c1Cc1n[nH]c(=S)n1NC(C)=O 50418633CC(=O)Nn1c(Cc2c(NC(=O)c3ccccc3)sc3CCCCc23)n[nH]c1=S 50418634CC(=O)Nn1c(Cc2c3CCCCc3sc2NCCC(O)=O)n[nH]c1=S 50418635Clc1ccc(cc1)C(=O)Nn1c(Cc2c(NC(=O)c3ccccc3)sc3CCCCc23)nnc1SCSc1nnc(Cc2c(NC(=O)c3ccccc3)sc3CCCCc23)n1NC(=O)c1ccc(Cl)cc1 50418636OC(=O)CCNc1sc2CCCCc2c1Cc1nnc(SCSc2nnc(Cc3c(NCCC(O)=O)sc4CCCCc34)n2NC(=O)c2ccc(Cl)cc2)n1NC(=O)c1ccc(Cl)cc1 50418637ClCC(=O)Nc1sc2CCCCc2c1Cc1nnc(SCSc2nnc(Cc3c(NC(=O)CCl)sc4CCCCc34)n2NC(=O)c2ccccc2)n1NC(=O)c1ccccc1 50418638CC(=O)Nc1sc2CCCCc2c1Cc1nnc(SCSc2nnc(Cc3c(NC(C)=O)sc4CCCCc34)n2NC(=O)c2ccccc2)n1NC(=O)c1ccccc1 50418639O=C(Nc1sc2CCCCc2c1Cc1nnc(SCSc2nnc(Cc3c(NC(=O)c4ccccc4)sc4CCCCc34)n2NC(=O)c2ccccc2)n1NC(=O)c1ccccc1)c1ccccc1 50418640OC(=O)CCNc1sc2CCCCc2c1Cc1nnc(SCSc2nnc(Cc3c(NCCC(O)=O)sc4CCCCc34)n2NC(=O)c2ccccc2)n1NC(=O)c1ccccc1 50418641CC(=O)Nn1c(Cc2c(NC(=O)CCl)sc3CCCCc23)nnc1SCSc1nnc(Cc2c(NC(=O)CCl)sc3CCCCc23)n1NC(C)=O 50418642CC(=O)Nc1sc2CCCCc2c1Cc1nnc(SCSc2nnc(Cc3c(NC(C)=O)sc4CCCCc34)n2NC(C)=O)n1NC(C)=O 50418643CC(=O)Nn1c(Cc2c(NC(=O)c3ccccc3)sc3CCCCc23)nnc1SCSc1nnc(Cc2c(NC(=O)c3ccccc3)sc3CCCCc23)n1NC(C)=O 50418644CC(=O)Nn1c(Cc2c(NCCC(O)=O)sc3CCCCc23)nnc1SCSc1nnc(Cc2c(NCCC(O)=O)sc3CCCCc23)n1NC(C)=O 50418645CC(=O)Nc1sc2CCCCc2c1CC(=O)NNC([S-])=S 50418646CC(=O)Nc1sc2CCCCc2c1Cc1nnc(SCC#N)n1NC(=O)c1ccc(Cl)cc1 50418647Clc1ccc(cc1)C(=O)Nn1c(Cc2c(NC(=O)c3ccccc3)sc3CCCCc23)nnc1SCC#N 50418648OC(=O)CCNc1sc2CCCCc2c1Cc1nnc(SCC#N)n1NC(=O)c1ccc(Cl)cc1 50418649ClCC(=O)Nc1sc2CCCCc2c1Cc1nnc(SCC#N)n1NC(=O)c1ccccc1 50418650CC(=O)Nc1sc2CCCCc2c1Cc1nnc(SCC#N)n1NC(=O)c1ccccc1 50418651O=C(Nc1sc2CCCCc2c1Cc1nnc(SCC#N)n1NC(=O)c1ccccc1)c1ccccc1 50418652OC(=O)CCNc1sc2CCCCc2c1Cc1nnc(SCC#N)n1NC(=O)c1ccccc1 50418653CC(=O)Nn1c(Cc2c(NC(=O)CCl)sc3CCCCc23)nnc1SCC#N 50418654CC(=O)Nc1sc2CCCCc2c1Cc1nnc(SCC#N)n1NC(C)=O 50418655CC(=O)Nn1c(Cc2c(NC(=O)c3ccccc3)sc3CCCCc23)nnc1SCC#N 50418656CC(=O)Nn1c(Cc2c(NCCC(O)=O)sc3CCCCc23)nnc1SCC#N 50418657COC(=O)CSc1nnc(Cc2c(NC(=O)CCl)sc3CCCCc23)n1NC(=O)c1ccc(Cl)cc1 50418658COC(=O)CSc1nnc(Cc2c(NC(C)=O)sc3CCCCc23)n1NC(=O)c1ccc(Cl)cc1 50418659COC(=O)CSc1nnc(Cc2c(NC(=O)c3ccccc3)sc3CCCCc23)n1NC(=O)c1ccc(Cl)cc1 50418660COC(=O)CSc1nnc(Cc2c3CCCCc3sc2NCCC(O)=O)n1NC(=O)c1ccc(Cl)cc1 50418661COC(=O)CSc1nnc(Cc2c(NC(=O)CCl)sc3CCCCc23)n1NC(=O)c1ccccc1 50418662COC(=O)CSc1nnc(Cc2c(NC(C)=O)sc3CCCCc23)n1NC(=O)c1ccccc1 50418663COC(=O)CSc1nnc(Cc2c(NCCC(O)=O)sc3CCCCc23)n1NC(=O)c1ccccc1 50418664COC(=O)CSc1nnc(Cc2c(NC(=O)CCl)sc3CCCCc23)n1NC(C)=O 50418665COC(=O)CSc1nnc(Cc2c(NC(C)=O)sc3CCCCc23)n1NC(C)=O 50418666COC(=O)CSc1nnc(Cc2c(NC(=O)c3ccccc3)sc3CCCCc23)n1NC(C)=O 50418667COC(=O)CSc1nnc(Cc2c(NCCC(O)=O)sc3CCCCc23)n1NC(C)=O 50418668NNC(=O)CSc1nnc(Cc2c(NC(=O)CCl)sc3CCCCc23)n1NC(=O)c1ccc(Cl)cc1 50418669CC(=O)Nc1sc2CCCCc2c1Cc1nnc(SCC(=O)NN)n1NC(=O)c1ccc(Cl)cc1 50418670NNC(=O)CSc1nnc(Cc2c(NC(=O)c3ccccc3)sc3CCCCc23)n1NC(=O)c1ccc(Cl)cc1 50418671NNC(=O)CSc1nnc(Cc2c(NC(=O)CCl)sc3CCCCc23)n1NC(=O)c1ccccc1 50418672CC(=O)Nc1sc2CCCCc2c1Cc1nnc(SCC(=O)NN)n1NC(=O)c1ccccc1 50418673NNC(=O)CSc1nnc(Cc2c(NC(=O)c3ccccc3)sc3CCCCc23)n1NC(=O)c1ccccc1 50418674NNC(=O)CSc1nnc(Cc2c(NCCC(O)=O)sc3CCCCc23)n1NC(=O)c1ccccc1 50418675CC(=O)Nn1c(Cc2c3CCCCc3sc2NC(=O)CCl)nnc1SCC(=O)NN 50418676CC(=O)Nc1sc2CCCCc2c1Cc1nnc(SCC(=O)NN)n1NC(C)=O 50418677CC(=O)Nn1c(Cc2c(NC(=O)c3ccccc3)sc3CCCCc23)nnc1SCC(=O)NN 50418678CC(=O)Nn1c(Cc2c3CCCCc3sc2NCCC(O)=O)nnc1SCC(=O)NN 50418679CC(=O)NNC(=O)CSc1nnc(Cc2c(NC(=O)c3ccccc3)sc3CCCCc23)n1NC(C)=O 50418680CC(=O)NNC(=O)CSc1nnc(Cc2c(NCCC(O)=O)sc3CCCCc23)n1NC(C)=O 50418681CC(=O)Nn1c(Cc2c(NC(=O)CCl)sc3CCCCc23)nnc1SCC(=O)NNC(=O)c1ccccc1 50418682CC(=O)Nc1sc2CCCCc2c1Cc1nnc(SCC(=O)NNC(=O)c2ccccc2)n1NC(C)=O 50418683CC(=O)Nn1c(Cc2c(NC(=O)c3ccccc3)sc3CCCCc23)nnc1SCC(=O)NNC(=O)c1ccccc1 50418684CC(=O)Nn1c(Cc2c(NCCC(O)=O)sc3CCCCc23)nnc1SCC(=O)NNC(=O)c1ccccc1 50418685CC(=O)Nn1c(Cc2c(NC(=O)CCl)sc3CCCCc23)nnc1SCC(=O)NNC(=O)CCl 50418686CC(=O)Nc1sc2CCCCc2c1Cc1nnc(SCC(=O)NNC(=O)CCl)n1NC(C)=O 50418687CC(=O)Nn1c(Cc2c(NC(=O)c3ccccc3)sc3CCCCc23)nnc1SCC(=O)NNC(=O)CCl 50418688CC(=O)Nn1c(Cc2c3CCCCc3sc2NCCC(O)=O)nnc1SCC(=O)NNC(=O)CCl 50418689CC(=O)NNC(=O)CSc1nnc(Cc2c(NC(=O)c3ccccc3)sc3CCCCc23)n1NC(=O)c1ccc(Cl)cc1 50418690CC(=O)NNC(=O)CSc1nnc(Cc2c3CCCCc3sc2NCCC(O)=O)n1NC(=O)c1ccc(Cl)cc1 50418691ClCC(=O)Nc1sc2CCCCc2c1Cc1nnc(SCC(=O)NNC(=O)c2ccccc2)n1NC(=O)c1ccc(Cl)cc1 50418692CC(=O)Nc1sc2CCCCc2c1Cc1nnc(SCC(=O)NNC(=O)c2ccccc2)n1NC(=O)c1ccc(Cl)cc1 50418693Clc1ccc(cc1)C(=O)Nn1c(Cc2c(NC(=O)c3ccccc3)sc3CCCCc23)nnc1SCC(=O)NNC(=O)c1ccccc1 50418694OC(=O)CCNc1sc2CCCCc2c1Cc1nnc(SCC(=O)NNC(=O)c2ccccc2)n1NC(=O)c1ccc(Cl)cc1 50418695ClCC(=O)NNC(=O)CSc1nnc(Cc2c(NC(=O)CCl)sc3CCCCc23)n1NC(=O)c1ccc(Cl)cc1 50418696ClCC(=O)NNC(=O)CSc1nnc(Cc2c(NC(=O)c3ccccc3)sc3CCCCc23)n1NC(=O)c1ccc(Cl)cc1 50418697OC(=O)CCNc1sc2CCCCc2c1Cc1nnc(SCC(=O)NNC(=O)CCl)n1NC(=O)c1ccc(Cl)cc1 50418698CC(=O)NNC(=O)CSc1nnc(Cc2c(NC(=O)CCl)sc3CCCCc23)n1NC(=O)c1ccccc1 50418699CC(=O)NNC(=O)CSc1nnc(Cc2c(NC(C)=O)sc3CCCCc23)n1NC(=O)c1ccccc1 50418700CC(=O)NNC(=O)CSc1nnc(Cc2c(NC(=O)c3ccccc3)sc3CCCCc23)n1NC(=O)c1ccccc1 50418701CC(=O)NNC(=O)CSc1nnc(Cc2c(NCCC(O)=O)sc3CCCCc23)n1NC(=O)c1ccccc1 50418702ClCC(=O)Nc1sc2CCCCc2c1Cc1nnc(SCC(=O)NNC(=O)c2ccccc2)n1NC(=O)c1ccccc1 50418703CC(=O)Nc1sc2CCCCc2c1Cc1nnc(SCC(=O)NNC(=O)c2ccccc2)n1NC(=O)c1ccccc1 50418704O=C(CSc1nnc(Cc2c(NC(=O)c3ccccc3)sc3CCCCc23)n1NC(=O)c1ccccc1)NNC(=O)c1ccccc1 50418705OC(=O)CCNc1sc2CCCCc2c1Cc1nnc(SCC(=O)NNC(=O)c2ccccc2)n1NC(=O)c1ccccc1 50418706ClCC(=O)NNC(=O)CSc1nnc(Cc2c(NC(=O)CCl)sc3CCCCc23)n1NC(=O)c1ccccc1 50418707CC(=O)Nc1sc2CCCCc2c1Cc1nnc(SCC(=O)NNC(=O)CCl)n1NC(=O)c1ccccc1 50418708OC(=O)CCNc1sc2CCCCc2c1Cc1nnc(SCC(=O)NNC(=O)CCl)n1NC(=O)c1ccccc1 50418709CC(=O)NNC(=O)CSc1nnc(Cc2c(NC(=O)CCl)sc3CCCCc23)n1NC(C)=O 50418710CC(=O)NNC(=O)CSc1nnc(Cc2c(NC(C)=O)sc3CCCCc23)n1NC(C)=O 50418711ClCC(=O)Nc1sc2CCCCc2c1Cc1nnc(SCC(=O)NN=Cc2ccccc2)n1NC(=O)c1ccc(Cl)cc1 50418712Clc1ccc(cc1)C(=O)Nn1c(Cc2c3CCCCc3sc2NC(=O)c2ccccc2)nnc1SCC(=O)NN=Cc1ccccc1 50418713OC(=O)CCNc1sc2CCCCc2c1Cc1nnc(SCC(=O)NN=Cc2ccccc2)n1NC(=O)c1ccc(Cl)cc1 50418714ClCC(=O)Nc1sc2CCCCc2c1Cc1nnc(SCC(=O)NN=Cc2ccccc2)n1NC(=O)c1ccccc1 50418715CC(=O)Nc1sc2CCCCc2c1Cc1nnc(SCC(=O)NN=Cc2ccccc2)n1NC(=O)c1ccccc1 50418716O=C(CSc1nnc(Cc2c3CCCCc3sc2NC(=O)c2ccccc2)n1NC(=O)c1ccccc1)NN=Cc1ccccc1 50418717OC(=O)CCNc1sc2CCCCc2c1Cc1nnc(SCC(=O)NN=Cc2ccccc2)n1NC(=O)c1ccccc1 50418718CC(=O)Nn1c(Cc2c(NC(=O)CCl)sc3CCCCc23)nnc1SCC(=O)NN=Cc1ccccc1 50418719CC(=O)Nc1sc2CCCCc2c1Cc1nnc(SCC(=O)NN=Cc2ccccc2)n1NC(C)=O 50418720CC(=O)Nn1c(Cc2c3CCCCc3sc2NC(=O)c2ccccc2)nnc1SCC(=O)NN=Cc1ccccc1 50418721CC(=O)Nn1c(Cc2c(NCCC(O)=O)sc3CCCCc23)nnc1SCC(=O)NN=Cc1ccccc1 50418722Nn1c(CSc2nnc(Cc3c4CCCCc4sc3NC(=O)CCl)n2NC(=O)c2ccc(Cl)cc2)n[nH]c1=S 50418723CC(=O)Nc1sc2CCCCc2c1Cc1nnc(SCc2n[nH]c(=S)n2N)n1NC(=O)c1ccc(Cl)cc1 50418724Nn1c(CSc2nnc(Cc3c4CCCCc4sc3NC(=O)c3ccccc3)n2NC(=O)c2ccc(Cl)cc2)n[nH]c1=S 50418725Nn1c(CSc2nnc(Cc3c(NCCC(O)=O)sc4CCCCc34)n2NC(=O)c2ccc(Cl)cc2)n[nH]c1=S 50418726CC(=O)Nc1sc2CCCCc2c1Cc1nnc(SCc2n[nH]c(=S)n2N)n1NC(=O)c1ccccc1 50418727Nn1c(CSc2nnc(Cc3c(NC(=O)c4ccccc4)sc4CCCCc34)n2NC(=O)c2ccccc2)n[nH]c1=S 50418728Nn1c(CSc2nnc(Cc3c4CCCCc4sc3NCCC(O)=O)n2NC(=O)c2ccccc2)n[nH]c1=S 50418729CC(=O)Nc1sc2CCCCc2c1Cc1nnc(SCc2n[nH]c(=S)n2N)n1NC(C)=O 50418730CC(=O)Nn1c(Cc2c3CCCCc3sc2NC(=O)c2ccccc2)nnc1SCc1n[nH]c(=S)n1N 50418731CC(=O)Nn1c(Cc2c(NCCC(O)=O)sc3CCCCc23)nnc1SCc1n[nH]c(=S)n1N 50418732CC(=O)Nc1sc2CCCCc2c1Cc1nnc(SCSc2nnc(Cc3c(NC(C)=O)sc4CCCCc34)n2NC(=O)c2ccc(Cl)cc2)n1NC(=O)c1ccc(Cl)cc1 50418733ClCC(=O)Nc1sc2CCCCc2c1Cc1nnc(SCSc2nnc(Cc3c(NC(=O)CCl)sc4CCCCc34)n2NC(=O)c2ccc(Cl)cc2)n1NC(=O)c1ccc(Cl)cc1 50418734ClCC(=O)Nc1sc2CCCCc2c1Cc1nnc(SCC#N)n1NC(=O)c1ccc(Cl)cc1 50418735COC(=O)CSc1nnc(Cc2c(NC(=O)c3ccccc3)sc3CCCCc23)n1NC(=O)c1ccccc1 50418736CC(=O)NNC(=O)CSc1nnc(Cc2c(NC(=O)CCl)sc3CCCCc23)n1NC(=O)c1ccc(Cl)cc1 50418737CC(=O)Nc1sc2CCCCc2c1Cc1nnc(SCC(=O)NNC(=O)CCl)n1NC(=O)c1ccc(Cl)cc1 50418738CC(=O)Nc1sc2CCCCc2c1Cc1nnc(SCC(=O)NN=Cc2ccccc2)n1NC(=O)c1ccc(Cl)cc1 50418739CC(=O)Nn1c(Cc2c(NC(=O)CCl)sc3CCCCc23)nnc1SCc1n[nH]c(=S)n1N 50418740NNC(=O)CSc1nnc(Cc2c3CCCCc3sc2NCCC(O)=O)n1NC(=O)c1ccc(Cl)cc1 50418741CC(=O)NNC(=O)CSc1nnc(Cc2c(NC(C)=O)sc3CCCCc23)n1NC(=O)c1ccc(Cl)cc1 50418742ClCC(=O)NNC(=O)CSc1nnc(Cc2c(NC(=O)c3ccccc3)sc3CCCCc23)n1NC(=O)c1ccccc1 50418743Nn1c(CSc2nnc(Cc3c4CCCCc4sc3NC(=O)CCl)n2NC(=O)c2ccccc2)n[nH]c1=S 50418744[S-]C(=S)NNC(=O)Cc1c(NC(=O)CCl)sc2CCCCc12 50420297CC(C)n1cnc2c(NCc3ccc(cc3)-c3ccccn3)nc(NC[C@@H](O)CO)nc12 50420298CC(C)n1cnc2c(NCc3ccc(cc3)-c3ccccn3)nc(N[C@@H]3CCC[C@H](O)[C@@H]3O)nc12 50420299CC(C)n1cnc2c(NCc3ccc(cc3)-c3ccccn3)nc(nc12)N1C[C@H](O)C[C@H]1CO 50420300CC(C)n1cnc2c(NCc3ccc(cc3)-c3ccccn3)nc(NCC[C@H](O)CO)nc12 50420301CC(C)[C@H](N)C(=O)OC[C@H](O)CNc1nc(NCc2ccc(cc2)-c2ccccn2)c2ncn(C(C)C)c2n1 50423711O[N-]c1c([nH]c2ccccc12)C1=c2ccc(cc2=[NH+]C1=O)[N+]([O-])=O 50423712Nc1ccc2C(C(=O)Nc2c1)c1[nH]c2ccccc2c1N=O 50423713O[N-]c1c([nH]c2ccc(Br)cc12)C1=c2ccc(cc2=[NH+]C1=O)[N+]([O-])=O 50423714Nc1ccc2C(C(=O)Nc2c1)=C1Nc2ccccc2C1=O 50423773C[C@]12O[C@@H](C[C@@]1(O)CO)n1c3ccccc3c3c4C(=O)NCc4c4c5ccccc5n2c4c13 50424255CC[C@@H](CO)Nc1nc(Nc2ccncn2)c2ncn(C(C)C)c2n1 50424256CC[C@H](CO)Nc1nc(Nc2ccncn2)c2ncn(C(C)C)c2n1 50424263CC(C)[C@@H](CO)Nc1nc(Nc2ccncc2)c2ncn(C(C)C)c2n1 50424264CC(C)[C@H](CO)Nc1nc(Nc2ccncc2)c2ncn(C(C)C)c2n1 50424265CC[C@@H](CO)Nc1nc(Nc2ccncc2)c2ncn(C(C)C)c2n1 50424266CC[C@H](CO)Nc1nc(Nc2ccncc2)c2ncn(C(C)C)c2n1 50424267CC(C)n1cnc2c(Nc3ccncc3)nc(Cl)nc12 50424268CC(C)n1c(nc2c(Nc3cccnc3)ncnc12)C(CO)CO 50424269CC(C)[C@@H](CO)Nc1nc(Nc2cccnc2)c2ncn(C(C)C)c2n1 50424270CC(C)[C@H](CO)Nc1nc(Nc2cccnc2)c2ncn(C(C)C)c2n1 50424271CC[C@@H](CO)Nc1nc(Nc2cccnc2)c2ncn(C(C)C)c2n1 50424272CC[C@H](CO)Nc1nc(Nc2cccnc2)c2ncn(C(C)C)c2n1 50424273CC(C)n1cnc2c(Nc3cccnc3)nc(Cl)nc12 50424274CC(C)[C@@H](CO)Nc1nc(Nc2ccccn2)c2ncn(C(C)C)c2n1 50424275CC(C)[C@H](CO)Nc1nc(Nc2ccccn2)c2ncn(C(C)C)c2n1 50424276CC[C@@H](CO)Nc1nc(Nc2ccccn2)c2ncn(C(C)C)c2n1 50424277CC[C@H](CO)Nc1nc(Nc2ccccn2)c2ncn(C(C)C)c2n1 50424278CC(C)n1cnc2c(Nc3ccccn3)nc(Cl)nc12 50424279CC(C)n1cnc2c(Nc3ccnnc3)nc(nc12)C(C)(C)CO 50424280CC(C)n1c(nc2c(Nc3ccnnc3)ncnc12)C(CO)CO 50424281CC(C)[C@@H](CO)Nc1nc(Nc2ccnnc2)c2ncn(C(C)C)c2n1 50424282CC(C)[C@H](CO)Nc1nc(Nc2ccnnc2)c2ncn(C(C)C)c2n1 50424283CC[C@@H](CO)Nc1nc(Nc2ccnnc2)c2ncn(C(C)C)c2n1 50424284CC[C@H](CO)Nc1nc(Nc2ccnnc2)c2ncn(C(C)C)c2n1 50424285CC(C)n1cnc2c(Nc3ccnnc3)nc(Cl)nc12 50424287CC(C)n1c(Nc2cncc(n2)C(C)(C)CO)nc2cncnc12 50424288CC(C)[C@H](CO)Nc1cncc(Nc2nc3cncnc3n2C(C)C)n1 50424289CC[C@H](CO)Nc1cncc(Nc2nc3cncnc3n2C(C)C)n1 50424291CC(C)n1c(nc2c(Nc3cncnc3)ncnc12)C(CO)CO 50424292CC(C)n1cnc2c(Nc3cncnc3)nc(nc12)C(C)(C)CO 50424293CC(C)[C@@H](CO)Nc1nc(Nc2cncnc2)c2ncn(C(C)C)c2n1 50424294CC(C)[C@H](CO)Nc1nc(Nc2cncnc2)c2ncn(C(C)C)c2n1 50424295CC[C@@H](CO)Nc1nc(Nc2cncnc2)c2ncn(C(C)C)c2n1 50424296CC[C@H](CO)Nc1nc(Nc2cncnc2)c2ncn(C(C)C)c2n1 50424297CC(C)n1cnc2c(Nc3cncnc3)nc(Nc3cncnc3)nc12 50424298CC(C)n1cnc2c(Nc3cncnc3)nc(Cl)nc12 50424299CC(C)n1cnc2c(Nc3ccncn3)nc(nc12)C(C)(C)CO 50424300CC(C)n1c(nc2c(Nc3ccncn3)ncnc12)C(CO)CO 50424301CC(C)[C@@H](CO)Nc1nc(Nc2ccncn2)c2ncn(C(C)C)c2n1 50424302CC(C)[C@H](CO)Nc1nc(Nc2ccncn2)c2ncn(C(C)C)c2n1 50426312COC(=O)c1ccc2[nH]c(C3C(=O)Nc4ccccc34)c(N=O)c2c1 50426313OC(=O)c1ccc2c(N=O)c([nH]c2c1)C1C(=O)Nc2ccccc12 50426314OC(=O)c1ccc2N\C(C(=O)c2c1)=C1/C(=O)Nc2ccccc12 50426316OC(=O)c1ccc2c(N=O)c([nH]c2c1)C1C(=O)Nc2c1cccc2C(F)(F)F 50426331Brc1cccc2C(C(=O)Nc12)c1[nH]c2ccc(CN=O)cc2c1N=O 50426332OCc1ccc2[nH]c(C3C(=O)Nc4c3cccc4Br)c(N=O)c2c1 50426334Brc1cccc2C(C(=O)Nc12)=C1Nc2ccc(CN=O)cc2C1=O 50426335OC(=O)c1ccc2[nH]c(C3C(=O)Nc4c3cccc4C(F)(F)F)c(N=O)c2c1 50426336OC(=O)c1ccc2[nH]c(C3C(=O)Nc4ccccc34)c(N=O)c2c1 50426338CN1C(=O)C(c2cccc(Br)c12)c1[nH]c2ccc(cc2c1N=O)C(O)=O 50426339COC(=O)c1ccc2c(N=O)c([nH]c2c1)C1C(=O)Nc2c1cccc2C(F)(F)F 50431282CC[C@H](CO)Nc1nc(NCc2cc(F)ccc2O)c2ncn(C(C)C)c2n1 50431283CC[C@@H](Nc1nc(NCc2cc(F)ccc2O)c2ncn(C(C)C)c2n1)C(C)O 50431284CC[C@@H](Nc1nc(NCc2cc(Cl)ccc2O)c2ncn(C(C)C)c2n1)C(C)O 50431285CC[C@H](CO)Nc1nc(NCc2cc(Cl)ccc2O)c2ncn(C(C)C)c2n1 50431286CC(C)n1cnc2c(NCc3cc(Cl)ccc3O)nc(NC3CCC(N)CC3)nc12 50431287CC(C)n1cnc2c(NCc3cc(Cl)ccc3O)nc(NC3CCC(O)CC3)nc12 50431288CC(C)CNc1nc(NCc2ccccc2O)c2ncn(C(C)C)c2n1 50431289CC(C)n1cnc2c(NCc3ccccc3O)nc(NCCC(C)(C)O)nc12 50431290CC(C)[C@H](Nc1nc(NCc2ccccc2N)c2ncn(C(C)C)c2n1)C(C)(C)O 50431292CC(C)n1cnc2c(NCc3ccccc3N)nc(NCC(C)(C)O)nc12 50431293CC(C)n1cnc2c(NCc3cc(Cl)ccc3O)nc(NCC(C)(C)O)nc12 50433369Nc1nc(Nc2ccc(cc2)S(N)(=O)=O)sc1C(=O)c1ccccc1[N+]([O-])=O 50437236NC1CCC(CC1)Nc1nc(NCc2ccc(nc2)-c2ccccc2O)c2ncn(C3CCCC3)c2n1 50439491Oc1cc2O\C(=C/c3ccc(O)c(O)c3)C(=O)c2c(O)c1 50440135COc1ccc(NC(=S)NC(=O)c2cn(nc2-c2ccc(OC)cc2)-c2ccccc2)cc1 50440136COc1ccc(NC(=S)NC(=O)c2cn(nc2-c2ccc(F)cc2)-c2ccccc2)cc1 50440137COc1ccc(NC(=S)NC(=O)c2cn(nc2-c2ccc(Cl)cc2)-c2ccccc2)cc1 50440138COc1ccc(NC(=S)NC(=O)c2cn(nc2-c2ccc(C)cc2)-c2ccccc2)cc1 50440139COc1ccc(NC(=S)NC(=O)c2cn(nc2-c2ccccc2)-c2ccccc2)cc1 50440393COc1cc(C)c(cc1O)-c1c2c(n3ccc4cc(O)c(OC)cc4c13)c(=O)oc1cc(O)c(OC)cc21 50440473Nc1nc(Nc2ccc(cc2)S(=O)(=O)NCCO)nc(OCC2CCCCC2)c1[N+](=O)[N-]C#N 50440474CNS(=O)(=O)c1ccc(Nc2nc(N)c(c(OCC3CCCCC3)n2)[N+](=O)[N-]C#N)cc1