14359OC(c1cnc(s1)[C@@H](Cc1ccc[n+]([O-])c1)c1ccc(OC(F)F)c(OC2CC2)c1)(C(F)(F)F)C(F)(F)F 14360OC(c1cnc(s1)[C@H](Cc1ccc[n+]([O-])c1)c1ccc(OC(F)F)c(OC2CC2)c1)(C(F)(F)F)C(F)(F)F 14361COc1ccc(cc1OC1CCCC1)C1CNC(=O)C1 14364CCNc1ncn(Cc2ccc(OC)c(OC3CCCC3)c2)c2nc(nc12)C(C)C 14365COc1ccc(Cn2cnc(N)c3nc(nc23)C(C)(C)OCc2ccccc2)cc1OC1CCCC1 14366COc1ccccc1COC(C)(C)c1nc2c(N)ncn(Cc3ccc(OC)c(OC4CCCC4)c3)c2n1 14367COc1cccc(COC(C)(C)c2nc3c(N)ncn(Cc4ccc(OC)c(OC5CCCC5)c4)c3n2)c1 14368COc1ccc(COC(C)(C)c2nc3c(N)ncn(Cc4ccc(OC)c(OC5CCCC5)c4)c3n2)cc1 14369COc1ccc(Cn2cnc(N)c3nc(nc23)C(C)(C)OCc2ccc(C)cc2)cc1OC1CCCC1 14370COc1ccc(Cn2cnc(N)c3nc(nc23)C(C)(C)OCc2ccc(Cl)cc2)cc1OC1CCCC1 14371COc1ccc(Cn2cnc(N)c3nc(nc23)C(C)(C)OCc2ccccc2F)cc1OC1CCCC1 14372COc1ccc(Cn2cnc(N)c3nc(nc23)C(C)(C)OCc2cccc(F)c2)cc1OC1CCCC1 14373COc1ccc(COC(C)(C)c2nc3c(N)ncn(Cc4ccc(OC)c(OC5CCCC5)c4)c3n2)cc1OC 14374COc1cc(COC(C)(C)c2nc3c(N)ncn(Cc4ccc(OC)c(OC5CCCC5)c4)c3n2)cc(OC)c1 14375COc1ccc(Cn2cnc(N)c3nc(nc23)C(C)(C)OCc2ccc(F)c(F)c2)cc1OC1CCCC1 14376COc1ccc(Cn2cnc(N)c3nc(nc23)C(C)(C)OCc2ccc3OCOc3c2)cc1OC1CCCC1 14377COc1ccc(Cn2cnc(N)c3nc(nc23)C(C)(C)OCc2ccc(cc2)C#N)cc1OC1CCCC1 14378COc1ccc(Cn2cnc(N)c3nc(nc23)C(C)(C)OCc2ccc(Cl)c(Cl)c2)cc1OC1CCCC1 14379COc1ccc(Cn2cnc(N)c3nc(nc23)C(C)(C)OCc2ccc(cc2)C(C)(C)C)cc1OC1CCCC1 14380COc1ccc(Cn2cnc(N)c3nc(nc23)C(C)(C)OCc2ccc(OC(F)(F)F)cc2)cc1OC1CCCC1 14381COC(=O)c1ccc(COC(C)(C)c2nc3c(N)ncn(Cc4ccc(OC)c(OC5CCCC5)c4)c3n2)cc1 14382COc1ccc(Cn2cnc(N)c3nc(nc23)C(C)(C)OCc2ccc(cc2)C(N)=O)cc1OC1CCCC1 14384COc1ccc(Cn2cnc(N)c3nc(nc23)C(C)(C)OCc2ccc(cc2)C(F)(F)F)cc1OC1CCCC1 14385COc1ccc(Cn2cnc(N)c3nc(nc23)C(C)(C)COc2cccs2)cc1OC1CCCC1 14386COc1ccc(Cn2cnc(N)c3nc(nc23)C(C)(C)COc2ccsc2)cc1OC1CCCC1 14387COc1ccc(Cn2cnc(N)c3nc(nc23)C(C)OCc2ccccc2)cc1OC1CCCC1 14388COc1ccc(COC(C)c2nc3c(N)ncn(Cc4ccc(OC)c(OC5CCCC5)c4)c3n2)cc1 14389COc1ccc(Cn2cnc(N)c3nc(nc23)C(C)OCc2ccc(F)cc2)cc1OC1CCCC1 14769COc1cc(ccc1OC(F)F)-c1ccc(=O)[nH]n1 14771COc1ccc(cc1OC1CCCC1)C(C)=NOC(N)=O 14772CCCOc1cc(ccc1OC)C1(C)CNC(=O)O1 14773COc1ccc(cc1OC1CCCC1)C1(CCC(CC1)C(O)=O)C#N 14774FC(F)Oc1ccc(cc1OCC1CC1)C(=O)Nc1c(Cl)cncc1Cl 14775COc1ccc(cc1OC1CCCC1)C(=O)Nc1c(Cl)cncc1Cl 14776CCCc1nc(C)c2n1nc([nH]c2=O)-c1cc(ccc1OCC)S(=O)(=O)N1CCN(CC)CC1 14777[H][C@]12Cc3c([nH]c4ccccc34)[C@H](N1C(=O)CN(C)C2=O)c1ccc2OCOc2c1 14785CCOC(=O)c1c(C)nn(c1C)-c1ccccc1 14786CCOC(=O)c1cn(nc1-c1ccc(Cl)cc1)-c1ccccc1 14794CCOC(=O)c1c(C)nn(c1C)-c1ccc(OC)cc1 14795CCOC(=O)c1c(C)nn(c1C)-c1ccc(cc1)[N+]([O-])=O 14796CCOC(=O)c1c(C)nn(c1C)-c1ccc(N)cc1 14797CCOC(=O)c1c(C)nn(c1C)-c1ccccc1Cl 14798CCOC(=O)c1c(C)nn(c1C)-c1cccc(c1)[N+]([O-])=O 30126COc1ccc(cc1OC)C1=NNC(=O)C2CC=CCC12 30128COc1ccc(F)c(CCC2CCC(CCNCCCCCN3N=C(C4CC=CCC4C3=O)c3ccc(OC)c(OC)c3)O2)c1 30129COc1ccc(F)c(CCCC2CCC(CCNCCCCCN3N=C(C4CC=CCC4C3=O)c3ccc(OC)c(OC)c3)O2)c1 31636CC(C)(C)C1CCc2c(C1)sc(NC(=O)c1ccncc1)c2C(N)=O 31637CC1CCc2c(C1)sc(NC(=O)c1ccccc1[N+]([O-])=O)c2C(N)=O 31638CC(C)(C)C1CCc2c(C1)sc(NC(=O)c1c(F)cccc1F)c2C(N)=O 31640CC1CCc2c(C1)sc(NC(=O)c1cccc(c1)[N+]([O-])=O)c2C(N)=O 31642NC(=O)c1c(NC(=O)c2ccccc2[N+]([O-])=O)sc2CCCCc12 31643CC1CCCc2sc(NC(=O)c3ccccc3[N+]([O-])=O)c(C(N)=O)c12 31644CC1(C)CCc2c(C1)sc(NC(=O)c1ccccc1[N+]([O-])=O)c2C(N)=O 31645CC1CCc2sc(NC(=O)c3ccccc3[N+]([O-])=O)c(C(N)=O)c2C1 31646CC(C)(C)C1CCc2sc(NC(=O)c3ccccc3[N+]([O-])=O)c(C(N)=O)c2C1 31647CCC1CCc2c(C1)sc(NC(=O)c1ccccc1[N+]([O-])=O)c2C(N)=O 31648CC(C)(C)C1CCc2c(C1)sc(NC(=O)c1ccccc1[N+]([O-])=O)c2C(N)=O 31649CCCC1CCc2c(C1)sc(NC(=O)c1ccccc1[N+]([O-])=O)c2C(N)=O 31650NC(=O)c1c(NC(=O)c2ccccc2[N+]([O-])=O)sc2CC(CCc12)c1ccccc1 31651Cc1cccc(C)c1C(=O)C1CCCc2sc(NC(=O)c3ccccc3[N+]([O-])=O)c(C(N)=O)c12 53163Cc1cccc(NNC2=c3cc(Br)ccc3=NC2=O)c1 50010981CCCCOc1cc(CC2CNC(=O)N2)ccc1OC 50017294C[C@H]1CN(Cc2ccc(c(CN3CCOCC3)c2)-c2cccc(Oc3ncc(F)cc3C(=O)N[C@@H]3CC[C@@H](CC3)NC(=O)c3nc(C)cs3)c2)C[C@@H](C)N1 50017295C[C@H]1CN(Cc2ccc(c(CN3CCOCC3)c2)-c2cccc(Oc3ncc(F)cc3C(=O)N[C@@H]3CC[C@@H](CC3)NC(=O)c3cc(C)ccc3O)c2)C[C@@H](C)N1 50017296Cc1cc(nn1C)C(=O)N[C@H]1CC[C@H](CC1)NC(=O)c1cc(F)cnc1Oc1cccc(c1)-c1ccc(O)cc1CN1CCOCC1 50017297Cc1cccc2nc(cn12)C(=O)N[C@H]1CC[C@H](CC1)NC(=O)c1cc(F)cnc1Oc1cccc(c1)-c1ccc(CN2CCC(CC2)N2CCCC2)cc1 50017298C[C@H]1CN(Cc2ccc(cc2)-c2cccc(Oc3ncc(F)cc3C(=O)N[C@@H]3CC[C@@H](CC3)NC(=O)c3cc4ccccn4n3)c2)C[C@@H](C)N1 50017299C[C@H]1CN(Cc2ccc(cc2)-c2cccc(Oc3ncc(F)cc3C(=O)N[C@@H]3CC[C@@H](CC3)NC(=O)c3cn4c(C)cccc4n3)c2)C[C@@H](C)N1 50017300Cc1cc(nn1C)C(=O)N[C@H]1CC[C@H](CC1)NC(=O)c1cc(F)cnc1Oc1cccc(c1)-c1ccc(O)cc1CN1CCCOCC1 50017301Cc1nc(cs1)C(=O)N[C@H]1CC[C@H](CC1)NC(=O)c1cc(F)cnc1Oc1cccc(c1)-c1ccc(O)cc1CN1CCOCC1 50017302CN(C)Cc1cc(O)ccc1-c1cccc(Oc2ncc(F)cc2C(=O)N[C@@H]2CC[C@@H](CC2)NC(=O)c2csc(C)n2)c1 50017303Cc1nc(cs1)C(=O)N[C@H]1CC[C@H](CC1)NC(=O)c1cc(F)cnc1Oc1cccc(c1)-c1ccc(O)cc1CN1CCCOCC1 50017304Cc1csc(n1)C(=O)N[C@H]1CC[C@H](CC1)NC(=O)c1cc(F)cnc1Oc1cccc(c1)-c1ccc(O)cc1CN1CCOCC1 50017305OCc1nc(cs1)C(=O)N[C@H]1CC[C@H](CC1)NC(=O)c1cc(F)cnc1Oc1cccc(c1)-c1ccc(O)cc1CN1CCOCC1 50017306CN(C)Cc1cc(O)ccc1-c1cccc(Oc2ncc(F)cc2C(=O)N[C@@H]2CC[C@@H](CC2)NC(=O)c2cccc(C)n2)c1 50017307Cc1cccc(n1)C(=O)N[C@H]1CC[C@H](CC1)NC(=O)c1cc(F)cnc1Oc1cccc(c1)-c1ccc(O)cc1CN1CCCOCC1 50017308Cc1cccc2nc(cn12)C(=O)N[C@H]1CC[C@H](CC1)NC(=O)c1cc(F)cnc1Oc1cccc(c1)-c1ccc(O)cc1CN1CCOCC1 50017310CN(C)Cc1cc(O)ccc1-c1cccc(Oc2ncc(F)cc2C(=O)N[C@@H]2CC[C@@H](CC2)NC(=O)c2cn3c(C)cccc3n2)c1 50017311Cc1cccc2nc(cn12)C(=O)N[C@H]1CC[C@H](CC1)NC(=O)c1cc(F)cnc1Oc1cccc(c1)-c1ccc(O)cc1CN1CCCOCC1 50017312CN(C)Cc1cc(O)ccc1-c1cccc(Oc2ncc(F)cc2C(=O)N[C@@H]2CC[C@@H](CC2)NC(=O)c2cn3cc(F)ccc3n2)c1 50017313Oc1ccc(c(CN2CCCOCC2)c1)-c1cccc(Oc2ncc(F)cc2C(=O)N[C@@H]2CC[C@@H](CC2)NC(=O)c2cn3cc(F)ccc3n2)c1 50017314Cc1cccc(O)c1C(=O)N[C@@H]1CC[C@@H](CC1)NC(=O)c1cc(F)cnc1Oc1cccc(c1)-c1ccc(O)cc1CN1CCOCC1 50017315Cc1cccc(O)c1C(=O)N[C@@H]1CC[C@@H](CC1)NC(=O)c1cc(F)cnc1Oc1cccc(c1)-c1ccc(O)cc1CN1CCCOCC1 50017316Oc1ccc(c(CN2CCOCC2)c1)-c1cccc(Oc2ncc(F)cc2C(=O)N[C@H]2CC[C@H](CC2)NC(=O)c2nc3ccccc3[nH]c2=O)c1 50017317Oc1ccc(c(CN2CCOCC2)c1)-c1cccc(Oc2ncc(F)cc2C(=O)N[C@H]2CC[C@H](CC2)NC(=O)c2ncccc2O)c1 50017318Oc1ccc(c(CN2CCOCC2)c1)-c1cccc(Oc2ncc(F)cc2C(=O)N[C@@H]2CC[C@@H](CC2)NC(=O)c2cncc(O)c2)c1 50017319Cc1cc(C)n2ncc(C(=O)N[C@H]3CC[C@H](CC3)NC(=O)c3cc(F)cnc3Oc3cccc(c3)-c3ccc(O)cc3CN3CCOCC3)c2n1 50017321CN(C)Cc1cc(O)ccc1-c1cccc(Oc2ncc(F)cc2C(=O)N[C@H]2CC[C@H](CC2)NC(=O)c2cccc3[nH]cnc23)c1 50017322CN(C)Cc1cc(O)ccc1-c1cccc(Oc2ncc(F)cc2C(=O)N[C@H]2CC[C@H](CC2)NC(=O)c2cccc3ocnc23)c1 50017323CN(C)Cc1cc(O)ccc1-c1cccc(Oc2ncc(F)cc2C(=O)N[C@H]2CC[C@H](CC2)NC(=O)c2cccc3oc(=O)[nH]c23)c1 50017324C[C@H]1CN(Cc2ccc(cc2)-c2cccc(Oc3ncc(F)cc3C(=O)N[C@@H]3CC[C@@H](CC3)NC(=O)c3cc(C)n(C)n3)c2)C[C@@H](C)N1 50017325CN(C)Cc1ccc(cc1)-c1cccc(Oc2ncc(F)cc2C(=O)N[C@@H]2CC[C@@H](CC2)NC(=O)c2csc(C)n2)c1 50017326Cc1nc(cs1)C(=O)N[C@H]1CC[C@H](CC1)NC(=O)c1cc(F)cnc1Oc1cccc(c1)-c1ccc(CN2CCCOCC2)cc1 50017327C[C@H]1CN(Cc2ccc(cc2)-c2cccc(Oc3ncc(F)cc3C(=O)N[C@@H]3CC[C@@H](CC3)NC(=O)c3nc(C)cs3)c2)C[C@@H](C)N1 50017328C[C@H]1CN(Cc2ccc(cc2)-c2cccc(Oc3ncc(F)cc3C(=O)N[C@@H]3CC[C@@H](CC3)NC(=O)c3csc(CO)n3)c2)C[C@@H](C)N1 50017329CN(C)Cc1ccc(cc1)-c1cccc(Oc2ncc(F)cc2C(=O)N[C@@H]2CC[C@@H](CC2)NC(=O)c2cn3c(C)cccc3n2)c1 50017330Cc1cccc2nc(cn12)C(=O)N[C@H]1CC[C@H](CC1)NC(=O)c1cc(F)cnc1Oc1cccc(c1)-c1ccc(CN2CCCOCC2)cc1 50017331C[C@H]1CN(Cc2ccc(cc2)-c2cccc(Oc3ncc(F)cc3C(=O)N[C@@H]3CC[C@@H](CC3)NC(=O)c3cn4cc(F)ccc4n3)c2)C[C@@H](C)N1 50017332C[C@H]1CN(Cc2ccc(cc2)-c2cccc(Oc3ncc(F)cc3C(=O)N[C@H]3CC[C@H](CC3)NC(=O)c3ncccc3O)c2)C[C@@H](C)N1 50017333C[C@H]1CN(Cc2ccc(cc2O)-c2cccc(Oc3ncc(F)cc3C(=O)N[C@@H]3CC[C@@H](CC3)NC(=O)c3cc(C)n(C)n3)c2)C[C@@H](C)N1 50017334C[C@H]1CN(Cc2cccc(c2)-c2cccc(Oc3ncc(F)cc3C(=O)N[C@@H]3CC[C@@H](CC3)NC(=O)c3cc(C)n(C)n3)c2)C[C@@H](C)N1 50017335C[C@H]1CN(Cc2cc(ccc2O)-c2cccc(Oc3ncc(F)cc3C(=O)N[C@@H]3CC[C@@H](CC3)NC(=O)c3cc(C)n(C)n3)c2)C[C@@H](C)N1 50017336C[C@H]1CN(Cc2cc(O)cc(c2)-c2cccc(Oc3ncc(F)cc3C(=O)N[C@@H]3CC[C@@H](CC3)NC(=O)c3cc(C)n(C)n3)c2)C[C@@H](C)N1 50017337C[C@H]1CN(Cc2cccc(c2O)-c2cccc(Oc3ncc(F)cc3C(=O)N[C@@H]3CC[C@@H](CC3)NC(=O)c3cc(C)n(C)n3)c2)C[C@@H](C)N1 50017338C[C@H]1CN(CCCc2ccc(cc2)-c2cccc(Oc3ncc(F)cc3C(=O)N[C@@H]3CC[C@@H](CC3)NC(=O)c3cc(C)n(C)n3)c2)C[C@@H](C)N1 50017339Cc1cc(nn1C)C(=O)N[C@H]1CC[C@H](CC1)NC(=O)c1cc(F)cnc1Oc1cccc(c1)-c1ccc(CCN2CCC(CC2)N2CCCC2)cc1 50017340Cc1ccc(O)c(c1)C(=O)N[C@H]1CC[C@H](CC1)NC(=O)c1cc(F)cnc1Oc1ccc(F)c(F)c1 50029951COc1ccc(cc1OC1CCCC1)[C@H]1CCN2[C@@H]1COC2=O 50029952COc1ccc(cc1OC1CCCC1)[C@H]1CCN2[C@H]1CNC2=O 50029953COc1ccc(cc1OC1CCCC1)[C@H]1CCN2[C@H]1COC2=O 50029954COc1ccc(cc1OC1CCCC1)[C@H]1CCN2[C@@H]1CNC2=O 50029955COc1ccc(cc1OC1CCCC1)[C@H]1CCN2[C@@H]1CCC2=O 50029956COc1ccc(CC2CNC(=O)N2)cc1OC1CCCC1 50029957COc1ccc(cc1OC1CCCC1)[C@H]1CCN2[C@H]1CCC2=O 50042058COc1ccc(cc1OC1CCCC1)[C@@H]1CNC(=O)C1 50048243COC(=O)[C@@H]1CN(C[C@H]1c1ccc(OC)c(OC2CCCC2)c1)C(=O)OC 50048245CCOC(=O)[C@@H]1CN(C[C@H]1c1ccc(OC)c(OC2CCCC2)c1)C(=O)OC 50048248COC(=O)N1C[C@H]([C@@H](C1)c1ccc(OC)c(OC2CCCC2)c1)C(C)=O 50062379COc1ccc(cc1OC1CCCC1)C(=O)NC(C)C(=O)NO 50062381COc1ccc(cc1OC1CCCC1)C1=NOC(C)(C1)C(=O)NO 50062383COc1ccc(cc1OC1CCCC1)C(=O)NCC(=O)NO 50062387COc1ccc(cc1OC1CCCC1)C1=NOC(C1)C(=O)NO 50064858COc1ccc(cc1OC1CCCC1)[C@H](Cc1ccncc1)c1ccccc1 50085135OC(=O)c1ccc(cc1)-c1cc2cccnc2c(n1)-c1cccc(c1)[N+]([O-])=O 50092350COc1ccc2c(Nc3c(Cl)cncc3Cl)nncc2c1OC1CCCC1 50098221CCCCNc1c(cnc2n(CC)ncc12)C(=O)OCC 50106185O=c1[nH]ncc2ccccc12 50108504OC(=O)c1ccc(cc1)-c1cc2cccnc2c(n1)-c1ccc2nonc2c1 50110029COc1ccc(cc1OC1CCOC1)C(C)Cn1cc[nH]c1=O 50110030COc1ccc(cc1OC1Cc2ccccc2C1)C(C)Cn1ccnc1NC#N 50110031COc1ccc(cc1OC1Cc2ccccc2C1)C(O)Cn1cc[nH]c1=O 50110032COc1ccc(cc1OC1CCCC1)C(C)C(C)n1cc[nH]c1=O 50110033COc1ccc(cc1OCCC1Cc2ccccc2C1)C(C)Cn1ccnc1NC#N 50110034CC(Cn1ccnc1NC#N)c1ccc(OC(F)F)c(OCCCCCc2ccccc2)c1 50110035COc1ccc(cc1OCC1CC1)C(C)Cn1ccnc1NC#N 50110036COc1ccc(CCn2cc[nH]c2=O)cc1OC1CCCC1 50110037COc1ccc(cc1OC1CCCC1)C(C)Cn1ccnc1NC#N 50110038COc1ccc(cc1OC1Cc2ccccc2C1)C(F)Cn1cc[nH]c1=O 50110039COc1ccc(cc1OCC1CC1)C(C)Cn1cc[nH]c1=O 50110040COc1ccc(cc1OC1CCCC1)C(C)Cn1cc[nH]c1=O 50110041COc1ccc(cc1OC1CCCC1)C1(Cn2cc[nH]c2=O)CC1 50110043COc1ccc(cc1OC1CCCC1)C(C)(C)Cn1cc[nH]c1=O 50110044COc1ccc(cc1OC1CCCC1)C(=O)Cn1cc[nH]c1=O 50110045COc1ccc(cc1OC1CCOC1)C(C)Cn1ccnc1NC#N 50110046CC(Cn1ccnc1NC#N)c1ccc(OC(F)F)c(OCC2CC2)c1 50110047FC(F)Oc1ccc(cc1OC1CCCC1)C1(Cn2cc[nH]c2=O)CC1 50110048COc1ccc(cc1OC1CCOC1)C(C)(F)Cn1cc[nH]c1=O 50110051COc1ccc(cc1OCCCCCc1ccccc1)C(C)Cn1ccnc1NC#N 50110052COc1ccc(cc1OC1CC2CCC1C2)C(C)Cn1cc[nH]c1=O 50114418COc1ccc(C(=O)Nc2c(Cl)cncc2Cl)c2ccc(nc12)C(F)(F)F 50174013CC(C)c1cc(-c2cccc(\C=C(\C(O)=O)c3ccc(cc3)S(C)(=O)=O)c2)c2ncccc2c1 50174014CC(C)c1cc(-c2cccc(CC(c3ccncc3)C(C)(C)O)c2)c2ncccc2c1 50174015CC(C)NC(=O)C(=C\c1cccc(c1)-c1cc(cc2cccnc12)C(C)(C)S(C)(=O)=O)\c1ccc(cc1)S(C)(=O)=O 50174016O=S(=O)(Nc1cccc(c1)-c1cc(Cc2ccncc2)cc2cccnc12)c1ccccc1 50174017COc1cccc(c1)-c1cc(Cc2ccncc2)cc2cccnc12 50174018CC(C)NC(=O)C(=C\c1cccc(c1)-c1cc(cc2cccnc12)C(C)C)\c1ccc(cc1)S(C)(=O)=O 50174019CC(C)c1cc(-c2cccc(c2)C(Cc2cc[n+]([O-])cc2)c2ccc(Cl)cc2)c2ncccc2c1 50174020OC(c1ncc(s1)[C@@H](Cc1ccc[n+]([O-])c1)c1ccc(OC(F)F)c(OC2CC2)c1)(C(F)(F)F)C(F)(F)F 50174021CC(C)NC(=O)C(=C/c1cccc(c1)-c1cc(cc2cccnc12)C(C)(C)C#N)\c1ccc(cc1)S(C)(=O)=O 50174022Cc1noc(n1)C(=C\c1cccc(c1)-c1cc(cc2cccnc12)C(C)(C)S(C)(=O)=O)\c1ccc(cc1)S(C)(=O)=O 50174023CC(C)c1cc(-c2cccc(\C=C(\c3nc(C)no3)c3ccccn3)c2)c2ncccc2c1 50174024CC(C)c1cc(-c2cccc(c2)C(Cc2ccncc2)c2ccc(Cl)cc2)c2ncccc2c1 50174025CC(C)c1cc(-c2cccc(\C=C(\c3nccs3)c3ccc(cc3)S(C)(=O)=O)c2)c2ncccc2c1 50174026Cc1noc(n1)C(=C/c1cccc(c1)-c1cc(cc2cccnc12)C(C)(C)S(C)(=O)=O)\c1ccc(cc1)S(C)(=O)=O 50174027CC(c1cc(-c2cccc(\C=C(\c3ncc(s3)C(C)(C)O)c3ccc(cc3)S(C)(=O)=O)c2)c2ncccc2c1)S(C)(=O)=O 50174028CC(C)c1cc(-c2cccc(\C=C(/c3ccc(cc3)S(C)(=O)=O)c3ccc(C)cn3)c2)c2ncccc2c1 50174029CC(C)NC(=O)C(=C\c1cccc(c1)-c1cc(cc2cccnc12)C(C)(C)C#N)\c1ccc(cc1)S(C)(=O)=O 50174030CC(C)c1cc(-c2cccc(\C=C(\c3nc(C)no3)c3ccc(cc3)S(C)(=O)=O)c2)c2ncccc2c1 50174031CC(C)c1cc(-c2cccc(\C=C(\c3ccc(cc3)C(C)(C)O)c3ccc(cc3)S(C)(=O)=O)c2)c2ncccc2c1 50176377C[C@@H](NC(=O)c1cccnc1Oc1ccc(F)cc1)c1cccs1 50183788CC(C)(c1cc(-c2cccc(c2)C(=O)Nc2ccncc2)c2ncccc2c1)S(C)(=O)=O 50183789CC(N(C(C)=O)c1ccc(cc1)S(C)(=O)=O)c1cccc(c1)-c1cc(cc2cccnc12)C(C)(C)S(C)(=O)=O 50183790CC(C)NC(=O)N(Cc1cc(ccc1Cl)-c1cc(cc2cccnc12)C(C)(C)S(C)(=O)=O)c1ccc(cc1)S(C)(=O)=O 50183791CC(C)OC(=O)N(Cc1cccc(c1)-c1cc(cc2cccnc12)C(C)(C)C#N)c1ccc(cc1)S(C)(=O)=O 50183792CC(C)NC(=O)N(Cc1cccc(c1)-c1cc(cc2cccnc12)C(C)(C)C#N)c1ccc(cc1)S(C)(=O)=O 50183793CC(N(C(=O)c1cccnc1)c1ccc(cc1)S(C)(=O)=O)c1cccc(c1)-c1cc(cc2cccnc12)C(C)(C)S(C)(=O)=O 50183794CC(C)NC(=O)N(Cc1cccc(c1)-c1cc(cc2cccnc12)C(C)(C)S(C)(=O)=O)c1ccc(cc1)S(C)(=O)=O 50183795CC(C)(C#N)c1cc(-c2cccc(CN(Cc3ccc(F)cc3)c3ccc(cc3)S(C)(=O)=O)c2)c2ncccc2c1 50183796CC(C)(c1cc(-c2cccc(c2)C(N)=O)c2ncccc2c1)S(C)(=O)=O 50183797CC(C)(c1cc(-c2cccc(c2)C(=O)Nc2c(Cl)cncc2Cl)c2ncccc2c1)S(C)(=O)=O 50183798CC(C)NC(=O)N(Cc1cc(ccc1F)-c1cc(cc2cccnc12)C(C)(C)S(C)(=O)=O)c1ccc(cc1)S(C)(=O)=O 50183799CC(N(C(=O)c1ccc(F)cc1)c1ccc(cc1)S(C)(=O)=O)c1cccc(c1)-c1cc(cc2cccnc12)C(C)(C)S(C)(=O)=O 50183800CC(C)NC(=O)N(C(C)c1cccc(c1)-c1cc(cc2cccnc12)C(C)(C)S(C)(=O)=O)c1ccc(cc1)S(C)(=O)=O 50183801CC(C)(c1cc(-c2cccc(c2)C(=O)Nc2ccc(cc2)S(C)(=O)=O)c2ncccc2c1)S(C)(=O)=O 50183802CC(N(C(=O)C1CC1)c1ccc(cc1)S(C)(=O)=O)c1cccc(c1)-c1cc(cc2cccnc12)C(C)(C)S(C)(=O)=O 50183803Cc1cc(no1)C(=O)N(Cc1cccc(c1)-c1cc(cc2cccnc12)C(C)(C)C#N)c1ccc(cc1)S(C)(=O)=O 50183804CC(N(C(=O)c1ccc(cc1)C(C)(C)O)c1ccc(cc1)S(C)(=O)=O)c1cccc(c1)-c1cc(cc2cccnc12)C(C)(C)S(C)(=O)=O 50183805CC(C)(C#N)c1cc(-c2cccc(CN(C(=O)Nc3ccccc3)c3ccc(cc3)S(C)(=O)=O)c2)c2ncccc2c1 50183806CC(C)(c1cc(-c2cccc(NC(=O)c3ccc(cc3)S(C)(=O)=O)c2)c2ncccc2c1)S(C)(=O)=O 50183807CC(C)(c1cc(-c2cccc(c2)C(=O)Nc2ccccc2)c2ncccc2c1)S(C)(=O)=O 50183808CC(C)(C#N)c1cc(-c2cccc(CN(C(=O)c3ccccc3)c3ccc(cc3)S(C)(=O)=O)c2)c2ncccc2c1 50202528CCc1nn(C2CCCC2)c-2c1CCn1c(nnc-21)-c1cccs1 50202530CCc1nn(C2CCCC2)c-2c1CCn1c-2nnc1-c1cccnc1 50202531CCc1nn(C2CCCC2)c-2c1CCn1c-2nnc1C(C)(C)C 50202532CCc1nn(C2CCCC2)c-2c1CCn1c-2nnc1-c1cccc(OC)c1 50202544CCc1nn(C2CCCC2)c-2c1CCn1c-2nnc1-c1ccccc1Cl 50216795NC(=O)c1noc(n1)[C@H](CCCC1CCCCC1)CC(=O)NO 50219268COc1ccc(-c2nc(C(=O)N3CC[C@H](C3)NC(=O)OC(C)(C)C)c(CN)o2)c2ccc(nc12)C(F)(F)F 50219269COc1cc(OC)nc(n1)N1CCN(CC1)C(=O)c1nc(oc1CN)-c1ccc(OC)c2nc(ccc12)C(F)(F)F 50219270COc1ccc(C(=O)Nc2c(Cl)c[n+]([O-])cc2Cl)c2ccc(nc12)C(F)(F)F 50219271COc1ccc(-c2nc(C(N)=O)c(CN)o2)c2ccc(nc12)C(F)(F)F 50219272COc1ccc(-c2nc(C(=O)N3CCC(O)(CC3)c3ccccc3)c(CN)o2)c2ccc(nc12)C(F)(F)F 50219273CO\N=C(\C1CCN(CC1)C(=O)c1nc(oc1CN)-c1ccc(OC)c2nc(ccc12)C(F)(F)F)c1ccccn1 50219274COc1ccc(-c2nc(C(=O)N3CCC4(CC3)N(CNC4=O)c3ccccc3)c(CN)o2)c2ccc(nc12)C(F)(F)F 50219275COc1ccc(-c2nc(C(=O)N3CCN(CC3)C(=O)OC(C)(C)C)c(CN)o2)c2ccc(nc12)C(F)(F)F 50219276COc1ccc(-c2nc(C(=O)N3CCN(CC3)c3ncccn3)c(CN)o2)c2ccc(nc12)C(F)(F)F 50219277COc1ccc(-c2nc(C(=O)N3CCN(CC3)S(=O)(=O)N(C)C)c(CN)o2)c2ccc(nc12)C(F)(F)F 50219278COc1ccc(-c2nc(C(=O)N3CCN(CC3)C(=O)c3cc(C)n[nH]3)c(CN)o2)c2ccc(nc12)C(F)(F)F 50219279CNCc1oc(nc1C(N)=O)-c1ccc(OC)c2nc(ccc12)C(F)(F)F 50219280COc1ccc(-c2nc(CCl)c(C)o2)c2ccc(nc12)C(F)(F)F 50219281COc1ccc(-c2nc(C(=O)N3CCN(CC3)C(=O)c3ccccn3)c(CN)o2)c2ccc(nc12)C(F)(F)F 50219282COc1ccc(-c2nc(C(O)=O)c(C)o2)c2ccc(nc12)C(F)(F)F 50219283COc1ccc(-c2nc(CN)c(o2)C(N)=O)c2ccc(nc12)C(F)(F)F 50219284COc1ccc(-c2nc(C(=O)N3CCCC3)c(CN)o2)c2ccc(nc12)C(F)(F)F 50219285COc1ccc(-c2nc(CN)c(C)o2)c2ccc(nc12)C(F)(F)F 50219286CCN(CC)C(=O)c1nc(oc1CN)-c1ccc(OC)c2nc(ccc12)C(F)(F)F 50219287COc1ccc(-c2nc(C(=O)N3CCCCC3)c(CN)o2)c2ccc(nc12)C(F)(F)F 50219288COc1ccc(-c2nc(C=O)c(C)o2)c2ccc(nc12)C(F)(F)F 50219289COc1ccc(-c2nc(C(N)=O)c(C)o2)c2ccc(nc12)C(F)(F)F 50219290COc1ccc(-c2nc(C(=O)N3CCC3)c(CN)o2)c2ccc(nc12)C(F)(F)F 50219291COc1ccc(-c2nc(CO)c(C)o2)c2ccc(nc12)C(F)(F)F 50219292CCc1coc(n1)-c1ccc(OC)c2nc(ccc12)C(F)(F)F 50219293COc1ccc(-c2nc(C(O)=O)c(CN)o2)c2ccc(nc12)C(F)(F)F 50219294CNC(=O)c1nc(oc1CN)-c1ccc(OC)c2nc(ccc12)C(F)(F)F 50219295COc1ccc(-c2nc(C)co2)c2ccc(nc12)C(F)(F)F 50232731CC(C)(c1cc(-c2cccc(c2)-c2ccc(cc2)C2CC2C(O)=O)c2ncccc2c1)S(C)(=O)=O 50236078COc1ccc(C=C2SC(S)=NC2=O)cc1OC1CCCC1 50236083COc1ccc(\C=C2/SC(=N)NC2=O)cc1OC1CCCC1 50240404CC(C)C(=O)c1c(nn2ccccc12)C(C)C 50250915Oc1ccc2cc(oc2c1)-c1cc(O)cc(O)c1 50274267[O-][n+]1cccc(c1)C#Cc1cccc(c1)-n1cc(C(=O)NC2CC2)c(=O)c2cccnc12 50285038COC(=O)[C@@H]1CN(C[C@H]1c1ccc(OC)c(OC2CCCC2)c1)C(=O)OCc1ccccc1 50285039COc1ccc(cc1OC1CCCC1)[C@@H]1CN(C[C@H]1NS(C)(=O)=O)C(=O)OCc1ccccc1 50285040COc1ccc(cc1OC1CCCC1)[C@@H]1CN(C[C@H]1NC(=O)OC(C)(C)C)C(=O)OC(C)(C)C 50285041COC(=O)N1C[C@@H](C#N)[C@@H](C1)c1ccc(OC)c(OC2CCCC2)c1 50285042COc1ccc(cc1OC1CCCC1)[C@@H]1CN(C[C@H]1CO)C(=O)OC(C)(C)C 50285043COC(=O)[C@@H]1CN(C[C@H]1c1ccc(OC)c(OC2CCCC2)c1)C=O 50285044COC(=O)N1C[C@H]([C@@H](C1)c1ccc(OC)c(OC2CCCC2)c1)C(=O)c1ccccc1 50285045COC(=O)[C@@H]1CN(C[C@H]1c1ccc(OC)c(OC2CCCC2)c1)C(=O)OC(C)C 50285046COC(=O)N1C[C@H]([C@@H](C1)c1ccc(OC)c(OC2CCCC2)c1)C(N)=O 50285047COC(=O)N1C[C@H]([C@@H](C1)c1ccc(OC)c(OC2CCCC2)c1)C(O)=O 50285048CCC(=O)N1C[C@H]([C@@H](C1)c1ccc(OC)c(OC2CCCC2)c1)C(=O)OC 50285049COc1ccc(cc1OC1CCCC1)[C@@H]1CN(C[C@H]1C(O)=O)C(=O)OC(C)(C)C 50285050COC(=O)N1C[C@H]([C@@H](C1)[N+]([O-])=O)c1ccc(OC)c(OC2CCCC2)c1 50285051COc1ccc(cc1OC1CCCC1)[C@@H]1CN(C[C@H]1NS(=O)(=O)c1ccccc1)C(=O)OCc1ccccc1 50285052COC(=O)N1C[C@H]([C@@H](C1)c1ccc(OC)c(OC2CCCC2)c1)C(=O)OC(C)C 50285053COC(=O)[C@@H]1CN(C[C@H]1c1ccc(OC)c(OC)c1)C(=O)OC(C)(C)C 50285054COC(=O)[C@@H]1CN(C[C@H]1c1ccc(OC)c(OCCCOc2ccccc2)c1)C(=O)OC(C)(C)C 50285055COC(=O)[C@@H]1CN(C[C@H]1c1ccc(OC)c(OC2CCCC2)c1)C(N)=O 50285056COC(=O)[C@@H]1CN(C[C@H]1c1ccc(OC)c(OC2CCCC2)c1)C(N)=S 50285057COC[C@@H]1CN(C[C@H]1c1ccc(OC)c(OC2CCCC2)c1)C(=O)OC(C)(C)C 50285059COC(=O)[C@@H]1CN(C[C@H]1c1ccc(OC)c(OC2CCCC2)c1)C(=O)OC(C)(C)C 50285060COC(=O)N1C[C@H]([C@@H](C1)c1ccc(OC)c(OC2CCCC2)c1)C(=O)OC(C)(C)C 50285061COc1ccc(cc1OC1CCCC1)[C@@H]1CN(C[C@H]1C(N)=O)C(=O)OC(C)(C)C 50285062CCC(=O)[C@@H]1CN(C[C@H]1c1ccc(OC)c(OC2CCCC2)c1)C(=O)OC 50285063COc1ccc(cc1OC1CCCC1)[C@@H]1CN(C[C@H]1NC(=O)OC(C)(C)C)C(=O)OCc1ccccc1 50300953CCCOCCn1c2cc(ncc2nc(N[C@H]2CC[C@H](O)CC2)c1=O)-c1ccc(OC)nc1 50308512CCCOc1cc(ccc1OC)[C@]1(C)CNC(=O)O1 50314556C(CNc1nnc(-c2ccccc2)c2c1cc1ccccn21)CN1CCN(CC1)c1ncccn1 50314557[O-][N+](=O)c1cccc(c1)-c1nnc(NCCCN2CCN(CC2)C(=O)c2cnccn2)c2cc3ccccn3c12 50314558O=C(N1CCN(CCCNc2nnc(-c3ccccc3)c3c2cc2ccccn32)CC1)c1cnccn1 50314559Cc1cccc(c1)-c1nnc(NCCCN2CCN(CC2)c2ncccn2)c2cc3ccccn3c12 50314560Brc1cccc(c1)-c1nnc(NCCCN2CCN(CC2)c2ncccn2)c2cc3ccccn3c12 50314561Clc1cccc(c1)-c1nnc(NCCCN2CCN(CC2)c2ncccn2)c2cc3ccccn3c12 50314562Fc1cccc(c1)-c1nnc(NCCCN2CCN(CC2)c2ncccn2)c2cc3ccccn3c12 50314563N#Cc1cccc(c1)-c1nnc(NCCCN2CCN(CC2)c2ncccn2)c2cc3ccccn3c12 50314564[O-][N+](=O)c1cccc(c1)-c1nnc(NCCCN2CCN(CC2)c2ncccn2)c2cc3ccccn3c12 50314565CC(=O)N1CCN(CCCNc2nnc(-c3cccc(F)c3)c3c2cc2ccccn32)CC1 50314566CCC(=O)N1CCN(CCCNc2nnc(-c3cccc(F)c3)c3c2cc2ccccn32)CC1 50314568Fc1cccc(c1)-c1nnc(NCCCN2CCN(CC2)C(=O)c2ccccc2)c2cc3ccccn3c12 50314569Cn1cccc1C(=O)N1CCN(CCCNc2nnc(-c3cccc(F)c3)c3c2cc2ccccn32)CC1 50314570Fc1cccc(c1)-c1nnc(NCCCN2CCN(CC2)C(=O)c2cccnc2)c2cc3ccccn3c12 50314571Fc1cccc(c1)-c1nnc(NCCCN2CCN(CC2)C(=O)c2ccccn2)c2cc3ccccn3c12 50314573Cc1cc2c(NCCCN3CCN(CC3)C(=O)c3ncccn3)nnc(-c3cccc(Cl)c3)c2n1C 50314574Cc1cc2c(NCCCN3CCN(CC3)C(=O)c3ncccn3)nnc(-c3cccc(F)c3)c2n1C 50314575Cc1cc2c(NCCCN3CCN(CC3)C(=O)c3ncccn3)nnc(-c3cccc(c3)[N+]([O-])=O)c2n1C 50314577Cc1cc2c(NCCCN3CCN(CC3)C(=O)c3cccnc3)nnc(-c3cccc(c3)[N+]([O-])=O)c2n1C 50314578Cc1cc2c(NCCCN3CCN(CC3)C(=O)c3ccccn3)nnc(-c3cccc(c3)[N+]([O-])=O)c2n1C 50314579Cc1cc2c(NCCCN3CCN(CC3)C(=O)c3cc[n-][o+]3)nnc(-c3cccc(c3)[N+]([O-])=O)c2n1C 50314580Cc1cc2c(NCCCN3CCN(CC3)C(=O)c3c[s+]n[n-]3)nnc(-c3cccc(c3)[N+]([O-])=O)c2n1C 50314581Cc1cc2c(NCCCN3CCN(CC3)C(=O)c3cncs3)nnc(-c3cccc(c3)[N+]([O-])=O)c2n1C 50314582Cc1cc2c(NCCCN3CCN(CC3)C(=O)c3ccnnc3)nnc(-c3cccc(c3)[N+]([O-])=O)c2n1C 50314583Cc1cc2c(NCCCN3CCN(CC3)C(=O)c3cnccn3)nnc(-c3cccc(c3)[N+]([O-])=O)c2n1C 50317598COc1ccc2c(Nc3c(Cl)cncc3Cl)ccnc2c1OC1CCCC1 50317599COc1ccc2c(Nc3c(Cl)cncc3Cl)nccc2c1OC1CCCC1 50317600COc1ccc2c(Nc3c(Cl)cncc3Cl)ncnc2c1OC1CCCC1 50317603COc1ccc2c(Nc3c(Cl)cncc3Cl)cc(=O)oc2c1OC1CCCC1 50317604COc1ccc2c(Nc3c(Cl)cncc3Cl)cc(=O)oc2c1OCC(O)=O 50317605COc1ccc2c(Nc3c(Cl)cncc3Cl)cc(=O)oc2c1OCCCC(O)=O 50317606COc1ccc2c(Nc3c(Cl)cncc3Cl)cc(=O)oc2c1OCCCCC(O)=O 50317607COc1ccc2c(Nc3c(Cl)cncc3Cl)cc(=O)oc2c1OCCCCCC(O)=O 50317608COc1ccc2c(Nc3c(Cl)cncc3Cl)cc(=O)oc2c1OCCCCCCC(O)=O 50317609COc1ccc2c(Nc3c(Cl)cncc3Cl)cc(=O)oc2c1OCCCCCCCC(O)=O 50317610COc1ccc2c(Nc3c(Cl)cncc3Cl)cc(=O)oc2c1OCCCCCCCCC(O)=O 50317611COc1ccc2c(Nc3c(Cl)cncc3Cl)cc(=O)oc2c1OCCCN(C)C 50317612COc1ccc2c(Nc3c(Cl)cncc3Cl)cc(=O)oc2c1OCCCCN(C)C 50317613COc1ccc2c(Nc3c(Cl)cncc3Cl)cc(=O)oc2c1OCCCCCN(C)C 50317614COc1ccc2c(Nc3c(Cl)cncc3Cl)cc(=O)oc2c1OCCCCCCN(C)C 50317615COc1ccc2c(Nc3c(Cl)cncc3Cl)cc(=O)oc2c1OCCCCCCCN(C)C 50317616COc1ccc2c(Nc3c(Cl)cncc3Cl)cc(=O)oc2c1OCCCCCCCCN(C)C 50325786CC(C)(O)CCc1ccc(OCc2cc(-c3cccc(OC(F)F)c3)c3ncccc3c2)cc1 50325787CS(=O)(=O)c1ccc(OCc2cc(-c3cccc(OC(F)F)c3)c3ncccc3c2)cc1 50325788OC(=O)Cc1ccc(OCc2cc(-c3cccc(OC(F)F)c3)c3ncccc3c2)cc1 50325789COc1cccc(c1)-c1cc(cc2cccnc12)C(C)(C)S(C)(=O)=O 50325790COC(=O)Cc1ccc(OCc2cc(-c3cccc(OC)c3)c3ncccc3c2)cc1 50325791COc1cccc(c1)-c1cc(COc2ccccc2Cl)cc2cccnc12 50325792COc1cccc(c1)-c1cc(COc2cccc(Cl)c2)cc2cccnc12 50325793COc1cccc(c1)-c1cc(COc2ccc(cc2)C(F)(F)F)cc2cccnc12 50325794COc1cccc(c1)-c1cc(COc2ccc(CCC#N)cc2)cc2cccnc12 50325795N#CCCc1ccc(OCc2cc(-c3ccccc3)c3ncccc3c2)cc1 50325796FC(F)(F)Oc1cccc(c1)-c1cc(COc2ccc(CCC#N)cc2)cc2cccnc12 50325797Fc1cccc(c1)-c1cc(COc2ccc(CCC#N)cc2)cc2cccnc12 50325798CCOc1cccc(c1)-c1cc(COc2ccc(CCC#N)cc2)cc2cccnc12 50325799Cc1cccc(c1)-c1cc(COc2ccc(CCC#N)cc2)cc2cccnc12 50325800FC(F)Oc1cccc(c1)-c1cc(COc2ccc(CCC#N)cc2)cc2cccnc12 50328090CC1(C)CCc2c(C1)c1c(nc2N2CCOCC2)sc2c(ncnc12)N(CCO)CCN1CCOCC1 50328091CC1(C)CCc2c(C1)c1c(nc2N2CCOCC2)sc2c(NCCN3CCOCC3)ncnc12 50328092CC1(C)CCc2c(C1)c1c(nc2-c2ccoc2)sc2c(NCCN3CCOCC3)ncnc12 50328093CC1(C)CCc2c(C1)c1c(nc2N2CCOCC2)sc2c(NCc3cccnc3)ncnc12 50328094CC1(C)CCc2c(C1)c1c(nc2-c2ccco2)sc2c(NCCN3CCOCC3)ncnc12 50328095CNc1nc2sc3c(NCCN4CCOCC4)ncnc3c2c2CC(C)(C)CCc12 50328096CC1(C)Cc2c(CO1)c(nc1sc3c(ncnc3c21)N(CCN1CCOCC1)Cc1cccnc1)N1CCOCC1 50328097CC1(C)Cc2c(CO1)c(nc1sc3c(NCc4cccnc4)ncnc3c21)N1CCOCC1 50328098CC(C)Cc1nc2sc3c(NCCN4CCOCC4)ncnc3c2c2CC(C)(C)CCc12 50328099CC1(C)CCc2c(C1)c1c(nc2N2CCCC2)sc2c(NCCN3CCOCC3)ncnc12 50328100CC1(C)CCc2c(C1)c1c(nc2N2CCOCC2)sc2c(NCc3ccncc3)ncnc12 50328101CC1(C)Cc2c(CO1)c(nc1sc3c(ncnc3c21)N(CCO)CCN1CCOCC1)N1CCOCC1 50328102CC1(C)CCc2c(C1)c1c(nc2N2CCOCC2)sc2c(NCCCN3CCCC3=O)ncnc12 50328103CN(C)c1nc2sc3c(NCCN4CCOCC4)ncnc3c2c2CC(C)(C)OCc12 50328104CC1(C)Cc2c(CO1)c(nc1sc3c(NCc4ccncc4)ncnc3c21)N1CCOCC1 50328105CC1(C)Cc2c(CO1)c(nc1sc3c(NCCN4CCOCC4)ncnc3c21)N1CCOCC1 50328106Cc1nc2sc3c(NCCN4CCOCC4)ncnc3c2c2CC(C)(C)CCc12 50328107COc1ccccc1CNc1ncnc2c1sc1nc(N3CCOCC3)c3COC(C)(C)Cc3c21 50328108CNc1nc2sc3c(NCCN4CCOCC4)ncnc3c2c2CC(C)(C)OCc12 50328109CCC1(C)Cc2c(CO1)c(nc1sc3c(NCCN4CCOCC4)ncnc3c21)N1CCOCC1 50328110CN1CCN(CC1)c1nc2sc3c(NCCN4CCOCC4)ncnc3c2c2CC(C)(C)CCc12 50328111CC1(C)Cc2c(CO1)c(nc1sc3c(NCCCN4CCCC4=O)ncnc3c21)N1CCOCC1 50328112COc1ccccc1CNc1ncnc2c1sc1nc(N3CCOCC3)c3CCC(C)(C)Cc3c21 50328113CC1(C)CCc2c1c1c(nc2N2CCOCC2)sc2c(NCCN3CCOCC3)ncnc12 50328114CC1(C)Cc2c(CO1)c(nc1sc3c(NCCN4CCCCC4)ncnc3c21)N1CCOCC1 50328115CC1(C)Cc2c(C1)c1c(nc2N2CCOCC2)sc2c(NCCN3CCOCC3)ncnc12 50328116CN(Cc1ccccc1)c1nc2sc3c(NCCN4CCOCC4)ncnc3c2c2CC(C)(C)CCc12 50328117CN1CCN(CC1)c1nc2sc3c(NCCN4CCOCC4)ncnc3c2c2CC(C)(C)OCc12 50328118C(CN1CCOCC1)Nc1ncnc2c1sc1nc(N3CCOCC3)c3COCCc3c21 50328119CN1Cc2c(CC1(C)C)c1c(nc2N2CCOCC2)sc2c(NCCN3CCOCC3)ncnc12 50335843CCn1c(O)c2Cc3c([nH]c4ccccc34)[C@@H](c3ccc(Cl)cc3Cl)n2c1=O 50344305CC(C)c1nn2ccccc2c1C1=NNC(=O)CC1C 50344314CC12CCc3nn4ccccc4c3C1=NN(Cc1ccccc1)C(=O)C2 50344318CC(C)c1nn2cccc3CC4CC(=O)N(Cc5ccccc5)N=C4c1c23 50344321COc1cccc2c(c(nn12)C(C)C)C1=NN(Cc2ccccc2)C(=O)CC1 50344325COc1ccc(-c2ccc(Cl)nn2)c2cc(nn12)C(C)C 50344326COc1ccc(-c2ccc(=O)[nH]n2)c2cc(nn12)C(C)C 50344327COc1ccc(-c2ccc(=O)n(Cc3ccccc3)n2)c2cc(nn12)C(C)C 50344328COc1ccc(C2=NNC(=O)CC2)c2cc(nn12)C(C)C 50344329COc1ccc(C2=NN(Cc3ccccc3)C(=O)CC2)c2cc(nn12)C(C)C 50346088COc1ccc(cc1OC1CCCC1)[C@]1(CC[C@@H](CC1)C(O)=O)C#N 50346089Cc1nc(nc(Nc2ccc(cc2)C(O)=O)c1CC=C)-c1ccccc1 50346090Cc1nc(nc(Nc2ccc(cc2)C(O)=O)c1C)-c1ccccc1 50346091CCc1c(C)nc(nc1Nc1ccc(cc1)C(O)=O)-c1ccccc1 50346092CCCc1c(C)nc(nc1Nc1ccc(cc1)C(O)=O)-c1ccccc1 50346096Cc1nc(nc(Nc2ccc(cc2)C(O)=O)c1C#N)-c1ccccc1 50346098Cc1nc(nc(Nc2ccc(cc2)C(O)=O)c1C=O)-c1ccccc1 50346099Cc1nc(nc(Nc2ccc(cc2)C(O)=O)c1CO)-c1ccccc1 50346100CCc1nc(nc(Nc2ccc(cc2)C(O)=O)c1CC=C)-c1ccccc1 50346102CCCc1nc(nc(Nc2ccc(cc2)C(O)=O)c1CC=C)-c1ccccc1 50346103Cc1nc(nc(Nc2ccc(cc2)C(O)=O)c1CC=C)-c1cccs1 50346104Cc1nc(nc(Nc2ccc(cc2)C(O)=O)c1CC=C)-c1ccsc1 50346105Cc1nc(cs1)-c1nc(C)c(CC=C)c(Nc2ccc(cc2)C(O)=O)n1 50346106Cc1nc(nc(Nc2ccc(cc2)C(O)=O)c1CC=C)-c1ccccn1 50346107Cc1nc(nc(Nc2ccc(cc2)C(O)=O)c1CC=C)-c1cnccn1 50346108Cc1ccc(cc1)-c1nc(C)c(CC=C)c(Nc2ccc(cc2)C(O)=O)n1 50346109Cc1cccc(c1)-c1nc(C)c(CC=C)c(Nc2ccc(cc2)C(O)=O)n1 50346110COc1ccc(cc1)-c1nc(C)c(CC=C)c(Nc2ccc(cc2)C(O)=O)n1 50346111Cc1ccc(s1)-c1nc(C)c(CC=C)c(Nc2ccc(cc2)C(O)=O)n1 50346112COc1ccc(s1)-c1nc(C)c(CC=C)c(Nc2ccc(cc2)C(O)=O)n1 50346113Cc1nc(nc(Nc2ccc(CC(O)=O)cc2)c1CC=C)-c1ccccc1 50346114Cc1ccc(cc1)-c1nc(C)c(CC=C)c(Nc2ccc(CC(O)=O)cc2)n1 50346115Cc1cccc(c1)-c1nc(C)c(CC=C)c(Nc2ccc(CC(O)=O)cc2)n1 50346116COc1ccc(cc1)-c1nc(C)c(CC=C)c(Nc2ccc(CC(O)=O)cc2)n1 50346117Cc1ccc(s1)-c1nc(C)c(CC=C)c(Nc2ccc(CC(O)=O)cc2)n1 50346118COc1ccc(s1)-c1nc(C)c(CC=C)c(Nc2ccc(CC(O)=O)cc2)n1 50346119CCc1c(C)nc(nc1Nc1ccc(CC(O)=O)cc1)-c1ccc(SC)s1 50346120CCc1c(C)nc(nc1Nc1ccc(CC(O)=O)cc1)-c1ccc(Br)s1 50346121CCc1c(C)nc(nc1Nc1ccc(CC(O)=O)cc1)-c1ccc(Cl)s1 50346122CCc1c(C)nc(nc1Nc1ccc(CC(O)=O)cc1)-c1cc(Br)c(C)s1 50346123CCc1c(C)nc(nc1Nc1ccc(CC(O)=O)cc1F)-c1ccc(F)s1 50347334OC(=O)C1CC1c1ccc(cc1)-c1cccc(c1)-n1cc(C(=O)NC2CC2)c(=O)c2cccnc12 50347335OC(=O)C1CC1c1cccc(c1)-c1cccc(c1)-n1cc(C(=O)NC2CC2)c(=O)c2cccnc12 50347336OC(=O)C1CC1c1ccccc1-c1cccc(c1)-n1cc(C(=O)NC2CC2)c(=O)c2cccnc12 50347337CC(C)(Cc1ccc(cc1)-c1cccc(c1)-n1cc(C(=O)NC2CC2)c(=O)c2cccnc12)C(O)=O 50347338CC(C)(CC(O)=O)c1ccc(cc1)-c1cccc(c1)-n1cc(C(=O)NC2CC2)c(=O)c2cccnc12 50347339O=C(NC1CC1)c1cn(-c2cccc(c2)-c2ccc(cc2)C2CC2c2nnn[nH]2)c2ncccc2c1=O 50347340CC(C)(C)NC(=O)c1cn(-c2cccc(c2)-c2ccc(cc2)C2CC2C(O)=O)c2ncccc2c1=O 50347341OC(=O)C1CC1c1ccc(cc1)-c1cccc(c1)-n1cc(C(=O)NC2(O)CC2)c(=O)c2cccnc12 50347342CC1(CC1)NC(=O)c1cn(-c2cccc(c2)-c2ccc(cc2)C2CC2C(O)=O)c2ncccc2c1=O 50347343OC(=O)C1CC1c1ccc(cc1)-c1cccc(c1)-n1cc(C(=O)NCC(F)(F)F)c(=O)c2cccnc12 50347344OC(=O)C1CC1c1ccc(cc1)-c1cccc(c1)-n1cc(C(=O)NCC2CC2)c(=O)c2cccnc12 50347345OC(=O)C1CC1c1ccc(cc1)-c1cccc(c1)-n1cc(C(=O)NC2CCC2)c(=O)c2cccnc12 50347346OC(=O)[C@@H]1C[C@H]1c1ccc(cc1)-c1cccc(c1)-n1cc(C(=O)NC2CC2)c(=O)c2cccnc12 50347347OC(=O)[C@H]1C[C@@H]1c1ccc(cc1)-c1cccc(c1)-n1cc(C(=O)NC2CC2)c(=O)c2cccnc12 50347348OC(=O)[C@@H]1C[C@H]1c1ccc(cc1F)-c1cccc(c1)-n1cc(C(=O)NC2CC2)c(=O)c2cccnc12 50347349OC(=O)[C@H]1C[C@@H]1c1ccc(cc1F)-c1cccc(c1)-n1cc(C(=O)NC2CC2)c(=O)c2cccnc12 50353691CC1(C)Cc2c(CO1)c(nc1oc3c(NCc4cccnc4)ncnc3c21)N1CCOCC1 50353692CC1(C)CCc2c(C1)c1c(nc2N2CCOCC2)oc2c(NCc3cccnc3)ncnc12 50353693CC1(C)CCc2c(C1)c1c(nc2N2CCOCC2)oc2c(NCCN3CCOCC3)ncnc12 50353694CC1(C)Cc2c(CO1)c(nc1oc3c(NCCN4CCOCC4)ncnc3c21)N1CCOCC1 50353695CC1(C)CCc2c(C1)c1c(nc2N2CCOCC2)oc2c(ncnc12)N(CCO)CCN1CCOCC1 50353696CC1(C)Cc2c(CO1)c(nc1oc3c(ncnc3c21)N(CCO)CCN1CCOCC1)N1CCOCC1 50353697CC1(C)CCc2c(NCCO)nc3oc4c(NCc5cccnc5)ncnc4c3c2C1 50353698CCNc1nc2oc3c(NCCN4CCOCC4)ncnc3c2c2CC(C)(C)CCc12 50353699CCN(C)c1nc2oc3c(NCCN4CCOCC4)ncnc3c2c2CC(C)(C)CCc12 50353700CC(C)Nc1nc2oc3c(NCCN4CCOCC4)ncnc3c2c2CC(C)(C)CCc12 50353701CCNc1nc2oc3c(NCCCN4CCCC4=O)ncnc3c2c2CC(C)(C)CCc12 50353702CCN(C)c1nc2oc3c(NCCCN4CCCC4=O)ncnc3c2c2CC(C)(C)CCc12 50353703CC(C)Nc1nc2oc3c(NCCCN4CCCC4=O)ncnc3c2c2CC(C)(C)CCc12 50353704CCN(C)c1nc2oc3c(NCc4cccnc4)ncnc3c2c2CC(C)(C)CCc12 50353705CCNc1nc2oc3c(NCc4cccnc4)ncnc3c2c2CC(C)(C)CCc12 50353706CC(C)Nc1nc2oc3c(NCc4cccnc4)ncnc3c2c2CC(C)(C)CCc12 50353707CC1(C)CCc2c(Nc3c(Cl)cncc3Cl)nc3oc4c(NCc5cccnc5)ncnc4c3c2C1 50363905COc1ccc(C2=NNC(=O)CC2C)c2nc(nn12)C(F)(F)F 50363906COc1ccc(C2=NNC(=O)CC2C)n2cc(nc12)C(F)(F)F 50363907COc1ccc(C2=NNC(=O)CC2C)c2oc(nc12)C(F)(F)F 50363908COc1ccc(C2=NNC(=O)CC2C)c2nc(oc12)C(F)(F)F 50363909COc1ccc(C2=NNC(=O)CC2C)c2sc(nc12)C(F)(F)F 50363910COc1ccc(C2=NNC(=O)CC2C)c2cc(sc12)C(F)(F)F 50363911COc1ccc(C2=NNC(=O)CC2C)c2ccc(nc12)C(F)(F)F 50363912COc1ccc(C2=NNC(=O)CC2C)c2[nH]c(nc12)C(F)(F)F 50363913COc1ccc(C2=NNC(=O)CC2C)c2cc(oc12)C(F)(F)F 50363914CCc1cc2c(ccc(OC)n2c1)C1=NNC(=O)CC1C 50365055COc1ccc(cc1OC)C1=NNC(=O)C2CCCCC12 50365056COc1ccc(cc1OC)C1=NN(CCNCC(O)c2ccc(O)c(NC=O)c2)C(=O)C2CCCCC12 50365057COc1ccc(cc1OC)C1=NN(CCCCNCC(O)c2ccc(O)c(NC=O)c2)C(=O)C2CCCCC12 50365058COc1ccc(cc1OC)C1=NN(CCCCNC[C@H](O)c2ccc(O)c(NC=O)c2)C(=O)C2CCCCC12 50365059COc1ccc(cc1OC)C1=NN(CCCCNC[C@@H](O)c2ccc(O)c(NC=O)c2)C(=O)C2CCCCC12 50365060COc1ccc(cc1OC)C1=NN(CCCCCNCC(O)c2ccc(O)c(NC=O)c2)C(=O)C2CCCCC12 50365061COc1ccc(cc1OC)C1=NN(CCCCCCNCC(O)c2ccc(O)c(NC=O)c2)C(=O)C2CCCCC12 50365480Oc1c(C#N)c(nc2ccncc12)-c1ccc(cc1)-c1ccccc1OC(F)(F)F 50366135COc1ccc2c(c[nH]c2c1)-c1nc2ccccc2cc1C#N 50366802COc1ccc(cc1OC1Cc2ccccc2C1)[C@H](C)Cn1ccnc1NC#N 50372899CCN1C(=S)S\C(=C/c2ccc(O)c(OC)c2)C1=O 50372900COc1ccc(\C=C2/SC(=S)N(C)C2=O)cc1OC1CCCC1 50372902CCOc1ccc(C=C2SC(S)=NC2=O)cc1OCC 50372904CCOc1ccc(C=C2SC(=S)NC2=O)cc1OC1CCCC1 50372905CCOc1cc(C=C2SC(S)=NC2=O)ccc1OC 50372906CCOc1ccc(C=C2SC(S)=NC2=O)cc1OC 50372907COc1ccc(\C=C2/CCNC2=O)cc1OC1CCCC1 50372908COc1ccc(C=C2SC(=O)NC2=O)cc1OC1CCCC1 50372911COc1ccc(\C=C2/SC(=S)N(CC(O)=O)C2=O)cc1OC1CCCC1 50372912COc1ccc(\C=C2/SC(=S)N(CC=C)C2=O)cc1OC1CCCC1 50372913COc1ccc(C=C2SC(=S)NC2=O)cc1OC1CCCCC1 50372914COc1ccc(C=C2SC(S)=NC2=O)cc1OCC=C 50379961COc1ccc(-c2nc(C(=O)NCc3c(F)cccc3F)c(o2)[C@H](C)N)c2ccc(nc12)C(F)(F)F 50379962COc1ccc(-c2nc(C(=O)NCc3ccccc3)c(CN)o2)c2ccc(nc12)C(F)(F)F 50379963COc1ccc(-c2nc(C(=O)NCc3ccc(F)cc3)c(CN)o2)c2ccc(nc12)C(F)(F)F 50379964COc1ccc(-c2nc(C(=O)NCc3ccc(Cl)cc3)c(CN)o2)c2ccc(nc12)C(F)(F)F 50379965COc1ccc(-c2nc(C(=O)NCc3cccc(F)c3)c(CN)o2)c2ccc(nc12)C(F)(F)F 50379966COc1ccc(-c2nc(C(=O)NCc3cccc(Cl)c3)c(CN)o2)c2ccc(nc12)C(F)(F)F 50379967COc1ccc(-c2nc(C(=O)NCc3ccccc3F)c(CN)o2)c2ccc(nc12)C(F)(F)F 50379968COc1ccc(-c2nc(C(=O)NCc3ccccc3Cl)c(CN)o2)c2ccc(nc12)C(F)(F)F 50379969COc1ccccc1CNC(=O)c1nc(oc1CN)-c1ccc(OC)c2nc(ccc12)C(F)(F)F 50379970COc1ccc(-c2nc(C(=O)NCc3c(F)cccc3F)c(CN)o2)c2ccc(nc12)C(F)(F)F 50379971COc1ccc(-c2nc(C(=O)NCc3c(F)cccc3Cl)c(CN)o2)c2ccc(nc12)C(F)(F)F 50379972COc1ccc(-c2nc(C(=O)NCc3ccc(F)cc3F)c(CN)o2)c2ccc(nc12)C(F)(F)F 50379973COc1ccc(-c2nc(C(=O)NCc3ccc(Cl)cc3F)c(CN)o2)c2ccc(nc12)C(F)(F)F 50379974COc1ccc(-c2nc(C(=O)NCc3ccc(Cl)cc3Cl)c(CN)o2)c2ccc(nc12)C(F)(F)F 50379975COc1ccc(-c2nc(C(=O)NCc3ccc(F)c(F)c3)c(CN)o2)c2ccc(nc12)C(F)(F)F 50379976COc1ccc(-c2nc(C(=O)NCc3ccc(Cl)cc3)c(o2)[C@H](C)N)c2ccc(nc12)C(F)(F)F 50379977COc1ccc(-c2nc(C(=O)NCc3cccc(F)c3)c(o2)[C@H](C)N)c2ccc(nc12)C(F)(F)F 50379978COc1ccc(-c2nc(C(=O)NCc3ccccc3F)c(o2)[C@H](C)N)c2ccc(nc12)C(F)(F)F 50379979COc1ccc(-c2nc(C(=O)NCc3c(F)cccc3Cl)c(o2)[C@H](C)N)c2ccc(nc12)C(F)(F)F 50379980COc1ccc(-c2nc(C(=O)NCc3ccc(F)cc3F)c(o2)[C@H](C)N)c2ccc(nc12)C(F)(F)F 50379981COc1ccc(-c2nc(C(=O)NCc3ccc(Cl)cc3F)c(o2)[C@H](C)N)c2ccc(nc12)C(F)(F)F 50379982COc1ccc(-c2nc(C(=O)NCc3ccc(Cl)cc3Cl)c(o2)[C@H](C)N)c2ccc(nc12)C(F)(F)F 50379983COc1ccc(-c2nc(C(=O)NCc3ccc(F)c(F)c3)c(o2)[C@H](C)N)c2ccc(nc12)C(F)(F)F 50379984COc1ccc(-c2nc(C(=O)NCc3c(F)cc(F)cc3F)c(o2)[C@H](C)N)c2ccc(nc12)C(F)(F)F 50379985COc1ccc(-c2nc(C(=O)N[C@H](CO)c3ccccc3)c(CN)o2)c2ccc(nc12)C(F)(F)F 50379986COc1ccc(-c2nc(C(=O)N[C@H](CO)c3ccccc3)c(o2)[C@H](C)N)c2ccc(nc12)C(F)(F)F 50379987COc1ccc(-c2nc(C(=O)N[C@H](CO)c3ccccc3)c(o2)[C@@H](C)N)c2ccc(nc12)C(F)(F)F 50379988COc1ccc(-c2nc(C(=O)NCc3ccc(cc3)C#N)c(CN)o2)c2ccc(nc12)C(F)(F)F 50379989COc1ccc(-c2nc(C(=O)NCc3ccc(cc3)S(C)(=O)=O)c(CN)o2)c2ccc(nc12)C(F)(F)F 50379990CC[C@H](N)c1oc(nc1C(=O)NCc1ccc(Cl)cc1)-c1ccc(OC)c2nc(ccc12)C(F)(F)F 50379991COc1ccc(-c2nc(C(=O)NCc3ccc(Cl)cc3)c(o2)[C@@H](N)CO)c2ccc(nc12)C(F)(F)F 50379992COc1ccc(-c2nc(C(=O)NCc3ccc(F)cc3F)c(o2)[C@@H](N)C(C)C)c2ccc(nc12)C(F)(F)F 50380675COc1cc2c(Nc3cccc4cccnc34)c(cnc2cc1-c1c(C)noc1C)C(N)=O 50380682COc1cc2c3n([C@H](C)c4ccccn4)c(=O)[nH]c3cnc2cc1-c1c(C)noc1C 50381089CC1(C)Cc2cnn(c2-c2cc(Br)ccc12)-c1ccccc1 50389205C[C@@H](O[C@H]1CC[C@H](O[C@@H]2CC[C@@H](OC(=O)[C@H](C)[C@@H](O)C(\C)=C\c3ccc4C(=O)C=CC(=O)c4c3)[C@H](C)O2)[C@H](C)O1)[C@H](C)[C@H](O)[C@@H](C)[C@H](O)[C@H](C)[C@H]1OC(=O)\C=C\[C@H](C)[C@@H](O)C[C@H](O)\C=C\CC[C@@H](C)[C@@H](O)[C@H](O)[C@@]2(O)O[C@H](C[C@@H](O)[C@@H]2O)C[C@H](C[C@@H](O)C[C@H](O)C[C@@H](O)[C@@H]2O[C@H]2[C@H]1C)OC(C)=O 50390612COc1ccc(C2=NNC(=O)C2(C)C)c2cc(nn12)C(F)F 50390613COc1ccc(C2=NNC(=O)C2(C)C)c2cc(nn12)C(F)(F)F 50390614COc1ccc(C2=NNC(=O)C2(C)C)c2cc(sc12)C(F)(F)F 50390615COc1ccc(C2=NNC(=O)C2(C)C)c2sc(nc12)C(F)(F)F 50390616COc1ccc(C2=NNC(=O)C2(C)C)c2[nH]c(nc12)C(F)(F)F 50390617COc1ccc(C2=NNC(=O)C2(C)C)n2cc(nc12)C(F)(F)F 50390618CCc1ccc2c(ccc(OC)c2n1)C1=NNC(=O)C1(C)C 50390619COc1ccc(C2=NNC(=O)C2(C)C)c2ccc(nc12)C(F)(F)F 50390620CCc1cc2c(ccc(OC)n2n1)C1=NNC(=O)CC1C 50390621CCc1cc2c(ccc(C)n2n1)C1=NNC(=O)C1(C)C 50390622CCc1cc2c(ccc(CC)n2n1)C1=NNC(=O)C1(C)C 50390623CCc1cc2c(ccc(OC)n2n1)C1=NNC(=O)C1(C)C 50390624CCc1cc2c(ccc(SC)n2n1)C1=NNC(=O)C1(C)C 50390625CCc1cc2c(ccc(NC)n2n1)C1=NNC(=O)C1(C)C 50390626CCc1cc2c(ccc(CO)n2n1)C1=NNC(=O)C1(C)C 50390627CCc1cc2c(ccc(C(C)O)n2n1)C1=NNC(=O)C1(C)C 50390628CCc1cc2c(ccc(C(C)=O)n2n1)C1=NNC(=O)C1(C)C 50390629COc1ccc(C2=NNC(=O)CC2C)c2cc(nn12)C(F)(F)F 50390630COc1ccc(C2=NNC(=O)C2(C)C)c2ccnn12 50390631COc1ccc(C2=NNC(=O)C2(C)C)c2cc(nn12)C1CC1 50390632COc1ccc(C2=NNC(=O)C2(C)C)c2cc(oc12)C(F)(F)F 50396755COc1cccc(c1)-c1nc(cc2cccnc12)N1CCC(CC1)C(O)=O 50396756OC(=O)C1CCN(CC1)c1cc2cccnc2c(n1)-c1cccc(OC(F)(F)F)c1 50396757OC(=O)C1CCN(CC1)c1cc2cccnc2c(n1)-c1cccc(F)c1 50396758OC(=O)C1CCN(CC1)c1cc2cccnc2c(n1)-c1cccc(Cl)c1 50396759OC(=O)C1CCN(CC1)c1cc2cccnc2c(n1)-c1cccc(c1)C#N 50396760CSc1cccc(c1)-c1nc(cc2cccnc12)N1CCC(CC1)C(O)=O 50396761COc1cccc(c1)-c1nc(cc2cccnc12)[C@H]1CC[C@@H](CC1)C(O)=O 50396762OC(=O)[C@H]1CC[C@@H](CC1)c1cc2cccnc2c(n1)-c1cccc(OC(F)(F)F)c1 50396763OC(=O)[C@H]1CC[C@@H](CC1)c1cc2cccnc2c(n1)-c1cccc(F)c1 50396764OC(=O)[C@H]1CC[C@@H](CC1)c1cc2cccnc2c(n1)-c1cccc(c1)C#N 50396765CSc1cccc(c1)-c1nc(cc2cccnc12)[C@H]1CC[C@@H](CC1)C(O)=O 50396783COc1ccc(\C=N\N(C)C(=O)c2ccc(O)cc2)cc1OC 50396784COc1ccc(cc1)C(=O)N(C)\N=C\c1ccc(OC)c(OC)c1 50396785Clc1ncnc2ccccc12 50397078COc1ccc(cc1OCCCCOc1ccc(cc1)-c1nnn[nH]1)C1=NN(C2CCCCCC2)C(=O)C1(C)C 50412387CCOC(=O)c1cnc2n(CC)ncc2c1Nc1ccccc1 50412388CCOC(=O)c1cnc2n(CC)ncc2c1NC(=O)c1ccccc1 50412389CCOC(=O)c1cnc2n(CC)ncc2c1N(C)C1CCOCC1 50412390CCOC(=O)c1cnc2n(CC)ncc2c1NCc1ccc(F)cc1 50412391CCOC(=O)c1cnc2n(CC)ncc2c1Nc1ccc(OC)cc1 50412392CCOC(=O)c1cnc2n(CC)ncc2c1NCC(C)C 50412393CCOC(=O)c1cnc2n(CC)ncc2c1NC1CCOCC1 50412394CCOC(=O)c1cnc2n(CC)ncc2c1NC1CCCCC1 50412395CCOC(=O)c1cnc2n(CC)ncc2c1N1CCCC1 50412396CCOC(=O)c1cnc2n(CC)ncc2c1NC1CCCC1 50412397CCOC(=O)c1cnc2n(ncc2c1NC1CCOCC1)-c1ccccc1 50412398CCOC(=O)c1cnc2n(CCO)ncc2c1NC1CCOCC1 50412399CCOC(=O)CCn1ncc2c(NC3CCOCC3)c(cnc12)C(=O)OCC 50412400CCOC(=O)c1cnc2n(Cc3ccccc3)ncc2c1NC1CCOCC1 50412401CCOC(=O)c1cnc2n(ncc2c1NC1CCOCC1)C(C)C 50412402CCCn1ncc2c(NC3CCOCC3)c(cnc12)C(=O)OCC 50412403CCOC(=O)c1cnc2n(C)ncc2c1NC1CCOCC1 50412404CCOC(=O)c1cnc2[nH]ncc2c1NC1CCOCC1 50412405CCn1ncc2c(NC3CCOCC3)c(cnc12)C(=O)NCC1CCCCC1 50412406CCn1ncc2c(NC3CCOCC3)c(cnc12)C(=O)NC1CC1 50412407CCn1ncc2c(NC3CCOCC3)c(cnc12)C(=O)NC1CCN(CC1)C(C)=O 50412408CCn1ncc2c(NC3CCOCC3)c(cnc12)C(=O)NC1CCCC1 50412409CCn1ncc2c(NC3CCOCC3)c(cnc12)C(=O)N1CCCC1 50412410CCn1ncc2c(NC3CCOCC3)c(cnc12)C(N)=O 50412411CCn1ncc2c(NC3CCOCC3)c(cnc12)C(=O)Nc1ccc(F)cc1 50412412CCC(CC)CNC(=O)c1cnc2n(CC)ncc2c1NC1CCOCC1 50412413CCn1ncc2c(NC3CCOCC3)c(cnc12)C(=O)N(C)Cc1ccccc1 50412414CCn1ncc2c(NC3CCOCC3)c(cnc12)C(=O)NCc1ccccc1 50413282CS(=O)(=O)c1ccc2ncc(C(N)=O)c(Nc3cccc(O)c3)c2c1 50413285CS(=O)(=O)c1ccc2ncc(C(N)=O)c(Nc3cccc(c3)C#N)c2c1 50413286CS(=O)(=O)c1ccc2ncc(C(N)=O)c(Nc3cccc4OCCc34)c2c1 50413287CS(=O)(=O)c1ccc2ncc(C(N)=O)c(Nc3cccc(c3)C(O)=O)c2c1 50413288CS(=O)(=O)c1ccc2ncc(C(N)=O)c(Nc3cccc(Cl)c3F)c2c1 50413289CS(=O)(=O)c1ccc2ncc(C(N)=O)c(Oc3cccc(Cl)c3)c2c1 50413290CN(c1cccc(Cl)c1)c1c(cnc2ccc(cc12)S(C)(=O)=O)C(N)=O 50413291COc1cccc(Nc2c(cnc3ccc(cc23)S(=O)(=O)c2ccccc2)C(N)=O)c1 50413292COc1cccc(Nc2c(CN)cnc3ccc(cc23)S(=O)(=O)c2ccccc2)c1 50413293CNC(=O)c1cnc2ccc(cc2c1Nc1cccc(OC)c1)S(C)(=O)=O 50413295COc1cccc(Nc2cc(nc3ccc(cc23)S(C)(=O)=O)C(N)=O)c1 50413296COc1cc(Nc2c(cnc3c(C)cc(cc23)S(C)(=O)=O)C(N)=O)ccc1F 50413297Cc1cc(cc2c(Nc3cccc(c3)C#N)c(cnc12)C(N)=O)S(C)(=O)=O 50413298COc1cccc(Nc2c(cnc3ccc(cc23)S(C)(=O)=O)C(N)=O)c1 50413299CS(=O)(=O)c1ccc2ncc(C(N)=O)c(Nc3cccc(Cl)c3)c2c1 50413300CS(=O)(=O)c1ccc2ncc(C(N)=O)c(Nc3cccnc3)c2c1 50413301COc1cc(Nc2c(cnc3ccc(cc23)S(C)(=O)=O)C(N)=O)ccc1F 50413303COc1cccc(Nc2c(cnc3ccc(cc23)S(C)(=O)=O)C#N)c1 50413306COc1cc(Nc2c(cnc3c(OC)cc(cc23)S(C)(=O)=O)C(N)=O)ccc1F 50413307CS(=O)(=O)c1ccc2ncc(C(N)=O)c(Nc3cccc(CN)c3)c2c1 50414989COc1cccc(Nc2c(cnc3ccc(cc23)S(=O)(=O)C2CCCC2)C(N)=O)c1 50414990COc1cccc(Nc2c(cnc3ccc(Sc4ccccc4)cc23)C(N)=O)c1 50414991COc1cccc(Nc2c(cnc3ccc(cc23)C(=O)N2CCOCC2)C(N)=O)c1 50414992COc1cccc(Nc2c(cnc3ccc(cc23)S(=O)(=O)N(C)C)C(N)=O)c1 50414993CCc1cccc(Nc2c(cnc3ccc(cc23)S(=O)(=O)c2ccccc2)C(N)=O)c1 50414994NC(=O)c1cnc2ccc(cc2c1Nc1cccc(c1)C#N)S(=O)(=O)c1ccccc1 50414995NC(=O)c1cnc2ccc(cc2c1NC1CCCCC1)S(=O)(=O)c1ccccc1 50414996NC(=O)c1cnc2ccc(cc2c1Nc1cccnc1)S(=O)(=O)c1ccccc1 50414997Cc1coc2CCCC(Nc3c(cnc4ccc(cc34)S(=O)(=O)c3ccccc3)C(N)=O)c12 50414998COc1ccc(cc1)S(=O)(=O)c1ccc2ncc(C(N)=O)c(Nc3cccc(OC)c3)c2c1 50414999COc1cccc(Nc2c(cnc3ccc(cc23)S(=O)(=O)c2cccc(c2)C(=O)N(C)C)C(N)=O)c1 50415000COc1cccc(Nc2c(cnc3ccc(cc23)S(=O)(=O)c2ccc(cc2)-c2ccoc2)C(N)=O)c1 50415002COc1cccc(Nc2c(cnc3ccccc23)C(N)=O)c1 50415003COc1cccc(Nc2c(cnc3ccc(cc23)C(=O)N(C)C)C(N)=O)c1 50415004COc1cccc(Nc2c(cnc3ccc(cc23)S(=O)(=O)N2CCOCC2)C(N)=O)c1 50415005NC(=O)c1cnc2ccc(cc2c1Nc1ccccc1)S(=O)(=O)c1ccccc1 50415006NC(=O)c1cnc2ccc(cc2c1Nc1ccc2ncsc2c1)S(=O)(=O)c1ccccc1 50415007COc1cccc(Nc2c(cnc3ccc(cc23)S(=O)(=O)c2ccc(cc2)C(C)(C)C)C(N)=O)c1 50415008COc1cccc(Nc2c(cnc3c(C)cc(cc23)S(=O)(=O)c2ccccc2)C(N)=O)c1 50415009COc1ccc(cc1)S(=O)(=O)c1cc(C)c2ncc(C(N)=O)c(Nc3cccc(OC)c3)c2c1 50415240Cc1cc(cc2C(Nc3cncc(Cl)c3)C(=NNc12)C(N)=O)S(C)(=O)=O 50415241CCn1nccc1NC1C(=NNc2c(C)cc(cc12)S(=O)(=O)CC)C(N)=O 50415242CS(=O)(=O)c1ccc2NN=C(C(Nc3cncc(Cl)c3)c2c1)C(N)=O 50415243CC(C)(C)S(=O)(=O)c1ccc2NN=C(C(Nc3cncc(F)c3)c2c1)C(N)=O 50415244CS(=O)(=O)c1cc(F)c2NN=C(C(Nc3cncc(F)c3)c2c1)C(N)=O 50415245Cc1cc(cc2c(Nc3cccc(c3)C#N)c(C(N)=O)c(=O)[nH]c12)S(C)(=O)=O 50415794CCn1ncc2c(Cl)c(cnc12)C(=O)NCc1ccc(C)cc1C 50425690CCOC(=O)C1=CN(Cc2ccc(OC)c(OC)c2)C=C(C1c1cccc(c1)[N+]([O-])=O)C(=O)OCC 50425691CCOC(=O)C1=CN(Cc2ccc(OC)c(OC)c2)C=C(C1c1c[nH]c2ccccc12)C(=O)OCC 50425692CCOC(=O)C1=CN(Cc2ccc(OC)c(OO)c2)C=C(C1c1cccc(F)c1)C(=O)OCC 50425693CCOC(=O)C1=CN(Cc2ccc(OC)c(OC)c2)C=C(C1c1ccc(Cl)cc1)C(=O)OCC 50428570COc1ccc(C2=NN(CCCCOc3ccc(cc3F)C3=NNC(=O)C3(C)C)C(=O)CC2C)c2cc(nn12)C(F)(F)F 50428571COc1ccc(C2=NN(CCCCOc3cccc(c3)C3=NNC(=O)C3(C)C)C(=O)CC2C)c2cc(nn12)C(F)(F)F 50428572COc1ccc(C2=NN(CCCCOc3cccc(c3)C3=NNC(=O)CC3C)C(=O)CC2C)c2cc(nn12)C(F)(F)F 50428573COc1ccc(C2=NN(CCCCOc3ccc(cc3)C3=NNC(=O)C3(C)C)C(=O)CC2C)c2cc(nn12)C(F)(F)F 50428574COc1ccc(C2=NN(CCCCOc3ccc(cc3)-c3ccc(=O)[nH]n3)C(=O)CC2C)c2cc(nn12)C(F)(F)F 50428575COc1ccc(C2=NN(CCCCOc3ccc(cc3)C3=NNC(=O)CC3)C(=O)CC2C)c2cc(nn12)C(F)(F)F 50428576COc1ccc(C2=NN(CCCCOc3ccc(cc3)-c3n[nH]c(=O)cc3C)C(=O)CC2C)c2cc(nn12)C(F)(F)F 50428577CCc1cc2c(ccc(OC)n2n1)C1=NN(CCCCOc2ccc(cc2)C2=NNC(=O)CC2C)C(=O)CC1C 50428578CCc1cc2c(ccc(OC)n2n1)C1=NN(CCCOc2ccc(cc2)C2=NNC(=O)CC2C)C(=O)CC1C 50428579COc1ccc(C2=NN(CCCCCOc3ccc(cc3)C3=NNC(=O)CC3C)C(=O)CC2C)c2cc(nn12)C(F)(F)F 50428580COc1ccc(C2=NN(CCCCOc3ccc(cc3)C3=NNC(=O)CC3C)C(=O)CC2C)c2cc(nn12)C(F)(F)F 50428581COc1ccc(C2=NN(CCCOc3ccc(cc3)C3=NNC(=O)CC3C)C(=O)CC2C)c2cc(nn12)C(F)(F)F 50428582COc1ccc(C2=NN(CCOc3ccc(cc3)C3=NNC(=O)CC3C)C(=O)CC2C)c2cc(nn12)C(F)(F)F 50428583COc1ccc(C2=NNC(=O)C[C@@H]2C)c2cc(nn12)C(F)(F)F 50428584COc1ccc(C2=NN(CCCCOc3ccc(C4=NNC(=O)C4(C)C)c(F)c3F)C(=O)C2(C)C)c2sc(nc12)C(F)(F)F 50428585COc1ccc(C2=NN(CCCCOc3ccc(C4=NNC(=O)C4(C)C)c(F)c3F)C(=O)C2(C)C)n2cc(nc12)C(F)(F)F 50428586COc1ccc(C2=NN(CCCCOc3ccc(C4=NNC(=O)CC4)c(F)c3F)C(=O)C2(C)C)c2sc(nc12)C(F)(F)F 50428587COc1ccc(C2=NN(CCCCOc3ccc(C4=NNC(=O)CC4)c(F)c3F)C(=O)C2(C)C)n2cc(nc12)C(F)(F)F 50428588CCc1cc2c(ccc(OC)n2n1)C1=NN(CCCCOc2ccc(cc2)C2=NNC(=O)CC2C)C(=O)C1(C)C 50428589CCc1cc2c(ccc(OC)n2n1)-c1ccc(=O)n(CCCCOc2ccc(cc2)C2=NNC(=O)CC2C)n1 50428590CCc1cc2c(ccc(OC)n2n1)C1=NN(CCCCOc2ccc(cc2)C2=NNC(=O)CC2C)C(=O)CC1 50428591COc1ccc(C2=NN(CCCCOc3ccc(C4=NNC(=O)CC4)c(F)c3F)C(=O)CC2C)c2cc(nn12)C(F)(F)F 50428592COc1ccc(C2=NN(CCCCOc3ccc(C4=NNC(=O)C4(C)C)c(F)c3F)C(=O)CC2C)c2cc(nn12)C(F)(F)F 50428593COc1ccc(C2=NN(CCCCOc3ccc(C4=NNC(=O)C4(C)C)c(F)c3)C(=O)CC2C)c2cc(nn12)C(F)(F)F 50429685COc1ccc(cc1OC)C1=NN(CCCCCCNCC(O)c2ccc(O)c(CO)c2)C(=O)C2CCCCC12 50429686COc1ccc(cc1OC)C1=NN(CCCCCNCC(O)c2ccc(O)c(CO)c2)C(=O)C2CCCCC12 50429687COc1ccc(cc1OC)C1=NN(CCCCNCC(O)c2ccc(O)c(CO)c2)C(=O)C2CCCCC12 50429688COc1ccc(cc1OC)C1=NN(CCNCC(O)c2ccc(O)c(CO)c2)C(=O)C2CCCCC12 50429689COc1ccc(cc1OCCCCCCNCC(O)c1ccc(O)c(CO)c1)C(=O)Nc1c(Cl)cncc1Cl 50429690COc1ccc(cc1OCCCCCNCC(O)c1ccc(O)c(CO)c1)C(=O)Nc1c(Cl)cncc1Cl 50429691COc1ccc(cc1OCCCCNCC(O)c1ccc(O)c(CO)c1)C(=O)Nc1c(Cl)cncc1Cl 50429692COc1ccc(cc1OCCCNCC(O)c1ccc(O)c(CO)c1)C(=O)Nc1c(Cl)cncc1Cl 50430301NS(=O)(=O)c1cc2nc(-c3cc(Br)ccc3F)n3c2c(c1)oc1ccccc31 50430302NS(=O)(=O)c1cc2nc(-c3cccc(Br)c3)n3c2c(c1)oc1ccccc31 50430303NS(=O)(=O)c1cc2nc(-c3ccccc3O)n3c2c(c1)oc1ccccc31 50451480COc1ccc(cc1OC1Cc2ccccc2C1)[C@@H](C)Cn1cc[nH]\c1=N/C#N