11[H][C@]1(CO)O[C@]2([H])O[C@]3([H])[C@@]([H])(CO)O[C@]([H])(O[C@]4([H])[C@@]([H])(CO)O[C@]([H])(O[C@]5([H])[C@@]([H])(CO)O[C@]([H])(O[C@]6([H])[C@@]([H])(CO)O[C@]([H])(O[C@]7([H])[C@@]([H])(CO)O[C@]([H])(O[C@]8([H])[C@@]([H])(CO)O[C@]([H])(O[C@@]1([H])[C@]([H])(O)[C@@]2([H])O)[C@]([H])(O)[C@@]8([H])O)[C@]([H])(O)[C@@]7([H])O)[C@]([H])(O)[C@@]6([H])O)[C@]([H])(O)[C@@]5([H])O)[C@]([H])(O)[C@@]4([H])O)[C@]([H])(O)[C@@]3([H])O 21COc1cc2c(Nc3ccc(Br)cc3F)ncnc2cc1OCC1CCN(C)CC1 2579CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13 3079Cc1ccc(Nc2ncc3cc(-c4c(Cl)cccc4Cl)c(=O)n(C)c3n2)cc1 3083Cn1c2nc(Nc3cccc(O)c3)ncc2cc(-c2c(Cl)cccc2Cl)c1=O 3084Cn1c2nc(Nc3ccc(O)cc3)ncc2cc(-c2c(Cl)cccc2Cl)c1=O 3085Cn1c2nc(Nc3cccc(CO)c3)ncc2cc(-c2c(Cl)cccc2Cl)c1=O 3532COc1cc2ncnc(Nc3cccc(Cl)c3)c2cc1OC 4552COc1cc(Nc2c(cnc3cc(OCCCN4CCN(C)CC4)c(OC)cc23)C#N)c(Cl)cc1Cl 4779Fc1ccc(Nc2ncnc3cc(OCCCN4CCOCC4)c(NC(=O)C=C)cc23)cc1Cl 4814CCN(CC)CCNC(=O)c1c(C)[nH]c(\C=C2/C(=O)Nc3ccc(F)cc23)c1C 5446COCCOc1cc2ncnc(Nc3cccc(c3)C#C)c2cc1OCCOC 5447COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCCN1CCOCC1 5655CN1CC[C@@H]([C@H](O)C1)c1c(O)cc(O)c2c1oc(cc2=O)-c1ccccc1Cl 6568CSc1cccc(Nc2ncc3cc(-c4c(Cl)cccc4Cl)c(=O)n(C)c3n2)c1 6569Cn1c2nc(Nc3ccc(F)cc3)ncc2cc(-c2c(Cl)cccc2Cl)c1=O 6866Nc1nc(Nc2ccc(cc2)S(N)(=O)=O)nn1C(=O)c1c(F)cccc1F 9503FC(F)(F)c1cccc(NC(=O)c2ccccc2NCc2ccncc2)c1 12107CN1CCN(CC1)c1ccc(cc1)C(=O)Nc1[nH]nc2CN(Cc12)C(=O)Cc1cccs1 12255CN1CCN(CCOc2cc(OC3CCOCC3)c3c(Nc4c5OCOc5ccc4Cl)ncnc3c2)CC1 12621COc1ccc(F)c(F)c1C(=O)c1cnc(NC2CCN(CC2)S(C)(=O)=O)nc1N 12985CO[C@@H](C(=O)N1Cc2n[nH]c(NC(=O)c3ccc(cc3)N3CCN(C)CC3)c2C1)c1ccccc1 12987CO[C@H](C(=O)N1Cc2n[nH]c(NC(=O)c3ccc(cc3)N3CCN(C)CC3)c2C1)c1ccccc1 13216Cc1nc(Nc2ncc(s2)C(=O)Nc2c(C)cccc2Cl)cc(n1)N1CCN(CCO)CC1 13336CS(=O)c1ccc(cc1)-c1nc(c([nH]1)-c1ccc(F)cc1)-c1ccncc1 13530CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(Nc3nccc(n3)-c3cccnc3)c2)CC1 13533Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(OCCN2CCOCC2)c2ccccc12)C(C)(C)C 13534CN1CCN(CC1)c1cc(Nc2cc(C)n[nH]2)nc(Sc2ccc(NC(=O)C3CC3)cc2)n1 15244Fc1ccc(Sc2ccc3c(-c4c(Cl)cccc4Cl)c(=O)ncn3n2)c(F)c1 16673CNC(=O)c1cc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(c3)C(F)(F)F)cc2)ccn1 21079Cc1ccc(F)c(NC(=O)Nc2ccc(cc2)-c2cccc3[nH]nc(N)c23)c1 24466COc1ccc2c(Oc3ccc(NC(=O)c4c(C)n(CC(C)(C)O)n(-c5ccccc5)c4=O)nc3)ccnc2c1 24773CC1(C)CNc2cc(NC(=O)c3cccnc3NCc3ccncc3)ccc12 25084Nc1nc(N)c2nc(-c3cccc(O)c3)c(nc2n1)-c1cccc(O)c1 25117CNC(=O)c1ccccc1Sc1ccc2c(\C=C\c3ccccn3)n[nH]c2c1 25118CN1CCN(CC1)c1ccc2nc([nH]c2c1)-c1c(N)c2c(F)cccc2[nH]c1=O 25121CC[C@H]1N(C2CCCC2)c2nc(Nc3ccc(cc3OC)C(=O)NC3CCN(C)CC3)ncc2N(C)C1=O 25617CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(Cl)cc23)c1F 25628OCCn1cc(c(n1)-c1ccncc1)-c1ccc2C(CCc2c1)N=O 26300CCN(CCO)CCCOc1ccc2c(Nc3cc(CC(=O)Nc4cccc(F)c4)n[nH]3)ncnc2c1 26373Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1C(=O)Nc1cncnc1 26474CN(c1ccc2c(C)n(C)nc2c1)c1ccnc(Nc2ccc(C)c(c2)S(N)(=O)=O)n1 27087O=C(NC1CC1)Nc1c[nH]nc1-c1nc2ccc(CN3CCOCC3)cc2[nH]1 31085CCN1CCN(Cc2ccc(NC(=O)Nc3ccc(Oc4cc(NC)ncn4)cc3)cc2C(F)(F)F)CC1 31088Cn1c(Nc2ccc(cc2)C(F)(F)F)nc2cc(Oc3ccnc(c3)-c3ncc([nH]3)C(F)(F)F)ccc12 31090CCOc1cc2ncc(C#N)c(Nc3ccc(F)c(Cl)c3)c2cc1NC(=O)\C=C\CN(C)C 31093OC(=O)c1ccc(Nc2ncc3CN=C(c4cc(Cl)ccc4-c3n2)c2c(F)cccc2F)cc1 31095Cc1[nH]c(\C=C2/C(=O)Nc3ccc(F)cc23)c(C)c1C(=O)NC[C@H](O)CN1CCOCC1 31829CCC(=O)Nc1ccc2ncnc(Nc3ccc(NC(=O)Nc4cc(nn4-c4cccc(C)c4)C(C)(C)C)cc3)c2c1 32102Cn1ncnc2c1nc(=O)n(C)c2=O 34671Cc1nn(C)c2nc(=O)n(C)c(=O)c2n1 34751COc1cc(OC)c(cc1OC)-c1c2cc(O)c(O)cc2oc2cc(=O)c(O)cc12 34905CCCc1nn(C)c2nc(=O)n(C)c(=O)c2n1 36408COc1ccc(cc1OC)-c1nn(C2CCC2)c2ncnc(N)c12 36409CC(C)n1nc(-c2cc3cc(O)ccc3[nH]2)c2c(N)ncnc12 38020CCC(C)(C)n1nnnc1C(N1CCCc2ccccc12)c1cccnc1 42546CCOC(=O)CCCCC(=O)c1[nH]c(=O)[nH]c1CSc1nnc2c3ccccc3n(C(C)C)c2n1 42775CC1NC(=O)NC1CCCCCC(=O)Nc1ccc(C)cc1 44685CCOC(=O)CCCCC(=O)c1[nH]c(=O)[nH]c1CSc1nc(-c2ccccc2)c(C#N)c(=O)[nH]1 63161CCCn1c2ccccc2c2nnc(SCc3[nH]c(=O)[nH]c3C(=O)CCCCC(=O)OCC)nc12 66175CC1NC(=O)NC1CCCCCC(=O)Nc1c(C)cccc1C 66184C[C@@H]1NC(=O)N[C@@H]1CCCCCC(O)=O 66219O=c1cc(OCc2ccccc2)cc[nH]1 81374Cc1cc(C)n2B(F)[N+]3=C(CCC(=O)NCCCCC(=O)NCCOc4ccc(Nc5ncnc(n5)-c5cccnc5Nc5cc(NC(=O)c6cccc(c6)C(F)(F)F)ccc5C)cc4)C=CC3=Cc12 81375Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1Nc1ncccc1-c1ncnc(Nc2ccc(OCCNC(=O)COCCOCCOCCOCCN)cc2)n1 81376Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1Nc1ncccc1-c1cc(Nc2ccc(OCCNC(=O)COCCOCCOCCOCCN)cc2)ncn1 83833[H]C12CC3([H])CC([H])(C1)CC(CNC(=O)CC1C[C@H](C(=O)N4CCN(CC4)C(=O)c4ccco4)[C@]4(CC)N(CCc5c4[nH]c4ccc(OC)cc54)C1=O)(C2)C3 87385N#CC12CCCCC1CC1CCCCC1(C#N)N2Cc1cccnc1 87391COc1cc(ccc1OC(C)=O)C(=O)Nc1ccc(O)cc1C(O)=O 87395Cc1oc2nc(SCCCC(=O)NCCO)nc(N)c2c1C 87396COC(=O)CCSCc1cn2cc(Cl)ccc2n1 87398CCc1nnc(NC(=O)CCc2nc(no2)C2=CCN(C)CC2)s1 87399CCOC(=O)CCCCC(=O)c1[nH]c(=O)[nH]c1CSc1nc2ccccc2[nH]1 87403COc1ccc(CCNc2cc(=O)[nH]c(N)n2)cc1 87404CCOC(=O)CCCCC(=O)c1[nH]c(=O)[nH]c1CN1CCOCC1 87408CCOC(=O)CCCCC(=O)c1[nH]c(=O)[nH]c1CSc1nc(C)cc(=O)[nH]1 87409CCOC(=O)CCCCC(=O)c1[nH]c(=O)[nH]c1Cn1cnc2ccccc12 87410COc1ccc2nc(NC(=O)CCc3nc(no3)C3=CCN(C)CC3)sc2c1 87413CCCCSCc1[nH]c(=O)[nH]c1C(=O)CCCCC(=O)OCC 87414CCOC(=O)CCCCC(=O)c1[nH]c(=O)[nH]c1CSc1nc(C)cc(C)n1 87415Cn1c2nc(-n3ccnc3)n(Cc3ccc(Cl)cc3Cl)c2c(=O)n(C)c1=O 87417CCCCN1C2NC(=O)NC2NC1=O 87419CCCCN1C2NC(=O)NC2N(C)C1=O 87421CCOC(=O)CCCCC(=O)c1[nH]c(=O)[nH]c1CSCCO 87423COc1cccc(CSc2nnc(CSc3nc4nc(C)cc(C)n4n3)s2)c1 87426Cc1[nH]c(=O)[nH]c1C(=O)CCCCC(O)=O 87427CCOC(=O)CCCCC(=O)c1[nH]c(=O)[nH]c1CSc1nnc2c3ccccc3n(CC=C)c2n1 87431CC(=O)Nc1ccc(NC(=O)C2CCN(CC2)C(=O)c2cccs2)cc1 87432CC1NC(=O)NC1CCCCCC(=O)Nc1ccc(F)cc1 87434CCc1cccc(NC(=O)CCCCCC2NC(=O)NC2C)c1 87443CCOC(=O)N1CCN(CC1)C(=O)Nc1ccc(NC(=O)N2CCN(CC2)C(=O)OCC)cc1 87446CC1NC(=O)NC1CCCCCC(=O)Nc1ccc(F)c(Cl)c1 87447CC1NC(=O)NC1CCCCCC(=O)Nc1cccc(F)c1C 87448CCOC(=O)CCCCC(=O)c1[nH]c(=O)[nH]c1C[n+]1ccc(C)cc1 87455COC(=O)Nc1csc2CCCCC(=O)Nc12 87466COc1ccc(cc1)C1c2c(Oc3nc[nH]c(=O)c13)nc[nH]c2=O 87470CCOc1ccc(CCNC(=O)CN2c3cc(C)ccc3Oc3ncccc3C2=O)cc1OCC 87475CSc1ccccc1OCc1cc(no1)C(=O)N1CCNC(=O)C1 87481CC12CCC(=O)N1C(CS2)C(=O)Nc1nnc(SCc2ccccc2F)s1 87482COc1ccc(CC(=O)Oc2ccc(C)cc2Br)cc1OC 87484COc1ccc2oc(C(=O)NCC(N(C)C)c3ccco3)c(C)c2c1 87485CN(C)C(CNC(=O)c1oc2c(Cl)cccc2c1C)c1ccco1 87486CCN(CC)C(=O)c1ccc(NC(=O)c2cc(ccc2OC)S(=O)(=O)N2CCCCCC2)cc1 87487CN(Cc1c(F)cccc1Cl)C(=O)CNC(=O)c1ccc2OCOc2c1 87488CCN(CC(=O)Nc1ccc(NC(C)=O)cc1)C(=O)c1ccccc1SCc1c(C)noc1C 87489O=C(NCC(N1CCCC1)c1ccco1)c1ccccc1Sc1ccccc1C#N 87490COc1ccc(Cl)cc1NC(=O)CN(C)C(=O)c1cc(nc2ccccc12)-c1ccncc1 87492COc1ccc(NC(=O)CN(C)C(=O)Cc2ccc(s2)S(=O)(=O)N2CCOCC2)cc1 87493Cc1c(oc2ccc(Br)cc12)C(=O)NCCN1CCOCC1 87495CC(C)n1nccc1NC(=O)C(C)OC(=O)c1ccccc1NCCO 87500COc1ccc(cc1C(=O)Nc1ccc(cc1)C(=O)N(C)C)S(=O)(=O)N1CCCCCC1 87502CN(C1CC1)C(=O)c1ccc(NC(=O)Cc2ccc(NC(=O)C3CCN(CC3)C(=O)C3CC3)cc2)cc1 87503CN(C1CC1)C(=O)c1ccc(NC(=O)Cc2ccc(NC(=O)C3CCN(CC3)C(=O)c3ccccc3)cc2)cc1 87508O=c1cc(SCc2ccccc2)nc[nH]1 87510CCOC(=O)N1CCC(CC1)NC(=O)CCc1nc(no1)C1=CCN(C)CC1 87519CN(CCc1ccccc1)C(=O)c1ccc(NC(=O)Cc2ccc(NC(=O)C3CCN(CC3)C(=O)C3CCCC3)cc2)cc1 87520O=C(Cc1ccc(NC(=O)C2CCN(CC2)C(=O)C2CCCCC2)cc1)Nc1ccc(cc1)C(=O)N1CCOCC1 87522O=C(Cc1ccc(NC(=O)C2CCN(CC2)C(=O)C2CCCC2)cc1)Nc1ccc(cc1)C(=O)N1CCOCC1 87527O=C(Cc1ccc(NC(=O)C2CCN(CC2)C(=O)c2ccccc2)cc1)Nc1ccc(cc1)C(=O)N1CCOCC1 87529CN(CCc1ccccc1)C(=O)c1ccc(NC(=O)Cc2ccc(NC(=O)C3CCN(CC3)C(=O)c3ccccc3)cc2)cc1 92347CCC(=O)Nc1ccc2ncnc(Nc3ccc(NC(=O)Nc4cc(nn4-c4cccc(N)c4)C(C)(C)C)cc3)c2c1 92348CN(C)CCCC(=O)Nc1ccc2ncnc(Nc3ccc(NC(=O)Nc4cc(nn4-c4cccc(N)c4)C(C)(C)C)cc3)c2c1 50004348Cc1nn(C)c2nnc(Nc3ccc(cc3)S(=O)(=O)N3CCNCC3)nc12 50004350Cc1nn(C)c2nnc(Nc3ccc(cc3)S(=O)(=O)N3CCCNCC3)nc12 50007080NCCNC(=O)c1ccc(cc1)S(=O)(=O)Oc1ccc(\C=C\[N+]([O-])=O)cc1 50020310CN1CCN(CCC(=O)Nc2c(C)[nH]c(\C=C3/C(=O)Nc4ccc(F)cc34)c2C)CC1 50027326Oc1ccc(C[C@H]2NCCc3cc(O)c(O)cc23)cc1O 50045408Nc1cccc(Nc2nccc(n2)-c2ccncc2)c1 50045424N(c1ccccc1)c1nccc(n1)-c1cccnc1 50045481N(c1cccc(c1)-n1ccnc1)c1nccc(n1)-c1cccnc1 50045485Clc1cccc(Nc2nccc(n2)-c2cccnc2)c1 50045526C(Cn1ccnc1)Oc1cccc(Nc2nccc(n2)-c2cccnc2)c1 50045528Nc1cccc(Nc2nccc(n2)-c2cccnc2)c1 50051304Cc1[nH]c2ncnc(Nc3cccc(C)c3)c2c1C 50051312Cc1[nH]c2ncnc(Nc3cccc(Br)c3)c2c1C 50051319Cc1[nH]c2ncnc(Nc3ccccc3)c2c1C 50056938Cc1c2cc(O)c(O)cc2oc2cc(=O)c(O)cc12 50059889CN[C@@H]1CC2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13 50067643CCCCN(CCCC)C(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](Cc1ccc(OP(O)(O)=O)cc1)NC(C)=O)C(C)C 50067644CCCCCCN(CCCCCC)C(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](Cc1ccc(OP(O)(O)=O)cc1)NC(C)=O)C(C)C 50067661CCCCCCN(CCCCCC)C(=O)[C@@H](C)NC(=O)[C@@H](NC(=O)[C@H](Cc1ccc(OP(O)(O)=O)cc1)NC(C)=O)C(C)C 50088898COc1cccc(c1)-c1cn(-c2ccc(CC(=O)NCCO)cc2)c2ncnc(N)c12 50088899COc1cccc(c1)-c1cn(-c2ccc(CNCCO)cc2)c2ncnc(N)c12 50088900Nc1ncnc2n(cc(-c3ccccc3)c12)-c1ccccc1 50088902Nc1ncnc2n(cc(-c3ccccc3)c12)-c1cccc(CO)c1 50088903COc1cccc(c1)-c1cn(-c2ccc(CCN(C)CCO)cc2)c2ncnc(N)c12 50088904COc1cccc(c1)-c1cn(-c2cccc(CO)c2)c2ncnc(N)c12 50088907Nc1ncnc2n(cc(-c3ccccc3)c12)-c1ccccc1CO 50088908COc1cccc(c1)-c1cn(-c2ccccc2)c2ncnc(N)c12 50088909Nc1ncnc2n(cc(-c3ccccc3)c12)-c1ccc(CO)cc1 50088910Nc1ncnc2n(cc(-c3cccc(Cl)c3)c12)-c1ccccc1 50088912Nc1ncnc2n(cc(-c3ccccc3)c12)-c1ccc(CNCCO)cc1 50088913COc1ccc(cc1)-c1cn(-c2ccccc2)c2ncnc(N)c12 50091935CC(C)(C)c1cc(NC(=O)Nc2cccc(Cl)c2Cl)n(n1)-c1cccc(N)c1 50097936Nc1ncnc2n(cc(-c3ccccc3)c12)C1CCC1 50097937Nc1ncnc2n(cc(-c3ccccc3)c12)C1CCC(O)C1 50097938Nc1ncnc2n(cc(-c3ccccc3)c12)C1CC(O)C1 50097939COc1cccc(c1)-c1cn(C2CCCC2)c2ncnc(N)c12 50097940COc1cccc(c1)-c1cn(C2CC(CNCCO)C2)c2ncnc(N)c12 50097941Nc1ncnc2n(cc(-c3ccc(O)cc3)c12)C1CCCC1 50097942Nc1ncnc2n(cc(-c3cccc(O)c3)c12)C1CCC1 50097944COc1cccc(c1)-c1cn(C2CC(C2)C(=O)NCCO)c2ncnc(N)c12 50097945COc1cccc(c1)-c1cn(C2CCC2)c2ncnc(N)c12 50097946COc1ccc(CC(CO)n2cc(-c3cccc(O)c3)c3c(N)ncnc23)cc1 50097947NA 50097948COc1ccc(CC(CO)n2cc(-c3cccc(OC)c3)c3c(N)ncnc23)cc1 50097951Nc1ncnc2n(cc(-c3ccc(O)cc3)c12)C1CCC1 50097953Nc1ncnc2n(cc(-c3ccccc3)c12)C(CO)Cc1ccc(O)cc1 50097954COc1ccc(cc1)-c1cn(C2CCCC2)c2ncnc(N)c12 50097955Nc1ncnc2n(cc(-c3ccccc3)c12)C1CCCC1 50097956Nc1ncnc2n(cc(-c3cccc(O)c3)c12)C1CCCC1 50097958CN(C)C(=O)CN1CCC(CC1)n1cc(-c2cccc(O)c2)c2c(N)ncnc12 50097959COCCNCCN1CCC(CC1)n1cc(-c2cccc(OC)c2)c2c(N)ncnc12 50097960COc1cccc(c1)-c1cn(C2CCN(CC(N)=O)C2)c2ncnc(N)c12 50097961COc1cccc(c1)-c1cn(C2CCN(CC(=O)N(C)C)CC2)c2ncnc(N)c12 50097962NC(=O)CN1CCC(C1)n1cc(-c2cccc(O)c2)c2c(N)ncnc12 50097963COCCN(C)CCN1CCC(CC1)n1cc(-c2cccc(OC)c2)c2c(N)ncnc12 50097964COc1cccc(c1)-c1cn(C2CCN(CC(N)=O)CC2)c2ncnc(N)c12 50097966COc1cccc(c1)-c1cn(C2CCN(C2)C(=O)OC(C)(C)C)c2ncnc(N)c12 50097967Nc1ncnc2n(cc(-c3cccc(O)c3)c12)C1CCN(CCO)CC1 50097968CC(C)(C)OC(=O)N1CCC(C1)n1cc(-c2cccc(O)c2)c2c(N)ncnc12 50097971COC(=O)CN1CCC(CC1)n1cc(-c2cccc(O)c2)c2c(N)ncnc12 50097972Nc1ncnc2n(cc(-c3cccc(O)c3)c12)C1CCNC1 50097973COc1cccc(c1)-c1cn(C2CCN(CCO)CC2)c2ncnc(N)c12 50097974COc1cccc(c1)-c1cn(C2CCN(CCN(C)CCO)CC2)c2ncnc(N)c12 50097978Nc1ncnc2n(cc(-c3ccc(O)cc3)c12)C1CCNC1 50097979NC(=O)CN1CCC(CC1)n1cc(-c2cccc(O)c2)c2c(N)ncnc12 50097980COC(=O)CN1CCC(CC1)n1cc(-c2cccc(OC)c2)c2c(N)ncnc12 50097987COc1cccc(c1)-c1cn(C2CCNC2)c2ncnc(N)c12 50097989COC(=O)CN1CCC(C1)n1cc(-c2cccc(OC)c2)c2c(N)ncnc12 50097991COC(=O)CN1CCC(C1)n1cc(-c2cccc(O)c2)c2c(N)ncnc12 50121980O=C(Nc1cccc(c1)-c1cncc2ccccc12)c1ccccc1NCc1ccncc1 50132704COCCN=NNc1ccc(cc1)C(=O)Nc1cccc(Nc2nccc(n2)-c2cccnc2)c1 50132705Nc1ccc(cc1)C(=O)Nc1cccc(Nc2nccc(n2)-c2cccnc2)c1 50132706COCCN=NNc1cccc(Nc2nccc(n2)-c2cccnc2)c1 50132707CN(C)\N=N\c1ccc(cc1)C(=O)Nc1ccc(C)c(Nc2nccc(n2)-c2cccnc2)c1 50142880CSc1nc(NCCc2ccccc2)c2cnn(CC(Cl)c3ccccc3)c2n1 50142882CCCCNc1nc(SCC)nc2n(CC(Cl)c3ccccc3)ncc12 50142883CCOCCNc1nc(SC)nc2n(CC(Cl)c3ccccc3)ncc12 50142885CSc1nc(NCc2ccccc2)c2cnn(CC(Cl)c3ccccc3)c2n1 50142887CC(C)(C)n1nc(-c2ccc(Cl)cc2)c2c(N)ncnc12 50142889CCCCNc1nc(SC)nc2n(CC(Cl)c3ccccc3)ncc12 50145411CCCNc1nc(SC)nc2n(CC(Cl)c3ccccc3)ncc12 50145415CCN(CC)c1nc(SC)nc2n(CC(Cl)c3ccccc3)ncc12 50155560Cc1ccc(NC(=O)Nc2cccc(Cl)c2)cc1Nc1nccc(n1)-c1cccnc1 50155561CN1CCN(CC1)C(=O)Nc1ccc(C)c(Nc2nccc(n2)-c2cccnc2)c1 50155562Cc1ccc(NC(=O)Nc2cccc(c2)N2CCCC2)cc1Nc1nccc(n1)-c1cccnc1 50155563CN(Cc1ccccc1NC(=O)Nc1ccc(C)c(Nc2nccc(n2)-c2cccnc2)c1)C1CCCCC1 50155567CN(C)c1cccc(NC(=O)Nc2ccc(C)c(Nc3nccc(n3)-c3cccnc3)c2)c1 50155568CCN(CC)c1cccc(NC(=O)Nc2ccc(C)c(Nc3nccc(n3)-c3cccnc3)c2)c1 50155574Cc1ccc(NC(=O)Nc2cccnc2)cc1Nc1nccc(n1)-c1cccnc1 50155575Cc1ccc(NC(=O)NCCN2CCCC2)cc1Nc1nccc(n1)-c1cccnc1 50161957CCOc1cc2ncc(C#N)c(Nc3ccc(OCc4ccccn4)c(Cl)c3)c2cc1NC(=O)\C=C\CN(C)C 50175491Cc1ccc(cc1)C(=O)Nc1ccc(C)c(Nc2nccc(n2)-c2cccnc2)c1 50175493O=C(Nc1cccc(Nc2nccc(n2)-c2cccnc2)c1)c1ccccc1 50178611CN1CCN(Cc2ccc(cc2Br)C(=O)Nc2ccc(C)c(Nc3nccc(n3)-c3cccnc3)c2)CC1 50178612CN(C)[C@H]1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)Nc2ccc(C)c(Nc3nccc(n3)-c3cncnc3)c2)C1 50178614CN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)Nc2ccc(C)c(Nc3nccc(n3)-c3cncnc3)c2)CC1 50178615CN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)Nc2ccc(C)c(Nc3nccc(n3)-c3cccnc3)c2)CC1 50178617CN1CCN(Cc2ccc(cc2F)C(=O)Nc2ccc(C)c(Nc3nccc(n3)-c3cccnc3)c2)CC1 50179207COc1cc2Cc3c(Nc4cccc(F)c4)[nH]nc3-c2cc1OC 50180753COC(=O)Nc1nc2ccc(cc2[nH]1)C(=O)c1ccccc1 50181670CN1CCN(CC1)c1ccc(NC(=O)c2cc(c[nH]c2=O)-c2ccc3OCOc3c2)cc1 50181672CN1CCN(CCc2ccc(NC(=O)c3cc(c[nH]c3=O)-c3ccc4OCOc4c3)cc2)CC1 50184807C[C@@H](O)COc1cn2ncnc(Oc3ccc4[nH]c(C)cc4c3F)c2c1C 50185169C1CCN(CC1)C1CCN(CC1)c1ccc2nc([nH]c2c1)-c1n[nH]c2ccc(Oc3ccccc3)cc12 50185170C1CCN(CC1)C1CCN(CC1)c1ccc2nc([nH]c2c1)-c1n[nH]c2ccccc12 50185178CC(C)(C)NC(=O)Nc1ccc2[nH]nc(-c3nc4ccc(cc4[nH]3)N3CCC(CC3)N3CCCCC3)c2c1 50185182C(Oc1ccc2[nH]nc(-c3nc4ccc(cc4[nH]3)N3CCC(CC3)N3CCCCC3)c2c1)c1ccccc1 50185184C(Oc1ccc2c(n[nH]c2c1)-c1nc2ccc(cc2[nH]1)N1CCC(CC1)N1CCCCC1)c1ccccc1 50186355COc1cccc(Oc2ccc3[nH]nc(-c4nc5ccc(cc5[nH]4)N4CCC(CC4)N4CCCCC4)c3c2)c1 50186356COc1cc2[nH]nc(-c3nc4ccc(cc4[nH]3)N3CCC(CC3)N3CCCCC3)c2cc1OCc1ccccc1 50186357COc1ccccc1Oc1ccc2[nH]nc(-c3nc4ccc(cc4[nH]3)N3CCC(CC3)N3CCCCC3)c2c1 50186358O=C(Nc1ccc2[nH]nc(-c3nc4ccc(cc4[nH]3)N3CCC(CC3)N3CCCCC3)c2c1)c1ccco1 50186359COc1ccc2[nH]nc(-c3nc4ccc(cc4[nH]3)N3CCC(CC3)N3CCCCC3)c2c1 50186360C(N1CCC(CC1)Nc1ccc2[nH]nc(-c3nc4ccc(cc4[nH]3)N3CCC(CC3)N3CCCCC3)c2c1)c1ccccc1 50186361C(Nc1ccc2[nH]nc(-c3nc4ccc(cc4[nH]3)N3CCC(CC3)N3CCCCC3)c2c1)c1ccco1 50186362C(Nc1ccc2[nH]nc(-c3nc4ccc(cc4[nH]3)N3CCC(CC3)N3CCCCC3)c2c1)c1nccs1 50186363COc1ccc(Oc2ccc3[nH]nc(-c4nc5ccc(cc5[nH]4)N4CCC(CC4)N4CCCCC4)c3c2)cc1 50186364C(Nc1ccc2[nH]nc(-c3nc4ccc(cc4[nH]3)N3CCC(CC3)N3CCCCC3)c2c1)c1ccccc1 50186365C(Oc1cc2[nH]nc(-c3nc4ccc(cc4[nH]3)N3CCC(CC3)N3CCCCC3)c2cc1OCc1ccccc1)c1ccccc1 50186757Oc1ccc(cc1)-c1ccccc1-c1cc(O)cc(O)c1 50186763COc1ccc(cc1)-c1ccccc1-c1cc(OC)cc(OC)c1 50186764COc1cc(OC)cc(\C=C\c2cccc(OC)c2O)c1 50187351Oc1ccc2[nH]c(cc2c1)C(=O)c1cc2cc(O)ccc2[nH]1 50187565Ic1ccccc1C(=O)Nc1nnc(CCc2ccccc2)s1 50187566Ic1ccc(cc1)C(=O)Nc1nnc(CCc2ccccc2)s1 50187569Ic1ccc(C=C2C(=O)NN(C2=O)c2ccc(I)cc2)cc1 50187571COc1cc(SC)ccc1C(=O)Nc1nnc(CCc2ccccc2)s1 50187572Clc1ccc(cc1Cl)N1NC(=O)C(=Cc2cccc(OCc3ccccc3)c2)C1=O 50187573Nc1ncnc2n[nH]c(-c3ccc(Cl)cc3)c12 50187574Cc1ccc(cc1C)N1NC(=O)C(=Cc2ccc(o2)-c2ccc(C)c(Cl)c2)C1=O 50187575Ic1ccc(cc1)N1NC(=O)C(=Cc2ccccc2)C1=O 50187579Brc1cc2OCOc2cc1C=C1C(=O)NN(C1=O)c1ccc(I)cc1 50193874Cc1cccc(C)c1-c1cc(C)c2nc(Nc3ccc(OCCN4CCCC4)cc3)nnc2c1 50193995C[C@@H]1CCN(C[C@@H]1N(C)c1ncnc2[nH]ccc12)C(=O)CC#N 50198782Cc1cc(cc2nnc(Nc3ccc(OCCN4CCCC4)cc3)nc12)-c1c(Cl)cccc1Cl 50198786Cc1cc(cc2nnc(Nc3ccc(cc3)S(=O)(=O)NCCN3CCCC3)nc12)-c1cc(N)ccc1Cl 50198813Cc1cc(cc2nnc(Nc3ccc(OCCN4CCCC4)cc3)nc12)-c1ccccc1Cl 50198826Cc1cc(cc2nnc(Nc3ccc(cc3)S(=O)(=O)NCCN3CCCC3)nc12)-c1c(O)cccc1Cl 50208746CN(C)C1CN(Cc2ccc(cc2C(F)(F)F)C(O)Nc2ccc(C)c(Nc3nccc(n3)-c3cncnc3)c2)C1 50208747CN(C)[C@@H]1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)Nc2ccc(C)c(Nc3nccc(n3)-c3cncnc3)c2)C1 50208748CN(C)C[C@@H]1CCN(Cc2ccc(cc2C(F)(F)F)C(O)Nc2ccc(C)c(Nc3nccc(n3)-c3cncnc3)c2)C1 50215054Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(-c2ccc(CN3CCOCC3)nc2)c2ccccc12)C(C)(C)C 50215557Cc1ccc(NC(=O)c2ccc(N)c(c2)C(F)(F)F)cc1Nc1nccc(n1)-c1cccnc1 50215558Cc1ccc(NC(=O)c2ccc(cc2)N(CCCl)CCCl)cc1Nc1nccc(n1)-c1cccnc1 50215559CN(CO)N=Nc1ccc(cc1)C(=O)Nc1ccc(C)c(Nc2nccc(n2)-c2cccnc2)c1 50215561CN=NNc1ccc(cc1Cl)C(=O)Nc1ccc(C)c(Nc2nccc(n2)-c2cccnc2)c1 50215562CN(CO)N=Nc1ccc(cc1C(F)(F)F)C(=O)Nc1ccc(C)c(Nc2nccc(n2)-c2cccnc2)c1 50215563CN(C)N=Nc1ccc(cc1C(F)(F)F)C(=O)Nc1ccc(C)c(Nc2nccc(n2)-c2cccnc2)c1 50215564CN(CCCl)Cc1ccc(cc1)C(=O)Nc1ccc(C)c(Nc2nccc(n2)-c2cccnc2)c1 50215565CN=NNc1ccc(cc1C(F)(F)F)C(=O)Nc1ccc(C)c(Nc2nccc(n2)-c2cccnc2)c1 50221516COc1cc2c(N[C@@H]3C[C@H]3c3ccccc3)c(cnc2cc1OCCCN1CCOCC1)C#N 50221517COCCOc1cc2ncc(C#N)c(N[C@@H]3C[C@H]3c3ccccc3)c2cc1OC 50221518COc1cc2ncc(C#N)c(N[C@@H]3C[C@H]3c3ccccc3)c2cc1OC 50221522NCc1ccc(cc1)-c1ccc2ncc(C#N)c(N[C@@H]3C[C@H]3c3ccccc3)c2c1 50221524COc1cc2c(N[C@@H]3C[C@H]3c3ccccc3)c(cnc2cc1OCCCc1cccnc1)C#N 50221527COc1cc2ncc(C#N)c(N[C@@H]3C[C@H]3c3ccccc3)c2cc1OCCCN1CCOCC1 50221528COc1cc2ncc(C#N)c(N[C@@H]3C[C@H]3c3ccccc3)c2cc1OCCCc1cccnc1 50221529N#Cc1cnc2cc(ccc2c1N[C@@H]1C[C@H]1c1ccccc1)-c1ccc(CN2CCOCC2)cc1 50221531COc1cc2c(N[C@@H]3C[C@H]3c3ccccc3)c(cnc2cc1OCCCN1CCN(C)CC1)C#N 50221546Cc1cc(cc2nnc(Nc3ccc(cc3)S(=O)(=O)NCCN3CCCC3)nc12)-c1c(Cl)ccc(O)c1Cl 50221547Cc1cc(cc2nnc(Nc3ccc(CCCN4CCCC4)cc3)nc12)-c1cc(O)ccc1Cl 50221548Cc1cc(cc2nnc(Nc3ccc(cc3)S(=O)(=O)NCCN3CCCC3)nc12)-c1cccc2[nH]ccc12 50221549Cc1cc(cc2nnc(Nc3ccc(cc3)S(=O)(=O)NCCN3CCCC3)nc12)-c1c(Cl)ccc(O)c1F 50221550Cc1cc(cc2nnc(Nc3ccc(cc3)S(=O)(=O)NCCN3CCCC3)nc12)-c1c(F)ccc(O)c1F 50221551Cc1cc(cc2nnc(Nc3ccc(cc3)S(=O)(=O)N3CCNCC3)nc12)-c1cc(O)ccc1Cl 50221552Cc1cc(cc2nnc(Nc3ccc(cc3)C(=O)N3CCS(=O)(=O)CC3)nc12)-c1cc(O)ccc1Cl 50221553Cc1cc(cc2nnc(Nc3ccc(cc3)S(=O)(=O)NCCN3CCCC3)nc12)-c1cc(O)ccc1Cl 50221554Cc1cc(cc2nnc(Nc3ccc(cc3)S(N)(=O)=O)nc12)-c1cc(O)ccc1Cl 50221555Cc1cc(cc2nnc(Nc3ccc(cc3)S(=O)(=O)CCCN3CCCC3)nc12)-c1cc(O)ccc1Cl 50221556Cc1cc(cc2nnc(Nc3ccc(cc3)S(=O)(=O)C3CCNCC3)nc12)-c1cc(O)ccc1Cl 50221557CN1CCN(CC1)C(=O)c1ccc(Nc2nnc3cc(cc(C)c3n2)-c2cc(O)ccc2Cl)cc1 50221558Cc1cc(cc2nnc(Nc3ccc(cc3)C(=O)NCCN3CCCC3)nc12)-c1cc(O)ccc1Cl 50221559CN(CCN1CCCC1)S(=O)(=O)c1ccc(Nc2nnc3cc(cc(C)c3n2)-c2cc(O)ccc2Cl)cc1 50221560CC(C)N(CCN1CCCC1)S(=O)(=O)c1ccc(Nc2nnc3cc(cc(C)c3n2)-c2cc(O)ccc2Cl)cc1 50221561CCN(CC)CCN1CCC(CC1)S(=O)(=O)c1ccc(Nc2nnc3cc(cc(C)c3n2)-c2cc(O)ccc2Cl)cc1 50221562Cc1cc(cc2nnc(Nc3ccc(cc3)S(=O)(=O)NCCN3CCCC3)nc12)-c1cc(O)ccc1Br 50221563Cc1cc(cc2nnc(Nc3ccc(cc3)C(=O)N3CCNCC3)nc12)-c1cc(O)ccc1Cl 50221564CN(CCN1CCOCC1)S(=O)(=O)c1ccc(Nc2nnc3cc(cc(C)c3n2)-c2cc(O)ccc2Cl)cc1 50221565CCN(CCN1CCCC1)S(=O)(=O)c1ccc(Nc2nnc3cc(cc(C)c3n2)-c2cc(O)ccc2Cl)cc1 50221566Cc1cc(cc2nnc(Nc3ccc(OCCN4CCCC4)cc3)nc12)-c1cc(O)ccc1Cl 50222913CC(C)NCc1ccc(Nc2cc(n[nH]2)-c2ccc(cc2)-c2ccc(O)cc2O)cc1 50224366ClC(Cn1ncc2c(Nc3cccc(Cl)c3)ncnc12)c1ccccc1 50224367CSc1nc(NCCc2ccccc2Cl)c2cnn(CC(Cl)c3ccccc3)c2n1 50224368CSc1nc(Nc2cccc(Cl)c2)c2cnn(CC(Cl)c3ccccc3)c2n1 50224369CCSc1nc(NCCc2ccccc2)c2cnn(CC(Cl)c3ccccc3)c2n1 50224370CSc1nc(NCc2ccccc2)c2cnn(CC(Cl)c3ccc(F)cc3)c2n1 50224371CCSc1nc(Nc2cccc(Cl)c2)c2cnn(CC(Cl)c3ccccc3)c2n1 50224372CSc1nc(NCc2ccc(F)cc2)c2cnn(CC(Cl)c3ccccc3)c2n1 50224373CSc1nc(NCCc2cccc(F)c2)c2cnn(CC(Cl)c3ccccc3)c2n1 50224374CSc1nc(NCc2ccccc2)c2cnn(CC(Cl)c3ccc(Cl)cc3)c2n1 50224376CCCSc1nc(Nc2cccc(Cl)c2)c2cnn(CC(Cl)c3ccccc3)c2n1 50224377CSc1nc(NCc2ccccc2F)c2cnn(CC(Cl)c3ccccc3)c2n1 50224379CSc1nc(NCCc2ccc(C)cc2)c2cnn(CC(Cl)c3ccccc3)c2n1 50224380CSc1nc(NCCc2cccc(Cl)c2)c2cnn(CC(Cl)c3ccccc3)c2n1 50224381CSc1nc(Nc2cccc(F)c2)c2cnn(CC(Cl)c3ccccc3)c2n1 50224382CSc1nc(Nc2cccc(Br)c2)c2cnn(CC(Cl)c3ccc(F)cc3)c2n1 50224383CSc1nc(NCCc2ccccc2)c2cnn(CC(Cl)c3ccc(Cl)cc3)c2n1 50224384CSc1nc(NCc2cccc(F)c2)c2cnn(CC(Cl)c3ccccc3)c2n1 50224385CSc1nc(Nc2ccccc2)c2cnn(CC(Cl)c3ccccc3)c2n1 50224387CSc1nc(NCc2ccccc2Cl)c2cnn(CC(Cl)c3ccccc3)c2n1 50224388CSc1nc(Nc2cccc(Br)c2)c2cnn(CC(Cl)c3ccccc3)c2n1 50225370Cc1nc(Nc2ncc(s2)C(=O)Nc2c(C)cccc2Cl)cc(n1)N1CCN(CCF)CC1 50229961CC(C)(C)n1nc(-c2cccc3ccccc23)c2c(N)ncnc12 50229973Cc1nc(N)sc1-c1ccnc(Nc2cccc(c2)[N+]([O-])=O)n1 50230100Fc1ccc(CSc2nnc(NC(=O)c3ccc(F)cc3)s2)cc1 50234144CCN(CC)CCOc1ccc(Nc2cc(NC(=O)Nc3c(Cl)cccc3Cl)ncn2)cc1 50236856COc1cc2nccc(Oc3ccc4c(cccc4c3)C(=O)NC3CC3)c2cc1OC 50237710Cc1cn(cn1)-c1cc(NC(=O)c2ccc(C)c(Nc3nccc(n3)-c3cccnc3)c2)cc(c1)C(F)(F)F 50240406CC(=O)Nc1ccc(C)c(Nc2nccc(n2)-c2cccnc2)c1 50240407Cc1ccc(NC(=O)c2ccccc2)cc1Nc1nccc(n1)-c1cccnc1 50241420CC(C)(C)N1CN(C(=N)c2cn[nH]c12)c1ccc(Cl)cc1 50242737Cc1[nH]c(\C=C2/C(=O)Nc3ccc(cc23)S(=O)(=O)Cc2c(Cl)cccc2Cl)c(C)c1C(=O)N1CCC[C@@H]1CN1CCCC1 50242742COc1cc(ccc1Nc1ncc(Cl)c(Nc2ccccc2S(=O)(=O)C(C)C)n1)N1CCC(CC1)N1CCN(C)CC1 50244385CCCP(=O)(CCC)c1ccc(Nc2nc(nc3n(\C=C\c4c(C)cccc4C)cnc23)C(C)C)cc1 50244386CCCP(=O)(CCC)c1ccc(Nc2nc(nc3n(\C=C/c4c(C)cccc4C)cnc23)C(C)C)cc1 50244387CCCP(=O)(CCC)c1ccc(Nc2nc(nc3n(\C=C\c4ccccc4)cnc23)C(C)C)cc1 50244388CCCP(=O)(CCC)c1ccc(Nc2nc(nc3n(\C=C/c4ccccc4)cnc23)C(C)C)cc1 50244430Cc1cccc(C)c1\C=C\n1cnc2c(Nc3ccc(cc3)P(C)(C)=O)ncnc12 50244524Cc1cccc(Cl)c1\C=C\n1cnc2c(Nc3ccc(cc3)P(C)(C)=O)ncnc12 50244525CP(C)(=O)c1ccc(Nc2ncnc3n(\C=C\c4ccccc4Cl)cnc23)cc1 50244526CP(C)(=O)c1ccc(Nc2ncnc3n(\C=C\c4cccc5[nH]ccc45)cnc23)cc1 50244527CP(C)(=O)c1ccc(Nc2ncnc3n(\C=C\c4cccc5[nH]ncc45)cnc23)cc1 50244570CCCP(=O)(CCC)c1ccc(Nc2ncnc3n(\C=C\c4c(C)cccc4C)cnc23)cc1 50244571CN(C)c1nc(Nc2ccc(cc2)P(C)(C)=O)c2ncn(\C=C\c3c(C)cccc3C)c2n1 50244572Cc1cccc(C)c1\C=C\n1cnc2c(Nc3ccc(cc3)P(C)(C)=O)nc(nc12)N1CCCC1 50244621Cc1cccc(C)c1\C=C\n1cnc2c(Nc3ccc(cc3)P(C)(C)=O)nc(nc12)N1CCOCC1 50244622CN1CCN(CC1)c1nc(Nc2ccc(cc2)P(C)(C)=O)c2ncn(\C=C\c3c(C)cccc3C)c2n1 50244623Cc1cccc(C)c1\C=C\n1cnc2c(Nc3ccc(cc3)P(C)(C)=O)nc(nc12)-n1ccnc1 50244624COc1nc(Nc2ccc(cc2)P(C)(C)=O)c2ncn(\C=C\c3c(C)cccc3C)c2n1 50244663CC(C)Oc1nc(Nc2ccc(cc2)P(C)(C)=O)c2ncn(\C=C\c3c(C)cccc3C)c2n1 50244664COCCOc1nc(Nc2ccc(cc2)P(C)(C)=O)c2ncn(\C=C\c3c(C)cccc3C)c2n1 50244666Cc1cccc(C)c1\C=C\n1cnc2c(Nc3ccc(cc3)P(C)(C)=O)nc(Oc3cccnc3)nc12 50244712CC(C)c1nc(Nc2ccc(cc2)P(C)(C)=O)c2ncn(\C=C\c3c(C)cccc3C)c2n1 50244713Cc1cccc(C)c1\C=C\n1cnc2c(Nc3ccc(cc3)P(C)(C)=O)nc(nc12)C1CCCC1 50247197CSc1nc(N2CCOCC2)c2cnn(CC(Cl)c3ccc(F)cc3)c2n1 50247198CSc1nc(NCc2ccc(F)cc2)c2cnn(CC(Cl)c3ccc(F)cc3)c2n1 50247199CSc1nc(NCc2ccccc2F)c2cnn(CC(Cl)c3ccc(F)cc3)c2n1 50247200CSc1nc(NCCc2ccccc2)c2cnn(CC(Cl)c3ccc(F)cc3)c2n1 50247201CSc1nc(N2CCOCC2)c2cnn(CC(Br)c3ccccc3)c2n1 50247202CSc1nc(NCc2ccccc2)c2cnn(CC(Br)c3ccccc3)c2n1 50247203CSc1nc(NCCc2ccccc2)c2cnn(CC(Br)c3ccccc3)c2n1 50247248CSc1nc(Nc2cccc(F)c2)c2cnn(CC(Cl)c3ccc(F)cc3)c2n1 50247249CCCNc1nc(SC)nc2n(CC(Cl)c3ccc(Cl)cc3)ncc12 50247250CCCCNc1nc(SC)nc2n(CC(Cl)c3ccc(Cl)cc3)ncc12 50247251CCN(CC)c1nc(SC)nc2n(CC(Cl)c3ccc(Cl)cc3)ncc12 50247252CSc1nc(N2CCOCC2)c2cnn(CC(Cl)c3ccc(Cl)cc3)c2n1 50247253CN(C)c1nc(NCc2ccccc2)c2cnn(CC(Cl)c3ccccc3)c2n1 50247254CCCNc1nc(nc2n(CC(Cl)c3ccccc3)ncc12)N(C)C 50247255CN(C)c1nc(N2CCOCC2)c2cnn(CC(Cl)c3ccccc3)c2n1 50247364CSc1nc(NCCc2ccccc2F)c2cnn(CC(Cl)c3ccccc3)c2n1 50247365CCCNc1nc(SC)nc2n(CC(Cl)c3ccc(F)cc3)ncc12 50247366CCCCNc1nc(SC)nc2n(CC(Cl)c3ccc(F)cc3)ncc12 50247367CCSc1nc(N(CC)CC)c2cnn(CC(Cl)c3ccccc3)c2n1 50247368CCCNc1nc(SCCC)nc2n(CC(Cl)c3ccccc3)ncc12 50247369CCCCNc1nc(SCCC)nc2n(CC(Cl)c3ccccc3)ncc12 50247370CCCSc1nc(N(CC)CC)c2cnn(CC(Cl)c3ccccc3)c2n1 50247371CCCSc1nc(NCc2ccccc2)c2cnn(CC(Cl)c3ccccc3)c2n1 50247385CCCNc1nc(SC)nc2n(CC(Br)c3ccccc3)ncc12 50247386CCCCNc1nc(SC)nc2n(CC(Br)c3ccccc3)ncc12 50247387CCOCCNc1nc(SC)nc2n(CC(Br)c3ccccc3)ncc12 50247388CSc1nc(N2CCCC2)c2cnn(CC(Br)c3ccccc3)c2n1 50247389CSc1nc(N2CCCCC2)c2cnn(CC(Br)c3ccccc3)c2n1 50247712CN(C)CCNC(=O)\C=C\c1ccc(\C=C2/Oc3ccccc3N(C)C2=O)s1 50247728CN1C(=O)\C(Oc2ccccc12)=C\c1ccc(\C=C\C(=O)NCc2cccnc2)s1 50247729CN1C(=O)\C(Oc2ccccc12)=C\c1ccc(\C=C\C(=O)NCc2ccncc2)s1 50247766O=C(Nc1ccc(cc1)N1CCOCC1)\C=C\c1ccc(\C=C2/Oc3ccccc3NC2=O)s1 50249542COc1cc(Nc2ncc(F)c(Nc3ccc4OC(C)(C)C(=O)Nc4n3)n2)cc(OC)c1OC 50255048OCc1ccc(o1)C(=O)NN=Cc1cc(C(O)=O)c(Nc2ccc(I)cc2F)c(F)c1F 50255049OC(=O)c1cc(C=NNC(=O)CS(=O)(=O)c2ccc(Cl)cc2)c(F)c(F)c1Nc1ccc(I)cc1F 50256927Cc1ccc(NCc2ccc(cc2)C(=O)Nc2ccccc2N)cc1Nc1nccc(n1)-c1cccnc1 50256928Cc1ccc(NCc2ccc(\C=C\C(=O)NO)cc2)cc1Nc1nccc(n1)-c1cccnc1 50256976Cc1ccc(NC(=O)c2ccc(cc2)C(=O)Nc2ccccc2N)cc1Nc1ncc(cn1)-c1cccnc1 50257031Nc1ccccc1NC(=O)c1ccc(cc1)C(=O)Nc1cccc(Nc2ncc(cn2)-c2cccnc2)c1 50257153Cc1ccc(NC(=O)c2ccc(cc2)C(=O)NO)cc1Nc1ncc(s1)-c1cccnc1 50257154ONC(=O)\C=C\c1ccc(cc1)C(=O)Nc1cccc(Nc2ncc(s2)-c2cccnc2)c1 50257155Cc1ccc(NC(=O)c2ccc(\C=C\C(=O)NO)cc2)cc1Nc1ncc(s1)-c1cccnc1 50257156ONC(=O)\C=C\c1ccc(s1)C(=O)Nc1cccc(Nc2ncc(s2)-c2cccnc2)c1 50257209Cc1ccc(NC(=O)c2ccc(\C=C\C(=O)NO)s2)cc1Nc1ncc(s1)-c1cccnc1 50260917Cc1ccn(-c2cccc(c2)C(F)(F)F)c(=O)c1-c1ccc2nc(N)ncc2c1 50262664O=C(Nc1ncc(Cc2ccccc2)s1)c1cccs1 50262665Fc1ccc(Cc2cnc(NC(=O)c3cccs3)s2)cc1 50262667COc1ccc-2c(Cc3sc(NC(=O)c4cccs4)nc-23)c1 50262668O=C(Nc1nnc(COc2ccccc2)s1)c1cccs1 50262669FC(F)(F)c1cccc(Cc2cnc(NC(=O)c3cccs3)s2)c1 50262670Clc1ccccc1Cc1cnc(NC(=O)c2cccs2)s1 50262671Fc1ccccc1Cc1cnc(NC(=O)c2cccs2)s1 50262714Clc1ccc(Cc2cnc(NC(=O)c3cccs3)s2)cc1 50262715Clc1cccc(Cc2cnc(NC(=O)c3cccs3)s2)c1 50262716FC(F)(F)c1ccc(Cl)c(Cc2cnc(NC(=O)c3cccs3)s2)c1 50262717Clc1ccc(Cc2cnc(NC(=O)c3cccs3)s2)c(Cl)c1 50262718COc1ccc(Cc2cnc(NC(=O)c3cccs3)s2)cc1 50262719Cc1ccc(Cc2cnc(NC(=O)c3cccs3)s2)cc1 50262720Fc1ccc(cc1)-c1cnc(NC(=O)c2cccs2)s1 50262721Clc1ccc(cc1)-c1cnc(NC(=O)c2cccs2)s1 50262722Cc1cccc(Cc2cnc(NC(=O)c3cccs3)s2)c1 50262723Clc1ccc(Cl)c(Cc2cnc(NC(=O)c3cccs3)s2)c1 50262724O=C(Nc1nnc(Cc2ccccc2)s1)c1cccs1 50277584CN1CCN(CC1)c1cc(Nc2cc(C)n[nH]2)nc(C=Cc2ccccc2)n1 50277623COc1c(NC(=O)Nc2ccc(-c3ccc(CN4CCOCC4)nc3)c3ccccc23)cc(cc1NS(C)(=O)=O)C(C)(C)C 50277639CCC(=O)Nc1ccc(Sc2nc(Nc3cc(C)n[nH]3)cc(n2)N2CCN(C)CC2)cc1 50287090Cc1ccc(NC(=O)c2ccc(Cl)cc2)cc1Nc1nccc(n1)-c1cccnc1 50287091Cc1ccc(NC(=O)c2ccc3ccccc3c2)cc1Nc1nccc(n1)-c1cccnc1 50287096COc1ccccc1C(=O)Nc1ccc(C)c(Nc2nccc(n2)-c2cccnc2)c1 50287097Cc1ccc(N)cc1Nc1nccc(n1)-c1cccnc1 50289742CC(=O)N[C@@H](Cc1ccc(OP(O)(O)=O)cc1)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCC1CCCCC1)C(N)=O 50289746CC[C@H](NC(=O)[C@H](Cc1ccc(cc1)C(F)(F)P(O)(O)=O)NC(C)=O)C(=O)N(C)CCCC1CCCCC1 50289747CC(=O)N[C@@H](Cc1ccc(cc1)C(F)(F)P(O)(O)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCC1CCCCC1)C(N)=O 50289748CC[C@H](C)[C@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](Cc1ccc(cc1)C(F)(F)P(O)(O)=O)NC(C)=O)C(=O)N[C@@H](CCC(O)=O)C(O)=O 50289750CN(CCCC1CCCCC1)C(=O)[C@H](CCC(O)=O)NC(=O)[C@H](Cc1ccc(cc1)C(F)(F)P(O)(O)=O)NC(C)=O 50290410OC(=O)c1cccc(Nc2nccc(n2)-c2cccnc2)c1 50290411O=C(Nc1cccc(Nc2nccc(n2)-c2cccnc2)c1)c1ccc(cc1)C#N 50290412Fc1ccc(cc1)C(=O)Nc1cccc(Nc2nccc(n2)-c2cccnc2)c1 50290413FC(F)C(F)(F)Oc1cccc(Nc2nccc(n2)-c2c[nH]c3ccccc23)c1 50290414OC(=O)c1ccccc1C(=O)Nc1cccc(Nc2nccc(n2)-c2cccnc2)c1 50290415NCCCNC(=O)c1cccc(Nc2nccc(n2)-c2cccnc2)c1 50290416NCCCn1ccc2c(cccc12)-c1ccnc(Nc2cccc(OC(F)(F)C(F)F)c2)n1 50290417O=C(Nc1cccc(Nc2nccc(n2)-c2cccnc2)c1)c1cccnc1 50290418COC(=O)c1cccc(Nc2nccc(n2)-c2cccnc2)c1 50290419O=C(Nc1cccc(Nc2nccc(n2)-c2cccnc2)c1)C1CCCCC1 50290421O=C(Nc1cccc(Nc2nccc(n2)-c2cccnc2)c1)c1ccncc1 50290422CN1CCN(Cc2ccc(cc2)C(=O)Nc2cccc(Nc3nccc(n3)-c3cccnc3)c2)CC1 50290424[O-][N+](=O)c1cccc(Nc2nccc(n2)-c2ccccn2)c1 50290427O=C(Nc1cccc(Nc2nccc(n2)-c2cccnc2)c1)c1cccs1 50290428O=C(Nc1cccc(Nc2nccc(n2)-c2cccnc2)c1)c1ccccn1 50290429COc1ccccc1C(=O)Nc1cccc(Nc2nccc(n2)-c2cccnc2)c1 50290430Cc1ccc(cc1)C(=O)Nc1cccc(Nc2nccc(n2)-c2cccnc2)c1 50290431CCCCCC(=O)Nc1cccc(Nc2nccc(n2)-c2cccnc2)c1 50293992Cc1cn(cn1)-c1cc(NC(=O)c2ccc(C)c(\C=C\n3cnc4cncnc34)c2)cc(c1)C(F)(F)F 50293993Cc1ccc(cc1\C=C\n1cnc2cncnc12)C(=O)Nc1cc(ccn1)C(F)(F)F 50293997Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1\C=C\n1cnc2c(Nc3ccncc3)ncnc12 50293999Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1\C=C\n1cnc2c(Nc3ccc(cc3)P(C)(C)=O)ncnc12 50294010Cc1ccc(cc1\C=C\n1cnc2c(NC3CC3)ncnc12)C(=O)Nc1cc(ccn1)C(F)(F)F 50294011Cc1cn(cn1)-c1cc(NC(=O)c2ccc(C)c(\C=C\n3cnc4c(NC5CC5)ncnc34)c2)cc(c1)C(F)(F)F 50294012Cc1ccc(cc1\C=C\n1cnc2c(NC3CC3)ncnc12)C(=O)Nc1cc(cc(c1)C(F)(F)F)-n1ccnc1 50297526COc1ccc(CNc2nc(SC)nc3n(CC(Cl)c4ccccc4)ncc23)cc1 50297527CSc1nc(NCCc2ccc(Cl)cc2)c2cnn(CC(Cl)c3ccccc3)c2n1 50298225CC(C)(C)n1nc(Cc2cccc3ccccc23)c2c(N)ncnc12 50299218COc1ccccc1-n1c(cn2c1nc1n(C)c(=O)[nH]c(=O)c21)-c1cc(O)ccc1C 50300026COCCOc1cc2ncnc(Nc3cccc(Cl)c3F)c2cc1NC(=O)[C@@H]1CCCN1C(=O)C=C 50300690CC(C)(C)c1cc(NC(=O)Nc2ccc(cc2)-c2cn3c(n2)sc2cc(OCCN4CCOCC4)ccc32)no1 50303221Cn1c2nc(Nc3ccc(I)cc3)ncc2cc(-c2c(Cl)cccc2Cl)c1=O 50303222Cn1c2nc(Nc3ccc(OC4OC(CO)C(O)C(O)C4O)cc3)ncc2cc(-c2c(Cl)cccc2Cl)c1=O 50303223Cn1c2nc(Nc3ccc(CCO)cc3)ncc2cc(-c2c(Cl)cccc2Cl)c1=O 50303224Cn1c2nc(Nc3ccc(N)cc3)ncc2cc(-c2c(Cl)cccc2Cl)c1=O 50303225CC(=O)Nc1ccc(Nc2ncc3cc(-c4c(Cl)cccc4Cl)c(=O)n(C)c3n2)cc1 50303226Cn1c2nc(Nc3ccc(NC(=O)CCl)cc3)ncc2cc(-c2c(Cl)cccc2Cl)c1=O 50303227CN1CCN(CC1)C(=O)c1ccc(Nc2ncc3cc(-c4c(Cl)cccc4Cl)c(=O)n(C)c3n2)cc1 50303228Cn1c2nc(Nc3ccc(NC(=O)CCNC(=O)OC(C)(C)C)cc3)ncc2cc(-c2c(Cl)cccc2Cl)c1=O 50303229Cn1c2nc(Nc3ccc(NCC(O)CO)cc3)ncc2cc(-c2c(Cl)cccc2Cl)c1=O 50303230Cn1c2nc(Nc3ccc(NC(=O)CCN)cc3)ncc2cc(-c2c(Cl)cccc2Cl)c1=O 50303231CCc1cccc(Nc2ncc3cc(-c4c(Cl)cccc4Cl)c(=O)n(C)c3n2)c1 50303232Cn1c2nc(Nc3cccc(COCC(O)CO)c3)ncc2cc(-c2c(Cl)cccc2Cl)c1=O 50303233Cn1c2nc(Nc3cccc(N)c3)ncc2cc(-c2c(Cl)cccc2Cl)c1=O 50303234CC(=O)Nc1cccc(Nc2ncc3cc(-c4c(Cl)cccc4Cl)c(=O)n(C)c3n2)c1 50306682C[C@@H](Oc1cc(cnc1N)-c1cnn(c1)C1CCNCC1)c1c(Cl)ccc(F)c1Cl 50307768COc1cc2ncnc(Nc3cccc(c3)C#C)c2cc1OCCCCCCC(=O)NO 50311985CN1C[C@@H]2C[C@H]1CN2c1ccc(cc1)-c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc(O)c1 50313643Cc1ccc(NC(=O)c2ccc(\C=C\C(=O)NO)cc2)cc1Nc1nc(cs1)-c1cccnc1 50313644Cc1cn(cn1)-c1cc(NC(=O)c2ccc(C)c(\C=C\N3CNc4c3ncnc4NC3CC3)c2)cc(c1)C(F)(F)F 50313645Nc1ncnc2n(nc(-c3cnc4[nH]ccc4c3)c12)C1CCCC1 50314344Cn1cc(\C=C2/Oc3cccc(O)c3C2=O)c2c(ccnc12)-c1ccc(cc1)C(=O)NCCO 50315231Fc1cc(cc(F)c1CN1CCOCC1)-c1cccc2ncc(nc12)-c1cnn(c1)C1CCNCC1 50317233COc1cc(Nc2c(cnc3cc(\C=C\CCN4CCN(C)CC4)c(OC)cc23)C#N)c(Cl)cc1Cl 50318870CCn1cnc2c(Nc3ccc(cc3)P(O)(=O)CP(O)(O)=O)nc(nc12)[C@H]1CC[C@H](N)CC1 50320203CC(C)COC(=O)Nc1ccc(cc1)-c1cnc2c(cnn2c1N)-c1ccc(cc1)N1CCN(C)CC1 50320700Fc1ccc(cc1)C(Cl)Cn1ncc2c(Nc3cccc(F)c3)ncnc12 50321649c1n[nH]cc1-c1cnc2ncc(cn12)-c1cn[nH]c1 50321650NCc1ccc(cc1)-c1cn2c(cnc2cn1)-c1cn[nH]c1 50321651OCc1ccc(cc1)-c1cn2c(cnc2cn1)-c1cn[nH]c1 50321738Nc1nc(SCC(=O)c2ccccc2)c(C#N)c(-c2ccsc2)c1C#N 50321943NS(=O)(=O)c1ccc(Nc2nc(nc3nc[nH]c23)N2CCOCC2)cc1 50322533Cc1cn(cn1)-c1cc(NC(=O)c2ccc(C)c(\C=C\n3cnc4c(N)ncnc34)c2)cc(c1)C(F)(F)F 50322534Cc1ccc(cc1C#Cn1cnc2c(NC3CC3)ncnc12)C(=O)Nc1cc(ccn1)C(F)(F)F 50322535CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc4cccnn34)cc2C(F)(F)F)CC1 50322536Cc1ccc(cc1\C=C\n1cnc2c(NC3CC3)ncnc12)C(=O)Nc1cc(on1)C(F)(F)F 50322537Cc1ccc(cc1C#Cn1cnc2c(NC3CC3)cccc12)C(=O)Nc1cc(on1)C(F)(F)F 50322538Cc1ccc(cc1C#Cc1cnc2c(N)cccn12)C(=O)Nc1cc(cc(c1)C(F)(F)F)-n1ccnc1 50322539CC(=O)Nc1cccn2c(cnc12)C#Cc1cc(ccc1C)C(=O)Nc1cc(cc(c1)C(F)(F)F)-n1ccnc1 50322540Cc1ccc(cc1C#Cc1cnc2ccccn12)C(=O)Nc1cc(cc(c1)C(F)(F)F)-n1ccnc1 50322541CN(C)Cc1nccn1-c1cc(NC(=O)c2ccc(C)c(c2)C#Cc2cnc3ccccn23)cc(c1)C(F)(F)F 50322542Cc1ccc(cc1C#Cc1cnc2ccccn12)C(=O)Nc1cc(cc(c1)C(F)(F)F)-n1cnc(CN2CCCC2)c1 50322543CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc4ccccn34)cc2C(F)(F)F)CC1 50322544CN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)Nc2ccc(C)c(c2)C#Cc2cnc3ccccn23)CC1 50322545CN1CCN(Cc2cc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc4ccccn34)cc(c2)C(F)(F)F)CC1 50322546Cc1ccc(cc1C#Cc1cnc2ccccn12)C(=O)Nc1ccc(CN2CCOCC2)c(c1)C(F)(F)F 50322547CN(C)[C@H]1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc4ccccn34)cc2C(F)(F)F)C1 50322548CN1CCCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc4ccccn34)cc2C(F)(F)F)CC1 50322549CN1CCC(CC1)Oc1ccc(NC(=O)c2ccc(C)c(c2)C#Cc2cnc3ccccn23)cc1C(F)(F)F 50322550CCN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc4ccccn34)cc2C(F)(F)F)CC1 50322551CC(C)N1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc4ccccn34)cc2C(F)(F)F)CC1 50322552Cc1ccc(cc1C#Cc1cnc2ccccn12)C(=O)Nc1ccc(CN2CCN(CCO)CC2)c(c1)C(F)(F)F 50322553Cc1ccc(cc1C#Cc1cnc2ccccn12)C(=O)Nc1ccc(CN2CCN(CCF)CC2)c(c1)C(F)(F)F 50322554Cc1ccc(cc1C#Cc1cnc2ccccn12)C(=O)Nc1ccc(CN2CCNCC2)c(c1)C(F)(F)F 50322555CC1CN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc4ccccn34)cc2C(F)(F)F)CCN1 50322556CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc4[nH]ccc4c3)cc2C(F)(F)F)CC1 50322557CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc4nc[nH]c4c3)cc2C(F)(F)F)CC1 50322558CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc4[nH]c(=O)[nH]c4c3)cc2C(F)(F)F)CC1 50322559CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc4NC(=O)COc4c3)cc2C(F)(F)F)CC1 50322560CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc4ncccn34)cc2C(F)(F)F)CC1 50322561CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc4cnccn34)cc2C(F)(F)F)CC1 50322562CCN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc4cccnn34)cc2C(F)(F)F)CC1 50322563Cc1ccc(cc1C#Cc1cnc2cccnn12)C(=O)Nc1ccc(CN2CCN(CCO)CC2)c(c1)C(F)(F)F 50322564Cc1ccc(cc1C#Cc1cnc2cccnn12)C(=O)Nc1ccc(CN2CCNCC2)c(c1)C(F)(F)F 50322565CN1CCN(Cc2ccc(NC(=O)c3cccc(c3)C#Cc3cnc4cccnn34)cc2C(F)(F)F)CC1 50322566CN1CCN(Cc2ccc(NC(=O)c3ccc(Cl)c(c3)C#Cc3cnc4cccnn34)cc2C(F)(F)F)CC1 50322567CN1CCN(Cc2ccc(NC(=O)c3ccc(F)c(c3)C#Cc3cnc4cccnn34)cc2C(F)(F)F)CC1 50322568CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc4cccnn34)cc2Cl)CC1 50322569CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc4cccnn34)cc2C2CC2)CC1 50322570Cc1ccc(cc1C#Cc1cnc2cccnn12)C(=O)Nc1cccc(c1)C(F)(F)F 50322571CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(CCc4cnc5cccnn45)c3)cc2C(F)(F)F)CC1 50322572CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(\C=C\c4cnc5cccnn45)c3)cc2C(F)(F)F)CC1 50322823CN(C)C\C=C\C(=O)Nc1cc2c(Nc3ccc(F)c(Cl)c3)ncnc2cc1O[C@H]1CCOC1 50323777CN1C(=O)N(Cc2cnc(Nc3ccc(C)nc3)nc12)c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C 50323778CN1C(=O)N(Cc2cnc(Nc3ccccc3)nc12)c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C 50325999NC(=O)c1cccc(c1)-c1cc(Nc2ccc(OC(F)(F)F)cc2)ncn1 50326061OC(=O)c1ccc(cc1)C(=O)C(\SCc1ccc(Br)cc1)=C/c1ccc(F)c(c1)[N+]([O-])=O 50326198CNc1nccc(n1)-c1cccnc1Oc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1C 50328120FC(F)(F)Oc1ccc(Nc2ncnc3n(Cc4ccccc4)ncc23)cc1 50328121FC(F)(F)Oc1ccc(Nc2ncnc3n(Cc4cccnc4)ncc23)cc1 50328122NC(=O)c1ccc(Cn2ncc3c(Nc4ccc(OC(F)(F)F)cc4)ncnc23)cc1 50328123FC(F)(F)Oc1ccc(Nc2ncnc3n(CC4CCOC4)ncc23)cc1 50328124CC(C)(C)n1ncc2c(Nc3ccc(OC(F)(F)F)cc3)ncnc12 50328125FC(F)(F)Oc1ccc(Nc2ncnc3n(Cc4ccncc4)ncc23)cc1 50328126Cc1nc(C)c(Cn2ncc3c(Nc4ccc(OC(F)(F)F)cc4)ncnc23)s1 50328127FC(F)(F)Oc1ccc(Nc2ncnc3n[nH]cc23)cc1 50328128OCCn1cc2c(Nc3ccc(OC(F)(F)F)cc3)ncnc2n1 50328129CCn1cc2c(Nc3ccc(OC(F)(F)F)cc3)ncnc2n1 50328130CCCn1cc2c(Nc3ccc(OC(F)(F)F)cc3)ncnc2n1 50328131FC(F)(F)Oc1ccc(Nc2ncnc3nn(cc23)C2CCCCC2)cc1 50328132NC(=O)Cn1cc2c(Nc3ccc(OC(F)(F)F)cc3)ncnc2n1 50328134FC(F)(F)Oc1ccc(Nc2ncnc3nn(Cc4cccnc4)cc23)cc1 50328135CS(=O)(=O)Nc1ccc(cc1)-c1cc(Nc2ccc(OC(F)(F)F)cc2)ncn1 50328136FC(F)(F)Oc1ccc(Nc2cc(ncn2)-c2cn[nH]c2)cc1 50328137Cn1cc(cn1)-c1cc(Nc2ccc(OC(F)(F)F)cc2)ncn1 50328138CN1CCN(CC1)C(=O)c1cc2c(Nc3ccc(OC(F)(F)F)cc3)ncnc2s1 50328139FC(F)(F)Oc1ccc(Nc2cc(NCCN3CCOCC3)ncn2)cc1 50328140FC(F)(F)Oc1ccc(Nc2cc(NCCCN3CCOCC3)ncn2)cc1 50328141FC(F)(F)Oc1ccc(Nc2cc(ncn2)N2CCOCC2)cc1 50328142FC(F)(F)Oc1ccc(Nc2cc(ncn2)-n2ccnc2)cc1 50328143NC(=O)c1cccc(Oc2cc(Nc3ccc(OC(F)(F)F)cc3)ncn2)c1 50328144NC(=O)c1cccc(Nc2cc(Nc3ccc(OC(F)(F)F)cc3)ncn2)c1 50328145NC(=O)c1ccc(cc1)-c1cc(Nc2ccc(OC(F)(F)F)cc2)ncn1 50328147FC(F)(F)Oc1ccc(Nc2cc(ncn2)-c2ccncc2)cc1 50328148NS(=O)(=O)c1cccc(c1)-c1cc(Nc2ccc(OC(F)(F)F)cc2)ncn1 50328149CS(=O)(=O)c1cccc(c1)-c1cc(Nc2ccc(OC(F)(F)F)cc2)ncn1 50328150Nc1cccc(c1)-c1cc(Nc2ccc(OC(F)(F)F)cc2)ncn1 50328151NS(=O)(=O)c1ccc(cc1)-c1cc(Nc2ccc(OC(F)(F)F)cc2)ncn1 50328152OCCNC(=O)c1cccc(c1)-c1cc(Nc2ccc(OC(F)(F)F)cc2)ncn1 50328153FC(F)(F)Oc1ccc(Nc2cc(ncn2)-c2cccc(c2)C(=O)NCCN2CCOCC2)cc1 50328154CNC(=O)c1cccc(c1)-c1cc(Nc2ccc(OC(F)(F)F)cc2)ncn1 50328155FC(F)(F)Oc1ccc(Nc2cc(ncn2)-c2cccc(c2)C(=O)N2CCOCC2)cc1 50328156CC(C)Cn1cc(cn1)-c1cc(Nc2ccc(OC(F)(F)F)cc2)ncn1 50328157Cc1c(cnn1-c1ccccc1)-c1cc(Nc2ccc(OC(F)(F)F)cc2)ncn1 50328158Cc1nn(C)c(C)c1-c1cc(Nc2ccc(OC(F)(F)F)cc2)ncn1 50328159FC(F)(F)Oc1ccc(Nc2cc(ncn2)-c2cnn(Cc3cccnc3)c2)cc1 50328160FC(F)(F)Oc1ccc(Nc2cc(ncn2)-c2cccc3[nH]ccc23)cc1 50328161FC(F)(F)Oc1ccc(Nc2cc(ncn2)-c2ccc3[nH]ccc3c2)cc1 50328162FC(F)(F)Oc1ccc(Nc2cc(ncn2)-c2ccnc3[nH]ccc23)cc1 50328163Cc1nc(cs1)-c1cc(Nc2ccc(OC(F)(F)F)cc2)ncn1 50328169FC(F)(F)c1ccc(Nc2cc(NCCN3CCOCC3)ncn2)cc1 50328171Cc1c(NCCN2CCOCC2)ncnc1Nc1ccc(OC(F)(F)F)cc1 50328172Cc1nc(NCCN2CCOCC2)cc(Nc2ccc(OC(F)(F)F)cc2)n1 50328180FC(F)(F)c1ccc(Nc2cc(ncn2)-c2ccncc2)cc1 50328181FC(F)(F)c1ccc(Nc2cc(ncn2)-c2ccncc2)cn1 50328183COC(=O)c1cc2c(Nc3ccc(OC(F)(F)F)cc3)ncnc2s1 50328184OCc1cc2c(Nc3ccc(OC(F)(F)F)cc3)ncnc2s1 50328187CCNC(=O)c1cc2c(Nc3ccc(OC(F)(F)F)cc3)ncnc2s1 50328188FC(F)(F)Oc1ccc(Nc2ncnc3sc(cc23)C(=O)N2CCNCC2)cc1 50328189FC(F)(F)Oc1ccc(Nc2ncnc3sc(cc23)C(=O)N2CCN(CC2)N2CCCC2)cc1 50328190OC1CCN(CC1)C(=O)c1cc2c(Nc3ccc(OC(F)(F)F)cc3)ncnc2s1 50328191Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1C(=O)c1cc2c(Nc3ccc(OC(F)(F)F)cc3)ncnc2s1 50328193Cn1ccc2c(Nc3ccc(OC(F)(F)F)cc3)ncnc12 50328194FC(F)(F)Oc1ccc(Nc2ncnc3n(CCN4CCOCC4)ccc23)cc1 50328195COc1ccc(Cn2ccc3c(Nc4ccc(OC(F)(F)F)cc4)ncnc23)cc1 50328196COCCCNC(=O)CCn1ccc2c(Nc3ccc(OC(F)(F)F)cc3)ncnc12 50328197NC(=O)CCn1ccc2c(Nc3ccc(OC(F)(F)F)cc3)ncnc12 50328198OCCn1ncc2c(Nc3ccc(OC(F)(F)F)cc3)ncnc12 50328199CCn1ncc2c(Nc3ccc(OC(F)(F)F)cc3)ncnc12 50328200CCCn1ncc2c(Nc3ccc(OC(F)(F)F)cc3)ncnc12 50328201FC(F)(F)Oc1ccc(Nc2ncnc3n(ncc23)C2CCCCC2)cc1 50328202NC(=O)Cn1ncc2c(Nc3ccc(OC(F)(F)F)cc3)ncnc12 50330905CN1C[C@@H]2C[C@H]1CN2c1cc(F)c(c(F)c1)-c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12 50331096COc1cc2c(Oc3ccc4[nH]c(C)cc4c3F)ncnc2cc1OCCCN1CCCC1 50331277COc1ccc2cc([nH]c2c1)-c1n[nH]c2cccnc12 50332294Cc1cnc(Nc2ccc(OCCN3CCCC3)cc2)nc1Nc1cccc(c1)S(=O)(=O)NC(C)(C)C 50332483ONC(=O)\C=C\c1ccc(o1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1 50332484Nc1ccccc1NC(=O)c1ccc(o1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1 50332485Nc1ccccc1NC(=O)c1ccc(s1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1 50332486Nc1ccccc1NC(=O)\C=C\c1ccc(o1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1 50332487Nc1ccccc1NC(=O)\C=C\c1cccc(c1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1 50332488Nc1ccccc1NC(=O)\C=C\c1ccc(cc1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1 50332489Nc1ccccc1NC(=O)CCc1ccc(cc1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1 50332490ONC(=O)c1ccc(o1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1 50332491ONC(=O)\C=C\c1ccc(s1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1 50332492ONC(=O)\C=C\c1ccc(cc1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1 50332493ONC(=O)c1ccc(s1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1 50332494ONC(=O)\C=C\c1cccc(c1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1 50339609CN(C)Cc1cc(cc(c1)C(F)(F)F)C(=O)N[C@@H]1CCc2ccc(Oc3ccnc4NC(=O)CCc34)cc2C1 50340954CC(=O)NC[C@H]1CC[C@@H](CC1)c1nc(-c2cc3ccccc3[nH]2)c2c(N)nccn12 50341117Cc1cn(cn1)-c1cc(NC(=O)c2ccc(C)c(Nc3nc(cs3)-c3cccnc3)c2)cc(c1)C(F)(F)F 50341118Cc1ccc(cc1Nc1nc(cs1)-c1cccnc1)C(=O)Nc1cc(cc(c1)C(F)(F)F)-n1ccnc1 50341119Cc1ncn(n1)-c1cc(NC(=O)c2ccc(C)c(Nc3nc(cs3)-c3cccnc3)c2)cc(c1)C(F)(F)F 50341120Cc1ccc(cc1Nc1nc(cs1)-c1cccnc1)C(=O)Nc1cc(cc(c1)C(F)(F)F)-c1cnn(C)c1 50341121Cc1ccc(cc1Nc1nc(cs1)-c1cccnc1)C(=O)Nc1cc(cc(c1)C(F)(F)F)-c1cn(C)nn1 50341123Cc1cn(cn1)-c1cc(C)cc(NC(=O)c2ccc(C)c(Nc3nc(cs3)-c3cccnc3)c2)c1 50341124CC(C)c1cc(NC(=O)c2ccc(C)c(Nc3nc(cs3)-c3cccnc3)c2)cc(c1)-n1cnc(C)c1 50341125Cc1cn(cn1)-c1cc(NC(=O)c2ccc(C)c(Nc3nc(cs3)-c3cccnc3)c2)cc(c1)C(C)(C)C 50341127Cc1cn(cn1)-c1cc(Cl)cc(NC(=O)c2ccc(C)c(Nc3nc(cs3)-c3cccnc3)c2)c1 50341128Cc1cn(cn1)-c1cc(NC(=O)c2cccc(Nc3nc(cs3)-c3cccnc3)c2)cc(c1)C(F)(F)F 50341129CCc1ccc(cc1Nc1nc(cs1)-c1cccnc1)C(=O)Nc1cc(cc(c1)C(F)(F)F)-n1cnc(C)c1 50341234Cc1ccc(NC(=O)c2ccc(CCl)cc2)cc1Nc1nccc(n1)-c1cccnc1 50343417ClC(Cn1ncc2c(NCc3ccncc3)ncnc12)c1ccc(Cl)cc1 50343418ClC(Cn1ncc2c(NCc3ccccn3)ncnc12)c1ccc(Cl)cc1 50343419CS(=O)(=O)c1nc(NCc2ccccc2)c2cnn(CC(Cl)c3ccccc3)c2n1 50343420CCCNc1nc(nc2n(\C=C/c3ccccc3)ncc12)S(C)(=O)=O 50343421OCCNc1nc(NCCc2ccccc2)c2cnn(\C=C/c3ccccc3)c2n1 50343422Fc1ccc(cc1)C(Cl)Cn1ncc2c(NCc3ccncc3)ncnc12 50343423Fc1ccc(cc1)C(Cl)Cn1ncc2c(NCc3ccccn3)ncnc12 50343424Fc1ccc(CNc2ncnc3n(CC(Cl)c4ccc(Cl)cc4)ncc23)cc1 50343425ClC(Cn1ncc2c(Nc3cccc(Cl)c3)nc(nc12)N1CCOCC1)c1ccccc1 50343426CCCNc1nc(SCCN2CCOCC2)nc2n(CC(Cl)c3ccccc3)ncc12 50343427ClC(Cn1ncc2c(NCc3ccccc3)nc(SCCN3CCOCC3)nc12)c1ccccc1 50343428Fc1ccc(CNc2nc(SCCN3CCOCC3)nc3n(CC(Cl)c4ccccc4)ncc23)cc1 50343429ClC(Cn1ncc2c(NCCc3ccccc3)nc(SCCN3CCOCC3)nc12)c1ccccc1 50343430ClC(Cn1ncc2c(Nc3cccc(Cl)c3)nc(SCCN3CCOCC3)nc12)c1ccccc1 50343431ClC(Cn1ncc2c(Nc3ccccc3)nc(SCCN3CCOCC3)nc12)c1ccccc1 50344664CC1(C)c2[nH]c3cc(ccc3c2C(=O)c2ccc(cc12)C1CCN(CC1)C1COC1)C#N 50345579CNC(=O)c1ncc(C#Cc2cc(ccc2C)C(=O)Nc2ccc(CN3CCN(CCO)CC3)c(c2)C(F)(F)F)n1C 50345580CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc(NC(C)=O)s3)cc2C(F)(F)F)CC1 50345581CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc(N)s3)cc2C(F)(F)F)CC1 50345582Cc1ccc(cc1C#Cc1cnc(C(N)=O)n1C)C(=O)Nc1ccc(CN2CCN(CC(O)=O)CC2)c(c1)C(F)(F)F 50345583COCCN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc(C(N)=O)n3C)cc2C(F)(F)F)CC1 50345584Cc1ccc(cc1C#Cc1cnc(C(N)=O)n1C)C(=O)Nc1ccc(CN2CCN(CCO)CC2)c(c1)C(F)(F)F 50345585CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc(C(=O)NCCO)n3C)cc2C(F)(F)F)CC1 50345586CNC(=O)c1ncc(C#Cc2cc(ccc2C)C(=O)Nc2ccc(CN3CCN(C)CC3)c(c2)C(F)(F)F)n1C 50345587CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc(C(N)=O)n3C)cc2C(F)(F)F)CC1 50345588CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc(C)n3C)cc2C(F)(F)F)CC1 50345589CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cncn3C)cc2C(F)(F)F)CC1 50345590CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc[nH]3)cc2C(F)(F)F)CC1 50345591CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc(NC4CC4)nc3)cc2C(F)(F)F)CC1 50345592CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3ccc(nc3)C(N)=O)cc2C(F)(F)F)CC1 50345593CCC(=O)Nc1ccc(cn1)C#Cc1cc(ccc1C)C(=O)Nc1ccc(CN2CCN(C)CC2)c(c1)C(F)(F)F 50345594CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3ccc(NC(C)=O)nc3)cc2C(F)(F)F)CC1 50345595CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cncnc3)cc2C(F)(F)F)CC1 50345596CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cccnc3)cc2C(F)(F)F)CC1 50345738CC(C)n1nc(-c2ccc3ccccc3c2)c2c(N)ncnc12 50345739COc1ccc2cc(ccc2c1)-c1nn(C(C)C)c2ncnc(N)c12 50345740CCOc1ccc2cc(ccc2c1)-c1nn(C(C)C)c2ncnc(N)c12 50345742CC(C)n1nc(-c2cnc3ccccc3c2)c2c(N)ncnc12 50347659CN(C[C@@H]1COCCO1)S(=O)(=O)Nc1ccc2ccc3ncc(cc3c(=O)c2c1)-c1cnn(C)c1 50349877CN1CCN(CC1)c1ccc(cc1)-c1cc2n(C)nc(N)c2c(=O)[nH]1 50349878Nc1n(nc2cc([nH]c(=O)c12)-c1ccccc1)-c1ccccc1 50354477CSc1nc(NCc2ccccc2F)c2cnn(CC(C)c3ccccc3)c2n1 50354478CSc1nc(NCc2ccc(F)cc2)c2cnn(CC(C)c3ccccc3)c2n1 50354479CSc1nc(NCc2ccccc2Cl)c2cnn(CC(C)c3ccccc3)c2n1 50354482Fc1cccc(CNc2ncnc3n(CCc4ccccc4)ncc23)c1 50354484CSc1nc(NCc2cccc(Br)c2)c2cnn(CC(Cl)c3ccccc3)c2n1 50354485Fc1cccc(CNc2ncnc3n(CC(Cl)c4ccccc4)ncc23)c1 50354486ClC(Cn1ncc2c(NCc3ccccc3)ncnc12)c1ccccc1 50354487Fc1ccccc1CNc1ncnc2n(CC(Cl)c3ccccc3)ncc12 50354488Fc1ccc(CNc2ncnc3n(CC(Cl)c4ccccc4)ncc23)cc1 50354489CSc1nc(Nc2cccc(Br)c2)c2cnn(CC(C)c3ccccc3)c2n1 50355393CCN1CCN(CC1)c1ccc(Nc2cc(ncn2)N(C)C(=O)Nc2c(Cl)c(OC)cc(OC)c2Cl)cc1 50355491Nc1nc(Nc2ccc(cc2)[C@H]2CC[C@@H](CC2)N2CCOCC2)nn1-c1ccccn1 50355494COc1cc(Oc2ccnc3cc(OC)c(OC)cc23)ccc1NC(=O)NC(C)c1nccs1 50355495CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(Nc3nc(cs3)-c3cccnc3)c2)CC1 50355496O=C(N1CCNCC1)c1ccc(\C=C\c2n[nH]c3ccccc23)cc1 50355498Cn1cc(cn1)-c1ccc2nnc(Sc3ccc4ncccc4c3)n2n1 50355499CN(C)CC(=O)N1CCC(CC1)c1ccc(NC(=O)c2ncc([nH]2)C#N)c(c1)C1=CCCCC1 50355501N#CC[C@H](C1CCCC1)n1cc(cn1)-c1ncnc2[nH]ccc12 50355502CN(C(=O)CN1CCN(C)CC1)c1ccc(cc1)N=C(C1C(=O)Nc2ccccc12)c1ccccc1 50355504COc1cc2c(Oc3ccc(NC(=O)C4(CC4)C(=O)NC4=CCC(F)C=C4)cc3F)ccnc2cc1OCCCN1CCOCC1 50357333CN(C)C\C=C\C(=O)N(C)c1cc2c(cc1F)nc(Nc1ccccc1C)c1cncn21 50358832CSc1cccc(c1)C(=O)Nc1ccc(C)c(Nc2nccc(n2)-c2cccnc2)c1 50372735Fc1ccc(cc1)C(Cl)Cn1ncc2c(NCc3cccc(Cl)c3)ncnc12 50372736Fc1ccc(cc1)C(Cl)Cn1ncc2c(NCc3ccccc3F)ncnc12 50372737Fc1ccc(cc1)C(Cl)Cn1ncc2c(NCc3cccc(F)c3)ncnc12 50372738Fc1ccc(CNc2ncnc3n(CC(Cl)c4ccc(F)cc4)ncc23)cc1 50372739Fc1ccc(cc1)C(Cl)Cn1ncc2c(NCc3ccccc3)ncnc12 50372740Fc1ccc(cc1)C(Cl)Cn1ncc2c(NCc3ccccc3Cl)ncnc12 50372741ClC(Cn1ncc2c(NCc3cccc(Cl)c3)ncnc12)c1ccc(Cl)cc1 50376003COc1cc2nccc(Oc3ccc4c(cccc4c3)C(N)=O)c2cc1OC 50376901Cc1cc(cc2nnc(Nc3ccc(OCC[N+]4([O-])CCCC4)cc3)nc12)-c1c(Cl)cccc1Cl 50378568CC1(C)CC(CC(C)(C)N1[O])NC(=O)c1cccc(c1)-c1cc2nccc(Nc3cccc(O)c3)n2n1 50378803Cn1c2nc(NCc3cccc(N)c3)ncc2cc(-c2c(Cl)cccc2Cl)c1=O 50378804Cn1c2nc(NCc3cccc(N)c3)ncc2cc(-c2ccccc2Cl)c1=O 50378805Cn1c2nc(NCc3cccc(N)c3)ncc2cc(-c2ccccc2)c1=O 50378806Cn1c2nc(NCc3cccc(N)c3)ncc2cc(-c2c(F)cccc2F)c1=O 50378807Cn1c2nc(NCc3cccc(N)c3)ncc2cc(-c2ccccc2Br)c1=O 50378808CSc1cccc(CNc2ncc3cc(-c4c(Cl)cccc4Cl)c(=O)n(C)c3n2)c1 50378809CCCCCCNc1cccc(CNc2ncc3cc(-c4c(Cl)cccc4Cl)c(=O)n(C)c3n2)c1 50378810Cn1c2nc(NCc3cccc(NC(=O)CN)c3)ncc2cc(-c2c(Cl)cccc2Cl)c1=O 50378811Cn1c2nc(NCc3cccc(c3)C(=O)CCCC[C@@H]3SC[C@@H]4NC(=O)N[C@H]34)ncc2cc(-c2c(Cl)cccc2Cl)c1=O 50378812Cn1c2nc(Nc3cccc(NC(=O)CN)c3)ncc2cc(-c2c(Cl)cccc2Cl)c1=O 50381716Nc1ncc(-c2cnn(CCO)c2)c2scc(-c3ccc(NC(=O)Nc4cccc(F)c4)cc3)c12 50381719C[C@@H](O)Cn1cc(cn1)-c1cnc(N)c2c(csc12)-c1ccc(NC(=O)Nc2cccc(F)c2)cc1 50382959COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C(F)(F)F)c3)c2cc1OC 50383191COc1cc2nccc(Oc3ccc(NC(=O)c4c(C)n(C)n(-c5ccccc5)c4=O)cc3F)c2cc1OC 50383376COc1ccc(cc1C)-c1nn(CC2CCNCC2)c2ncnc(N)c12 50383382CC(C)n1nc(-c2cc3c(Cl)cccc3[nH]2)c2c(N)ncnc12 50385915C[C@@H](Oc1cc(ccc1C(N)=O)-c1cc(cnc1N)-c1cc(CN(C)C)cs1)\C=C/C(F)(F)F 50388030OCCNC(=O)Nc1nc2ccc(cc2[nH]1)C(=O)c1ccccc1 50388031O=C(NCCC1CCNCC1)Nc1nc2ccc(cc2[nH]1)C(=O)c1ccccc1 50388032O=C(NCCC1CCCNC1)Nc1nc2ccc(cc2[nH]1)C(=O)c1ccccc1 50388033NCCC(=O)Nc1nc2ccc(cc2[nH]1)C(=O)c1ccccc1 50389704CCOc1ccc2cc(ccc2c1)-c1nn(CC2CCN(C)CC2)c2ncnc(N)c12 50390208C(Cc1ccccc1)Nc1ncnc2n(\C=C/c3ccccc3)ncc12 50390444C[C@H](NC(=O)c1cc(cnc1N)-c1cnn(c1)C1CCOCC1)c1c(Cl)ccc(F)c1Cl 50392791CC(C)Oc1cc(n[nH]1)-n1cnc2ccc(N[C@@H](C)c3ccc(F)cn3)nc12 50393034Cc1ccc(O)cc1-n1c2ncnc(N)c2c2CCCCc2c1=O 50399363CC(C)c1ccc(cc1-n1cc(nn1)-c1cnc2[nH]ncc2c1)C(=O)Nc1ccc(CN2CCN(C)CC2)c(c1)C(F)(F)F 50399364CN1CCN(Cc2ccc(NC(=O)c3ccc(C4CC4)c(c3)-n3cc(nn3)-c3cnc4[nH]ncc4c3)cc2C(F)(F)F)CC1 50399365CCc1ccc(cc1-n1cc(nn1)-c1cnc2[nH]ncc2c1)C(=O)Nc1ccc(CN2CCN(C)CC2)c(c1)C(F)(F)F 50399366CN1CCN(Cc2ccc(NC(=O)c3ccc(Br)c(c3)-n3cc(nn3)-c3cnc4[nH]ncc4c3)cc2C(F)(F)F)CC1 50399367CN1CCN(Cc2ccc(NC(=O)c3ccc(Cl)c(c3)-n3cc(nn3)-c3cnc4[nH]ncc4c3)cc2C(F)(F)F)CC1 50399368CN1CCN(Cc2ccc(NC(=O)c3ccc(F)c(c3)-n3cc(nn3)-c3cnc4[nH]ncc4c3)cc2C(F)(F)F)CC1 50399369CN1CCN(Cc2ccc(NC(=O)c3cccc(c3)-n3cc(nn3)-c3cnc4[nH]ncc4c3)cc2C(F)(F)F)CC1 50399370Cc1ncn(n1)-c1cc(NC(=O)c2ccc(C)c(c2)-n2cc(nn2)-c2cnc3[nH]ncc3c2)cc(c1)C(F)(F)F 50399371Cc1ccc(cc1-n1cc(nn1)-c1cnc2[nH]ncc2c1)C(=O)Nc1cc(cc(c1)C(F)(F)F)-n1cncn1 50399372Cc1cn(cn1)-c1cc(NC(=O)c2ccc(C)c(c2)-n2cc(nn2)-c2cnc3[nH]ncc3c2)cc(c1)C(F)(F)F 50399373CN1C[C@H]2CN(Cc3ccc(NC(=O)c4ccc(C)c(c4)-n4cc(nn4)-c4cnc5[nH]ncc5c4)cc3C(F)(F)F)C[C@H]2C1 50399374CN(C)C1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)-n3cc(nn3)-c3cnc4[nH]ncc4c3)cc2C(F)(F)F)CC1 50399375CN1CCN(CC1)C1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)-n3cc(nn3)-c3cnc4[nH]ncc4c3)cc2C(F)(F)F)CC1 50399376CN1CCCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)-n3cc(nn3)-c3cnc4[nH]ncc4c3)cc2C(F)(F)F)CC1 50399377Cc1ccc(cc1-n1cc(nn1)-c1cnc2[nH]ncc2c1)C(=O)Nc1ccc(CN2CCOCC2)c(c1)C(F)(F)F 50399378Cc1ccc(cc1-n1cc(nn1)-c1cnc2[nH]ncc2c1)C(=O)Nc1ccc(CN2CCCCC2)c(c1)C(F)(F)F 50399379CN(C)[C@@H]1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)-n3cc(nn3)-c3cnc4[nH]ncc4c3)cc2C(F)(F)F)C1 50399380CN(C)[C@H]1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)-n3cc(nn3)-c3cnc4[nH]ncc4c3)cc2C(F)(F)F)C1 50399381Cc1ccc(cc1-n1cc(nn1)-c1cnc2[nH]ncc2c1)C(=O)Nc1ccc(CN2CCCC2)c(c1)C(F)(F)F 50399382CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)-n3cc(nn3)-c3cnc4[nH]nc(C)c4c3)cc2C(F)(F)F)CC1 50399383CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)-n3cc(nn3)-c3cnc4[nH]ncc4c3)cc2C(F)(F)F)CC1 50399384CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)-n3cc(nn3)-c3ccc4[nH]ncc4c3)cc2C(F)(F)F)CC1 50399385CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)-n3cc(nn3)-c3ccc4[nH]ccc4c3)cc2C(F)(F)F)CC1 50399386CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)-n3cc(nn3)-c3cnc4[nH]ccc4c3)cc2C(F)(F)F)CC1 50399387CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)-n3cc(nn3)-c3cnc4ncnn4c3)cc2C(F)(F)F)CC1 50399388CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)-n3cc(nn3)-c3cnc(nc3)N3CCCCC3)cc2C(F)(F)F)CC1 50399389CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)-n3cc(nn3)-c3cnc(NCc4ccccc4)nc3)cc2C(F)(F)F)CC1 50399390CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)-n3cc(nn3)-c3cnc(NC4CCCCC4)nc3)cc2C(F)(F)F)CC1 50399391CC(C)Nc1ncc(cn1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1ccc(CN2CCN(C)CC2)c(c1)C(F)(F)F 50399392CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)-n3cc(nn3)-c3cnc(NC4CC4)nc3)cc2C(F)(F)F)CC1 50399393CCNc1ncc(cn1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1ccc(CN2CCN(C)CC2)c(c1)C(F)(F)F 50399394CNc1ncc(cn1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1ccc(CN2CCN(C)CC2)c(c1)C(F)(F)F 50399395CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)-n3cc(nn3)-c3cnc(N)nc3)cc2C(F)(F)F)CC1 50399396CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)-n3cc(nn3)-c3cnc4ccccn34)cc2C(F)(F)F)CC1 50399397CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)-n3cc(nn3)-c3cnn4cccnc34)cc2C(F)(F)F)CC1 50399398CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)-n3cc(nn3)-c3cnc4ncccn34)cc2C(F)(F)F)CC1 50399399CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)-n3cc(nn3)-c3cnc4cccnn34)cc2C(F)(F)F)CC1 50423656CO[C@H]1[C@@H](C[C@H]2O[C@@]1(C)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13)N(C)C(=O)c1ccccc1 50423773C[C@]12O[C@@H](C[C@@]1(O)CO)n1c3ccccc3c3c4C(=O)NCc4c4c5ccccc5n2c4c13 50425385Cc1cn(cn1)-c1cc(F)cc(NC(=O)c2ccc(C)c(Nc3nccc(n3)-c3cccnc3)c2)c1 50425386Cc1cn(cn1)-c1cccc(NC(=O)c2ccc(C)c(Nc3nccc(n3)-c3cccnc3)c2)c1 50425387Cc1cn(cn1)-c1cc(C)cc(NC(=O)c2ccc(C)c(Nc3nccc(n3)-c3cccnc3)c2)c1 50425780CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc4[nH]ncc4c3)cc2C(F)(F)F)CC1 50425781CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc4ncnn4c3)cc2C(F)(F)F)CC1 50425782CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc4n(C)ncc4c3)cc2C(F)(F)F)CC1 50425783CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3ccc4[nH]ncc4c3)cc2C(F)(F)F)CC1 50425784COc1n[nH]c2ncc(cc12)C#Cc1cc(ccc1C)C(=O)Nc1ccc(CN2CCN(C)CC2)c(c1)C(F)(F)F 50425785CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc4[nH]nc(-c5ccccc5)c4c3)cc2C(F)(F)F)CC1 50425786CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc4[nH]nc(C5CC5)c4c3)cc2C(F)(F)F)CC1 50425787CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc4[nH]nc(C)c4c3)cc2C(F)(F)F)CC1 50425788CN1CCN(Cc2ccc(NC(=O)c3ccc(Cl)c(c3)C#Cc3cnc4[nH]ncc4c3)cc2C(F)(F)F)CC1 50425789CN1CCN(Cc2ccc(NC(=O)c3ccc(C4CC4)c(c3)C#Cc3cnc4[nH]ncc4c3)cc2C(F)(F)F)CC1 50425790CCc1ccc(cc1C#Cc1cnc2[nH]ncc2c1)C(=O)Nc1ccc(CN2CCN(C)CC2)c(c1)C(F)(F)F 50425791CN1CCN(Cc2ccc(NC(=O)c3cccc(c3)C#Cc3cnc4[nH]ncc4c3)cc2C(F)(F)F)CC1 50425832COc1ccc(CCNc2ncc(C(=O)NCCCN3CCCC3=O)c(NC3CCCC3)n2)cc1OC 50425862CN(C)C1CCC(CC1)Nc1nc(Nc2cc(Cl)cc(Cl)c2)ncc1-c1cc(C)no1 50425864CN(C)C1CCC(CC1)Nc1nc(Nc2cc(Cl)cc(Cl)c2)ncc1C(=O)NC1CCN(C)CC1 50425865CN1CCC(CC1)NC(=O)c1cnc(NCc2cc(Cl)ccc2Cl)nc1NC1CCCC1 50427740Cc1ccc(NC(=O)c2ccc(Cn3ccnc3)c(c2)C(F)(F)F)cc1C#Cc1cncnc1 50427741Cc1ccc(NC(=O)c2ccc(CN3CCN(CCO)CC3)c(c2)C(F)(F)F)cc1C#Cc1cnc2ccccn12 50427742CN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)Nc2ccc(C)c(c2)C#Cc2cnc3cccnn23)CC1 50427743CN1CCN(Cc2ccc(NC(=O)Nc3cc(C#Cc4ccc(N)nc4)n(C)n3)cc2C(F)(F)F)CC1 50427744CN1CCN(Cc2ccc(NC(=O)Nc3cc(C#Cc4cccnc4)n(C)n3)cc2C(F)(F)F)CC1 50427745CN1CCN(Cc2ccc(NC(=O)Nc3cc(C#Cc4cnc5ccccn45)n(C)n3)cc2C(F)(F)F)CC1 50427746Cc1ccc(NC(=O)c2ccc(Cn3ccnc3)c(c2)C(F)(F)F)cc1C#Cc1ncc(Nc2ccccc2)cn1 50427747CN1CCN(Cc2ccc(NC(=O)Nc3cc(C#Cc4cnc5cccnn45)n(C)n3)cc2C(F)(F)F)CC1 50427748CN1CCN(Cc2ccc(NC(=O)Nc3cc(C#Cc4cnc5cnccn45)n(C)n3)cc2C(F)(F)F)CC1 50427749CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cncc4nccn34)cc2C(F)(F)F)CC1 50427750CN1CCN(Cc2ccc(NC(=O)Nc3cc(C#Cc4cncc5nccn45)n(C)n3)cc2C(F)(F)F)CC1 50428741CCCCn1c(cn2c1nc1n(C)c(=O)[nH]c(=O)c21)-c1cc(ccc1C)-c1cccc2[nH]ncc12 50428742CCCCn1c(cn2c1nc1n(C)c(=O)[nH]c(=O)c21)-c1ccc(F)cc1C 50428743CCCCn1c(cn2c1nc1n(C)c(=O)[nH]c(=O)c21)-c1ccccc1C 50431279Fc1ccc(cc1)-n1cccc(C(=O)Nc2ccc(Oc3ncnc4nc[nH]c34)c(F)c2)c1=O 50431280Fc1cccc(c1)-n1cccc(C(=O)Nc2ccc(Oc3ncnc4nc[nH]c34)c(F)c2)c1=O 50431812[O-][N+](=O)c1ccccc1-c1n[nH]cc1C=C1C(=O)Nc2ccccc12 50432859Sc1ccccc1C(=O)Nc1cccc(Nc2nccc(n2)-c2cccnc2)c1 50432860CCCCCCC(=O)Nc1cccc(Nc2nccc(n2)-c2cccnc2)c1 50432861CN1CCN(CC1)c1ccc(cc1)C(=O)Nc1[nH]nc2sc(cc12)C(=O)NC(C)(C)c1ccccc1 50432862CC(C)(NC(=O)c1cc2c(NC(=O)c3ccc(CN4CCCCC4)cc3)[nH]nc2s1)c1ccccc1 50432863CN(C)C1CN(Cc2ccc(cc2C(F)(F)F)C(=O)Nc2ccc(C)c(Nc3nccc(n3)-c3cncnc3)c2)C1 50432864CN(C)CC1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)Nc2ccc(C)c(Nc3nccc(n3)-c3cncnc3)c2)C1 50432865CN1CCN(Cc2ccc(cc2I)C(=O)Nc2ccc(C)c(Nc3nccc(n3)-c3cccnc3)c2)CC1 50432866CN1CCN(Cc2ccc(cc2Cl)C(=O)Nc2ccc(C)c(Nc3nccc(n3)-c3cccnc3)c2)CC1 50432867Cc1ccc(NC(=O)NCc2cccc(Cl)c2)cc1Nc1nccc(n1)-c1cccnc1 50432870COCCN=NNc1cccc(Nc2cc(ncn2)-c2cccnc2)c1 50432872Cc1cccc(Nc2nccc(n2)-c2cccnc2)c1 50432873NCCCCNC(=O)c1cccc(Nc2nccc(n2)-c2cccnc2)c1 50432892C[C@@H](Oc1c[nH]c(=O)c(c1)C(=O)Nc1ccc(cc1)N1CCN(C)CC1)c1c(Cl)ccc(F)c1Cl 50433223COc1ccc(cc1Nc1nccc(n1)-c1cccnc1)C(=O)Nc1cccc(c1)C(F)(F)F 50433224COc1ccc(cc1Nc1nccc(n1)-c1cccnc1)C(=O)Nc1ccncc1 50433225COc1ccc(cc1Nc1nccc(n1)-c1cccnc1)C(=O)Nc1ccc(OCCN2CCCCC2)cc1 50433226COc1ccc(cc1Nc1nccc(n1)-c1cccnc1)C(=O)Nc1ccc(OCCN2CCCC2)cc1 50433227COc1ccc(cc1Nc1nccc(n1)-c1cccnc1)C(=O)Nc1nccs1 50433228COc1ccc(cc1Nc1nccc(n1)-c1cccnc1)C(=O)Nc1ccc(OCCN2CCOCC2)cc1 50433229COc1ccc(cc1Nc1nccc(n1)-c1cccnc1)C(=O)Nc1cccc(Cl)c1 50433230COc1ccc(cc1Nc1nccc(n1)-c1cccnc1)C(=O)Nc1ccc(OCCCN2CCOCC2)cc1 50433231COc1ccc(cc1Nc1nccc(n1)-c1cccnc1)C(=O)Nc1ccc(Br)cc1 50433232COc1ccc(cc1Nc1nccc(n1)-c1cccnc1)C(=O)Nc1ccc(F)c(Cl)c1 50433233COc1ccc(cc1Nc1nccc(n1)-c1cccnc1)C(=O)Nc1ncccn1 50433234COc1ccc(cc1Nc1nccc(n1)-c1cccnc1)C(=O)Nc1cccc(F)c1 50433235COc1ccc(cc1Nc1nccc(n1)-c1cccnc1)C(=O)Nc1ccc(OCCN(C)C)cc1 50433236CCN(CC)CCOc1ccc(NC(=O)c2ccc(OC)c(Nc3nccc(n3)-c3cccnc3)c2)cc1 50433237COc1ccc(cc1Nc1nccc(n1)-c1cccnc1)C(=O)Nc1ccc(OCCCN(C)C)cc1 50433806NC(N)=NCCC[C@@H]1NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC1=O 50434582Cc1ccc(NC(=O)c2ccc(CN3CCNCC3)cc2)cc1Nc1nccc(n1)-c1cccnc1 50436570ClC(Cn1ncc2c(Nc3ccccc3)ncnc12)c1ccc(I)cc1 50436571Cc1ccc(cc1)C(Cl)Cn1ncc2c(Nc3ccccc3)ncnc12 50436572FC(F)(F)c1cc(CNc2ncnc3n(CC(Cl)c4ccc(Br)cc4)ncc23)cc(c1)C(F)(F)F 50436573COc1cccc(CNc2ncnc3n(CC(Cl)c4ccc(Br)cc4)ncc23)c1 50436574ClC(Cn1ncc2c(NCc3cccc(Br)c3)ncnc12)c1ccc(Br)cc1 50436575ClC(Cn1ncc2c(NCc3ccc(Br)cc3)ncnc12)c1ccc(Br)cc1 50436576Fc1ccc(F)c(CNc2ncnc3n(CC(Cl)c4ccc(Br)cc4)ncc23)c1 50436577Fc1ccc(CNc2ncnc3n(CC(Cl)c4ccc(Br)cc4)ncc23)cc1 50436578ClC(Cn1ncc2c(NCc3ccc(Cl)c(Cl)c3)ncnc12)c1ccc(Br)cc1 50436579ClC(Cn1ncc2c(NCc3cc(Cl)ccc3Cl)ncnc12)c1ccc(Br)cc1 50436580ClC(Cn1ncc2c(NCc3ccc(Cl)cc3)ncnc12)c1ccc(Br)cc1 50436581ClC(Cn1ncc2c(NCc3ccccc3Cl)ncnc12)c1ccc(Br)cc1 50436582ClC(Cn1ncc2c(NCc3cccc(Cl)c3)ncnc12)c1ccc(Br)cc1 50436583ClC(Cn1ncc2c(NCc3ccccc3)ncnc12)c1ccc(Br)cc1 50436584ClC(Cn1ncc2c(Nc3ccccc3)ncnc12)c1ccc(Br)cc1 50436585ClC(Cn1ncc2c(Nc3ccccc3)ncnc12)c1ccccc1 50436586Fc1cccc(Nc2ncnc3n(CC(Cl)c4ccccc4)ncc23)c1 50436587ClC(Cn1ncc2c(Nc3cccc(Br)c3)ncnc12)c1ccccc1 50436588Fc1ccc(cc1)C(Cl)Cn1ncc2c(Nc3cccc(Br)c3)ncnc12 50436589Fc1ccc(cc1)C(Cl)Cn1ncc2c(Nc3cccc(Cl)c3)ncnc12 50436590Fc1cccc(CNc2ncnc3n(CC(Cl)c4ccc(Br)cc4)ncc23)c1 50436850CC(C)Oc1cc(C2CCNCC2)c(C)cc1Nc1ncc(Cl)c(Nc2ccccc2S(=O)(=O)C(C)C)n1 50437147CC(C)(C)c1cc(NC(=O)Nc2cccc(Nc3ncnc4ccccc34)c2)n(n1)-c1cccc(N)c1 50437148CC(C)(C)c1cc(NC(=O)Nc2cccc(Nc3ncnc4ccccc34)c2)n(n1)-c1cccc(c1)[N+]([O-])=O 50437149CC(C)(C)c1cc(NC(=O)Nc2ccc(Nc3ncnc4ccc(NC(=O)CCN5CCOCC5)cc34)cc2)n(n1)-c1cccc(N)c1 50437150CN1CCN(CCC(=O)Nc2ccc3ncnc(Nc4ccc(NC(=O)Nc5cc(nn5-c5cccc(N)c5)C(C)(C)C)cc4)c3c2)CC1 50437151CC(C)(C)c1cc(NC(=O)Nc2ccc(Nc3ncnc4ccc(N)cc34)cc2)n(n1)-c1cccc(NC(=O)OCC2c3ccccc3-c3ccccc23)c1 50437152CC(C)(C)c1cc(NC(=O)Nc2ccc(Nc3ncnc4ccccc34)cc2)n(n1)-c1cccc(N)c1 50437153CC(C)(C)c1cc(NC(=O)Nc2ccc(Nc3ncnc4ccc(N)cc34)cc2)n(n1)-c1cccc(N)c1 50437154CC(C)(C)c1cc(NC(=O)Nc2ccc(Nc3ncnc4ccccc34)cc2)n(n1)-c1cccc(c1)[N+]([O-])=O 50437155CC(C)(C)c1cc(NC(=O)Nc2ccc(Nc3ncnc4ccc(cc34)[N+]([O-])=O)cc2)n(n1)-c1cccc(c1)[N+]([O-])=O 50437405Nc1ncnc2n(nc(-c3ccc(Cl)cc3)c12)-c1cccc(c1)-c1cnnn1CCCCCC(=O)NO 50437676Oc1cc(OCC(=O)NCCN2CCOCC2)cc2oc(cc(=O)c12)-c1ccccc1 50437677Oc1cc(OCC(=O)NCc2ccccc2)cc2oc(cc(=O)c12)-c1ccccc1 50437678COc1cccc(NC(=O)COc2cc(O)c3c(c2)oc(cc3=O)-c2ccccc2)c1 50437680Oc1cc(OCC(=O)Nc2cccc(Br)c2)cc2oc(cc(=O)c12)-c1ccccc1 50437681Oc1cc(OCC(=O)Nc2ccc(Br)cc2)cc2oc(cc(=O)c12)-c1ccccc1 50437682Cc1ccc(NC(=O)COc2cc(O)c3c(c2)oc(cc3=O)-c2ccccc2)cc1 50437683Cc1cccc(NC(=O)COc2cc(O)c3c(c2)oc(cc3=O)-c2ccccc2)c1 50437684Oc1cc(OCC(=O)Nc2ncccc2F)cc2oc(cc(=O)c12)-c1ccccc1 50437686Cc1cc(NC(=O)COc2cc(O)c3c(c2)oc(cc3=O)-c2ccccc2)ncc1Br 50437687Oc1cc(OCC(=O)Nc2cc(Br)ccn2)cc2oc(cc(=O)c12)-c1ccccc1 50437688Oc1cc(OCC(=O)Nc2ccc(Br)cn2)cc2oc(cc(=O)c12)-c1ccccc1 50437689Cc1ccnc(NC(=O)COc2cc(O)c3c(c2)oc(cc3=O)-c2ccccc2)c1 50437690Cc1ccc(NC(=O)COc2cc(O)c3c(c2)oc(cc3=O)-c2ccccc2)nc1 50437691Cc1cccc(NC(=O)COc2cc(O)c3c(c2)oc(cc3=O)-c2cc(F)ccc2F)n1 50437692Cc1cccc(NC(=O)COc2cc(O)c3c(c2)oc(cc3=O)-c2ccccc2)n1 50439333C1COc2cc3ncnc(Nc4cccc(c4)-c4ccccc4)c3cc2OC1 50439334C1COc2cc3c(Nc4cccc(c4)-c4ccccc4)ncnc3cc2O1 50439335C1Oc2cc3ncnc(Nc4cccc(c4)-c4ccccc4)c3cc2O1 50439463C1CNCC2(C1)CCN(CC2)c1ncnc2nc[nH]c12 50441518Oc1ccc(NS(=O)(=O)c2ccc(cc2)[N+]([O-])=O)cc1Sc1nnc[nH]1 50441567CN1CCN(Cc2ccc(cc2)-c2cnc3[nH]cc(-c4ccc5[nH]ccc5c4)c3c2)CC1 50443993CCN(CC)CCCNC(=O)Nc1cc2c(Nc3ccc(F)c(Cl)c3)ncnc2cc1O[C@H]1CCOC1 50444656Cc1ccc(NC(=O)c2ccc(CN3CCN(Cc4ccc(I)cc4)CC3)cc2)cc1Nc1nccc(n1)-c1cccnc1 50444657Cc1ccc(NC(=O)c2ccc(CN3CCN(CCO)CC3)cc2)cc1Nc1nccc(n1)-c1cccnc1 50444658Cc1ccc(NC(=O)c2ccc(CN3CCN(CCF)CC3)cc2)cc1Nc1nccc(n1)-c1cccnc1 50446982C[C@H](Nc1nc(Nc2cn(C)cn2)c2cc[nH]c2n1)c1ncc(F)cn1 50447512CN1CCN(CC1)c1ccc(Nc2ncc3cc(C#N)c(=O)n(C4CCCC4)c3n2)cc1 50447756COc1ccc(cc1OC)S(=O)(=O)Nc1cc(Sc2ncnc3nc[nH]c23)c(O)c2ccccc12