1898CNC(=O)c1ccc2[C@H]3CCCN([C@H]3Cc2c1)C(=O)c1ccc2nc[nH]c2c1 8528Cc1noc(n1)[C@]12CC3CC(C1)[C@H](NC(=O)N1CCN(c4ccc(cn4)N4CCN(CC4)S(=O)(=O)C4CC4)c4ccccc14)C(C3)C2 13738CC(C)C1(C)SC(Nc2ccccc2C(F)(F)F)=NC1=O 13740CC(C)C1(C)SC(NCc2ccccc2)=NC1=O 13741CC(C)C1(C)SC(N[C@@H](C)c2ccccc2)=NC1=O 13742CC(C)C1(C)SC(N[C@H](C)c2ccccc2)=NC1=O 13743CC(C)C1(C)SC(N[C@@H](C)c2ccc(cc2)C(F)(F)F)=NC1=O 13744CC(C)C1(C)SC(N[C@@H](C)c2cccc(c2)C(F)(F)F)=NC1=O 13745CC(C)C1(C)SC(N[C@@H](C)c2ccccc2C(F)(F)F)=NC1=O 13746CC(C)C1(C)SC(N[C@@H](C)c2ccccc2F)=NC1=O 13747CC(C)C1(C)SC(N[C@@H](C)c2ccccc2Cl)=NC1=O 13748CC(C)C1(C)SC(N[C@@H](C)c2ccccc2Br)=NC1=O 13749CC(C)[C@]1(C)SC(N[C@@H](C)c2ccccc2F)=NC1=O 13750CC(C)[C@@]1(C)SC(N[C@@H](C)c2ccccc2F)=NC1=O 13751C[C@H](NC1=NC(=O)C(C)(S1)C(C)(C)F)c1ccccc1F 13752C[C@H](NC1=NC(=O)C(C)(S1)C(F)(F)F)c1ccccc1F 13753C[C@H](NC1=NC(=O)[C@@](C)(S1)C(F)(F)F)c1ccccc1F 13754C[C@H](NC1=NC(=O)[C@](C)(S1)C(F)(F)F)c1ccccc1F 13755CC(C)(Oc1ccccc1)C(=O)N[C@H]1C2C[C@@H]3C[C@@H]1C[C@](C3)(C2)C(O)=O 13756CC(C)(Oc1ccccc1)C(=O)N[C@H]1C2C[C@@H]3C[C@@H]1C[C@](C3)(C2)C(N)=O 13757CC(C)(Oc1ccccc1Cl)C(=O)N[C@H]1C2C[C@@H]3C[C@@H]1C[C@](C3)(C2)C(O)=O 13758CC(C)(Oc1cccc(Cl)c1)C(=O)N[C@H]1C2C[C@@H]3C[C@@H]1C[C@](C3)(C2)C(O)=O 13759CC(C)(Oc1ccc(Cl)cc1)C(=O)N[C@H]1C2C[C@@H]3C[C@@H]1C[C@](C3)(C2)C(O)=O 13760CC(C)(Oc1ccc(Cl)cc1)C(=O)N[C@H]1C2C[C@@H]3C[C@@H]1C[C@](C3)(C2)C(N)=O 13761COc1ccc(OC(C)(C)C(=O)N[C@H]2C3C[C@@H]4C[C@@H]2C[C@](C4)(C3)C(N)=O)cc1 13762CC(C)(Oc1ccc(Cl)cc1)C(=O)N[C@H]1C2C[C@@H]3C[C@@H]1C[C@](C3)(C2)C(=O)NCc1ccc(cc1)C(O)=O 13763CC(C)(Oc1ccc(Cl)cc1)C(=O)N[C@H]1C2C[C@@H]3C[C@@H]1C[C@](C3)(C2)C(=O)NCc1ccc(cc1)C(=O)NS(C)(=O)=O 13764CC(C)(Oc1ccc(Cl)cc1)C(=O)N[C@H]1C2C[C@@H]3C[C@@H]1C[C@](C3)(C2)C(=O)NCc1ccc(cc1)-c1nnn[nH]1 13765CC(C)(Oc1ccc(Cl)cc1)C(=O)N[C@H]1C2C[C@@H]3C[C@@H]1C[C@](C3)(C2)C(=O)NCc1ccc(cc1)S(N)(=O)=O 13766CC(C)(Oc1ccc(Cl)cc1)C(=O)N[C@H]1C2C[C@@H]3C[C@@H]1C[C@](C3)(C2)C(=O)NCc1cncs1 13767CC(C)(Oc1ccc(Cl)cc1)C(=O)N[C@H]1C2C[C@@H]3C[C@@H]1C[C@](C3)(C2)C(=O)NCc1ccncc1 13768CC(C)(Oc1ccc(Cl)cc1)C(=O)N[C@H]1C2C[C@@H]3C[C@@H]1C[C@](C3)(C2)C(=O)NCC(N)=O 13769CNC(=O)NC(=O)[C@@]12C[C@@H]3CC(C1)[C@H](NC(=O)C(C)(C)Oc1ccc(Cl)cc1)[C@H](C3)C2 13770CC(C)(Oc1ccc(Cl)cc1)C(=O)N[C@H]1C2C[C@@H]3C[C@@H]1C[C@](CO)(C3)C2 13771CC(C)(Oc1ccc(Cl)cc1)C(=O)N[C@H]1C2C[C@@H]3C[C@@H]1C[C@](COCC(O)=O)(C3)C2 13772CC(C)(Oc1ccc(F)cc1Cl)C(=O)N[C@H]1C2C[C@@H]3C[C@@H]1C[C@](C3)(C2)c1nnn[nH]1 13773CC(C)(Oc1ccccc1Cl)C(=O)N[C@H]1C2C[C@@H]3C[C@@H]1C[C@](C3)(C2)C(=O)NS(C)(=O)=O 13774CC(C)(Oc1ccccc1Cl)C(=O)N[C@H]1C2C[C@@H]3C[C@@H]1C[C@](C3)(C2)C(=O)NS(=O)(=O)c1ccccc1 22451CCC1(C)SC(NC2CCCCC2)=NC1=O 22453CCCC1(C)SC(NC2CCCCC2)=NC1=O 22454CCC1(C)SC(NCC2CCCCC2)=NC1=O 22455CCCC1(C)SC(NCC2CCCCC2)=NC1=O 22456CCC1(C)SC(NC2CCCCCC2)=NC1=O 22457CCCC1(C)SC(NC2CCCCCC2)=NC1=O 22458CCC1(C)SC(NC2CCCCCCC2)=NC1=O 22459CCCC1(C)SC(NC2CCCCCCC2)=NC1=O 22460CCC1(C)SC(NC2C(C)(C)C2(C)C)=NC1=O 22461CCCC1(C)SC(NC2C(C)(C)C2(C)C)=NC1=O 22462CCC1(C)SC(NC23CCC(CC2)C3)=NC1=O 22463CCCC1(C)SC(NC23CCC(CC2)C3)=NC1=O 22464CCC1(C)SC(NC2C3CCC2CC3)=NC1=O 22465CCCC1(C)SC(NC2C3CCC2CC3)=NC1=O 22466CCC1(C)SC(NC23CC4CC2CC(C3)C4)=NC1=O 22467CCCC1(C)SC(NC23CC4CC2CC(C3)C4)=NC1=O 22468CCC1(C)SC(NC23CC4CC(CC(C4)C2)C3)=NC1=O 22469CCCC1(C)SC(NC23CC4CC(CC(C4)C2)C3)=NC1=O 22470CCC1(CC)SC(NC2CCCCCCC2)=NC1=O 22471O=C1N=C(NC2CCCCCCC2)SC11CCCC1 22472CCC1(CC)SC(NC23CC4CC2CC(C3)C4)=NC1=O 22473O=C1N=C(NC23CC4CC2CC(C3)C4)SC11CCCC1 22474CCC1(CC)SC(NC23CC4CC(CC(C4)C2)C3)=NC1=O 22475O=C1N=C(NC23CC4CC(CC(C4)C2)C3)SC11CCCC1 25902NS(=O)(=O)c1cc(C(O)=O)c(NCc2ccco2)cc1Cl 28361C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@@H](CC1)c1cccnc1)C(F)(F)F 28363C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@H](CC#N)CC1)C(F)(F)F 28364C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@@H]1CC[C@H](CC#N)CC1)C(F)(F)F 28365C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@H](CCC#N)CC1)C(F)(F)F 28366C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@@H]1CC[C@H](CCC#N)CC1)C(F)(F)F 28367CC(C)(C[C@H]1CC[C@@H](CC1)N(C1CC1)C(=O)c1ccc(cc1)[C@](C)(O)C(F)(F)F)C#N 28368CC(C)(C[C@H]1CC[C@H](CC1)N(C1CC1)C(=O)c1ccc(cc1)[C@](C)(O)C(F)(F)F)C#N 28369C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@H](CC2(CC2)C#N)CC1)C(F)(F)F 28370C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)C1CCC(CC(N)=O)CC1)C(F)(F)F 28371C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@H](CCC(N)=O)CC1)C(F)(F)F 28372C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@@H]1CC[C@H](CCC(N)=O)CC1)C(F)(F)F 28373CC(C)(C[C@H]1CC[C@@H](CC1)N(C1CC1)C(=O)c1ccc(cc1)[C@](C)(O)C(F)(F)F)C(N)=O 28374C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@H](CC2(CC2)C(N)=O)CC1)C(F)(F)F 28375C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC2(CC2)C#N)CC1)C(F)(F)F 28376C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC2(CC2)C(N)=O)CC1)C(F)(F)F 29828Fc1ccc2OC3(CCN(CC3)C(=O)C3(CC3)c3ccccc3)CC(=O)c2c1 29829Clc1ccc(cc1)C1(CC1)C(=O)N1CCCC2(CCc3ccccc23)C1 29830Clc1ccc(cc1)C1(CC1)C(=O)N1CCC2(CCc3ccccc23)C1 29831Clc1ccc(cc1)C1(CC1)C(=O)N1CCC2(CC1)C=Cc1ccccc21 29832Clc1ccc(cc1)C1(CC1)C(=O)N1CCC2(C1)CCCc1ccccc21 29833Clc1ccc(cc1)C1(CC1)C(=O)N1CCC2(C1)CCCCC2 29834Fc1ccc(cc1)C1(CC1)C(=O)N1CCC2(C1)CCCCC2 29835Fc1ccc(CC(=O)N2CCC3(C2)CCCCC3)cc1 29836Clc1ccc(CC(=O)N2CCC3(C2)CCCCC3)cc1 29837O=C(N1CCC2(C1)CCCCC2)C1(CC1)c1ccccn1 29838O=C(N1CCC2(C1)CCCCC2)C1(CC1)c1ccncc1 29839CC(C)(C(=O)N1CCC2(C1)CCCCC2)c1ccccc1 29840O=C(N1CCC2(C1)CCCCC2)C1(CC1)c1ccccc1 29841CCN(CC)C(=O)Cc1cccc(NS(=O)(=O)c2cccc(Cl)c2C)n1 29843Cc1c(Cl)cccc1S(=O)(=O)Nc1cccc(CC(=O)N2CCCCC2)n1 29849Cc1cccc(NS(=O)(=O)c2cccc(Cl)c2C)n1 29850Cc1cccc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)n1 29854Cc1cccc(NS(=O)(=O)c2ccc3ccccc3c2)n1 29856Cc1cccc(NS(=O)(=O)c2ccc(cc2)-c2ccccc2)n1 29857Cc1cccc(NS(=O)(=O)c2ccc(cc2)-c2ccc(F)cc2)n1 29858Cc1cccc(NS(=O)(=O)c2ccc(cc2)-c2ccc(Cl)cc2)n1 29859Cc1ccc(cc1)-c1ccc(cc1)S(=O)(=O)Nc1cccc(C)n1 29860Cc1cccc(NS(=O)(=O)c2ccc(cc2)-c2ccc(cc2)C#N)n1 29861CCc1cccc(NS(=O)(=O)c2ccc(cc2)-c2ccc(cc2)C#N)n1 29862O=S(=O)(Nc1cccc(n1)C1CC1)c1ccc(cc1)-c1ccc(cc1)C#N 29863CC(C)c1cccc(NS(=O)(=O)c2ccc(cc2)-c2ccc(cc2)C#N)n1 29864Nc1cccc(NS(=O)(=O)c2ccc(cc2)-c2ccc(cc2)C#N)n1 29865CNc1cccc(NS(=O)(=O)c2ccc(cc2)-c2ccc(cc2)C#N)n1 29866CCNc1cccc(NS(=O)(=O)c2ccc(cc2)-c2ccc(cc2)C#N)n1 32530FC(F)(F)c1cccnc1N1CCN(CC1)S(=O)(=O)c1ccccc1 32546FC(F)(F)c1cccnc1N1CCN(CC1)S(=O)(=O)c1ccc2ccccc2c1 32547FC(F)(F)c1cccnc1N1CCN(CC1)S(=O)(=O)c1cccc2ccccc12 32573C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(cc1)C(C)(C)C)c1ccc(cc1)[N+]([O-])=O 47119C[C@H](N1CC[C@@](CCCNS(C)(=O)=O)(OC1=O)c1ccc(F)cc1)c1ccc(cc1)-c1ccc(=O)n(C)c1 47120NA 47121NA 47123NA 72094O=C(CSc1nnc(-c2ccccc2)c(n1)-c1ccccc1)N1CCc2ccccc12 97725Clc1ccc(cc1)C1(CC1)C(=O)N1CCC2(CC12)c1c[nH]c2ncccc12 99290Oc1ccc(cc1)C(=O)N1CCCC2[C@@H]1CCc1ccccc21 99291O=C(N1CCCC2[C@@H]1CCc1ccccc21)c1ccc2nc[nH]c2c1 99292O=C(N1CCC[C@@H]2[C@H]1CCc1ccccc21)c1ccc2nc[nH]c2c1 99293O=C(N1CCCC2[C@H]1CCc1ccccc21)c1ccc2nc[nH]c2c1 99294NC(=O)c1ccc(cc1)C(=O)N1CCCC2[C@@H]1CCc1ccccc21 99295COc1cccc2C3CCCN([C@H]3CCc12)C(=O)c1ccc2nc[nH]c2c1 99296Oc1cccc2C3CCCN([C@H]3CCc12)C(=O)c1ccc2nc[nH]c2c1 99297COc1cccc2CC[C@H]3C(CCCN3C(=O)c3ccc4nc[nH]c4c3)c12 99298COc1cccc2CC[C@@H]3C(CCCN3C(=O)c3ccc4nc[nH]c4c3)c12 99299C[C@]12CCCN([C@H]1CCc1ccccc21)C(=O)c1ccc2nc[nH]c2c1 99300C[C@]12CCCN([C@@H]1CCc1ccccc21)C(=O)c1ccc2nc[nH]c2c1 99301COc1cccc2C3CCCN([C@@H]3CCc12)C(=O)c1ccc2nc[nH]c2c1 99302Oc1cccc2CC[C@H]3C(CCCN3C(=O)c3ccc4nc[nH]c4c3)c12 99303COc1ccc2CC[C@H]3C(CCCN3C(=O)c3ccc4nc[nH]c4c3)c2c1 99304COc1ccc2CC[C@@H]3C(CCCN3C(=O)c3ccc4nc[nH]c4c3)c2c1 99305Oc1ccc2CC[C@H]3C(CCCN3C(=O)c3ccc4nc[nH]c4c3)c2c1 99306Oc1ccc2CC[C@@H]3C(CCCN3C(=O)c3ccc4nc[nH]c4c3)c2c1 99307Oc1cccc2CC[C@@H]3C(CCCN3C(=O)c3ccc4nc[nH]c4c3)c12 99308Oc1cccc2C3CCCN([C@@H]3CCc12)C(=O)c1ccc2nc[nH]c2c1 99309Fc1cc(F)c2CC[C@H]3C(CCCN3C(=O)c3ccc4nc[nH]c4c3)c2c1 99310Fc1cc(F)c2CC[C@@H]3C(CCCN3C(=O)c3ccc4nc[nH]c4c3)c2c1 99311COc1ccc2C3CCCN([C@H]3CCc2c1)C(=O)c1ccc2nc[nH]c2c1 99312COc1ccc2C3CCCN([C@@H]3CCc2c1)C(=O)c1ccc2nc[nH]c2c1 99313Oc1ccc2C3CCCN([C@@H]3CCc2c1)C(=O)c1ccc2nc[nH]c2c1 99314Oc1ccc2C3CCCN([C@H]3CCc2c1)C(=O)c1ccc2nc[nH]c2c1 99315Fc1cccc2CC[C@@H]3C(CCCN3C(=O)c3ccc4nc[nH]c4c3)c12 99316Fc1cccc2CC[C@H]3C(CCCN3C(=O)c3ccc4nc[nH]c4c3)c12 99317O=C(N1CCCC2[C@H]1CCc1cc(ccc21)-c1ccccc1)c1ccc2nc[nH]c2c1 99318O=C(N1CCCC2[C@@H]1CCc1cc(ccc21)-c1ccccc1)c1ccc2nc[nH]c2c1 99319O=C(N1CCCC2[C@@H]1CCc1ccccc21)c1ccc2[nH]cnc2n1 99320O=C(N1CCCC2[C@@H]1CCc1ccccc21)c1ccc2nccn2c1 99321O=C(N1CCCC2[C@@H]1CCc1ccccc21)c1ccc2[nH]c(=O)sc2c1 99322COC(=O)c1ccc2C3CCCN([C@H]3CCc2c1)C(=O)c1ccc2nc[nH]c2c1 99323OCc1ccc2C3CCCN([C@H]3CCc2c1)C(=O)c1ccc2nc[nH]c2c1 99324OC(=O)c1ccc2C3CCCN([C@H]3CCc2c1)C(=O)c1ccc2nc[nH]c2c1 99325CNC(=O)c1ccc2C3CCCN([C@H]3CCc2c1)C(=O)c1ccc2nc[nH]c2c1 99326NC(=O)c1ccc2C3CCCN([C@H]3CCc2c1)C(=O)c1ccc2nc[nH]c2c1 99327CN(C)C(=O)c1ccc2C3CCCN([C@H]3CCc2c1)C(=O)c1ccc2nc[nH]c2c1 99328O=C(N1CCCC1)c1ccc2C3CCCN([C@H]3CCc2c1)C(=O)c1ccc2nc[nH]c2c1 99329O=C(N1CCOCC1)c1ccc2C3CCCN([C@H]3CCc2c1)C(=O)c1ccc2nc[nH]c2c1 99330CC(C)(O)c1ccc2C3CCCN([C@H]3CCc2c1)C(=O)c1ccc2nc[nH]c2c1 99331O=C(N1CCCC2[C@@H]1CCc1cc(ccc21)C#N)c1ccc2nc[nH]c2c1 99332Nc1nc2ccc(cc2s1)C(=O)N1CCCC2[C@@H]1CCc1ccccc21 99333Cc1ccc(cc1O)C(=O)N1CCCC2[C@@H]1CCc1ccccc21 99334COc1ccc(cc1N)C(=O)N1CCCC2[C@@H]1CCc1ccccc21 99335Cc1cc2cc(ccc2[nH]1)C(=O)N1CCCC2[C@@H]1CCc1ccccc21 99336Cn1c2ccc(cc2[nH]c1=O)C(=O)N1CCCC2[C@@H]1CCc1ccccc21 99337O=C(N1CCCC2[C@@H]1CCc1ccccc21)c1ccc2cc[nH]c2c1 99338O=C(N1CCCC2[C@@H]1CCc1ccccc21)c1ccc2NC(=O)Cc2c1 99339O=C(N1CCCC2[C@@H]1CCc1ccccc21)c1ccc2CC(=O)Nc2c1 99340Cn1cnc2cc(ccc12)C(=O)N1CCCC2[C@@H]1CCc1ccccc21 99341Cn1nnc2cc(ccc12)C(=O)N1CCCC2[C@@H]1CCc1ccccc21 99342COc1cccc2C3CCCN([C@H]3CCc12)C(=O)c1cn(C)c2ccccc12 99343Oc1ccc(cc1F)C(=O)N1CCCC2[C@@H]1CCc1ccccc21 99344Cc1nc2ccc(cc2[nH]1)C(=O)N1CCCC2[C@@H]1CCc1ccccc21 99345Nc1ccc(cc1Cl)C(=O)N1CCCC2[C@@H]1CCc1ccccc21 99346Nc1nc2ccc(cc2[nH]1)C(=O)N1CCCC2[C@@H]1CCc1ccccc21 99347O=C(N1CCCC2[C@@H]1CCc1ccccc21)c1ccc2ncsc2c1 99348Oc1cc(ccc1Cl)C(=O)N1CCCC2[C@@H]1CCc1ccccc21 99350O=C(N1CCCC2[C@@H]1CCc1ccccc21)c1ccc2[nH]c(=O)[nH]c2c1 99351Cn1cnc2ccc(cc12)C(=O)N1CCCC2[C@@H]1CCc1ccccc21 99352Nc1cc(ccc1F)C(=O)N1CCCC2[C@@H]1CCc1ccccc21 99353O=C(N1CCCC2[C@@H]1CCc1ccccc21)c1ccn2ccnc2c1 99354O=C(N1CCCC2[C@@H]1CCc1ccccc21)c1ccc2[nH]ncc2c1 99355CC1(C)C(=O)Nc2ccc(cc12)C(=O)N1CCCC2[C@@H]1CCc1ccccc21 99356Nc1ccc(cc1)C(=O)N1CCCC2[C@@H]1CCc1ccccc21 99358O=C(N1CCCC2[C@@H]1CCc1ccccc21)c1ccc2[nH]ccc2c1 99359O=C(N1CCCC2[C@@H]1CCc1ccccc21)c1c[nH]c2ccccc12 99360Oc1c(Cl)cc(cc1Cl)C(=O)N1CCCC2[C@@H]1CCc1ccccc21 99361O=C(N1CCCC2[C@@H]1CCc1ccccc21)c1ccc2nn[nH]c2c1 99362Cn1cc(C(=O)N2CCCC3[C@@H]2CCc2ccccc32)c2ccccc12 99363COc1ccc(cc1O)C(=O)N1CCCC2[C@@H]1CCc1ccccc21 99364Oc1ccc(cc1Cl)C(=O)N1CCCC2[C@@H]1CCc1ccccc21 99365Nc1cc(ccc1Cl)C(=O)N1CCCC2[C@@H]1CCc1ccccc21 99366Cc1ccc(cc1N)C(=O)N1CCCC2[C@@H]1CCc1ccccc21 99367COc1cc(ccc1N)C(=O)N1CCCC2[C@@H]1CCc1ccccc21 99368Nc1ccc(cc1F)C(=O)N1CCCC2[C@@H]1CCc1ccccc21 99369O=C(N1CCCC2[C@@H]1CCc1ccccc21)c1ccc2[nH]c(=O)cnc2c1 99370Cn1cc(C(=O)N2CCCC3[C@@H]2CCc2c(O)cccc32)c2ccccc12 99371O=C(N1CCCC2[C@@H]1CCc1cc(Cc3ccccc3)ccc21)c1ccc2nc[nH]c2c1 99372O=C(N1CCCC2[C@@H]1CCc1cc(CC3CCCCC3)ccc21)c1ccc2nc[nH]c2c1 99373OCc1cccc2CC[C@H]3C(CCCN3C(=O)c3ccc4nc[nH]c4c3)c12 99374COc1ccc(Cc2cccc3CC[C@H]4C(CCCN4C(=O)c4ccc5nc[nH]c5c4)c23)cc1 99375CC1(C)C[C@H]2C(CCCN2C(=O)c2ccc3nc[nH]c3c2)c2ccccc12 99376NC(=O)c1cccc2CC[C@H]3C(CCCN3C(=O)c3ccc4nc[nH]c4c3)c12 99377O=C(N1CCCC2[C@@H]1CCc1cccc(C#N)c21)c1ccc2nc[nH]c2c1 99378COc1ccc(Oc2ccc3C4CCCN([C@H]4CCc3c2)C(=O)c2ccc3nc[nH]c3c2)cc1 99379O=C(N1CCCC2[C@H]1CCc1ccc(cc21)C#N)c1ccc2nc[nH]c2c1 99380O=C(N1CCCC2[C@@H]1CCc1ccc(cc21)C#N)c1ccc2nc[nH]c2c1 99381Cc1ccc(Oc2cccc3CC[C@H]4C(CCCN4C(=O)c4ccc5nc[nH]c5c4)c23)nn1 99382O=C(N1CCCC2[C@@H]1Cc1ccccc21)c1ccc2nc[nH]c2c1 99383O=C(N1CCC[C@H]2[C@@H]1Cc1ccccc21)c1ccc2nc[nH]c2c1 99384O=C(N1CCC[C@@H]2[C@H]1Cc1ccccc21)c1ccc2nc[nH]c2c1 99385NC(=O)c1ccc(cc1)C(=O)N1CCCC2[C@@H]1Cc1ccccc21 99386Brc1ccc2C[C@H]3C(CCCN3C(=O)c3ccc4nc[nH]c4c3)c2c1 99387OC(=O)c1ccc2C[C@H]3C(CCCN3C(=O)c3ccc4nc[nH]c4c3)c2c1 99388OC(=O)c1ccc2C3CCCN([C@H]3Cc2c1)C(=O)c1ccc2nc[nH]c2c1 99389NC(=O)c1ccc2C[C@H]3C(CCCN3C(=O)c3ccc4nc[nH]c4c3)c2c1 99390CNC(=O)c1ccc2C3CCCN([C@H]3Cc2c1)C(=O)c1ccc2nc[nH]c2c1 99391O=C(N1CCCC2[C@@H]1Cc1ccccc21)c1ccc2[nH]cnc2n1 99392O=C(N1CCCC2[C@@H]1Cc1ccccc21)c1ccc2[nH]c(=O)sc2c1 99393O=C(N1CCCC2[C@@H]1Cc1ccccc21)c1ccc2nccn2c1 99394CC[C@]12CCCN([C@@H]1CCc1ccccc21)C(=O)c1ccc2nc[nH]c2c1 99395O=C(N1CCCC2[C@@H]1Cc1ccc(cc21)C#N)c1ccc2nc[nH]c2c1 99396O=C(N1CCC[C@H]2[C@@H]1Cc1ccc(cc21)C#N)c1ccc2nc[nH]c2c1 99397O=C(N1CCC[C@@H]2[C@H]1Cc1ccc(cc21)C#N)c1ccc2nc[nH]c2c1 99398Nc1nc2ccc(cc2s1)C(=O)N1CCCC2[C@@H]1Cc1ccccc21 99399Cc1ccc(cc1O)C(=O)N1CCCC2[C@@H]1Cc1ccccc21 99400COc1ccc(cc1N)C(=O)N1CCCC2[C@@H]1Cc1ccccc21 99401Cc1cc2cc(ccc2[nH]1)C(=O)N1CCCC2[C@@H]1Cc1ccccc21 99402Cn1c2ccc(cc2[nH]c1=O)C(=O)N1CCCC2[C@@H]1Cc1ccccc21 99403O=C(N1CCCC2[C@@H]1Cc1ccccc21)c1ccc2cc[nH]c2c1 99404O=C(N1CCCC2[C@@H]1Cc1ccccc21)c1ccc2NC(=O)Cc2c1 99405O=C(N1CCCC2[C@@H]1Cc1ccccc21)c1ccc2CC(=O)Nc2c1 99406Cn1cnc2cc(ccc12)C(=O)N1CCCC2[C@@H]1Cc1ccccc21 99407Cn1nnc2cc(ccc12)C(=O)N1CCCC2[C@@H]1Cc1ccccc21 99408Oc1ccc2[C@H]3CCCN([C@H]3Cc2c1)C(=O)c1ccc2nc[nH]c2c1 99409Cc1cc(ccc1O)C(=O)N1CCCC2[C@@H]1Cc1ccccc21 99410Cc1nc2ccc(cc2[nH]1)C(=O)N1CCCC2[C@@H]1Cc1ccccc21 99411Nc1ccc(cc1Cl)C(=O)N1CCCC2[C@@H]1Cc1ccccc21 99412O=C(N1CCCC2[C@@H]1Cc1ccccc21)c1ccc2cn[nH]c2c1 99413Nc1nc2ccc(cc2[nH]1)C(=O)N1CCCC2[C@@H]1Cc1ccccc21 99414O=C(N1CCCC2[C@@H]1Cc1ccccc21)c1ccc2ncsc2c1 99415Oc1cc(ccc1Cl)C(=O)N1CCCC2[C@@H]1Cc1ccccc21 99416O=C(N1CCCC2[C@@H]1Cc1ccccc21)c1cnc2nc[nH]c2c1 99417O=C(N1CCCC2[C@@H]1Cc1ccccc21)c1ccc2[nH]c(=O)[nH]c2c1 99418Cn1cnc2ccc(cc12)C(=O)N1CCCC2[C@@H]1Cc1ccccc21 99419Nc1cc(ccc1F)C(=O)N1CCCC2[C@@H]1Cc1ccccc21 99420O=C(N1CCCC2[C@@H]1Cc1ccccc21)c1ccn2ccnc2c1 99421O=C(N1CCCC2[C@@H]1Cc1ccccc21)c1ccc2[nH]ncc2c1 99422Nc1ccc(cc1)C(=O)N1CCCC2[C@@H]1Cc1ccccc21 99423Oc1ccc(cc1)C(=O)N1CCCC2[C@@H]1Cc1ccccc21 99424O=C(N1CCCC2[C@@H]1Cc1ccccc21)c1ccc2[nH]ccc2c1 99425O=C(N1CCCC2[C@@H]1Cc1ccccc21)c1c[nH]c2ccccc12 99426Oc1c(Cl)cc(cc1Cl)C(=O)N1CCCC2[C@@H]1Cc1ccccc21 99427O=C(N1CCCC2[C@@H]1Cc1ccccc21)c1ccc2nn[nH]c2c1 99428Cn1cc(C(=O)N2CCCC3[C@@H]2Cc2ccccc32)c2ccccc12 99429COc1ccc(cc1O)C(=O)N1CCCC2[C@@H]1Cc1ccccc21 99430Oc1ccc(cc1Cl)C(=O)N1CCCC2[C@@H]1Cc1ccccc21 99431Nc1cc(ccc1Cl)C(=O)N1CCCC2[C@@H]1Cc1ccccc21 99432Cc1ccc(cc1N)C(=O)N1CCCC2[C@@H]1Cc1ccccc21 99433COc1cc(ccc1N)C(=O)N1CCCC2[C@@H]1Cc1ccccc21 99434Nc1ccc(cc1F)C(=O)N1CCCC2[C@@H]1Cc1ccccc21 99435C[C@H]1CCN([C@H]2Cc3ccccc3[C@@H]12)C(=O)c1ccc2nc[nH]c2c1 99436O=C(N1CCCC2[C@@H]1Cc1ccccc21)c1ccc2[nH]c(=O)cnc2c1 99437O=C(N1CCC[C@H]2[C@@H]1Cc1cc(ccc21)C#N)c1ccc2nc[nH]c2c1 99438COc1ccc2C[C@H]3[C@H](CCCN3C(=O)c3ccc4nc[nH]c4c3)c2c1 99439Oc1ccc2C[C@H]3[C@H](CCCN3C(=O)c3ccc4nc[nH]c4c3)c2c1 99440Nc1ccc2[C@H]3CCCN([C@H]3Cc2c1)C(=O)c1ccc2nc[nH]c2c1 99441Cc1cc(cc2[nH]cnc12)C(=O)N1CCC[C@H]2[C@@H]1Cc1ccc(cc21)C#N 99442Cc1cc2nc[nH]c2cc1C(=O)N1CCC[C@H]2[C@@H]1Cc1ccc(cc21)C#N 99443COC(=O)c1ccc2C[C@H]3[C@H](CCCN3C(=O)c3ccc4nc[nH]c4c3)c2c1 99444O=C(N1CCC[C@H]2[C@@H]1Cc1ccc(cc21)C#C)c1ccc2nc[nH]c2c1 99445OCc1ccc2C[C@H]3[C@H](CCCN3C(=O)c3ccc4nc[nH]c4c3)c2c1 99446CC(C)(O)c1ccc2C[C@H]3[C@H](CCCN3C(=O)c3ccc4nc[nH]c4c3)c2c1 99447O=C(N1CCC[C@H]2[C@@H]1Cc1ccc(cc21)-c1ccccc1)c1ccc2nc[nH]c2c1 99448O=C(N1CCC[C@H]2[C@@H]1Cc1ccc(cc21)C#Cc1ccccc1)c1ccc2nc[nH]c2c1 99449O=C(N1CCC[C@H]2[C@@H]1Cc1ccc(cc21)-c1ccoc1)c1ccc2nc[nH]c2c1 99450CC#Cc1ccc2C[C@H]3[C@H](CCCN3C(=O)c3ccc4nc[nH]c4c3)c2c1 99451Cn1cc(cn1)-c1ccc2C[C@H]3[C@H](CCCN3C(=O)c3ccc4nc[nH]c4c3)c2c1 99452Cc1ccc2C[C@H]3[C@H](CCCN3C(=O)c3ccc4nc[nH]c4c3)c2c1 99453O=C(N1CCC[C@H]2[C@@H]1Cc1ccc(cc21)C1CCOCC1)c1ccc2nc[nH]c2c1 99454O=C(N1CCC[C@H]2[C@@H]1Cc1ccc(cc21)C1CCCC1)c1ccc2nc[nH]c2c1 99455CC(=O)Nc1ccc2[C@H]3CCCN([C@H]3Cc2c1)C(=O)c1ccc2nc[nH]c2c1 99456CS(=O)(=O)Nc1ccc2[C@H]3CCCN([C@H]3Cc2c1)C(=O)c1ccc2nc[nH]c2c1 99457Oc1cc2[C@H]3CCCN([C@H]3Cc2cc1[N+]([O-])=O)C(=O)c1ccc2nc[nH]c2c1 99458Nc1cc2C[C@H]3[C@H](CCCN3C(=O)c3ccc4nc[nH]c4c3)c2cc1O 99459Cc1nc2cc3C[C@H]4[C@H](CCCN4C(=O)c4ccc5nc[nH]c5c4)c3cc2o1 99460O=C(N1CCC[C@H]2[C@@H]1Cc1cc3ncoc3cc21)c1ccc2nc[nH]c2c1 99461COc1cc2[C@H]3CCCN([C@H]3Cc2cc1C)C(=O)c1ccc2nc[nH]c2c1 99462Cc1cc2C[C@H]3[C@H](CCCN3C(=O)c3ccc4nc[nH]c4c3)c2cc1O 99463Cc1cc2C[C@H]3[C@H](CCCN3C(=O)c3ccc4nc[nH]c4c3)c2cc1C#N 99464Cc1c2[C@H]3CCCN([C@H]3Cc2ccc1C#N)C(=O)c1ccc2nc[nH]c2c1 99465Cc1cc2C[C@@H]3[C@@H](CCCN3C(=O)c3ccc4nc[nH]c4c3)c2cc1C#N 102426OC(=O)N1CCN(c2ccc(cn2)N2CCN(CC2)C2CCOCC2)c2ccccc12 102427CC(C)(C)N1CCN(CC1)c1ccc(nc1)N1CCN(C(=O)N[C@H]2C3CC4CC2C[C@@](CNS(C)(=O)=O)(C4)C3)c2ccccc12 102428NC(=O)C[C@]12CC3CC(C1)[C@H](NC(=O)N1CCN(c4ccc(cn4)N4CCN(CC4)S(=O)(=O)C4CC4)c4ccccc14)C(C3)C2 102429NC[C@]12CC3CC(C1)[C@H](NC(=O)N1CCN(c4ccc(cn4)N4CCN(CC4)S(=O)(=O)C4CC4)c4ccccc14)C(C3)C2 102430NC(=O)C[C@]12CC3CC(C1)[C@H](NC(=O)N1CCN(c4ccc(cn4)N4CCN(CC4)S(=O)(=O)C4CC4)c4ccccc14)C(C3)C2 102431CC(C)(C)N1CCN(CC1)c1ccc(nc1)N1CCN(C(=O)N[C@H]2C3CC4CC2C[C@@](C4)(C3)C(O)C(F)(F)F)c2ccccc12 102432CC(C)(C)N1CCN(CC1)c1ccc(nc1)N1CCN(C(=O)N[C@H]2C3CC4CC2C[C@@](Cc2nn[nH]n2)(C4)C3)c2ccccc12 102433CONC(=O)[C@]12CC3CC(C1)[C@H](NC(=O)N1CCN(c4ccc(cn4)N4CCN(CC4)S(=O)(=O)C4CC4)c4ccccc14)C(C3)C2 102434CC(C)(C)N1CCN(CC1)c1ccc(nc1)N1CCN(C(=O)N[C@H]2C3CC4CC2C[C@@](C4)(C3)NS(C)(=O)=O)c2ccccc12 107468C[C@H](N1CC[C@@](CC(C)(C)O)(OC1=O)c1ccccc1)c1ccc(cc1)-c1cnc(=O)n(C)c1 107469C[C@H](N1CC[C@@](CC(C)(C)C#N)(OC1=O)c1ccccc1)c1ccc(cc1)-c1ccc(=O)n(C)n1 107470C[C@H](N1CC[C@@](CCCO)(OC1=O)c1ccc(F)cc1)c1ccc(cc1)-c1cc(=O)n(C)cn1 107471C[C@H](N1CC[C@@](CCCO)(OC1=O)c1ccc(F)cc1)c1ccc(cc1)-c1ccc(=O)n(C)n1 107472C[C@H](N1CC[C@@](CCCO)(OC1=O)c1ccc(F)cc1)c1ccc(cc1)-c1ccn(C)c(=O)n1 107473C[C@H](N1CC[C@@](CC(C)(C)O)(OC1=O)c1ccc(F)cc1)c1ccc(cc1)-c1ccc(=O)n(C)n1 107474CCn1nc(ccc1=O)-c1ccc(cc1)[C@H](C)N1CC[C@@](CC(C)(C)O)(OC1=O)c1ccccc1 107475CC(C)n1nc(ccc1=O)-c1ccc(cc1)[C@H](C)N1CC[C@@](CC(C)(C)O)(OC1=O)c1ccccc1 107476C[C@H](N1CC[C@@](CC(C)(C)O)(OC1=O)c1ccccc1)c1ccc(cc1)-c1ccc(=O)n(CC(F)(F)F)n1 107477C[C@H](N1CC[C@@](CC(C)(C)O)(OC1=O)c1ccccc1)c1ccc(cc1)-c1cc(C)c(=O)n(C)n1 107479C[C@H](N1CC[C@@](CC(C)(C)O)(OC1=O)c1ccccc1)c1ccc(cc1)-c1ccc(=O)n(CC2CC2)n1 107480C[C@H](N1CC[C@@](CC(C)(C)O)(OC1=O)c1ccccc1)c1ccc(cc1)-c1ccc(=O)n(n1)C1CC1 107481OCC[C@@]1(CCN(C(=O)O1)c1cccc(c1)-c1ccc(F)cc1F)c1ccccc1 107482OCCC1(CCN(C(=O)O1)c1cccc(n1)-c1ccc(F)cc1F)c1ccccc1F 107483OCC[C@@]1(CCN(C(=O)O1)c1cccc(n1)-c1ccc(F)cc1)c1ccccc1 107484C[C@H](N1CC[C@@](CC(C)(C)O)(OC1=O)c1ccc(F)cc1)c1ccc(cc1)-c1ccc(F)cc1F 107485C[C@H](N1CC[C@@](CCC(N)=O)(OC1=O)c1ccccc1)c1ccc(cc1)-c1ccc(F)cc1 107486C[C@H](N1CC[C@@](CC(C)(C)O)(OC1=O)c1ccccc1)c1ccc(cc1)-c1ccc(F)cc1 107487C[C@H](N1CC[C@@](CC(C)(C)O)(OC1=O)c1ccc(F)cc1)c1ccc(Br)cc1 107488C[C@H](N1CC[C@@](CCO)(OC1=O)c1ccc(F)cc1)c1ccc(OC(F)F)cc1 107489C[C@H](N1CC[C@@](CC(C)(C)O)(OC1=O)c1ccccc1)c1ccc(Br)cc1 107491C[C@H](N1CC[C@@](CC(C)(C)O)(OC1=O)c1ccccc1)c1ccc(cc1)-c1c[nH]c(=O)cn1 107492C[C@H](N1CC[C@@](CC(C)(C)C#N)(OC1=O)c1ccccc1)c1ccc(cc1)-c1ccc(=O)[nH]n1 107493C[C@H](N1CC[C@@](CCCO)(OC1=O)c1ccc(F)cc1)c1ccc(cc1)-c1ccc(=O)[nH]n1 107494C[C@H](N1CC[C@@](CCCO)(OC1=O)c1ccc(F)cc1)c1ccc(cc1)-c1cc[nH]c(=O)n1 107495C[C@H](N1CC[C@@](CCCO)(OC1=O)c1ccc(F)cc1)c1ccc(cc1)-c1cc(=O)[nH]cn1 107496C[C@H](N1CC[C@@](CCCO)(OC1=O)c1ccccc1)c1ccc(cc1)-c1ccc(=O)n(C)n1 107577C[C@H](N1CC[C@@](CC(C)(C)O)(OC1=O)c1ccccc1)c1ccc(cc1)-c1ccc(=O)[nH]c1 107578C[C@H](N1CC[C@@](CC(C)(C)O)(OC1=O)c1ccccc1)c1ccc(cc1)-c1cc[nH]c(=O)c1 107579C[C@H](N1CC[C@@](CC(C)(C)N)(OC1=O)c1ccccc1)c1ccc(cc1)-c1ccc(=O)n(C)c1 107580C[C@H](N1CC[C@@](CC(C)(C)NC(C)=O)(OC1=O)c1ccccc1)c1ccc(cc1)-c1ccc(=O)n(C)c1 107581COC(=O)NC(C)(C)C[C@@]1(CCN([C@@H](C)c2ccc(cc2)-c2ccc(=O)n(C)c2)C(=O)O1)c1ccccc1 107582C[C@H](N1CC[C@@](CC(C)(C)NS(C)(=O)=O)(OC1=O)c1ccccc1)c1ccc(cc1)-c1ccc(=O)[nH]c1 107583C[C@H](N1CC[C@@](CC(C)(C)NS(C)(=O)=O)(OC1=O)c1ccccc1)c1ccc(cc1)-c1ccc(=O)n(C)c1 107584C[C@H](N1CC[C@@](CC(C)(C)N(C)S(C)(=O)=O)(OC1=O)c1ccccc1)c1ccc(cc1)-c1ccc(=O)n(C)c1 107585C[C@H](N1CC[C@@](CC(C)(C)C#N)(OC1=O)c1ccccc1)c1ccc(cc1)-c1cc[nH]c(=O)c1 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107664C[C@H](N1CC[C@@](CC(C)(C)O)(OC1=O)c1ccccc1)c1ccc(cc1)-c1ccn(C)c(=O)c1 107665CC(C)n1cc(ccc1=O)-c1ccc(cc1)[C@H](C)N1CC[C@@](CC(C)(C)O)(OC1=O)c1ccccc1 107666C[C@H](N1CC[C@@](CC(C)(C)C#C)(OC1=O)c1ccccc1)c1ccc(cc1)-c1ccc(=O)[nH]c1 107667CC(C)n1cc(ccc1=O)-c1ccc(cc1)[C@H](C)N1CC[C@@](CC(C)(C)C#C)(OC1=O)c1ccccc1 107669CC(C)[C@@]1(CC(C)(C)O)CCN([C@@H](C)c2ccc(cc2)-c2ccn(C3CC3)c(=O)c2)C(=O)O1 107670CCCn1cc(ccc1=O)-c1ccc(cc1)[C@H](C)N1CC[C@@](CC(C)(C)O)(OC1=O)c1ccccc1 107671C[C@H](N1CC[C@@](CC(C)(C)O)(OC1=O)c1ccccc1)c1ccc(cc1)-c1ccc(=O)n(CC(C)(C)C)c1 108085C[C@H](N1CC[C@@](CC(C)(C)O)(OC1=O)c1ccccc1)c1ccc(cc1)-c1ccc2nc(C)cn2n1 108086C[C@H](N1CC[C@@](CC(C)(C)O)(OC1=O)c1ccccc1)c1ccc(cc1)-c1ccc2nc(C)nn2c1 108088C[C@H](N1CC[C@@](CC(C)(C)O)(OC1=O)c1ccccc1)c1ccc(cc1)-c1ccn2nc(C)nc2c1 108089C[C@H](N1CC[C@@](CC(C)(C)O)(OC1=O)c1ccccc1)c1ccc(cc1)-c1ccn2ncnc2c1 108090COc1nc2ccc(cn2n1)-c1ccc(cc1)[C@H](C)N1CC[C@@](CC(C)(C)O)(OC1=O)c1ccccc1 108091C[C@H](N1CC[C@@](CC(C)(C)O)(OC1=O)c1ccccc1)c1ccc(cc1)-c1ccc2nccn2n1 108092C[C@H](N1CC[C@@](CC(C)(C)O)(OC1=O)c1ccccc1)c1ccc(cc1)-c1ccc2ncnn2c1 108093CC(C)[C@@]1(CC(C)(C)O)CCN([C@@H](C)c2ccc(cc2)-c2ccc3nc(C)nn3c2)C(=O)O1 108094CC(C)(O)C[C@@]1(CCN([C@H]2CCCN(C2)c2ccc3ncnn3c2)C(=O)O1)c1ccccc1 119209CCCSc1nc(ccc1C(=O)NC1CCCCC1)N1CCC(C1)C(O)=O 119210CCCSc1nc(OC2CCC(CC2)C(O)=O)ccc1C(=O)NC1CCCCC1 119211CCCSc1nc(NCCC(O)=O)ccc1C(=O)NC1CCCCC1 119212CCCSc1nc(ccc1C(=O)NC1CCCCC1)N1CCCC(C1)C1(CC1)C(O)=O 119213OC(=O)C[C@H]1CCN(C1)c1ccc(C(=O)NC2CCCCC2)c(SC2CCCC2)n1 119214CCCSc1nc(ccc1C(=O)NC1C2CC3CC(C2)CC1C3)N1CC[C@@H](C1)OCC(O)=O 119215CCCSc1nc(ccc1C(=O)NC1C2CC3CC(C2)CC1C3)N1CCOC(C1)C(O)=O 119216CCSc1nc(ccc1C(=O)NC1C2CC3CC(C2)CC1C3)N1CC[C@H](C1)C(O)=O 119217CCSc1nc(ccc1C(=O)NC1C2CC3CC(C2)CC1C3)N1C[C@H]2[C@@H](C1)[C@@H]2C(O)=O 119218CSc1nc(ccc1C(=O)NC1C2CC3CC(C2)CC1C3)N1C[C@H]2[C@@H](C1)[C@@H]2C(O)=O 119219CCCSc1nc(NC2CC[C@@H](CC2)C(O)=O)ccc1C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 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142007Cc1ncc(cn1)-c1ccc(cc1)C1(CC1)c1nnc2C[C@](C)(CO)SCCn12 142008Cc1ccc(nn1)-c1ccc(c(F)c1)C1(CC1)c1nnc2C[C@](C)(CO)SCCn12 142009CC(C)(O)CC1(CCN(C(=O)O1)C(C)(C)C#Cc1ccc(F)cc1)c1ccccc1 142010CC(=C)CC1(CCN(C(=O)O1)C(C)(C)C#Cc1ccc2n(C)c(=O)ccc2c1)c1ccccc1 142011CC(C)(C)CC1(CCN(C(=O)O1)C(C)(C)c1cn(nn1)-c1ccccc1)c1ccccc1 142013CC(C)(O)CC1(CCN(C(=O)O1)C(C)(C)c1ccc(Br)cc1)c1ccccc1 142014CC(=C)CC1(CCN(C(=O)O1)C(C)(C)C#Cc1ccc(F)cc1)c1ccccc1 142015CC(=C)CC1(CCN(C(=O)O1)C(C)(C)c1cn(nn1)-c1ccccc1)c1ccccc1 142016CC(=C)CC1(CCN(C(=O)O1)C1(CC1)c1ccc(cc1)-c1ccn(C)c(=O)c1)c1ccccc1 142017Cn1ccc(cc1=O)-c1ccc(cc1)C(C)(C)N1CCC(CC(C)(C)O)(OC1=O)c1ccccc1 142018CC(C)(O)CC1(CCN(C(=O)O1)C(C)(C)c1ccc(cc1)-c1ccn(C2CC2)c(=O)c1)c1ccccc1 50016982NC(=O)[C@@]12CC3CC(C[C@](C3)(C1)NC(=O)CN1CCCN(c3c(Cl)cc(Cl)cc3Cl)S1(=O)=O)C2 50016983[H][C@@]12CN(C[C@]1([H])[C@H]2C(O)=O)c1ccc(C(=O)NC23CC4CC(CC(C4)C2)C3)c(SC)n1 50016984[H][C@]12CCCC[C@@]1([H])N(CCC2)C(=O)c1csc(c1)C1CCN(CC1)C(=O)CCNS(C)(=O)=O 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50018794[H][C@@]12CC[C@@](C)(c3c1c(=O)n(-c1ccccc1)n3Cc1ccccc1)C2(C)C 50018795[H][C@@]12CC[C@@](C)(c3c1c(=O)n(-c1ccccc1)n3CC)C2(C)C 50018797[H][C@@]12CC[C@@](C)(c3c1c(=O)n(-c1ccccc1C(F)(F)F)n3C)C2(C)C 50018798[H][C@@]12CC[C@@](C)(c3c1c(=O)n(-c1ccccc1F)n3C(C)C)C2(C)C 50018799[H][C@@]12CC[C@@](C)(c3c1c(=O)n(-c1ccc(F)cc1F)n3CCc1ccccc1)C2(C)C 50018802[H][C@@]12CC[C@@](C)(c3c1c(=O)n(-c1ccccc1Cl)n3C)C2(C)C 50018803[H][C@@]12CC[C@@](C)(c3c1c(=O)n(Cc1cccc(c1)-c1ccccc1C)n3C)C2(C)C 50018804[H][C@@]12CC[C@@](C)(c3c1c(=O)n(-c1ccccc1F)n3CCC)C2(C)C 50018806[H][C@@]12CC[C@@](C)(c3c1c(=O)n(-c1ccccc1F)n3CC=C)C2(C)C 50018807[H][C@@]12CC[C@@](C)(c3c1c(=O)n(-c1cccc(OC)c1)n3C)C2(C)C 50018808[H][C@@]12CC[C@@](C)(c3c1c(=O)n(-c1ccccc1)n3C)C2(C)C 50018809[H][C@@]12CC[C@@](C)(c3c1c(=O)n(Cc1ccccc1)n3C)C2(C)C 50018810[H][C@]12CC[C@](C)(c3c1c(=O)n(-c1ccccc1)n3C)C2(C)C 50018811[H][C@@]12CC[C@@](C)(c3c1c(=O)n(-c1ccc(C)cc1)n3C)C2(C)C 50018812[H][C@@]12CC[C@@](C)(c3c1c(=O)n(-c1ccccn1)n3C)C2(C)C 50052665O=C(NCc1cccnc1)C12CC3CC(CC(C3)C1)C2 50067028COc1cc(\C=C\C(=O)\C=C\c2ccc(O)c(OC)c2)ccc1O 50067040COc1cc(C=CC(=O)CC(=O)C=Cc2ccc(O)c(OC)c2)ccc1O 50067044Oc1ccc(\C=C\C(=O)\C=C\c2ccc(O)cc2)cc1 50117900CN1CCN(CC1)C(=O)Cc1csc(NS(=O)(=O)c2cccc(Cl)c2C)n1 50117901CCN(CC)C(=O)Cc1csc(NS(=O)(=O)c2cccc(Cl)c2C)n1 50148911C[C@@H]1CC[C@@]2(CC[C@]3(C)C(=CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@@]34C)[C@@H]2[C@H]1C)C(O)=O 50167716FC(F)(F)c1ccc(cc1)-c1coc(NS(=O)(=O)c2ccccc2)n1 50167718FC(F)(F)c1ccc(cc1)C(=O)CS(=O)(=O)c1ccccc1 50167720O=S(=O)(Nc1nc(co1)-c1ccc(cc1)-c1ccccc1)c1ccccc1 50174278COc1ccc(cn1)-c1noc(n1)C12CCC(CC1)(CC2)c1nnc(-c2ccccc2C(F)(F)F)n1C 50174279Clc1ccc(cc1)-c1noc(n1)C12CCC(CC1)(CC2)c1nnc2CCCCCCn12 50174280Cc1noc(n1)C12CCC(CC1)(CC2)c1nnc2CCCCCCn12 50174281CCCCCC12CCC(CC1)(CC2)c1nnc(-c2ccccc2C(F)(F)F)n1C 50174282Cn1c(nnc1C12CCC(CC1)(CC2)c1nc(c[nH]1)-c1ccc(F)cc1)-c1ccccc1C(F)(F)F 50174283Cn1c(nnc1C12CCC(CC1)(CC2)c1nc(no1)-c1ccc(Cl)cc1)-c1ccccc1C(F)(F)F 50174284Cn1c(nnc1C12CCC(CC1)(CC2)c1nc(no1)-c1ccc(cc1)S(C)(=O)=O)-c1ccccc1C(F)(F)F 50174285CCCCCC12CCC(CC1)(CC2)c1nnc2CCCCCCn12 50174286Cn1c(nnc1C12CCC(CC1)(CC2)c1nc(no1)-c1ccc(F)cc1)-c1ccccc1S(C)(=O)=O 50174287Cn1c(nnc1C12CCC(CC1)(CC2)c1nc(no1)-c1ccc(=O)n(C)c1)-c1ccccc1C(F)(F)F 50174288Cn1c(nnc1C12CCC(CC1)(CC2)c1nnc([nH]1)-c1ccc(F)cc1)-c1ccccc1C(F)(F)F 50174289C(C1CC1)c1noc(n1)C12CCC(CC1)(CC2)c1nnc2CCCCCCn12 50174290COc1cc(O)ccc1-c1nnc(n1C)C12CCC(CC1)(CC2)c1nc(no1)-c1ccc(F)cc1 50174291COc1ccc(-c2nnc(n2C)C23CCC(CC2)(CC3)c2nc(no2)-c2ccc(F)cc2)c(Cl)c1 50174292Cn1c(nnc1C12CCC(CC1)(CC2)c1nnc(o1)-c1ccc(F)cc1)-c1ccccc1C(F)(F)F 50174293Cn1c(nnc1C12CCC(CC1)(CC2)c1nc(no1)-c1ccc(F)cc1)-c1ccccc1Cl 50174294COC(=O)C12CCC(CC1)(CC2)c1nnc2CCCCCCn12 50174295Cn1c(nnc1C12CCC(CC1)(CC2)c1nc(no1)-c1ccc(cc1)S(=O)(=O)C(F)(F)F)-c1ccccc1C(F)(F)F 50174296Cn1c(nnc1C12CCC(CC1)(CC2)c1noc(n1)-c1ccc(F)cc1)-c1ccccc1C(F)(F)F 50174297Cn1c(nnc1C12CCC(CC1)(CC2)c1nc(no1)-c1ccc(F)cc1F)-c1ccccc1C(F)(F)F 50174298Cn1c(nnc1C12CCC(CC1)(CC2)c1nc(no1)-c1ccc(F)cc1)-c1ccccc1C(F)(F)F 50174299Cn1c(nnc1C12CCC(CC1)(CC2)c1nc(no1)-c1ccc(cc1)C(O)C(F)(F)F)-c1ccccc1C(F)(F)F 50174300Cn1c(nnc1C12CCC(CC1)(CC2)c1nc(no1)-c1ccc(F)cc1)-c1ccccc1OC(F)F 50174301Cn1c(nnc1C12CCC(CC1)(CC2)c1nc(no1)-c1cccc(c1)S(C)(=O)=O)-c1ccccc1C(F)(F)F 50185127CC1(C)[C@H](CC[C@@]2(C)[C@H]1CC[C@]1(C)[C@@H]2C(=O)C=C2[C@@H]3C[C@](C)(CC[C@]3(C)CC[C@@]12C)C(O)=O)O[C@H]1O[C@@H]([C@@H](O)[C@H](O)[C@H]1O[C@@H]1O[C@@H]([C@@H](O)[C@H](O)[C@H]1O)C(O)=O)C(O)=O 50188385CC(=O)O[C@H]1CC[C@@]2(C)[C@@H](CC[C@]3(C)[C@@H]2C(=O)C=C2[C@@H]4C[C@](C)(CC[C@]4(C)CC[C@@]32C)C(O)=O)C1(C)C 50188386COC(=O)[C@@]1(C)CC[C@]2(C)CC[C@]3(C)C(=CC(=O)[C@@H]4[C@@]5(C)CC[C@H](Oc6ccccc6C(O)=O)C(C)(C)[C@@H]5CC[C@@]34C)[C@@H]2C1 50188387CC1(C)[C@@H](N)CC[C@@]2(C)[C@H]1CC[C@]1(C)[C@@H]2C(=O)C=C2[C@@H]3C[C@](C)(CC[C@]3(C)CC[C@@]12C)C(O)=O 50188388C[C@H]1C[C@@]2(C)CC[C@@](C)(C[C@@]2(C)C2=CC(=O)[C@@H]3[C@@]4(C)CC[C@H](O)C(C)(C)[C@@H]4CC[C@@]3(C)[C@]12C)C(=O)N[C@H](Cc1ccccc1)C(O)=O 50188389COc1ccc(CCNC(=O)C23CCC(C)(C(=O)C2=O)C3(C)C)cc1OC 50188390CC(CCC(O)=O)C1CC[C@@]2(C)C3=C(C(=O)C[C@]12C)[C@@]1(C)CCC(OC(C)=O)C(C)(C)[C@@H]1CC3=O 50188391COCCC1C(C(C(=O)c2ccc(OC)c(C)c2)C(=O)C1=O)c1ccc(Cl)cc1Cl 50192671CC(C)(Oc1ccc(Cl)cc1)C(=O)NC1CCCC(CCC1)C#N 50192672CC(C)(N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(=O)N[C@H]1C2CCCC1C[C@H](C2)C(N)=O 50192673CC(C)(Oc1ccc(Cl)cc1)C(=O)N[C@H]1C2CC3CC1CC(O)(C2)O3 50192674CC(C)(N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(=O)NC12CCC(CC1)(CC2)C(N)=O 50192675CC(C)(Oc1ccc(Cl)cc1)C(=O)N[C@H]1C2COCC1C[C@H](C2)C(N)=O 50192676CC(C)(N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(=O)N[C@H]1C2CCCC1C[C@H](C2)C(O)=O 50192677CC(C)(N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(=O)NC1CC[C@H]2[C@@H](CC1)[C@@H]2C(N)=O 50192678CCOC(=O)[C@@H]1[C@H]2CCC(CC[C@@H]12)NC(=O)C(C)(C)Oc1ccc(Cl)cc1 50192679CC(C)(Oc1ccc(Cl)cc1)C(=O)N[C@H]1C2CCCC1C[C@H](C2)C(N)=O 50192680CC(C)(N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(=O)NC1CC2CC(C1)CC(C2)C(N)=O 50192681CC(C)(N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(=O)NC1CCCC(CCC1)C#N 50192682CC(C)(N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(=O)N[C@H]1C2CCC1C[C@H](C2)C(O)=O 50192683CC(C)(N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(=O)N[C@@H]1C2CCCC1C[C@H](C2)C(N)=O 50192684CC(C)(Oc1ccc(cn1)C#N)C(=O)N[C@@H]1C2CCCC1C[C@H](C2)C(N)=O 50192685CC(C)(Oc1ccc(Cl)cc1)C(=O)N[C@@H]1C2CCCC1C[C@H](C2)C(O)=O 50192686CC(C)(Oc1ccc(Cl)cc1)C(=O)NC12CCC(CC1)(CC2)C(N)=O 50192687CC(C)(Oc1ccc(Cl)cc1)C(=O)N[C@H]1C2CCCC1C[C@H](C2)C(O)=O 50192785CC(C)(Oc1ccc(cn1)C#N)C(=O)N[C@H]1C2C[C@@H]3C[C@H]1C[C@](CC(N)=O)(C3)C2 50192786CC(C)(Oc1ccc(cn1)N1CCOCC1)C(=O)N[C@H]1C2C[C@@H]3C[C@H]1C[C@](CC(N)=O)(C3)C2 50192787CC(C)(Oc1ccc(Cl)cc1)C(=O)N[C@H]1C2C[C@@H]3C[C@H]1C[C@](C3)(C2)c1nnc(N)[nH]1 50192788CC(C)(Oc1ccc(Cl)cc1)C(=O)N[C@H]1C2C[C@@H]3C[C@H]1C[C@](C3)(C2)c1nc(=O)o[nH]1 50192789CC(C)(Oc1ccc(Cl)cc1)C(=O)N[C@H]1C2C[C@@H]3C[C@H]1C[C@](Cc1nnn[nH]1)(C3)C2 50192790CC(C)(Oc1ccc(Cl)cc1)C(=O)N[C@H]1C2C[C@@H]3C[C@H]1C[C@](C3)(C2)C(=N)NO 50192791CC(C)(Oc1ccc(Br)cn1)C(=O)N[C@H]1C2C[C@@H]3C[C@H]1C[C@](CC(N)=O)(C3)C2 50192792CC(C)(Oc1ccc(cn1)-n1cccn1)C(=O)N[C@H]1C2C[C@@H]3C[C@H]1C[C@](CC(N)=O)(C3)C2 50192793CC(C)(Oc1ccc(Cl)cc1)C(=O)N[C@H]1C2C[C@@H]3C[C@H]1C[C@](CCC(O)=O)(C3)C2 50192794CN1CCN(CC1)c1ccc(OC(C)(C)C(=O)N[C@H]2C3C[C@@H]4C[C@H]2C[C@](CC(N)=O)(C4)C3)nc1 50192795CNc1ccc(cn1)C(C)(C)C(=O)N[C@H]1C2C[C@@H]3C[C@H]1C[C@](CC(N)=O)(C3)C2 50192796CC(C)(Oc1ccc(Cl)cc1)C(=O)N[C@H]1C2C[C@@H]3C[C@H]1C[C@](C3)(C2)c1nc(C#N)c(N)o1 50192797CC(C)(Oc1ccc(Cl)cc1)C(=O)N[C@H]1C2C[C@@H]3C[C@H]1C[C@](C3)(C2)c1ncc[nH]1 50192798CC(C)(C(=O)N[C@H]1C2C[C@@H]3C[C@H]1C[C@](CC(N)=O)(C3)C2)c1ccc(cn1)C#N 50192799CC(C)(C(=O)N[C@H]1C2C[C@@H]3C[C@H]1C[C@](CC(N)=O)(C3)C2)c1ccc(nc1)N1CCOCC1 50192800CC(C)(Oc1ccc(Cl)cc1)C(=O)N[C@H]1C2C[C@@H]3C[C@H]1C[C@](C3)(C2)c1ccno1 50192801CC(C)(Oc1ccc(Cl)cc1)C(=O)N[C@H]1C2C[C@@H]3C[C@H]1C[C@](CC(O)=O)(C3)C2 50193783CCOC(=O)[C@@H]1[C@H]2CCC(CC[C@@H]12)N1CC(COc2ccc(cn2)C#N)C(C)(C)C1=O 50193784CC1(C)C(COc2ccc(cc2)-n2ccnc2)CN([C@H]2C3CC4CC2C[C@](C4)(C3)C(N)=O)C1=O 50193785CC1(C)C(COc2ccc(cn2)C#N)CN([C@H]2C3CCCC2C[C@H](C3)C(N)=O)C1=O 50193786CC1(C)C(COc2ccc(cn2)C#N)CN([C@H]2C3CC4CC2C[C@](C4)(C3)C(N)=O)C1=O 50193787CC1(C)C(COc2ccc(cn2)C(F)(F)F)CN([C@H]2C3CC4CC2C[C@](C4)(C3)C(=N)NO)C1=O 50193788CC1(C)C(COc2ccc(cn2)C#N)CN([C@@H]2C3CCCC2C[C@H](C3)C(N)=O)C1=O 50193789CC1(C)C(COc2ccc(cc2)-n2cncn2)CN([C@H]2C3CC4CC2C[C@](C4)(C3)C(N)=O)C1=O 50193790CC1(C)C(COc2ccc(cn2)C#N)CN(C2CCCCCC2)C1=O 50193791CC1(C)C(COc2ccc(cn2)C(F)(F)F)CN([C@H]2C3CC4CC2C[C@](C4)(C3)C(N)=N)C1=O 50193792O=C1C(Cc2ccccc2)CCN1C1CCCCC1 50193793C[C@@H]1[C@@H](COc2ccc(cn2)C#N)CN(C2CCCCCC2)C1=O 50193794O[C@@]12CC3CC(C1)[C@@H](C(C3)C2)N1CCC(Cc2ccccc2)C1=O 50193795CC1(C)C(COc2ccc(cn2)C#N)CN(C1=O)C12CCC(CC1)(CC2)C(N)=O 50193796CC1(C)C(COc2ccc(cn2)C(F)(F)F)CN([C@H]2C3CC4CC2C[C@](C4)(C3)c2nnn[nH]2)C1=O 50193797NC(=O)[C@@]12CC3CC(C1)[C@@H](C(C3)C2)N1CCC(Cc2ccccc2)C1=O 50193798O=C1CC(COc2ccc(cn2)C#N)CN1C1CCCCCC1 50193799O=C1C(Cc2ccccc2)CCN1[C@H]1C2CC3CC(C2)CC1C3 50193800CC1(C)C(COc2ccc(cn2)C#N)CN(C2CCCN(CC2)C(N)=O)C1=O 50195286NC(=O)[C@@]12CC3CC(C1)[C@H](NC(=O)C1(CCCC1)N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(C3)C2 50195287NC(=O)[C@@]12C[C@H]3CC(C1)[C@@H](NC(=O)C1(CC1)N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(C3)C2 50195288OC(=O)[C@@]12CC3CC(C1)[C@H](NC(=O)C(C1CC1)N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(C3)C2 50195289O[C@@]12C[C@H]3CC(C1)[C@H](NC(=O)C1(CC1)N1CCCCC1)C(C3)C2 50195290CC(C)(N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(=O)N[C@H]1C2C[C@H]3CC1C[C@](C3)(C2)C(O)=O 50195291CC(C)(N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(=O)N[C@H]1C2C[C@H]3CC1C[C@](C3)(C2)C(N)=O 50195292NC(=O)[C@@]12C[C@H]3CC(C1)[C@H](NC(=O)C1(CC1)N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(C3)C2 50195293CCC(N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)C(O)=O 50195294OC(=O)[C@@]12C[C@H]3CC(C1)[C@H](NC(=O)C1(CC1)N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(C3)C2 50195295OC(=O)[C@@]12CC3CC(C1)[C@H](NC(=O)C1(CCCC1)N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(C3)C2 50195296OC(=O)[C@@]12C[C@H]3CC(C1)[C@@H](NC(=O)C1(CC1)N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(C3)C2 50195297O[C@@]12C[C@H]3CC(C1)[C@@H](NC(=O)C1(CC1)N1CCCCC1)C(C3)C2 50195298CCC(N1CCCC(F)(F)C1)C(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)C(N)=O 50195299NC(=O)[C@@]12CC3CC(C1)[C@H](NC(=O)C1(CCC1)N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(C3)C2 50195300OC(=O)[C@@]12CC3CC(C1)[C@H](NC(=O)C1(CCC1)N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(C3)C2 50195301NC(=O)[C@@]12CC3CC(C1)[C@H](NC(=O)C(C1CC1)N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(C3)C2 50195302CCC(N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)C(N)=O 50195303CCC(N1CCCC(F)(F)C1)C(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)C(O)=O 50195304CC(C)(N1CCCCC1)C(=O)N[C@H]1C2C[C@H]3CC1C[C@](O)(C3)C2 50195481CCOC(=O)[C@@H]1CC[C@@H](CC1)N(C1CC1)C(=O)c1cc(Cl)c(N)c(Cl)c1 50195482C[C@H]1CN(C[C@@H](C)N1C(=O)c1cc(Cl)c(N)c(Cl)c1)c1ccccn1 50195483CN(C(=O)c1cc(Cl)c(N)c(Cl)c1)C12CC3CC(CC(C3)C1)C2 50195484C[C@@H]1CC(C[C@@H](C)N1C(=O)c1cc(Cl)c(N)c(Cl)c1)N1CCNC1=O 50195485Nc1c(Cl)cc(cc1Cl)C(=O)N(C1CC1)C1CCCCC1 50195486CCOC(=O)CN1C[C@H](C)N([C@H](C)C1)C(=O)c1cc(Cl)c(N)c(Cl)c1 50195487Nc1c(Cl)cc(cc1Cl)C(=O)N(C1CC1)C1CCCC1 50195488CN(C)CCNC(=O)[C@@H]1CC[C@@H](CC1)N(C1CC1)C(=O)c1cc(Cl)c(N)c(Cl)c1 50195489Nc1c(Cl)cc(cc1Cl)C(=O)N(C1CC1)[C@H]1CC[C@H](CC1)C(=O)N1CCCC1 50195490Nc1c(Cl)cc(cc1Cl)C(=O)N(C1CC1)[C@H]1CC[C@H](CC1)C(=O)NCC(O)=O 50195491Nc1c(Cl)cc(cc1Cl)C(=O)N1CC2CC1CN(Cc1ccccc1)C2 50195492C[C@@H]1C[C@@H](CCN1C(=O)c1cc(Cl)c(N)c(Cl)c1)n1c2ccccc2oc1=O 50195493CN1CCN(CC1)C(=O)[C@@H]1CC[C@@H](CC1)N(C1CC1)C(=O)c1cc(Cl)c(N)c(Cl)c1 50195494Nc1c(Cl)cc(cc1Cl)C(=O)N1CCCN(Cc2ccccc2)CCC1 50195495C[C@@H]1CC(C[C@@H](C)N1C(=O)c1cc(Cl)c(N)c(Cl)c1)n1c2ccccc2oc1=O 50195496C[C@H]1CCC[C@@H](C)N1C(=O)c1cc(Cl)c(N)c(Cl)c1 50195497C[C@H]1CN(C[C@@H](C)N1C(=O)c1cc(Cl)c(N)c(Cl)c1)c1ncccc1N 50195498COC(=O)CN(C)C(=O)[C@@H]1CC[C@@H](CC1)N(C1CC1)C(=O)c1cc(Cl)c(N)c(Cl)c1 50195499COc1ccccc1N1C[C@H](C)N([C@H](C)C1)C(=O)c1cc(Cl)c(N)c(Cl)c1 50195501Nc1c(Cl)cc(cc1Cl)C(=O)N1CCCCC1 50195502Nc1c(Cl)cc(cc1Cl)C(=O)N(C1CC1)[C@H]1CC[C@H](CC1)C(=O)NCC1CCCCC1 50195503Nc1c(Cl)cc(cc1Cl)C(=O)N(C1CC1)[C@H]1CC[C@H](CC1)C(=O)NCc1ccccc1 50195504CC12CC(CC(C)(C)C1)N(C2)C(=O)c1cc(Cl)c(N)c(Cl)c1 50195505CCOC(=O)c1cccnc1N1C[C@H](C)N([C@H](C)C1)C(=O)c1cc(Cl)c(N)c(Cl)c1 50195506Nc1c(Cl)cc(cc1Cl)C(=O)N1C2CC3CC(C2)CC1C3 50195507C[C@H]1CN(C[C@@H](C)N1C(=O)c1cc(Cl)c(N)c(Cl)c1)c1ccc(cn1)C(F)(F)F 50197399CC(C)(Oc1ccccc1Cl)C(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)S(N)(=O)=O 50197400COc1cc(F)ccc1OC(C)(C)C(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)S(C)(=O)=O 50197401CC(C)(Oc1ccccc1)C(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)S(N)(=O)=O 50197402CC(C)(Oc1ccc(Cl)cc1)C(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)S(N)(=O)=O 50197403CC(C)(Oc1ccccc1C(F)(F)F)C(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)S(C)(=O)=O 50197404CC(C)(Oc1c(Cl)cc(F)cc1Cl)C(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)S(N)(=O)=O 50197405CC(C)(Oc1ccc(Cl)cc1)C(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)S(C)(=O)=O 50197406CN(C)S(=O)(=O)[C@@]12CC3CC(C1)[C@H](NC(=O)C(C)(C)Oc1ccc(Cl)cc1)C(C3)C2 50197407CC(C)(Oc1ccc(F)cc1Cl)C(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)S(=O)(=O)CCCN1CCOCC1 50197408CC(C)(Oc1cccc(Cl)c1)C(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)S(N)(=O)=O 50197409CCS(=O)(=O)[C@@]12CC3CC(C1)[C@H](NC(=O)C(C)(C)Oc1ccc(F)cc1Cl)C(C3)C2 50197410CC(C)(Oc1ccccc1OC(F)(F)F)C(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)S(N)(=O)=O 50197411CC(C)(C(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)S(N)(=O)=O)c1ccccc1 50197412CC(C)(Oc1ccc(F)cc1Cl)C(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)S(=O)(=O)CC(N)=O 50197413CC(C)(Oc1cccc(Cl)c1)C(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)S(C)(=O)=O 50197414CC(C)(Oc1ccc(F)cc1Cl)C(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)S(C)(=O)=O 50197415CC(=O)NS(=O)(=O)[C@@]12CC3CC(C1)[C@H](NC(=O)C(C)(C)Oc1ccc(Cl)cc1)C(C3)C2 50197416CC(C)(Oc1ccc(F)cc1Cl)C(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)S(N)(=O)=O 50197417CC(C)(Oc1ccc(Cl)cc1F)C(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)S(C)(=O)=O 50197418CC(C)(Oc1ccccc1Cl)C(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)S(C)(=O)=O 50197419CNS(=O)(=O)[C@@]12CC3CC(C1)[C@H](NC(=O)C(C)(C)Oc1ccc(Cl)cc1)C(C3)C2 50202085C[C@H](N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50202086O[C@@]12CC3CC(C1)[C@H](NC(=O)CN1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(C3)C2 50202087CC(N1CCc2ccc3OCOc3c2CC1)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50202088FC(F)(F)c1ccc(nc1)N1CCN(CC(=O)NC2C3CC4CC(C3)CC2C4)CC1 50202089O[C@]12CC3CC(C1)[C@H](NC(=O)CN1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(C3)C2 50202090NA 50202091O=C(CN1CCN(CC1)c1ncccc1C#N)NC1C2CC3CC(C2)CC1C3 50202092FC(F)(F)c1ccc(nc1)N1CCN(CC(=O)N[C@H]2C3CC4CC2C[C@](F)(C4)C3)CC1 50202093CC(N1CC(C1)Oc1ccccc1F)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50202094O[C@@]12CC3CC(C1)[C@H](NC(=O)CN1CC[C@@H](C1)C(F)(F)F)C(C3)C2 50202095NA 50202096CC(N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(=O)N[C@H]1C2C[C@]3(O)CC1C[C@](F)(C2)C3 50202097CC(C)(N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50202098OC12CC3CC(CC(C3)C1NC(=O)CN1CCN(CC1)c1ccc(cn1)C(F)(F)F)C2 50202099FC(F)(F)c1ccc(nc1)N1CCN(CC(=O)N[C@H]2C3CC4CC2C[C@@](F)(C4)C3)CC1 50202100CC(N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(=O)N[C@H]1C2C[C@@]3(O)CC1C[C@@](F)(C2)C3 50202101CC(N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(=O)N[C@H]1C2C[C@]3(O)CC1C[C@](O)(C2)C3 50202102CC(N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50202103CC(C)(N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(=O)N[C@H]1C2C[C@]3(O)CC1C[C@](O)(C2)C3 50202104CO[C@@]12CC3CC(C1)[C@H](NC(=O)C(C)N1CCN(CC1)c1ccc(cn1)C(F)(F)F)C(C3)C2 50202105Clc1ccc(cc1)N1CCN(CC(=O)NC2C3CC4CC(C3)CC2C4)CC1 50202106NA 50207756Cc1ccc(cc1)C12CC3CC(CC(C3)(C1)C(=O)N1CCN(CC1)S(=O)(=O)Cc1ccccc1)C2 50207760Cc1ccc(cc1)C12CC3CC(CC(C3)(C1)C(=O)N1CCN(CCO)CC1)C2 50207765CCN1CCN(CC1)C(=O)CC12CC3CC(CC(C3)C1)C2 50207767OCCN1CCN(CC1)C(=O)C12CC3CC(CC(C3)C1)C2 50207768CN1CCN(CC1)C(=O)C12CC3CC(C1)CC(C3)(C2)c1ccc(C)cc1 50207769Cc1ccc(cc1)C12CC3CC(CC(C3)(C1)C(=O)N1CCN(CCc3ccccc3)CC1)C2 50207770CCN1CCN(CC1)C(=O)C12CC3CC(C1)CC(C3)(C2)c1ccc(OC)cc1 50207772O=C(N1CCCCC1)C12CC3CC(CC(C3)C1)C2 50207773COCCN1CCN(CC1)C(=O)C12CC3CC(C1)CC(C3)(C2)c1ccc(C)cc1 50207774O=C(N1CCN(Cc2ccncc2)CC1)C12CC3CC(CC(C3)C1)C2 50207776CCN1CCN(CC1)C(=O)C12CC3CC(CC(C3)C1)C2 50207777Cc1ccc(cc1)C12CC3CC(CC(C3)(C1)C(=O)N1CCN(CC1)c1ccccc1)C2 50207779Cc1ccc(cc1)C12CC3CC(CC(C3)(C1)C(=O)N1CCN(Cc3ccncc3)CC1)C2 50207781Cc1ccc(cc1)C12CC3CC(CC(C3)(C1)C(=O)N1CCN(CC1)C(C#N)c1ccccc1)C2 50207783O=C(N1CCNCC1)C12CC3CC(CC(C3)C1)C2 50207784OC12CC3CC(C1)CC(C3)(C2)C(=O)N1CCCCC1 50207786O=C(N1CCc2ccccc2C1)C12CC3CC(CC(C3)C1)C2 50207787O=C(N1CCC2CCCCC2C1)C12CC3CC(CC(C3)C1)C2 50207788O=C(N1CCCC1)C12CC3CC(CC(C3)C1)C2 50207789Cc1ccc(cc1)C12CC3CC(CC(C3)(C1)C(=O)N1CCN(Cc3ccccc3)CC1)C2 50207790CCN1CCN(CC1)C(=O)C12CC3CC(CC(Cc4ccccc4)(C3)C1)C2 50207795O=C(N1CCCc2ccccc12)C12CC3CC(CC(C3)C1)C2 50207797CCN1CCN(CC1)C(=O)Cc1ccccc1 50207799O=C(C1C2CC3CC(C2)CC1C3)N1CCCCC1 50207800CN1CCN(CC1)C(=O)C12CC3CC(CC(C3)C1)C2 50207803O=C(N1CCN(Cc2ccccc2)CC1)C12CC3CC(CC(C3)C1)C2 50210881FC(F)(F)c1cccc(c1)C(=O)N1CCC(CC1)n1c2ccccc2[nH]c1=O 50210882FC(F)(F)c1ccccc1C(=O)N1CCC(CC1)n1c2ccccc2[nH]c1=O 50210884COc1cc(ccc1C)C(=O)N1CCC(CC1)n1c2ccccc2[nH]c1=O 50210885Cc1ccc(cc1F)C(=O)N1CCC(CC1)n1c2ccccc2[nH]c1=O 50210886Cc1ccc(cc1C)C(=O)N1CCC(CC1)n1c2ccccc2[nH]c1=O 50210887Cc1cccc(C(=O)N2CCC(CC2)n2c3ccccc3[nH]c2=O)c1C 50210888COc1cccc(c1)C(=O)N1CCC(CC1)n1c2ccccc2[nH]c1=O 50210889CC(C)(C)c1ccc(cc1)C(=O)N1CCC(CC1)n1c2ccccc2[nH]c1=O 50210890COc1cc(ccc1C)C(=O)N1CCC(CC1)n1c2ccccc2sc1=O 50210891FC(F)(F)c1ccc(cc1)C(=O)N1CCC(CC1)n1c2ccccc2[nH]c1=O 50210892COc1cc(ccc1C)C(=O)N1CCC(CC1)n1c2cccc(C)c2[nH]c1=O 50210894COc1cc(ccc1C)C(=O)N1CCC(CC1)n1c2ccc(Cl)cc2[nH]c1=O 50210895COc1cc(ccc1C)C(=O)N1CCC(CC1)n1c2ccc(F)cc2[nH]c1=O 50210896COc1cc(Cl)nc(c1)C(=O)N1CCC(CC1)n1c2ccccc2[nH]c1=O 50210897O=C(N1CCC(CC1)n1c2ccccc2[nH]c1=O)c1ccc2OCOc2c1 50210898COc1cc(ccc1C)C(=O)N1CCC(CC1)n1c2ccccc2oc1=O 50210899COc1cc(ccc1N)C(=O)N1CCC(CC1)n1c2ccccc2[nH]c1=O 50210900Fc1ccccc1C(=O)N1CCC(CC1)n1c2ccccc2[nH]c1=O 50210901COc1cc(ccc1C)C(=O)N1CCC(CC1)n1c2ccccc2n(C)c1=O 50210902COc1cc(ccc1C)C(=O)N1CCC(CC1)N1C(=O)Cc2ccccc12 50210903O=C(N1CCC(CC1)n1c2ccccc2[nH]c1=O)c1ccc2ccoc2c1 50210904COc1cc(ccc1C)C(=O)N1CCC(CC1)n1c2ccc(Cl)cc2n(C)c1=O 50210905COc1cc(ccc1C)C(=O)N1CCC(CC1)n1c2ccc(C)c(C)c2[nH]c1=O 50212522CCOC(=O)CC(C)(C)C(=O)CS(=O)(=O)c1ccccc1 50212524O=C(N(Cc1ccccc1)S(=O)(=O)c1ccccc1)c1ccccc1 50212525Fc1ccc(cc1)C(=O)CS(=O)(=O)c1ccccc1 50212526COc1ccc(OC)c(c1)C(=O)CS(=O)(=O)c1ccccc1 50212529O=C(CS(=O)(=O)c1ccccc1)c1ccc(s1)-c1ccccc1 50212530Cc1ccc(cc1)C(=O)CS(=O)(=O)c1ccccc1 50212531Clc1ccc(cc1)C(=O)CS(=O)(=O)c1ccccc1 50212532Clc1ccc(cc1Cl)C(=O)CS(=O)(=O)c1ccccc1 50212533O=C(CS(=O)(=O)c1ccccc1)c1ccsc1 50212534COc1cccc(c1)C(=O)CS(=O)(=O)c1ccccc1 50212535COc1ccc(cc1)C(=O)CS(=O)(=O)c1ccccc1 50212538O=C(CS(=O)(=O)c1ccccc1)C(c1ccccc1)c1ccccc1 50212543Clc1ccc(-c2ccc(o2)C(=O)CS(=O)(=O)c2ccccc2)c(Cl)c1 50212544CCN(CC)c1ccc(cc1)C(=O)CS(=O)(=O)c1ccccc1 50212547Cc1ccc(C(=O)CS(=O)(=O)c2ccccc2)c(C)c1 50212548Cc1c(sc2ccccc12)C(=O)CS(=O)(=O)c1ccccc1 50212551[O-][N+](=O)c1ccc(cc1)C(=O)CS(=O)(=O)c1ccccc1 50216900C[C@@H](NC1=NC(=O)C2(CCN(Cc3ccccc3)CC2)O1)c1ccccc1 50216901O=C1N=C(NC2CCCCCCC2)OC11CCCC1 50216902CCC1(CC)OC(NC23CC4CC(CC(C4)C2)C3)=NC1=O 50216903CC(C)C1(C)OC(NC2CCCCCC2)=NC1=O 50216904CC(C)C1(C)OC(NC23CC4CC(CC(C4)C2)C3)=NC1=O 50216907CCC1(CC)OC(NC23CC4CC(CC(O)(C4)C2)C3)=NC1=O 50216908CCC1(CC)OC(N[C@@H](C)c2ccc(Br)cc2)=NC1=O 50216909CC(C)C1(C)OC(NC23CC4CC(CC(O)(C4)C2)C3)=NC1=O 50216910CC(C)C1(C)OC(NC2C3CC4CC(C3)CC2C4)=NC1=O 50216911O=C1N=C(NC2C3CC4CC(C3)CC2C4)OC11CCCC1 50216912CC1(OC(NC2CCCCCCC2)=NC1=O)C(F)(F)F 50216913CC(C)C1(C)OC(N[C@H](C)c2ccccc2)=NC1=O 50216914CC(C)C1(C)OC(NC2CCCCCCC2)=NC1=O 50216915CC1(OC(NC2C3CC4CC(C3)CC2C4)=NC1=O)C(F)(F)F 50216916CCC1(CC)OC(N[C@@H](C)c2ccccc2C(F)(F)F)=NC1=O 50216917CCC1(CC)OC(NC2CCCCCCC2)=NC1=O 50216918C[C@H](NC1=NC(=O)C2(CCN(Cc3ccccc3)CC2)O1)c1ccccc1C(F)(F)F 50216919CCC1(CC)OC(NCc2ccccc2)=NC1=O 50216920CC(C)C1(C)OC(N[C@@H](C)c2ccccc2)=NC1=O 50216921O=C1N=C(NC23CC4CC(CC(C4)C2)C3)OC11CCCC1 50216922CC(C)C1(C)OC(N[C@@H](C)c2ccccc2C(F)(F)F)=NC1=O 50216924O=C1N=C(NC2CCCCCC2)OC11CCOCC1 50216925CCC1(CC)OC(NC2Cc3ccccc3C2)=NC1=O 50216926C[C@H](NC1=NC(=O)C2(CCN(Cc3ccccc3)CC2)O1)c1ccccc1 50216927CCC1(CC)OC(N[C@@H](C)c2ccccc2)=NC1=O 50216928O=C1N=C(NC23CC4CC(CC(C4)C2)C3)OC11CCOCC1 50216929CCC1(CC)OC(NCCc2ccccc2)=NC1=O 50216931CCC1(CC)OC(NC2C3CC4CC(C3)CC2C4)=NC1=O 50222205C[C@@H]1CC[C@@]2(CC[C@]3(C)C(=CC[C@@H]4[C@@]5(C)C[C@@H](O)[C@H](O)C(C)(C)[C@@H]5CC[C@@]34C)[C@@H]2[C@H]1C)C(O)=O 50224200CC(C)c1sc(Nc2ccc(F)cc2F)nc1O 50224201CC(C)c1sc(Nc2ccc(F)cc2)nc1O 50224202Oc1nc(Nc2ccccc2F)sc1C1CCCCC1 50224203Oc1nc(Nc2ccccc2Cl)sc1C1CCCCC1 50224204CC(C)c1sc(Nc2ccccn2)nc1O 50224205CC(C)c1sc(Nc2c(Cl)cccc2Cl)nc1O 50224206CC(C)c1sc(Nc2ccccc2)nc1O 50224207CC(C)c1sc(Nc2ccccc2F)nc1O 50224208CC(C)c1sc(Nc2ccccc2Cl)nc1O 50224209COc1ccccc1Nc1nc(O)c(s1)C(C)C 50224210CC(C)c1sc(Nc2ccc(cc2)C2CCCCC2)nc1O 50224211CC(C)c1sc(Nc2cccc3cnccc23)nc1O 50224212CC(C)c1sc(Nc2ccccc2C(F)(F)F)nc1O 50224213CC(C)c1sc(Nc2ccccc2C)nc1O 50224214CC(C)c1sc(Nc2ccc3n[nH]cc3c2)nc1O 50224215CC(C)c1sc(Nc2cccc3[nH]ccc23)nc1O 50224216Oc1nc(Nc2ccccc2Cl)sc1C1CCCC1 50224217CC(C)c1sc(Nc2cc(F)ccc2F)nc1O 50224220Cc1sc(Nc2ccccc2Cl)nc1O 50224221Oc1nc(Nc2ccccc2F)sc1C1CCCC1 50224222CC(C)c1sc(Nc2ccc(Cl)cc2Cl)nc1O 50224223CC(C)c1sc(Nc2ccc(Oc3ccccc3)cc2)nc1O 50224224CC(C)c1sc(Nc2ccncc2)nc1O 50224225CC(C)c1sc(Nc2ccc3sc(C)nc3c2)nc1O 50233538CC1(C)[C@@H](O)CC[C@@]2(C)[C@H]1CC[C@]1(C)[C@@H]2C(=O)C=C2[C@@H]3C[C@](C)(CC[C@]3(C)CC[C@@]12C)C(O)=O 50239276Cn1c(nnc1C12CC3CC(CC(C3)C1)C2)-c1ccccc1 50239401C1C2CC3CC1CC(C2)(C3)c1nnc2CCCCCn12 50239407Clc1ccc(cc1)C1(CCC1)c1nnc2CCCCCCn12 50241490O=C(Nc1cccc(c1)C(=O)N1CCC[C@H]2CCCC[C@H]12)c1ccccc1 50243595CCN(C1CCCCC1)C(=O)c1ccc(cc1)[C@](C)(O)C(F)(F)F 50243596C[C@](O)(c1ccc(cc1)C(=O)N(CC(F)(F)F)C1CCCCC1)C(F)(F)F 50243631CC(O)(c1ccc(cc1)C(=O)N(CC1CC1)C1CCCCC1)C(F)(F)F 50243632C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)C1CCCCC1)C(F)(F)F 50243633C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@@H](CC1)c1ccccc1)C(F)(F)F 50243634C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@H](CC1)c1ccccc1)C(F)(F)F 50243635C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@@H](CC1)c1ccc(cc1)C#N)C(F)(F)F 50243671C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@H](F)CC1)C(F)(F)F 50243672C[C@H]1CCCCN1S(=O)(=O)c1ccc(cc1)C(C)(O)C(F)(F)F 50244290CCOc1cc(CNc2c(C)[nH][nH]c2=S)cc(Br)c1OCC(=O)NC1CCCCC1 50244328Cc1ccc(cc1)S(=O)(=O)NN=C1C=C[C@H]2[C@@H]3CC=C4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]12C 50247012CC1(C)[C@H](CC[C@@]2(C)[C@H]1CC[C@]1(C)[C@@H]2C(=O)C=C2[C@@H]3C[C@](C)(CC[C@]3(C)CC[C@@]12C)C(O)=O)OC(=O)CCC(O)=O 50247925C[C@@H]1CN(CC2(CC2)C(N)=O)CCN1S(=O)(=O)c1ccc(cc1)[C@@](C)(O)C(F)(F)F 50248020C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@H](CC1)c1cccnc1)C(F)(F)F 50248066C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@H](CC1)c1ccc(cc1)C#N)C(F)(F)F 50248067C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@](CC1)(C#N)c1ccccc1)C(F)(F)F 50248101C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@](CC1)(C#N)c1ccc(cc1)C#N)C(F)(F)F 50248102C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@](CC1)(C#N)c1cccnc1)C(F)(F)F 50248133C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@](CC1)(C#N)C1CC1)C(F)(F)F 50248134C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@@](O)(CC1)c1ccccc1)C(F)(F)F 50248163C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@](O)(CC1)c1ccccc1)C(F)(F)F 50248164C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@@](O)(CC1)c1cccnc1)C(F)(F)F 50248165C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@@](O)(CC1)c1ccccn1)C(F)(F)F 50248166C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@@](C)(O)CC1)C(F)(F)F 50248209CC(C)[C@@]1(O)CC[C@@H](CC1)N(C1CC1)C(=O)c1ccc(cc1)[C@](C)(O)C(F)(F)F 50248210C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@](O)(CC2CC2)CC1)C(F)(F)F 50248211C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@@](O)(CC1)C1CC1)C(F)(F)F 50248252C[C@@H]1CN(CCc2ccncc2)CCN1S(=O)(=O)c1ccc(cc1)C(C)(O)C(F)(F)F 50248253C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(cc1)C(C)(C)C)C(c1ccccc1)c1ccncc1 50248254C[C@@H]1CN(Cc2ccnc3ccccc23)CCN1S(=O)(=O)c1ccc(cc1)C(C)(C)C 50248255C[C@@H]1CN(CCc2ccncc2)CCN1S(=O)(=O)c1ccc(cc1)C(C)(C)O 50248307C[C@@H]1CN(CCc2ccncc2)CCN1S(=O)(=O)c1ccc(cc1)C(C)(C)F 50248308CC(N1CCN([C@H](C)C1)S(=O)(=O)c1ccc(cc1)C(C)(C)C)c1ccncc1 50248309C[C@@H]1CN(CCc2ccncc2)CCN1S(=O)(=O)c1ccc(cc1)C(C)(C)C 50248310C[C@@H]1CN(CCCc2ccncc2)CCN1S(=O)(=O)c1ccc(cc1)C(C)(C)C 50248311C[C@@H]1CN(Cc2ccncc2)CCN1S(=O)(=O)c1ccc(cc1)C(C)(C)C 50248370C[C@@H]1CN(CCc2ccncc2)CCN1S(=O)(=O)c1ccc(cc1)C(C)(F)C(F)(F)F 50248371CC(O)c1ccc(cc1)S(=O)(=O)N1CCN(CCc2ccncc2)C[C@H]1C 50248372CC(F)c1ccc(cc1)S(=O)(=O)N1CCN(CCc2ccncc2)C[C@H]1C 50248373C[C@@H]1CN(CCc2ccncc2)CCN1S(=O)(=O)c1ccc(cc1)C(C)(F)F 50248425C[C@@H]1CN(CCc2ccncc2)CCN1S(=O)(=O)c1ccc(cc1)C1(CO)CC1 50248426C[C@@H]1CN(CCc2ccncc2)CCN1S(=O)(=O)c1ccc(cc1)C1(CN2CCOCC2)CC1 50248427C[C@@H]1CN(CCc2cccnc2)CCN1S(=O)(=O)c1ccc(cc1)C(C)(O)C(F)(F)F 50248428C[C@@H]1CN(CCc2ccccn2)CCN1S(=O)(=O)c1ccc(cc1)C(C)(O)C(F)(F)F 50248469C[C@@H]1CN(CC(F)(F)c2ccncc2)CCN1S(=O)(=O)c1ccc(cc1)C(C)(O)C(F)(F)F 50248470C[C@@H]1CN(CC(F)(F)c2cccnc2)CCN1S(=O)(=O)c1ccc(cc1)C(C)(O)C(F)(F)F 50248471C[C@@H]1CN(CC2(CC2)c2ccncc2)CCN1S(=O)(=O)c1ccc(cc1)C(C)(O)C(F)(F)F 50248472C[C@@H]1CN(CC2(CC2)c2cccnc2)CCN1S(=O)(=O)c1ccc(cc1)C(C)(O)C(F)(F)F 50248518C[C@@H]1CN(CC2(CCC2)c2ccncc2)CCN1S(=O)(=O)c1ccc(cc1)C(C)(O)C(F)(F)F 50248519C[C@@H]1CN(CC2(CCC2)c2cccnc2)CCN1S(=O)(=O)c1ccc(cc1)C(C)(O)C(F)(F)F 50248520C[C@@H]1CN(CC2(CCCC2)c2ccncc2)CCN1S(=O)(=O)c1ccc(cc1)C(C)(O)C(F)(F)F 50248521C[C@@H]1CN(CC2(CCCC2)c2cccnc2)CCN1S(=O)(=O)c1ccc(cc1)C(C)(O)C(F)(F)F 50248566C[C@@H]1CN(CC2(CC2)C(N)=O)CCN1S(=O)(=O)c1ccc(cc1)C(C)(O)C(F)(F)F 50248567C[C@@H]1CN(CC2(CCC2)C(N)=O)CCN1S(=O)(=O)c1ccc(cc1)C(C)(O)C(F)(F)F 50248568C[C@@H]1CN(CC2(CC2)c2ccc(cc2)C(N)=O)CCN1S(=O)(=O)c1ccc(cc1)C(C)(O)C(F)(F)F 50248569C[C@@H]1CN(CC2(CC2)C(N)=O)CCN1S(=O)(=O)c1ccc(cc1)[C@](C)(O)C(F)(F)F 50249080Cc1ccc(c(C)c1)S(=O)(=O)Nc1cc(Cl)c(O)c2ccccc12 50249081Cc1cccc(OCC(=O)NN=Cc2c(C)cc(O)cc2O)c1 50249082Cc1ccc(CSc2nnc(s2)N2C(C(C(=O)c3cc4ccccc4o3)C(=O)C2=O)c2ccccc2F)cc1 50249501Cc1cc(O)cc(O)c1C=NNC(=O)C1COc2ccccc2O1 50249525CC1(C)CC(O)CC(C)(CNS(=O)(=O)c2ccc3oc4ccccc4c3c2)C1 50249526CC(O)c1cccc(NC(=O)C(C)Oc2ccc(Br)cc2Br)c1 50249527CCCc1oc2ccc(NS(=O)(=O)c3cc(C)ccc3C)cc2c1C(=O)OCC 50249528CC(Sc1nnc(CNc2ccccc2)n1CC=C)C(=O)NN=Cc1cc(Br)ccc1O 50252104CCNC(=O)N1CCN(CC1)c1cccc(c1)S(=O)(=O)N1CCN(C[C@H]1C)c1ccc(F)cc1C(F)(F)F 50252153FC(F)(F)c1cccnc1N1CCN(CC1)S(=O)(=O)c1ccc(Cl)c(Cl)c1 50252154FC(F)(F)c1ccccc1N1CCN(CC1)S(=O)(=O)c1ccc(Cl)c(Cl)c1 50252155Fc1ccc(N2CCN(CC2)S(=O)(=O)c2ccc(Cl)c(Cl)c2)c(c1)C(F)(F)F 50252156C[C@H]1CN([C@H](C)CN1c1ncccc1Cl)S(=O)(=O)c1ccc(Cl)c(Cl)c1 50252157C[C@H]1CN(C[C@@H](C)N1S(=O)(=O)c1ccc(Cl)c(Cl)c1)c1ncccc1Cl 50252200FC(F)(F)c1cccnc1N1CCN(C(=O)C1)S(=O)(=O)c1ccc(Cl)c(Cl)c1 50252201FC(F)(F)c1cccnc1N1CCN(CC1=O)S(=O)(=O)c1ccc(Cl)c(Cl)c1 50252202C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(Cl)c(Cl)c1)c1ccccc1C(F)(F)F 50252203C[C@@H]1CN(CCN1S(=O)(=O)c1cccc(c1)N1CCCCC1)c1ccc(F)cc1C(F)(F)F 50252243C[C@@H]1CN(CCN1S(=O)(=O)c1cccc(c1)N1CCOCC1)c1ccc(F)cc1C(F)(F)F 50252244C[C@@H]1CN(CCN1S(=O)(=O)c1cccc(c1)N1CCN(C)CC1)c1ccc(F)cc1C(F)(F)F 50252245CCN1CCN(CC1)c1cccc(c1)S(=O)(=O)N1CCN(C[C@H]1C)c1ccc(F)cc1C(F)(F)F 50252246CC(C)N1CCN(CC1)c1cccc(c1)S(=O)(=O)N1CCN(C[C@H]1C)c1ccc(F)cc1C(F)(F)F 50252313COC(=O)N1CCN(CC1)c1cccc(c1)S(=O)(=O)N1CCN(C[C@H]1C)c1ccc(F)cc1C(F)(F)F 50252315C[C@@H]1CN(CCN1S(=O)(=O)c1cccc(c1)N1CC[C@@H](O)C1)c1ccc(F)cc1C(F)(F)F 50252316C[C@@H]1CN(CCN1S(=O)(=O)c1cccc(c1)N1CCCC1)c1ccc(F)cc1C(F)(F)F 50252367C[C@@H]1CN(CCN1S(=O)(=O)c1cccc(c1)N1CCC(O)C1)c1ccc(F)cc1C(F)(F)F 50252368C[C@@H]1CN(CCN1S(=O)(=O)c1cccc(c1)N1CC[C@H](O)C1)c1ccc(F)cc1C(F)(F)F 50252369COC(=O)C1CCN(C1)c1cccc(c1)S(=O)(=O)N1CCN(C[C@H]1C)c1ccc(F)cc1C(F)(F)F 50252370C[C@@H]1CN(CCN1S(=O)(=O)c1cccc(c1)N1CCC(C1)C(O)=O)c1ccc(F)cc1C(F)(F)F 50252436C[C@@H]1CN(CCN1S(=O)(=O)c1cccc(c1)N1CCC(C1)C(N)=O)c1ccc(F)cc1C(F)(F)F 50252437C[C@@H]1CN(CCN1S(=O)(=O)c1cccc(c1)N1CCCC1C(O)=O)c1ccc(F)cc1C(F)(F)F 50252438C[C@@H]1CN(CCN1S(=O)(=O)c1cccc(c1)-n1cncn1)c1ccc(F)cc1C(F)(F)F 50252439C[C@@H]1CN(CCN1S(=O)(=O)c1cccc(c1)-n1cnnc1)c1ccc(F)cc1C(F)(F)F 50252476C[C@@H]1CN(CCN1S(=O)(=O)c1cccc(c1)-n1ccnc1)c1ccc(F)cc1C(F)(F)F 50252477C[C@@H]1CN(CCN1S(=O)(=O)c1cccc(c1)-n1cccn1)c1ccc(F)cc1C(F)(F)F 50252478C[C@@H]1CN(CCN1S(=O)(=O)c1cccc(OC(C)(C)C(O)=O)c1)c1ccc(F)cc1C(F)(F)F 50260623Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccccc1 50260624Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(O)cc1 50260625Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccccc1O 50260666Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1cccc(O)c1 50260667Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(OC(F)(F)F)cc1 50260668Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccccc1OC(F)(F)F 50260669Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1cccc(OC(F)(F)F)c1 50260670Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(Cl)cc1 50260704Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccccc1Cl 50260705Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1cccc(Cl)c1 50260706Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(F)cc1 50260707Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccccc1F 50260708Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1cccc(F)c1 50260745Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1)C(F)(F)F 50260746Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccccc1C(F)(F)F 50260747Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(I)cc1 50260748Cc1ccccc1-c1nnc(n1C)C1(CCC1)c1ccc(Cl)cc1 50260749COc1ccccc1-c1nnc(n1C)C1(CCC1)c1ccc(Cl)cc1 50260793Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(Cl)cc1Cl 50260794Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(O)c(F)c1 50260795COc1ccc(cc1F)-c1nnc(n1C)C1(CCC1)c1ccc(Cl)cc1 50260796Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(OC2CC2)cc1 50260797Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1)-c1ccccc1 50260822Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1cccc(c1)-c1ccccc1 50260823Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1)-c1ccc(F)cc1 50260824Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(Cc2ccccc2)cc1 50260825Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1)C(C)(C)C 50260878Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(Oc2ccccc2)cc1 50260879Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1)-n1ccnc1 50260880Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1Cl)-c1ccccc1 50260881Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1)-n1cccc1 50260882Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1)-c1nccs1 50260908Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1Cl)-c1cccnc1 50260909Cc1nc2ccccc2n1-c1ccc(-c2nnc(n2C)C2(CCC2)c2ccc(Cl)cc2)c(Cl)c1 50260910Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1Cl)-c1ccncc1 50260911CCSc1ccccc1-c1ccc(-c2nnc(n2C)C2(CCC2)c2ccc(Cl)cc2)c(Cl)c1 50260936Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1Cl)-c1ccccn1 50260937Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1Cl)-c1ccc(cc1)S(C)(=O)=O 50260938Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1Cl)-n1ccnc1 50260939Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1Cl)-c1cccc(c1)S(C)(=O)=O 50260964Cc1nccn1-c1ccc(-c2nnc(n2C)C2(CCC2)c2ccc(Cl)cc2)c(Cl)c1 50260965Cc1cn(c(C)n1)-c1ccc(-c2nnc(n2C)C2(CCC2)c2ccc(Cl)cc2)c(Cl)c1 50260966Cc1cn(c(n1)C1CC1)-c1ccc(-c2nnc(n2C)C2(CCC2)c2ccc(Cl)cc2)c(Cl)c1 50260967Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1Cl)-n1ccnc1C(F)(F)F 50261007CSc1nccn1-c1ccc(-c2nnc(n2C)C2(CCC2)c2ccc(Cl)cc2)c(Cl)c1 50261008Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1Cl)-n1ccnc1S(C)(=O)=O 50261009CCS(=O)(=O)c1ccc(cc1)-c1ccc(-c2nnc(n2C)C2(CCC2)c2ccc(Cl)cc2)c(Cl)c1 50261010CCS(=O)(=O)c1ccccc1-c1ccc(-c2nnc(n2C)C2(CCC2)c2ccc(Cl)cc2)c(Cl)c1 50261050CCS(=O)(=O)c1cccc(c1)-c1ccc(-c2nnc(n2C)C2(CCC2)c2ccc(Cl)cc2)c(Cl)c1 50263346CC(C)n1c(nnc1C1(CC1)c1ccc(F)cc1)-c1ccc(OC(F)(F)F)cc1 50264832Oc1ccc(\C=C2/CCC\C(=C/c3ccc(O)cc3)C2=O)cc1 50266759Fc1ccc(\C=C\C(=O)\C=C\c2ccc(F)cc2)cc1 50273397C[C@H](NC1=NC(=O)C(C)(S1)c1ccc(cc1)C(O)=O)c1ccc(F)cc1 50273398C[C@H](NC1=NC(=O)C(C)(S1)c1ccc(cc1)C(N)=O)c1ccc(F)cc1 50273399C[C@H](NC1=NC(=O)C(C)(Cc2ccc(cc2)C(N)=O)S1)c1ccc(F)cc1 50273400C[C@H](NC1=NC(=O)C(C)(S1)c1ccc(cc1)C(=O)N1CCOCC1)c1ccc(F)cc1 50273401C[C@H](NC1=NC(=O)C(C)(S1)C(C)(C)O)c1ccc(Br)cc1 50273402C[C@H](NC1=NC(=O)C(C)(S1)C(C)(C)O)c1ccc(C)cc1 50273403C[C@H](NC1=NC(=O)C(C)(S1)C(C)(C)O)c1ccc(Cl)cc1 50273404C[C@H](NC1=NC(=O)C(C)(S1)C(C)(C)O)c1ccccc1 50273405C[C@H](NC1=NC(=O)C(C)(S1)C(C)(C)O)c1cccc(F)c1 50273449C[C@H](NC1=NC(=O)C(C)(S1)c1ccc(cc1)C(=O)NC1CC1)c1ccc(F)cc1 50273450C[C@H](NC1=NC(=O)C(C)(S1)c1ccc(cc1)C(=O)NC1CCCC1)c1ccc(F)cc1 50273451CNC(=O)c1ccc(cc1)C1(C)SC(N[C@@H](C)c2ccc(F)cc2)=NC1=O 50273452C[C@H](NC1=NC(=O)C(C)(S1)c1ccc(cc1)C(=O)N1CCCC1)c1ccc(F)cc1 50273453C[C@H](NC1=NC(=O)C(C)(S1)c1ccc(CC(N)=O)cc1)c1ccc(F)cc1 50273454C[C@H](NC1=NC(=O)C(C)(S1)C(C)(C)O)c1ccccc1F 50273455C[C@H](NC1=NC(=O)C(C)(S1)C(C)(C)O)c1ccccc1Cl 50273456C[C@H](NC1=NC(=O)C(C)(S1)C(C)(C)O)c1ccccc1C(F)(F)F 50273457C[C@H](NC1=NC(=O)[C@](C)(S1)C(C)(C)O)c1ccc(F)cc1 50273458C[C@H](NC1=NC(=O)[C@@](C)(S1)C(C)(C)O)c1ccc(F)cc1 50273821COC(=O)c1ccc(cc1)C1(C)SC(N[C@@H](C)c2ccc(F)cc2)=NC1=O 50273822C[C@H](NC1=NC(=O)C(C)(S1)c1ccc(F)cc1)c1ccc(F)cc1 50273823C[C@H](NC1=NC(=O)C(C)(S1)c1ccc(cc1)C(C)(C)C(N)=O)c1ccc(F)cc1 50273824C[C@H](NC1=NC(=O)C(C)(S1)c1ccc(CCC(N)=O)cc1)c1ccc(F)cc1 50273825C[C@H](NC1=NC(=O)C(C)(S1)c1ccc(cc1)C1(CC1)C(N)=O)c1ccc(F)cc1 50273826C[C@H](NC1=NC(=O)C(C)(S1)c1ccc(cc1)C(C)(C)O)c1ccc(F)cc1 50273827C[C@H](NC1=NC(=O)C(C)(S1)c1ccc(CCO)cc1)c1ccc(F)cc1 50273855C[C@H](NC1=NC(=O)C(C)(S1)c1ccc(CO)cc1)c1ccc(F)cc1 50273856C[C@H](NC1=NC(=O)C(C)(CC(C)(C)O)S1)c1ccc(F)cc1 50273857C[C@H](NC1=NC(=O)C(C)(S1)C(C)(C)O)c1ccc(F)cc1 50273858C[C@H](NC1=NC(=O)C(C)(S1)C1(O)CCC1)c1ccc(F)cc1 50273859C[C@H](NC1=NC(=O)C(C)(S1)C1(O)CCCC1)c1ccc(F)cc1 50273860C[C@H](NC1=NC(=O)C(C)(S1)C(C)(C)O)c1ccc(cc1)C#N 50273861O=C(Nc1cccc(c1)C(=O)N1CCC[C@@H]2CCCC[C@@H]12)c1ccccc1 50273862Cc1cccc(c1)C(C)(C)C(=O)NC1C2CC3CC1CC(O)(C3)C2 50294764CC(C)(CC(=O)NC1CC1)CC(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50294765Fc1ccc(NC(=O)CC2(CC(=O)NC3C4CC5CC(C4)CC3C5)CCCC2)cc1 50294766O=C(CC1(CC(=O)NC2C3CC4CC(C3)CC2C4)CCCC1)NCc1ccccc1 50294767COc1ccccc1NC(=O)CC1(CC(=O)NC2C3CC4CC(C3)CC2C4)CCCC1 50294768COc1ccc(NC(=O)CC2(CC(=O)NC3C4CC5CC(C4)CC3C5)CCCC2)cc1 50294769Fc1ccc(CNC(=O)CC2(CC(=O)NC3C4CC5CC(C4)CC3C5)CCCC2)cc1 50294770O=C(CC1(CC(=O)NC2C3CC4CC(C3)CC2C4)CCCC1)NCc1ccccn1 50294771CC(C)CNC(=O)CC1(CC(=O)NC2C3CC4CC(C3)CC2C4)CCCC1 50294772CCN1CCN(CC1)C(=O)CC1(CC(=O)NC2C3CC4CC(C3)CC2C4)CCCC1 50294773O=C(CC1(CC(=O)N2CCCC2)CCCC1)NC1C2CC3CC(C2)CC1C3 50294774O=C(CC1(CC(=O)NC2C3CC4CC(C3)CC2C4)CCCC1)NC1CC1 50294776CC(C)(CC(=O)NC1CC1)CC(=O)NC1C2CC3CC(C2)CC1C3 50294777O=C(CC1(CC(=O)NC2C3CC4CC(C3)CC2C4)CCCCC1)NC1CC1 50294778CC(C)(CC(=O)NC1C2CC3CC(C2)CC1C3)Cc1nc(no1)-c1ccc(Cl)cc1 50294779CC(C)(CC(=O)NC1C2CC3CC(C2)CC1C3)Cc1nc(no1)-c1ccccn1 50294780CC(C)(CC(=O)NC1C2CC3CC(C2)CC1C3)Cc1nc(no1)C1CC1 50294781CC(C)c1noc(CC(C)(C)CC(=O)NC2C3CC4CC(C3)CC2C4)n1 50294783CC(C)(CC(=O)NC1CC1)CC(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)C(N)=O 50294784OC(=O)CC1(CC(=O)NCc2ccc(F)cc2Cl)CCCC1 50294785CC(C)(CC(=O)NC1CC1)CC(=O)N[C@H]1C2CC3CC1C[C@@](O)(C3)C2 50294786OC(=O)CC1(CC(=O)NC2C3CC4CC(C3)CC2C4)CCCC1 50295368C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(Br)cc1)c1ccc(F)cc1C(F)(F)F 50295369C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(cc1)C#N)c1ccc(F)cc1C(F)(F)F 50295370C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(cc1Cl)C(N)=O)c1ccc(F)cc1C(F)(F)F 50295371COc1ccc(cc1)S(=O)(=O)N1CCN(C[C@H]1C)c1ccc(F)cc1C(F)(F)F 50295372C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(OC(F)(F)F)cc1)c1ccc(F)cc1C(F)(F)F 50295373C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(cc1)N1CCCCC1)c1ccc(F)cc1C(F)(F)F 50295374C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(cc1)N1CCOCC1)c1ccc(F)cc1C(F)(F)F 50295375C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(cc1)C(N)=O)c1ccc(F)cc1C(F)(F)F 50295376C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(cc1)-c1nnn[nH]1)c1ccc(F)cc1C(F)(F)F 50295377C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(Br)cc1Cl)c1ccc(F)cc1C(F)(F)F 50295378C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(cc1Cl)N(C)C)c1ccc(F)cc1C(F)(F)F 50295379C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(cc1Cl)N1CCCC1)c1ccc(F)cc1C(F)(F)F 50295380C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(cc1Cl)N1CCCCC1)c1ccc(F)cc1C(F)(F)F 50295381C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(cc1Cl)N1CCC(F)CC1)c1ccc(F)cc1C(F)(F)F 50295382C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(cc1Cl)N1CCC(F)(F)CC1)c1ccc(F)cc1C(F)(F)F 50295383C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(cc1Cl)N1CCC(CC1)N(C)C)c1ccc(F)cc1C(F)(F)F 50295384C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(cc1Cl)N1CCC(O)CC1)c1ccc(F)cc1C(F)(F)F 50295385C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(cc1Cl)N1CCC(CC1)C(O)=O)c1ccc(F)cc1C(F)(F)F 50295386C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(cc1Cl)N1CCC(CC1)C(N)=O)c1ccc(F)cc1C(F)(F)F 50295387C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(cc1Cl)N1CCOCC1)c1ccc(F)cc1C(F)(F)F 50295388C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(cc1F)N1CCOCC1)c1ccc(F)cc1C(F)(F)F 50295390C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(NC(=O)N2CCOCC2)cc1Cl)c1ccc(F)cc1C(F)(F)F 50295391C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(cc1Cl)N1CCN(C)CC1)c1ccc(F)cc1C(F)(F)F 50295392C[C@H]1CN(CCN1)c1ccc(c(Cl)c1)S(=O)(=O)N1CCN(C[C@H]1C)c1ccc(F)cc1C(F)(F)F 50295393C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(cc1Cl)N1CCS(=O)(=O)CC1)c1ccc(F)cc1C(F)(F)F 50295394C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(cc1Cl)N1CCNC(=O)C1)c1ccc(F)cc1C(F)(F)F 50295395C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(cc1Cl)N1CCNCC1=O)c1ccc(F)cc1C(F)(F)F 50295396C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(cc1Cl)-n1cncn1)c1ccc(F)cc1C(F)(F)F 50295397C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(OC(C)(C)C)cc1Cl)c1ccc(F)cc1C(F)(F)F 50295398C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(O)cc1Cl)c1ccc(F)cc1C(F)(F)F 50295399C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(OC(F)F)cc1Cl)c1ccc(F)cc1C(F)(F)F 50295400CCOc1ccc(c(Cl)c1)S(=O)(=O)N1CCN(C[C@H]1C)c1ccc(F)cc1C(F)(F)F 50295401COCCOc1ccc(c(Cl)c1)S(=O)(=O)N1CCN(C[C@H]1C)c1ccc(F)cc1C(F)(F)F 50295402C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(OCCN(C)C)cc1Cl)c1ccc(F)cc1C(F)(F)F 50295403C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(cc1Cl)C#N)c1ccc(F)cc1C(F)(F)F 50297203COc1ccc(cc1)C(=O)N1CCCC(CC1)c1ccccc1 50297204COc1ccc(cc1)S(=O)(=O)N1CCC=C(CC1)c1ccccc1 50297205CC(C)(C)c1ccc(cc1)S(=O)(=O)N1CCC=C(CC1)c1ccccc1 50297206Cc1ccc(cc1)S(=O)(=O)N1CCC=C(CC1)c1ccccc1 50297207CCc1ccc(cc1)S(=O)(=O)N1CCC=C(CC1)c1ccccc1 50297208Clc1ccc(c(Cl)c1)S(=O)(=O)N1CCC=C(CC1)c1ccccc1 50297209Cc1ccc(cc1)S(=O)(=O)N1CCCC(=CC1)c1ccccc1 50297210COc1ccc(cc1)S(=O)(=O)N1CCCC(=CC1)c1ccccc1 50297211CC(C)(C)c1ccc(cc1)S(=O)(=O)N1CCCC(=CC1)c1ccccc1 50297212CC(C)(C)c1ccc(cc1)S(=O)(=O)N1CCCC(O)(CC1)c1ccccc1 50297213CCc1ccc(cc1)S(=O)(=O)N1CCCC(O)(CC1)c1ccccc1 50297214OC1(CCCN(CC1)S(=O)(=O)c1ccc(Cl)cc1)c1ccccc1 50297215COc1ccc(cc1)S(=O)(=O)N1CCCC(O)(CC1)c1ccccc1 50297216CC(C)(C)c1ccc(cc1)S(=O)(=O)N1CCCC(C)(O)CC1 50297217CC(C)(C)c1ccc(cc1)S(=O)(=O)N1CCCC(O)(CC1)C1CC1 50297218CC(C)(C)c1ccc(cc1)S(=O)(=O)N1CCCC(O)CC1 50297219COC1(C)CCCN(CC1)S(=O)(=O)c1ccc(cc1)C(C)(C)C 50297220COC1CCCN(CC1)S(=O)(=O)c1ccc(cc1)C(C)(C)C 50297221COC1(CCCN(CC1)S(=O)(=O)c1ccc(cc1)C(C)(C)C)C1CC1 50297222COC1(CCCN(CC1)S(=O)(=O)c1ccc(cc1)C(C)(C)C)c1ccccc1 50297223COC(C)(C)c1ccc(cc1)S(=O)(=O)N1CCCC(C)(CC1)OC 50297224COC1(C)CCCN(CC1)S(=O)(=O)c1ccc(cc1)C(C)(C)O 50297905CCN(CC)C(=O)c1ccc(CNS(=O)(=O)c2cccc(Cl)c2)cc1 50297906Clc1cccc(c1)S(=O)(=O)NCc1ccc(cc1)C(=O)NC1CCCCC1 50297907Clc1cccc(c1)S(=O)(=O)NCc1ccc(cc1)C(=O)NC1CCCC1 50297908Clc1cccc(c1)S(=O)(=O)NCc1ccc(cc1)C(=O)NC1CCCCCC1 50297909CN(C1CCCCCC1)C(=O)c1ccc(CNS(=O)(=O)c2cccc(Cl)c2)cc1 50297910CCCN(C1CCCCCC1)C(=O)c1ccc(CNS(=O)(=O)c2cccc(Cl)c2)cc1 50297911CCCCN(C1CCCCCC1)C(=O)c1ccc(CNS(=O)(=O)c2cccc(Cl)c2)cc1 50297912Clc1cccc(c1)S(=O)(=O)NCc1ccc(cc1)C(=O)NC12CC3CC(CC(C3)C1)C2 50297914C[C@H]1CN(C[C@@H](C)O1)C(=O)c1ccc(CNS(=O)(=O)c2cccc(Cl)c2)cc1 50297915C[C@H]1CN(C[C@@H](C)O1)C(=O)c1ccc(CNS(=O)(=O)c2ccc(Cl)cc2)cc1 50297916C[C@H]1CN(C[C@@H](C)O1)C(=O)c1ccc(CNS(=O)(=O)c2ccccc2Cl)cc1 50297917C[C@H]1CN(C[C@@H](C)O1)C(=O)c1ccc(CNS(=O)(=O)c2cccc(c2)C(F)(F)F)cc1 50297918C[C@H]1CN(C[C@@H](C)O1)C(=O)c1ccc(CNS(=O)(=O)c2ccc(F)c(Cl)c2)cc1 50297921Clc1cccc(c1)S(=O)(=O)NCc1ccc(cc1)C(=O)N1CCCCC1 50297922Clc1cccc(c1)S(=O)(=O)NCc1ccc(cc1)C(=O)N1CCCC1 50306409NA 50306410NA 50306411O=C(NC1C2CC3CC(C2)CC1C3)N1CCCC(Cc2ccccc2)C1 50306412O=C(NC1C2CC3CC(C2)CC1C3)N1CCC(Cc2ccccc2)CC1 50306413NA 50306414NA 50306415NA 50306416O=C(NC1C2CC3CC(C2)CC1C3)N1CCCC2(Cc3ccccc3C2)C1 50306417O=C(NC1C2CC3CC(C2)CC1C3)N1CCC2(CCc3ccccc23)CC1 50306418NC(=O)C1(CCN(CC1)C(=O)NC1C2CC3CC(C2)CC1C3)c1ccccc1 50306419NA 50306420NA 50306421NA 50306422Cc1cccc2c1C(CC(O)=O)CC21CCN(CC1)C(=O)NC1C2CC3CC(C2)CC1C3 50306423Cc1ccc2c(c1)C(CC(O)=O)CC21CCN(CC1)C(=O)NC1C2CC3CC(C2)CC1C3 50306424NA 50306425Cc1cccc2C(CC(O)=O)CC3(CCN(CC3)C(=O)NC3C4CC5CC(C4)CC3C5)c12 50306426OC(=O)CC1CC2(CCN(CC2)C(=O)NC2C3CC4CC(C3)CC2C4)c2ccc(Cl)cc12 50306427OC(=O)CC1CC2(CCN(CC2)C(=O)NC2C3CC4CC(C3)CC2C4)c2cc(Cl)ccc12 50306428NA 50306429OC(=O)CC1CC2(CCN(CC2)C(=O)NC2C3CC4CC(C3)CC2C4)c2c1cccc2Br 50306430NA 50306431NA 50306432CS(=O)(=O)NC(=O)CC1CC2(CCN(CC2)C(=O)NC2C3CC4CC(C3)CC2C4)c2c1cccc2Br 50306433NA 50306434OCCC1CC2(CCN(CC2)C(=O)NC2C3CC4CC(C3)CC2C4)c2c1cccc2Br 50307106COC(=O)[C@]12CC[C@@H](C)[C@H](C)[C@H]1C1=CC[C@@H]3[C@@]4(C)C[C@@H](O)[C@@H](O)C(C)(C)[C@@H]4CC[C@@]3(C)[C@]1(C)CC2 50307107COC(=O)[C@]12CC[C@@H](C)[C@@](C)(O)[C@H]1C1=CC[C@@H]3[C@@]4(C)C[C@@H](O)[C@H](O)C(C)(C)[C@@H]4CC[C@@]3(C)[C@]1(C)CC2 50307108C[C@@H]1CC[C@@]2(CC[C@]3(C)C(=CC(=O)[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@@]34C)[C@@H]2[C@H]1C)C(O)=O 50307109C[C@@H]1CC[C@@]2(CC[C@]3(C)C(=CC(=O)[C@@H]4[C@@]5(C)CC[C@H](OC(C)=O)C(C)(C)[C@@H]5CC[C@@]34C)[C@@H]2[C@H]1C)C(O)=O 50309934OC1=C(N(CC(=O)c2ccccc2)S(=O)(=O)c2ccccc12)C(=O)c1ccccc1 50309936CN1C(C(=O)c2ccccc2)=C(O)c2ccccc2S1(=O)=O 50309937CN1C(C(=O)c2ccccc2)=C(OCC(=O)c2ccccc2)c2ccccc2S1(=O)=O 50309938CCOC(=O)C1=C(O)c2ccccc2S(=O)(=O)N1C 50309939OC1=C(N(Cc2ccccc2)S(=O)(=O)c2ccccc12)C(=O)c1ccccc1 50309940OC1=C(N(CCc2ccccc2)S(=O)(=O)c2ccccc12)C(=O)c1ccccc1 50309941FC(F)(F)S(=O)(=O)OC1=C(N(CC(=O)c2ccccc2)S(=O)(=O)c2ccccc12)C(=O)c1ccccc1 50309942CCOC(=O)C1=C(O)c2ccccc2S(=O)(=O)N1CC(=O)c1ccccc1 50309943OC1=C(N(CC(=O)c2ccc(cc2)-c2ccccc2)S(=O)(=O)c2ccccc12)C(=O)c1ccccc1 50309944OC1=C(N(CC(=O)c2ccc(cc2)[N+]([O-])=O)S(=O)(=O)c2ccccc12)C(=O)c1ccccc1 50309945COC(=O)c1ccc(cc1)C(=O)CN1C(C(=O)c2ccccc2)=C(O)c2ccccc2S1(=O)=O 50309946OC1=C(N(CC(=O)c2ccc(cc2)C#N)S(=O)(=O)c2ccccc12)C(=O)c1ccccc1 50309947OC(=O)c1ccc(cc1)C(=O)CN1C(C(=O)c2ccccc2)=C(O)c2ccccc2S1(=O)=O 50313285CN1C[C@@H]2C[C@H]1CN2S(=O)(=O)c1ccc(cc1)C(C)(C)C 50313286CN1C[C@@H]2C[C@H]1CN2S(=O)(=O)c1ccc(CC(C)(C)C)cc1 50313287CCc1ccc(cc1)S(=O)(=O)N1C[C@@H]2C[C@H]1CN2C 50313288COc1ccc(cc1)S(=O)(=O)N1C[C@@H]2C[C@H]1CN2C 50313289CN1C[C@@H]2C[C@H]1CN2S(=O)(=O)c1ccc(Cl)cc1 50313290CC(C)(C)OC(=O)N1C[C@@H]2C[C@H]1CN2S(=O)(=O)c1ccc(cc1)C(C)(C)C 50313291CC(C)(C)c1ccc(cc1)S(=O)(=O)N1C[C@@H]2C[C@H]1CN2 50313292CC(C)(C)c1ccc(cc1)S(=O)(=O)N1C[C@@H]2C[C@H]1CN2C1CC2CCC1C2 50313293CC(C)(C)c1ccc(cc1)S(=O)(=O)N1C[C@@H]2C[C@H]1CN2C1CCCCC1 50313294CC(C)(C)c1ccc(cc1)S(=O)(=O)N1C[C@@H]2CC[C@H](C1)N2 50313295CC(C)(C)OC(=O)N1[C@H]2CC[C@@H]1CN(C2)S(=O)(=O)c1ccc(cc1)C(C)(C)C 50313296CN1[C@H]2CC[C@@H]1CN(C2)S(=O)(=O)c1ccc(cc1)C(C)(C)C 50313297CC(C)(C)c1ccc(cc1)S(=O)(=O)N1C[C@@H]2CC[C@H](C1)N2C1CCCC1 50313298CC(C)(C)c1ccc(cc1)S(=O)(=O)N1[C@H]2CC[C@@H]1CC(O)(O)C2 50313299CC(C)(C)c1ccc(cc1)S(=O)(=O)N1[C@@H]2CC[C@@]1(C)CC(O)(O)C2 50313300CC(C)(C)c1ccc(cc1)S(=O)(=O)N1[C@H]2CC[C@@H]1CC(O)C2 50313301COC1C[C@@H]2CC[C@H](C1)N2S(=O)(=O)c1ccc(cc1)C(C)(C)C 50313302CC(C)(C)c1ccc(cc1)S(=O)(=O)N1[C@H]2CC[C@@H]1CC(C)(O)C2 50313303COC1(C)C[C@@H]2CC[C@H](C1)N2S(=O)(=O)c1ccc(cc1)C(C)(C)C 50313304CC(C)(C)c1ccc(cc1)S(=O)(=O)N1[C@H]2CC[C@@H]1CC(O)(C2)C(F)(F)F 50313305COC1(C[C@@H]2CC[C@H](C1)N2S(=O)(=O)c1ccc(cc1)C(C)(C)C)C(F)(F)F 50313306CCOC1C[C@@H]2CC[C@H](C1)N2S(=O)(=O)c1ccc(cc1)C(C)(C)C 50313307CC(C)(C)c1ccc(cc1)S(=O)(=O)N1[C@H]2CC[C@@H]1C\C(C2)=N\OCc1ccccc1 50313308CO\N=C1/C[C@@H]2CC[C@H](C1)N2S(=O)(=O)c1ccc(cc1)C(C)(C)C 50313309CC(C)(C)c1ccc(cc1)S(=O)(=O)N1[C@H]2CC[C@@H]1CC(C2)N=O 50313310CC(C)(C)c1ccc(cc1)S(=O)(=O)N1C[C@@H]2C[C@H]1CN2C1CCCC1 50315878Brc1cccc(\C=C2/CC\C(=C/c3cccc(Br)c3)C2=O)c1 50317206O=C(N1CCCCC1)C12CC3CC(C1)CC(C3)(C2)c1ccccc1 50317207CCN(C1CCCCC1)C(=O)CN1CCc2conc2CC1 50317208CCN(CC(=O)NC1C2CC3CC(C2)CC1C3)C1CCCCC1 50317209CCN1CCC[C@@H]1C(=O)NC1C2CC3CC(C2)CC1C3 50317210CN1CCC[C@@H]1C(=O)NC1C2CC3CC(C2)CC1C3 50317211CCCN1CCC[C@@H]1C(=O)NC1C2CC3CC(C2)CC1C3 50317212CC(C)N1CCC[C@@H]1C(=O)NC1C2CC3CC(C2)CC1C3 50317213O=C(NC1C2CC3CC(C2)CC1C3)[C@H]1CCCN1CC1CCCC1 50317214CC(C)CN1CCC[C@@H]1C(=O)NC1C2CC3CC(C2)CC1C3 50317215O=C(NC1C2CC3CC(C2)CC1C3)[C@H]1CCCN1CC1CCC1 50317216O=C(NC1C2CC3CC(C2)CC1C3)[C@H]1CCCN1CC1CCCCC1 50317217FC(F)(F)CN1CCC[C@@H]1C(=O)NC1C2CC3CC(C2)CC1C3 50317218FC(F)(F)CCN1CCC[C@@H]1C(=O)NC1C2CC3CC(C2)CC1C3 50317219Clc1ccc(CN2CCC[C@@H]2C(=O)NC2C3CC4CC(C3)CC2C4)cc1 50317220O=C(NC1C2CC3CC(C2)CC1C3)[C@H]1CCCN1Cc1ccc(cc1)C#N 50317221O=C(NC1C2CC3CC(C2)CC1C3)[C@H]1CCCN1Cc1cccc(c1)C#N 50317222OCCN1CCC[C@@H]1C(=O)NC1C2CC3CC(C2)CC1C3 50317223O=C(NC1C2CC3CC(C2)CC1C3)[C@H]1CCCN1c1ccccn1 50317224O=C(NC1C2CC3CC(C2)CC1C3)[C@H]1CCCN1CC1CCOCC1 50317225OC1(CN2CCC[C@@H]2C(=O)NC2C3CC4CC(C3)CC2C4)CCCC1 50317226OC1(CN2CCC[C@@H]2C(=O)NC2C3CC4CC(C3)CC2C4)CCCCC1 50319310CC(C)(C)C(=O)CSc1cnnn1-c1ccccc1 50319311O=C(CSc1cnnn1-c1ccccc1)c1ccccc1 50319312Fc1ccc(cc1)C(=O)CSc1cnnn1-c1ccccc1 50319313Fc1cccc(c1)C(=O)CSc1cnnn1-c1ccccc1 50319314COc1ccc(cc1)C(=O)CSc1cnnn1-c1ccccc1 50319315COc1cccc(c1)C(=O)CSc1cnnn1-c1ccccc1 50319316COc1ccc(cc1OC)C(=O)CSc1cnnn1-c1ccccc1 50319317O=C(CSc1cnnn1-c1ccccc1)Cc1ccccc1 50319318O=C(CSc1cnnn1-c1ccccc1)c1ccco1 50319319O=C(CSc1cnnn1-c1ccccc1)c1cccs1 50319320COc1ccc(cc1OC)C(=O)CSc1cnnn1C 50319321COc1ccc(cc1OC)C(=O)CSc1cnnn1C(C)C 50319322COc1ccc(cc1OC)C(=O)CSc1cnnn1C(C)(C)C 50319323COc1ccc(cc1OC)C(=O)CSc1cnnn1-c1ccccc1C 50319324COc1ccc(cc1OC)C(=O)CSc1cnnn1-c1cccc(C)c1 50319325COc1ccc(cc1OC)C(=O)CSc1cnnn1-c1ccc(C)cc1 50319326COc1ccc(cc1OC)C(=O)CSc1cnnn1-c1ccc(C)cc1C 50319327COc1ccc(cc1OC)C(=O)CSc1cnnn1-c1ccccc1OC 50319328COc1ccc(cc1OC)C(=O)CSc1cnnn1-c1ccc(Cl)cc1 50319329COc1ccc(cc1OC)C(=O)CSc1cnnn1Cc1ccccc1 50319330COc1ccc(cc1OC)C(=O)CSc1cnnn1Cc1cccs1 50319331COc1ccc(cc1OC)C(=O)CSc1cnnn1C1CCCCC1 50319332Clc1ccc(cc1)-n1nncc1CCC(=O)c1ccccc1 50319333Clc1cccc(c1)-n1nncc1CCC(=O)c1ccccc1 50319334Cc1ccc(cc1)-n1nncc1CCC(=O)c1ccccc1 50319335Cc1cccc(c1)-n1nncc1CCC(=O)c1ccccc1 50319336Cc1ccccc1-n1nnnc1CCC(=O)c1ccccc1 50319337O=C(CCc1cnnn1Cc1ccccc1)c1ccccc1 50319338CC(C)(C)C(=O)CS(=O)c1cnnn1-c1ccccc1 50319339CC(C)(C)C(=O)CS(=O)(=O)c1cnnn1-c1ccccc1 50319340O=C(COc1cnnn1-c1ccccc1)c1ccccc1 50319341O=C(CCc1cnnn1-c1ccccc1)c1ccccc1 50319342COc1ccccc1-n1nncc1CCC(=O)c1ccccc1 50319343COc1cccc(c1)-n1nncc1CCC(=O)c1ccccc1 50319344COc1ccc(cc1)-n1nncc1CCC(=O)c1ccccc1 50319345O=C(CCc1cnnn1-c1ccc(cc1)C#N)c1ccccc1 50319346O=C(CCc1nnnn1-c1cccnc1)c1ccccc1 50319347O=C(CCc1nnnn1C1CCc2ccccc12)c1ccccc1 50319348O=C(CCc1cnnn1C1CCCc2ccccc12)c1ccccc1 50319349O=C(CCc1nnnn1C1CC1)c1ccccc1 50319350O=C(CCc1cnnn1C1CCCC1)c1ccccc1 50319351O=C(CCc1cnnn1C1CCCCC1)c1ccccc1 50319352O=C(CCc1cnnn1[C@@]12CC3CC(CC(C3)C1)C2)c1ccccc1 50319353O=C(CCc1cnnn1C1CCOCC1)c1ccccc1 50319354O=C(CCc1nnnn1-c1ccccc1)Cc1ccccc1 50319355O=C(CCc1nnnn1-c1ccccc1)CCc1ccccc1 50319356Fc1cccc(c1)C(=O)CCc1cnnn1-c1ccccc1 50319357Fc1ccc(cc1)C(=O)CCc1nnnn1-c1ccccc1 50319358Clc1cccc(c1)C(=O)CCc1cnnn1-c1ccccc1 50319359Clc1ccc(cc1)C(=O)CCc1cnnn1-c1ccccc1 50319360COc1cccc(c1)C(=O)CCc1cnnn1-c1ccccc1 50319362O=C(CCc1nnnn1-c1ccccc1)C1CCCCC1 50319363O=C(CCn1nnnc1-c1ccccc1)c1ccccc1 50319364COc1ccccc1-c1nnnn1CCC(=O)c1ccccc1 50319365COc1ccc(cc1)-c1nnnn1CCC(=O)c1ccccc1 50319366O=C(CCn1nnnc1-c1ccc2OCOc2c1)c1ccccc1 50319367Clc1ccccc1-n1nncc1CCC(=O)c1ccccc1 50319368Clc1cccc(c1)-c1nnnn1CCC(=O)c1ccccc1 50319370O=C(CCn1nnnc1-c1cccnc1)c1ccccc1 50319371O=C(CCn1nnnc1-c1cnccn1)c1ccccc1 50319372O=C(CCn1nnnc1-c1ncccn1)c1ccccc1 50319373O=C(CCc1cnnn1-c1ccsc1)c1ccccc1 50319659CC(C)c1sc(NC2CC3CCC2C3)nc1O 50319660CC(C)c1sc(N[C@H]2C[C@@H]3CC[C@H]2C3)nc1O 50319661CC(C)c1sc(N[C@@H]2C[C@H]3CC[C@@H]2C3)nc1O 50319664CC(C)C1(C)SC(N[C@H]2C[C@@H]3CC[C@H]2C3)=NC1=O 50319665CC(C)[C@]1(C)SC(N[C@H]2C[C@@H]3CC[C@H]2C3)=NC1=O 50319666CC(C)[C@]1(C)SC(N[C@@H]2C[C@H]3CC[C@@H]2C3)=NC1=O 50319667CC(C)[C@@]1(C)SC(N[C@H]2C[C@@H]3CC[C@H]2C3)=NC1=O 50319668CC(C)[C@@]1(C)SC(N[C@@H]2C[C@H]3CC[C@@H]2C3)=NC1=O 50321134Fc1ccc(cc1)C(=O)C1CCN(CC1)C(=O)c1ccccc1F 50321137Fc1ccc(cc1)C(=O)C1CCN(CC1)C(=O)c1cccc(c1)C(F)(F)F 50321138Fc1ccc(cc1)C(=O)C1CCN(CC1)C(=O)c1ccc(cc1)-c1ccccc1 50321139CC(=O)c1ccc(cc1)C(=O)N1CCC(CC1)C(=O)c1ccc(F)cc1 50321140Fc1ccc(cc1)C(=O)C1CCN(CC1)C(=O)c1ccc(cc1)C(F)(F)F 50321141Fc1ccc(cc1)C(=O)C1CCN(CC1)C(=O)c1ccc(F)c(F)c1 50321142Cc1cccc(c1)C(=O)N1CCC(CC1)C(=O)c1ccc(F)cc1 50321150[O-][N+](=O)c1ccc(cc1)C(=O)N1CCC(CC1)C(=O)c1ccc(F)cc1 50321151Fc1ccc(cc1)C(=O)C1CCN(CC1)C(=O)c1ccccc1 50321153Fc1ccc(cc1)C(=O)C1CCN(CC1)C(=O)c1cccc(Br)c1 50321154Fc1ccc(cc1)C(=O)C1CCN(CC1)C(=O)c1cccc(Cl)c1 50321155Fc1ccc(cc1)C(=O)C1CCN(CC1)C(=O)c1cccc(OC(F)(F)F)c1 50321158COc1cccc(c1)C(=O)N1CCC(CC1)C(=O)c1ccc(F)cc1 50321161Cc1ccc(cc1)C(=O)N1CCC(CC1)C(=O)c1ccc(F)cc1 50321163Fc1ccc(cc1)C(=O)C1CCN(CC1)C(=O)c1ccc(Cl)cc1 50321164Fc1ccc(cc1)C(=O)C1CCN(CC1)C(=O)c1ccc(Br)cc1 50321166Cc1ccccc1C(=O)N1CCC(CC1)C(=O)c1ccc(F)cc1 50321167Fc1ccc(cc1)C(=O)C1CCN(CC1)C(=O)c1ccc(OC(F)(F)F)cc1 50321168Fc1ccc(cc1)C(=O)C1CCN(CC1)C(=O)c1ccc(F)cc1Cl 50321169Fc1ccc(cc1)C(=O)C1CCN(CC1)C(=O)c1ccc(Cl)c(Cl)c1 50321171CN(C)c1cccc(c1)C(=O)N1CCC(CC1)C(=O)c1ccc(F)cc1 50321173Fc1ccc(cc1)C(=O)C1CCN(CC1)C(=O)c1ccc(Cl)c(c1)C(F)(F)F 50321175Fc1ccc(cc1)C(=O)C1CCN(CC1)C(=O)c1ccccc1Cl 50329187CON[C@@H]1CC[C@@]2(C)[C@@H](CC[C@]3(C)[C@@H]2C(=O)C=C2[C@@H]4C[C@](C)(CC[C@]4(C)CC[C@@]32C)C(O)=O)C1(C)C 50329188CON[C@H]1CC[C@@]2(C)[C@@H](CC[C@]3(C)[C@@H]2C(=O)C=C2[C@@H]4C[C@](C)(CC[C@]4(C)CC[C@@]32C)C(O)=O)C1(C)C 50329189CC(=O)N[C@H]1CC[C@@]2(C)[C@@H](CC[C@]3(C)[C@@H]2C(=O)C=C2[C@@H]4C[C@](C)(CC[C@]4(C)CC[C@@]32C)C(O)=O)C1(C)C 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50329318NC(=O)[C@@]12CC3CC(C1)[C@H](OC(=O)N1CC[C@@H](C1)Nc1ccc(cn1)C#N)C(C3)C2 50331328CC(O)(c1ccc(cc1)S(=O)(=O)c1ccccc1)C(F)(F)F 50331329CC(O)(c1ccc(cc1)S(=O)(=O)c1ccccc1Cl)C(F)(F)F 50331330Cc1ccccc1S(=O)(=O)c1ccc(cc1)C(C)(O)C(F)(F)F 50331331CC(O)(c1ccc(cc1)S(=O)(=O)c1cccc(Cl)c1)C(F)(F)F 50331332COc1ccc(cc1)S(=O)(=O)c1ccc(cc1)C(C)(O)C(F)(F)F 50331333CC(O)(c1ccc(cc1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F 50331334CC(O)(c1ccc(cc1)S(=O)(=O)c1ccc(cc1)[N+]([O-])=O)C(F)(F)F 50331335CC(C)(O)c1ccc(cc1)S(=O)(=O)c1ccccc1Cl 50331336CC(C)(F)c1ccc(cc1)S(=O)(=O)c1ccccc1Cl 50331337CC(C)(C)c1ccc(cc1)S(=O)(=O)c1ccccc1Cl 50331339CC(O)(c1ccc(cc1)S(=O)(=O)c1ccccc1F)C(F)(F)F 50331340CC(O)(c1ccc(cc1)S(=O)(=O)c1ccccc1C(F)(F)F)C(F)(F)F 50331341CCc1ccccc1S(=O)(=O)c1ccc(cc1)C(C)(O)C(F)(F)F 50331342CC(C)c1ccccc1S(=O)(=O)c1ccc(cc1)C(C)(O)C(F)(F)F 50331343CC(O)(c1ccc(cc1)S(=O)(=O)c1ccccc1C1CC1)C(F)(F)F 50331344CC(C)(C)c1ccccc1S(=O)(=O)c1ccc(cc1)C(C)(O)C(F)(F)F 50331345CC(O)(c1ccc(cc1)S(=O)(=O)c1ccccc1C#N)C(F)(F)F 50331346CC(O)(c1ccc(cc1)S(=O)(=O)c1ccccc1-c1ccc(F)cc1)C(F)(F)F 50331347CC(C)(O)c1ccccc1S(=O)(=O)c1ccc(cc1)C(C)(O)C(F)(F)F 50331349CC(O)(c1ccc(cc1)S(=O)(=O)c1ccc(Cl)cc1Cl)C(F)(F)F 50331350CC(O)(c1ccc(cc1)S(=O)(=O)c1ccc(Br)cc1Cl)C(F)(F)F 50331351CC(O)(c1ccc(cc1)S(=O)(=O)c1ccc(cc1Cl)C#N)C(F)(F)F 50331352CC(O)(c1ccc(cc1)S(=O)(=O)c1ccc(cc1Cl)[N+]([O-])=O)C(F)(F)F 50331353CC(O)(c1ccc(cc1)S(=O)(=O)c1ccc(cc1Cl)-c1ccc(cc1)C#N)C(F)(F)F 50331354CC(O)(c1ccc(cc1)S(=O)(=O)c1ccc(cc1Cl)-c1ccncc1)C(F)(F)F 50331355CC(O)(c1ccc(cc1)S(=O)(=O)c1ccc(N)cc1Cl)C(F)(F)F 50331356CC(O)(c1ccc(cc1)S(=O)(=O)c1ccc(cc1Cl)C(N)=O)C(F)(F)F 50331357CC(O)(c1ccc(cc1)S(=O)(=O)c1ccc(NC(N)=O)cc1Cl)C(F)(F)F 50331358CC(O)(c1ccc(cc1)S(=O)(=O)c1ccc(CC2(CC2)C#N)cc1Cl)C(F)(F)F 50331359CC(O)(c1ccc(cc1)S(=O)(=O)c1ccc(CC2(CC2)C(N)=O)cc1Cl)C(F)(F)F 50331360C[C@@](O)(c1ccc(cc1)S(=O)(=O)c1ccc(cc1Cl)-c1ccc(cc1)C#N)C(F)(F)F 50331361C[C@](O)(c1ccc(cc1)S(=O)(=O)c1ccc(cc1Cl)-c1ccc(cc1)C#N)C(F)(F)F 50331362C[C@@](O)(c1ccc(cc1)S(=O)(=O)c1ccc(cc1C1CC1)-c1ccc(cc1)C#N)C(F)(F)F 50331363C[C@](O)(c1ccc(cc1)S(=O)(=O)c1ccc(cc1C1CC1)-c1ccc(cc1)C#N)C(F)(F)F 50331364C[C@@](O)(c1ccc(cc1)S(=O)(=O)c1ccc(cc1CCF)-c1ccc(cc1)C#N)C(F)(F)F 50331365C[C@](O)(c1ccc(cc1)S(=O)(=O)c1ccc(cc1CCF)-c1ccc(cc1)C#N)C(F)(F)F 50334672C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@@](CCO)(CC1)c1ccccc1)C(F)(F)F 50334673C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@@](CCC(N)=O)(CC1)c1ccccc1)C(F)(F)F 50334674C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@@](CNS(C)(=O)=O)(CC1)c1ccccc1)C(F)(F)F 50334675C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@@](COC(N)=O)(CC1)c1ccccc1)C(F)(F)F 50334676CC(=O)NC[C@@]1(CC[C@@H](CC1)N(C1CC1)C(=O)c1ccc(cc1)[C@](C)(O)C(F)(F)F)c1ccccc1 50334677C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@@](CCC(N)=O)(CC1)c1ccccc1F)C(F)(F)F 50334678C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@@](CCC(N)=O)(CC1)c1ccc(F)cc1)C(F)(F)F 50334679C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@@](CCC(N)=O)(CC1)c1ccccn1)C(F)(F)F 50334680C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@@](COC(N)=O)(CC1)c1ccccc1F)C(F)(F)F 50334681C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@@](COC(N)=O)(CC1)c1ccc(F)cc1)C(F)(F)F 50334682C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@@](COC(N)=O)(CC1)c1ccccn1)C(F)(F)F 50334683C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@@](COC(N)=O)(CC1)c1ccc(F)cn1)C(F)(F)F 50334684C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@@](COC(N)=O)(CC1)c1cscn1)C(F)(F)F 50334685C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@@](CO)(CC1)c1ccccc1)C(F)(F)F 50334686C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@@](CC#N)(CC1)c1ccccc1)C(F)(F)F 50334687C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@@](CCC#N)(CC1)c1ccccc1)C(F)(F)F 50334688C[C@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@@](CC(N)=O)(CC1)c1ccccc1)C(F)(F)F 50334689O=C(NC1C2CC3CC(C2)CC1C3)C1SCCN1Cc1ccccc1 50334690O=C(NC1C2CC3CC(C2)CC1C3)C1NCCS1 50334691CC(C)(C)OC(=O)N1CCSC1C(=O)NC1C2CC3CC(C2)CC1C3 50334692O=C(NC1C2CC3CC(C2)CC1C3)C1SCCN1C(=O)c1ccccc1 50334693O=C(NC1C2CC3CC(C2)CC1C3)C1SCCN1C(=O)Nc1ccccc1 50334694O=C(NC1C2CC3CC(C2)CC1C3)C1SCCN1S(=O)(=O)c1ccccc1 50334695Cc1ccc(cc1)S(=O)(=O)N1CCSC1C(=O)NC1C2CC3CC(C2)CC1C3 50334696COc1ccc(cc1)S(=O)(=O)N1CCSC1C(=O)NC1C2CC3CC(C2)CC1C3 50334697CC(C)(C)c1ccc(cc1)S(=O)(=O)N1CCSC1C(=O)NC1C2CC3CC(C2)CC1C3 50334698Fc1ccc(cc1)S(=O)(=O)N1CCSC1C(=O)NC1C2CC3CC(C2)CC1C3 50334699Fc1ccccc1S(=O)(=O)N1CCSC1C(=O)NC1C2CC3CC(C2)CC1C3 50334700Clc1ccc(cc1)S(=O)(=O)N1CCSC1C(=O)NC1C2CC3CC(C2)CC1C3 50334701Clc1ccc(cc1Cl)S(=O)(=O)N1CCSC1C(=O)NC1C2CC3CC(C2)CC1C3 50334702OC12CC3CC(C1)C(NC(=O)C1SCCN1S(=O)(=O)c1ccc(Cl)c(Cl)c1)C(C3)C2 50334703COC(=O)C12CC3CC(C1)C(NC(=O)C1SCCN1S(=O)(=O)c1ccc(Cl)c(Cl)c1)C(C3)C2 50334704NC(=O)C12CC3CC(C1)C(NC(=O)C1SCCN1S(=O)(=O)c1ccc(Cl)c(Cl)c1)C(C3)C2 50334705NC(=O)C12CC3CC(C1)C(NC(=O)C1SCCN1S(=O)(=O)c1ccccc1)C(C3)C2 50334706Cc1ccc(cc1)S(=O)(=O)N1CCSC1C(=O)NC1C2CC3CC1CC(C3)(C2)C(N)=O 50334707COc1ccc(cc1)S(=O)(=O)N1CCSC1C(=O)NC1C2CC3CC1CC(C3)(C2)C(N)=O 50334708NC(=O)C12CC3CC(C1)C(NC(=O)C1SCCN1S(=O)(=O)c1ccccc1F)C(C3)C2 50334709NC(=O)C12CC3CC(C1)C(NC(=O)C1SCCN1S(=O)(=O)c1cccc(F)c1)C(C3)C2 50334710NC(=O)C12CC3CC(C1)C(NC(=O)C1SCCN1S(=O)(=O)c1ccc(F)cc1)C(C3)C2 50334712NC(=O)C12CC3CC(C1)C(NC(=O)[C@H]1SCCN1S(=O)(=O)c1ccccc1F)C(C3)C2 50334713NC(=O)C12CC3CC(C1)C(NC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccccc1F)C(C3)C2 50334714NC(=O)C12CC3CC(C1)C(NC(=O)[C@H]1CCCN1S(=O)(=O)c1ccccc1F)C(C3)C2 50335195CC(=O)c1cc2ccc(OS(=O)(=O)C(F)(F)F)cc2oc1=O 50335196CC(=O)c1cc2ccc(cc2oc1=O)-c1ccccc1 50335197CC(=O)c1cc2ccc(cc2oc1=O)-c1ccc(C)cc1 50335198COc1ccc(cc1)-c1ccc2cc(C(C)=O)c(=O)oc2c1 50335199CC(=O)c1cc2ccc(cc2oc1=O)-c1ccc(O)cc1 50335200COc1cc(c(Br)c(OC)c1OC)-c1nc2sc3c(O)cccc3c2c(=O)n1Cc1ccccc1 50339805C[C@]12CC[C@@](C)(C[C@H]1C1=CC(=O)[C@@H]3[C@@]4(C)CC[C@H](Oc5nc(=O)o[nH]5)C(C)(C)[C@@H]4CC[C@@]3(C)[C@]1(C)CC2)C(O)=O 50339806CC(=O)O[C@H]1CC[C@@]2(C)[C@@H](CC[C@]3(C)[C@@H]2C(=O)C=C2[C@@H]4C[C@](C)(CC[C@]4(C)CC[C@@]32C)NC(N)=O)C1(C)C 50339807CC(=O)O[C@H]1CC[C@@]2(C)[C@@H](CC[C@]3(C)[C@@H]2C(=O)C=C2[C@@H]4C[C@](C)(CC[C@]4(C)CC[C@@]32C)NC(=O)NS(=O)(=O)C(F)(F)F)C1(C)C 50339811CN(O)C(=O)[C@@]1(C)CC[C@]2(C)CC[C@]3(C)C(=CC(=O)[C@@H]4[C@@]5(C)CC[C@H](Oc6nc(=O)o[nH]6)C(C)(C)[C@@H]5CC[C@@]34C)[C@@H]2C1 50339812CC1(C)[C@@H](O)CC[C@@]2(C)[C@H]1CC[C@]1(C)[C@@H]2C(=O)C=C2[C@@H]3C[C@](C)(CC[C@]3(C)CC[C@@]12C)NC(N)=O 50340371CCS(=O)CCC12CCC(CC1)(CC2)c1nnc(-c2ccccc2C(F)(F)F)n1C 50340372CC(C)S(=O)(=O)CCC12CCC(CC1)(CC2)c1nnc(-c2ccccc2C(F)(F)F)n1C 50340373Cn1c(nnc1C12CCC(CCS(=O)(=O)c3ccccc3)(CC1)CC2)-c1ccccc1C(F)(F)F 50340374CCCS(=O)(=O)CCC12CCC(CC1)(CC2)c1nnc(-c2ccccc2C(F)(F)F)n1C 50340375Cn1c(nnc1C12CCC(CCS(=O)(=O)C(C)(C)C)(CC1)CC2)-c1ccccc1C(F)(F)F 50340376Cn1c(nnc1C12CCC(CCS(=O)(=O)c3ccc(F)cc3)(CC1)CC2)-c1ccccc1C(F)(F)F 50340377Cn1c(nnc1C12CCC(CCS(=O)(=O)C(F)(F)F)(CC1)CC2)-c1ccccc1C(F)(F)F 50340378CCS(=O)(=O)CCC12CCC(CC1)(CC2)c1nnc(-c2ccccc2C(F)(F)F)n1C 50340379CCS(=O)(=O)CCC12CCC(CC1)(CC2)c1nnc(-c2ccccc2Cl)n1C 50340380CCCS(=O)(=O)NCC12CCC(CC1)(CC2)c1nnc(-c2ccccc2C(F)(F)F)n1C 50340381CCS(=O)(=O)CCC12CCC(CC1)(CC2)c1nnc(-c2ccccc2Br)n1C 50340382Cn1c(nnc1C12CCC(CCS(C)(=O)=O)(CC1)CC2)-c1ccccc1C(F)(F)F 50340383CC(O)CCCC12CCC(CC1)(CC2)c1nnc2CCCCCCn12 50340384CCS(=O)(=O)NCC12CCC(CC1)(CC2)c1nnc(-c2ccccc2C(F)(F)F)n1C 50340385CCS(=O)(=O)CCC12CCC(CC1)(CC2)c1nnc(-c2ccccc2C)n1C 50340386CCS(=O)(=O)CC12CCC(CC1)(CC2)c1nnc(-c2ccccc2C(F)(F)F)n1C 50340387Cn1c(nnc1C12CCC(CNS(C)(=O)=O)(CC1)CC2)-c1ccccc1C(F)(F)F 50340388CCS(=O)(=O)CCC12CCC(CC1)(CC2)c1nnc(-c2ccccc2F)n1C 50340389Cn1c(nnc1C12CCC(COc3ccc(Cl)cc3)(CC1)CC2)-c1ccccc1C(F)(F)F 50340390CCS(=O)(=O)CCC12CCC(CC1)(CC2)c1nnc(-c2cccc(Cl)c2)n1C 50340392Cn1c(nnc1C12CCC(CCS(=O)(=O)CC(F)(F)F)(CC1)CC2)-c1ccccc1C(F)(F)F 50340393CCS(=O)(=O)CCC12CCC(CC1)(CC2)c1nnc(-c2ccc(Cl)cc2)n1C 50340394CC(=O)CCCC12CCC(CC1)(CC2)c1nnc(-c2ccccc2C(F)(F)F)n1C 50340395COCCCCC12CCC(CC1)(CC2)c1nnc(-c2ccccc2C(F)(F)F)n1C 50340398CCOCC12CCC(CC1)(CC2)c1nnc(-c2ccccc2C(F)(F)F)n1C 50340399Cn1c(nnc1C12CCC(COc3ccc(cc3)S(C)(=O)=O)(CC1)CC2)-c1ccccc1C(F)(F)F 50340400CCSCCC12CCC(CC1)(CC2)c1nnc(-c2ccccc2C(F)(F)F)n1C 50340401CCS(=O)(=O)CCCC12CCC(CC1)(CC2)c1nnc(-c2ccccc2C(F)(F)F)n1C 50340402CCS(=O)(=O)CCCCC12CCC(CC1)(CC2)c1nnc(-c2ccccc2C(F)(F)F)n1C 50340403CCS(=O)(=O)CCC12CCC(CC1)(CC2)c1nnc(-c2ccc(O)cc2Cl)n1C 50340431O=C(N1CCC(CC1)c1cnc[nH]1)N1CCCc2ccccc12 50340432CC1COc2ccccc2N1C(=O)N1CCC(CC1)c1cnc[nH]1 50340433COc1ccc(cc1)-c1cnc(nc1)N1CCN(C(=O)N2CCC(C2)c2cn[nH]c2)c2ccccc12 50340434O=C(N1CCC(CC1)c1ccn[nH]1)N1CCCc2ccccc12 50340435O=C(N1CCC(CC1)c1cn[nH]c1)N1CCCc2ccccc12 50340436O=C(N1CCC(CC1)c1cccnc1)N1CCCc2ccccc12 50340437O=C(N1[C@H]2CC[C@@H]1C[C@@H](C2)c1ccn[nH]1)N1CCCc2ccccc12 50340438O=C(N1CCC(C1)c1cn[nH]c1)N1CCCc2ccccc12 50340439CC1(C)CCN(C(=O)N2CCC(C2)c2cn[nH]c2)c2ccccc12 50340440O=C(N1CCC(C1)c1cn[nH]c1)N1CCC2(CC2)c2ccccc12 50340441O=C(N1CCC(C1)c1cn[nH]c1)N1CCOc2ccccc12 50340442O=C(N1CCC(C1)c1cn[nH]c1)N1CCNc2ccccc12 50340443CN1CCN(C(=O)N2CCC(C2)c2cn[nH]c2)c2ccccc12 50340444NC(=O)c1ccc(cc1)N1CCN(C(=O)N2CCC(C2)c2cn[nH]c2)c2ccccc12 50340445O=C(N1CCC(C1)c1cn[nH]c1)N1CCN(c2ccc(cc2)C#N)c2ccccc12 50340446O=C(NC1CC1)c1ccc(cc1)N1CCN(C(=O)N2CCC(C2)c2cn[nH]c2)c2ccccc12 50340447O=C(NC1CC1)c1ccc(CN2CCN(C(=O)N3CCC(C3)c3cn[nH]c3)c3ccccc23)cc1 50340448Cn1cc(cn1)C1CCN(CC1)C(=O)N1CCCc2ccccc12 50340452O=C(N1CCC(CC1)c1ncon1)N1CCCc2ccccc12 50340454Cc1noc(n1)C1CCN(CC1)C(=O)N1CCCc2ccccc12 50340457O=C(N1[C@H]2CC[C@@H]1C[C@H](C2)c1ccn[nH]1)N1CCCc2ccccc12 50340792CC(=O)Nc1ccc(cc1)-c1nnc(n1C)C1(CCC1)c1ccc(Cl)cc1 50340793Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(NC(=O)c2cnccn2)cc1 50340794Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(NC(=O)c2cccs2)cc1 50340795Cc1cc(C(=O)Nc2ccc(cc2)-c2nnc(n2C)C2(CCC2)c2ccc(Cl)cc2)c(C)o1 50340796Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(NC(=O)c2ccno2)cc1 50340797Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1)-c1ccon1 50340799Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1F)-c1cccnc1 50340800COc1cc(ccc1-c1nnc(n1C)C1(CCC1)c1ccc(Cl)cc1)-c1cccnc1 50340801Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1O)-c1cccnc1 50340802Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1F)-c1cnccn1 50340803Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1OC(F)F)-c1cnccn1 50340804Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1C(N)=O)-c1cnccn1 50340805Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1C(N)=O)C(N)=O 50340808Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(NC(=O)c2cnccn2)cc1Cl 50340809C1C2CC3CC1CC(C2)(C3)c1nnc2CCCCCCn12 50340810Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1)C(O)=O 50340811Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1)C(N)=O 50340812Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1)-c1cncnc1 50340813Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1)-c1cnc(N)nc1 50340814Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1)-c1cnc(=O)[nH]c1 50340815COc1ncc(-c2ccc(cc2)-c2nnc(n2C)C2(CCC2)c2ccc(Cl)cc2)c(OC)n1 50340816Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1)-c1cnccn1 50340817Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1)-c1cc(=O)[nH]cn1 50340818Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1)-c1ccc(Cl)nn1 50340819Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1)-c1ccc(N)nn1 50340820Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1)-c1cnoc1 50340821Cc1noc(C)c1-c1ccc(cc1)-c1nnc(n1C)C1(CCC1)c1ccc(Cl)cc1 50340822CCNC(=O)c1ccc(cc1)-c1nnc(n1C)C1(CCC1)c1ccc(Cl)cc1 50340823Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1)C(=O)NC(C)(C)C 50340824Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1)C(=O)NC1CC1 50340825Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1)C(=O)NC1CCC1 50340826Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1)C(=O)N1CCC1 50340827Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1)C(=O)N1CCCC1 50340828Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1)C(=O)N1CCOCC1 50340829Cn1c(nnc1C1(CCC1)c1ccc(Cl)cc1)-c1ccc(cc1Cl)C(O)=O 50340831NA 50348280Clc1cccc(Cl)c1SCc1cccn2c(nnc12)C1CCCCC1 50348281Clc1cccc(Cl)c1OCc1cccn2c(nnc12)C1CCCCC1 50348282Clc1cccc(Cl)c1OCc1cccn2c(nnc12)C1CCCCCC1 50348283Clc1cccc(Cl)c1COc1cccn2c(nnc12)C1CCCCCC1 50348284Clc1cccc(Cl)c1COCc1cccn2c(nnc12)C1CCCCCC1 50348285Clc1cccc(Cl)c1Oc1cccn2c(nnc12)C1CCCCCC1 50348286Clc1cccc(Cl)c1S(=O)(=O)Cc1cccn2c(nnc12)C1CCCCCC1 50348287Clc1cccc(Cl)c1S(=O)(=O)NCc1cccn2c(nnc12)C1CCCCCC1 50348288Clc1cccc(Cl)c1S(=O)(=O)Nc1cccn2c(nnc12)C1CCCCCC1 50348289Clc1cc(Cl)cc(SCc2cccn3c(nnc23)C2CCCCCC2)c1 50348290Cc1c(Cl)cccc1S(=O)(=O)NCc1cccn2c(nnc12)C1CCCCCC1 50348291Cc1c(Cl)cccc1Oc1cccn2c(nnc12)C1CCCCCC1 50348292Cc1c(Cl)cccc1Oc1cccn2c(nnc12)C12CCC(CC1)C2 50348293COC1(CCCCCC1)c1nnc2c(Oc3cccc(Cl)c3C)cccn12 50348294COC12CC3CC(C1)CC(C3)(C2)c1nnc2c(Oc3cccc(Cl)c3C)cccn12 50348295Cc1c(Cl)cccc1Oc1cccn2c(nnc12)[C@]12CCC(C[C@H]1O)C2(C)C 50348296Cc1c(Cl)cccc1Oc1cccn2c(CC3CC4CCC3C4)nnc12 50348297Cc1c(Cl)cccc1Oc1cccn2c(nnc12)C1CCC(F)(F)CC1 50348298Cc1c(Cl)cccc1Oc1cccn2c(nnc12)C1CCC(C)(O)CC1 50348299Cc1c(Cl)cccc1Oc1cccn2c(nnc12)C1CCC(=O)CC1 50348300Cc1c(Cl)cccc1Oc1cccn2c(nnc12)C1CCOCC1 50348304Cc1c(Cl)cccc1Oc1cccn2c(nnc12)C12CCC(N)(CC1)CC2 50348305Cc1c(Cl)cccc1Oc1cccn2c(nnc12)C1CCCCCC1O 50348306Cc1c(Cl)cccc1Oc1cccn2c(nnc12)C12CC3CC(CC(O)(C3)C1)C2 50348307COC12CCC(CC1)(CC2)c1nnc2c(Oc3cccc(Cl)c3C)cccn12 50348308Cc1c(Cl)cccc1Oc1cccn2c(nnc12)C12CCC(F)(CC1)CC2 50348309Cc1c(Cl)cccc1Oc1cccn2c(nnc12)C12CCC(O)(CC1)CC2 50353386C[C@H](N1CC[C@@](CCO)(OC1=O)c1ccc(F)cc1)c1ccc(cc1)-c1ccc(F)cc1F 50353387C[C@H](N1CC[C@@](CCC(N)=O)(OC1=O)c1ccc(F)cc1)c1ccc(cc1)-c1ccc(F)cc1F 50353388C[C@H](N1CC[C@@](CC(N)=O)(OC1=O)c1ccc(F)cc1)c1ccc(cc1)-c1ccc(F)cc1F 50353389C[C@H](N1CC[C@@](CCCO)(OC1=O)c1ccc(F)cc1)c1ccc(cc1)-c1ccc(F)cc1F 50353390C[C@H](N1CC[C@@](CCO)(OC1=O)c1ccc(F)cc1)c1ccc(cc1)-c1ccc(F)cc1 50353391C[C@H](N1CC[C@@](CCNS(N)(=O)=O)(OC1=O)c1ccc(F)cc1)c1ccc(cc1)-c1ccc(F)cc1F 50353392C[C@H](N1CC[C@@](CCCO)(OC1=O)c1ccccc1)c1ccc(cc1)-c1ccc(F)cc1 50353393C[C@H](N1CC[C@@](CCCO)(OC1=O)c1ccccc1F)c1ccc(cc1)-c1ccc(F)cc1 50353394C[C@H](N1CC[C@@](CCCO)(OC1=O)c1ccc(F)cc1)c1ccc(cc1)-c1ccc(F)cc1 50353395C[C@H](N1CC[C@@](CCCNS(C)(=O)=O)(OC1=O)c1ccc(F)cc1)c1ccc(cc1)-c1ccc(F)cc1F 50353396C[C@H](N1CC[C@@](CCCO)(OC1=O)c1cccc(F)c1)c1ccc(cc1)-c1ccc(F)cc1 50353397C[C@H](N1CC[C@@](CCNC(N)=O)(OC1=O)c1ccc(F)cc1)c1ccc(cc1)-c1ccc(F)cc1F 50353398C[C@H](N1CC[C@@](CCCNC(N)=O)(OC1=O)c1ccc(F)cc1)c1ccc(cc1)-c1ccc(F)cc1F 50353399C[C@H](N1CC[C@@](CCN)(OC1=O)c1ccc(F)cc1)c1ccc(cc1)-c1ccc(F)cc1F 50353400CC[C@H](N1CC[C@@](CCCO)(OC1=O)c1ccccc1)c1ccc(cc1)-c1ccc(F)cc1 50353401CNC(=O)NCC[C@@]1(CCN([C@@H](C)c2ccc(cc2)-c2ccc(F)cc2F)C(=O)O1)c1ccc(F)cc1 50353402CNC(=O)NCCC[C@@]1(CCN([C@@H](C)c2ccc(cc2)-c2ccc(F)cc2F)C(=O)O1)c1ccc(F)cc1 50353403C[C@H](N1CC[C@@](CCNC(C)=O)(OC1=O)c1ccc(F)cc1)c1ccc(cc1)-c1ccc(F)cc1F 50353404C[C@H](N1CC[C@@](CCNS(C)(=O)=O)(OC1=O)c1ccc(F)cc1)c1ccc(cc1)-c1ccc(F)cc1F 50353405C[C@H](N1CC[C@@](CCCO)(OC1=O)c1ccccc1)c1ccc(cc1)-c1ccc(F)cc1F 50353406C[C@H](N1CC[C@@](CCO)(OC1=O)c1ccccc1)c1ccc(cc1)-c1ccc(F)cc1F 50353407C[C@H](N1CC[C@@](CCO)(OC1=O)c1ccccc1)c1ccc(cc1)-c1ccc(F)cc1 50353408OCCC1(CCN(C(=O)O1)c1cccc(c1)-c1ccc(F)cc1F)c1ccccc1 50353409CNC(=O)CC[C@@]1(CCN([C@@H](C)c2ccc(cc2)-c2ccc(F)cc2F)C(=O)O1)c1ccc(F)cc1 50353410CCNC(=O)NCC[C@@]1(CCN([C@@H](C)c2ccc(cc2)-c2ccc(F)cc2F)C(=O)O1)c1ccc(F)cc1 50353411CC1(CCN(C(=O)O1)c1cccc(c1)-c1ccccc1)c1ccccc1 50353412Fc1ccc(c(F)c1)-c1cccc(c1)N1CCC(CC=C)(OC1=O)c1ccccc1 50353413CC1(CCN(C(=O)O1)c1cccc(c1)-c1cccc(F)c1)c1ccccc1 50353414CC1(CCN(C(=O)O1)c1cccc(c1)-c1ccccc1F)c1ccccc1 50353415CC1(CCN(C(=O)O1)c1cccc(c1)-c1ccc(F)cc1)c1ccccc1 50353416CC1(CCN(C(=O)O1)c1cccc(c1)-c1ccc(F)cc1F)c1ccccc1 50353417C[C@H](N1CC[C@@](CCCN)(OC1=O)c1ccc(F)cc1)c1ccc(cc1)-c1ccc(F)cc1F 50353418OCCCC1(CCN(C(=O)O1)c1cccc(c1)-c1ccc(F)cc1F)c1ccccc1 50353419Cc1cccc(c1)N1CC[C@@H](OC1=O)c1ccccc1 50353420CC1(CCN(C(=O)O1)c1ccc(cc1)C(F)(F)F)c1ccccc1 50353421CC1(CCN(Cc2ccc(Br)cc2)C(=O)O1)c1ccccc1 50353422Cc1cccc(c1)N1CC[C@H](OC1=O)c1ccccc1 50353423CC1(CCN(C(=O)O1)c1ccc(Cl)cc1)c1ccccc1 50353424CC1(CCN(C(=O)O1)c1ccccc1)c1ccccc1 50353425Cc1cccc(c1)N1CCC(C)(OC1=O)c1ccccc1 50353426CC1(CCN(C(=O)O1)c1cccc(Cl)c1)c1ccccc1 50353427CC1(CCN(C(=O)O1)c1ccccc1Cl)c1ccccc1 50353428CC1(CCN(C(=O)O1)c1cccc(Br)c1)c1ccccc1 50353430C[C@@H](N1CC[C@@](CCO)(OC1=O)c1ccc(F)cc1)c1ccc(cc1)-c1ccc(F)cc1F 50354740O=S(=O)(N1CCC(=CC1)c1ccccc1)c1ccc2ccccc2c1 50354741FC(F)(F)c1cnc(N2CCN(CC2)S(=O)(=O)c2ccc3ccccc3c2)c(Cl)c1 50354742Fc1cccc(Cl)c1CSc1nnc(-c2ccco2)n1-c1ccc(OCc2ccccc2)cc1 50354743Clc1ccc(c(Cl)c1)S(=O)(=O)C(=C\c1ccc2OCCc2c1)\C#N 50354744Clc1ccc(Cl)c(c1)S(=O)(=O)Nc1cccc(CCc2ccccn2)c1 50354745Fc1cccc(Cl)c1CN1CCCN(CC1)S(=O)(=O)c1ccc2ccccc2c1 50354746CN(Cc1ccccc1)S(=O)(=O)c1ccc(Oc2cccc(Cl)c2C#N)cc1 50356333OC(=O)CC1(C2CC3CC(C2)CC1C3)c1ccc(F)cc1 50356334OC(=O)CC1(CCc2ccccc2)C2CC3CC(C2)CC1C3 50356335OC(=O)CC1(Cc2cccc(Cl)c2)C2CC3CC(C2)CC1C3 50356336OC(=O)CC1(Cc2ccccc2Cl)C2CC3CC(C2)CC1C3 50356337OC(=O)CC1(Cc2ccccc2)C2CC3CC(C2)CC1C3 50356338OC(=O)CC1(C2CC3CC(C2)CC1C3)c1ccccc1 50356339OC(=O)CC1(C2CC3CC(C2)CC1C3)c1cccc(c1)C#N 50356340OC(=O)CC1(C2CC3CC(C2)CC1C3)c1cccc(Cl)c1 50356341OC(=O)CC1(C2CC3CC(C2)CC1C3)c1ccc(Cl)cc1 50356342Cc1ccc(cc1)C1(CC(O)=O)C2CC3CC(C2)CC1C3 50356343COc1ccc(cc1)C1(CC(O)=O)C2CC3CC(C2)CC1C3 50356344OC(=O)CC1(C2CC3CC(C2)CC1C3)c1cccc(F)c1 50356345CC1(O)C2CC3CC(C2)C(CC(O)=O)(C1C3)c1ccc(F)cc1 50356346OC1C2CC3CC1CC(C2)C3(CC(O)=O)c1ccc(F)cc1 50356347OC(=O)CC1(C2CC3CC1CC(O)(C3)C2)c1ccc(F)cc1 50356348OC1C2CC3CC(C2)C(CC(O)=O)(C1C3)c1ccc(F)cc1 50356349COC12CC3CC(C1)C(CC(O)=O)(C(C3)C2)c1ccc(F)cc1 50356350OC(=O)CC1(C2CC3CC1CC(F)(C3)C2)c1ccc(F)cc1 50356351OC(=O)CC1(C2CC3CC1CC(C2)O3)c1ccc(F)cc1 50356352OC1CC2CCCC(C1)C2(CC(O)=O)c1ccc(F)cc1 50356353OC(=O)CC1(C2CCCC1COC2)c1ccc(F)cc1 50356354OC(=O)CC1(C2CCCC1CCC2)c1ccc(F)cc1 50356355OC(=O)CC1(CC2(C1)CCCCC2)c1ccc(F)cc1 50356356NA 50356357OC(=O)CC1(CC2CCC(C2)C1)c1ccc(F)cc1 50356358OC(=O)CC1(CC2CCC1C2)c1ccc(F)cc1 50356359OC(=O)CC1(CCCCC1)c1ccc(F)cc1 50356360OC(=O)CC1(C2CC3CC(C2)CC1(O)C3)c1ccc(F)cc1 50356361OC(=O)CCC1(C2CC3CC(C2)CC1C3)c1ccc(F)cc1 50356362OC(=O)C1(C2CC3CC(C2)CC1C3)c1ccc(F)cc1 50356363OC(=O)CC1(C#N)C2CC3CC(C2)CC1C3 50356364OC(=O)CC1C2CC3CC(C2)CC1C3 50356365O=C(N1CCC(CCSc2ncc[nH]2)CC1)C12CC3CC(CC(C3)C1)C2 50356429CS(=O)(=O)c1ccccc1CSc1[nH]c(=O)c(C#N)c2CCCCc12 50356430O=c1[nH]c(SCc2ccccc2-c2ccccc2)c2CCCCc2c1C#N 50356431COc1ccccc1CSc1[nH]c(=O)c(C#N)c2CCCCc12 50356432Clc1ccc(CSc2[nH]c(=O)c(C#N)c3CCCCc23)cc1 50356433Clc1cccc(CSc2[nH]c(=O)c(C#N)c3CCCCc23)c1 50356434O=c1[nH]c(SCc2ccccc2)c2CCCCc2c1C#N 50356435Clc1ccccc1CSc1[nH]c(=O)c(C#N)c2CCCCc12 50356436Clc1ccccc1CSc1nc(-c2ccccc2)c(C#N)c(=O)[nH]1 50356437Fc1ccc2c(C#N)c(=O)[nH]c(OCc3ccccc3Cl)c2c1 50356438Fc1ccc2c(C#N)c(=O)[nH]c(SCc3cccnc3C#N)c2c1 50356439Fc1ccc2c(C#N)c(=O)[nH]c(SCc3ccccc3Cl)c2c1 50356440Clc1ccccc1CSc1[nH]c(=O)c(C#N)c2ccc(cc12)C#N 50356441Fc1ccc2c(SCc3ccccc3Cl)[nH]c(=O)c(C#N)c2c1 50356442Fc1cccc2c(C#N)c(=O)[nH]c(SCc3ccccc3Cl)c12 50356443Fc1cccc2c(SCc3ccccc3Cl)[nH]c(=O)c(C#N)c12 50356444Clc1ccccc1CSc1[nH]c(=O)c(C#N)c2ccccc12 50356445O=c1[nH]c(SCc2cccnc2C#N)c2COCCc2c1C#N 50356446Clc1ccccc1CSc1[nH]c(=O)c(C#N)c2CCOCc12 50356447Clc1ccccc1CSc1[nH]c(=O)c(C#N)c2CCN(Cc3ccccc3)Cc12 50356448O=c1[nH]c(SCc2ccccc2)c2CCc3ccccc3-c2c1C#N 50356449O=c1[nH]c(SCc2cccnc2C#N)c2CCCCc2c1C#N 50356450O=c1[nH]c(SCC2CCC2)c2CCCCc2c1C#N 50356451Clc1ccccc1COc1[nH]c(=O)c(C#N)c2CCCCc12 50356452Clc1ccccc1CCSc1[nH]c(=O)c(C#N)c2CCCCc12 50356453O=c1[nH]c(-c2ccccc2)c2CCCCc2c1C#N 50356454Clc1ccccc1Sc1[nH]c(=O)c(C#N)c2CCCCc12 50356455Clc1ccccc1CS(=O)(=O)c1[nH]c(=O)c(C#N)c2CCCCc12 50356457Clc1ccccc1CSc1[nH]c(=O)c(-c2ccc(cc2)C#N)c2CCCCc12 50356458Clc1ccccc1CSc1[nH]c(=O)c(Br)c2CCCCc12 50356459Clc1ccccc1CSc1[nH]c(=O)cc2CCCCc12 50356460Fc1ccc(cc1CSc1[nH]c(=O)c(C#N)c2CCCCc12)C#N 50356461Clc1cccc(Cl)c1CSc1[nH]c(=O)c(C#N)c2CCCCc12 50356462O=c1[nH]c(SCc2ccccc2C#N)c2CCCCc2c1C#N 50358118COc1cccc(-c2ccc(s2)C(=O)N(C)Cc2cccc(O)c2)c1F 50359991CC1(C)[C@H](CC[C@@]2(C)[C@H]1CC[C@]1(C)[C@@H]2C(=O)C=C2[C@@H]3C[C@](C)(CC[C@]3(C)CC[C@@]12C)C(O)=O)O[C@@H]1O[C@@H]([C@@H](O)[C@H](O[C@@H]2O[C@@H]([C@@H](O)[C@H](O)[C@H]2O)C(O)=O)[C@H]1O)C(O)=O 50371796Cc1ccccc1C(=O)Nc1ccc2nc(SCC(=O)NCc3ccccc3)sc2c1 50371797Oc1ccc(NC(=O)CN2C(=O)C3C(C2=O)C2(Br)c4ccccc4C3c3ccccc23)cc1 50371798COc1cc(\C=C2\S\C(NC2=O)=N/c2ccccc2Cl)ccc1OC(=O)c1ccccc1 50371801Cc1cc(NS(=O)(=O)c2ccc(NC(=O)c3ccc(cc3)C(=O)C(=O)c3ccccc3)cc2)nc(C)n1 50371802Brc1ccccc1C(=O)Nc1ccc2nc(SCC(=O)NCCc3ccccc3)sc2c1 50371804Cc1ccc(cc1)S(=O)(=O)N(CC(=O)Nc1ccc2OCOc2c1)c1ccccc1Cl 50371805Cc1ccc2oc(C(=O)c3ccccc3)c(-c3cnc-4c(COc5ccccc-45)c3)c2c1 50371806Cc1ccc(cc1)C(=O)COC(=O)C(Cc1ccccc1)N1C(=O)c2ccccc2C1=O 50371808CCOc1cc(\C=N\NC(=O)c2ccc(C)cc2OC)ccc1OC(=O)c1ccc(Cl)cc1 50371809COc1cccc(c1)C(=O)COC(=O)c1ccccc1NC(=O)c1ccccc1 50377712Cn1c(nnc1-c1ccccc1C(F)(F)F)-c1ccccc1OC(F)(F)F 50377713Cn1c(nnc1-c1ccccc1[N+]([O-])=O)-c1ccc(Cl)cc1Cl 50377714CCS(=O)(=O)CCCc1ccc(-c2nnc(-c3ccccc3C(F)(F)F)n2C)c(Cl)c1 50377715CCS(=O)(=O)CCCc1ccc(-c2nnc(-c3ccccc3C(F)(F)F)n2C)c(C)c1 50377716CCS(=O)(=O)CCc1ccc(-c2nnc(-c3ccccc3C(F)(F)F)n2C)c(C)c1 50377717Cn1c(nnc1-c1ccccc1Cl)-c1ccc(cc1)S(C)(=O)=O 50377718Cn1c(nnc1-c1ccccc1S(C)(=O)=O)-c1ccccc1Cl 50377719CCCCCc1ccc(cc1)-c1nnc(-c2ccccc2)n1C 50377720CCCCc1ccc(cc1)-c1nnc(-c2ccccc2)n1C 50377721CCCCCc1ccc(cc1)-c1nnc(-c2ccccc2Cl)n1C 50377722CCCCCc1ccc(cc1)-c1nnc(-c2ccccc2C(F)(F)F)n1C 50377723Cc1ccc2ccccc2c1-c1nnc(-c2ccccc2C(F)(F)F)n1C 50377724COc1c(ccc2ccc(Cl)cc12)-c1nnc(-c2ccccc2S(C)(=O)=O)n1C 50377725COc1c(cc(Cl)c2ccccc12)-c1nnc(-c2ccccc2C(F)(F)F)n1C 50377726Cn1c(nnc1-c1cc2ccccc2cc1Cl)-c1ccccc1C(F)(F)F 50377727Cn1c(nnc1-c1ccccc1C(F)(F)F)-c1ccc2ccc(Cl)cc2c1O 50377728COc1c(cc2ccccc2c1Cl)-c1nnc(-c2ccccc2C(F)(F)F)n1C 50377729Cc1ccc2ccc(cc2c1)-c1nnc(-c2ccccc2C(F)(F)F)n1C 50377730CNc1c(ccc2ccccc12)-c1nnc(-c2ccccc2C(F)(F)F)n1C 50377731Cn1c(nnc1-c1ccccc1C(F)(F)F)-c1ccc2ccccc2c1 50377732Cn1c(nnc1-c1ccccc1C(F)(F)F)-c1ccc2ccccc2c1F 50377733Cn1ccc2cc(ccc12)-c1nnc(-c2ccccc2)n1C 50377734Cn1ccc2c(cccc12)-c1nnc(-c2ccccc2)n1C 50377735Cn1c(nnc1-c1cccc2n(C)ccc12)-c1ccccc1C(F)(F)F 50377736Cn1c(nnc1-c1cccc2n(C)ccc12)-c1ccccc1Cl 50377737Cn1c(nnc1-c1cccc2n(C)ccc12)-c1ccc(O)cc1 50377738Cn1c(nnc1-c1ccccc1Cl)-c1ccc(Cl)c(Cl)c1 50377739Cn1c(nnc1-c1ccccc1C(F)(F)F)-c1cc(Cl)cc(Cl)c1 50377740Cn1c(nnc1-c1ccc(Cl)cc1Cl)-c1ccccc1 50377741Cn1c(nnc1-c1ccccc1C(F)(F)F)-c1ccccc1 50377742Cn1c(nnc1-c1ccccc1Cl)-c1ccc(cc1F)C(F)(F)F 50377743Cn1c(nnc1-c1ccc(Cl)cc1Cl)-c1ccccc1F 50377744Cn1c(nnc1-c1ccccc1C(F)(F)F)-c1ccc(Cl)cc1F 50377745Cn1c(nnc1-c1cccc(c1C(F)(F)F)C(F)(F)F)-c1ccccc1C(F)(F)F 50377746Cn1c(nnc1-c1ccccc1C(F)(F)F)-c1ccc(Cl)cc1Cl 50377747Cn1c(nnc1-c1ccccc1C(F)(F)F)-c1ccccc1C(F)(F)F 50377748Cn1c(nnc1-c1ccc(Cl)cc1Cl)-c1ccc(Cl)cc1Cl 50377749Cn1c(nnc1-c1ccccc1Cl)-c1ccccc1Cl 50377750Cn1c(nnc1-c1ccccc1Br)-c1ccccc1Cl 50377751Cn1c(nnc1-c1ccccc1C(F)(F)F)-c1ccccc1Cl 50377752Cn1c(nnc1-c1ccc(Cl)cc1Cl)-c1ccc(Cl)cc1 50377753Cn1c(nnc1-c1ccccc1Cl)-c1ccccc1 50377754Cn1c(nnc1-c1ccccc1C(F)(F)F)-c1cccc(F)c1F 50377755Cn1c(nnc1-c1ccc(F)cc1Cl)-c1ccccc1Cl 50377756Cn1c(nnc1-c1ccccc1C(F)(F)F)-c1ccccc1Br 50377757Cn1c(nnc1-c1ccccc1C(F)(F)F)-c1ccc(F)cc1Cl 50377864FC(F)(F)c1ccc(cc1)C1(CCC1)c1nnc2CCCCCCn12 50377865Cc1ccc(cc1)C1(CCC1)c1nnc2CCCCCCn12 50377866Cc1cccc(c1)C1(CCC1)c1nnc2CCCCCCn12 50377867Fc1ccc(cc1)C1(CCC1)c1nnc2CCCCCCn12 50377868Fc1cccc(c1)C1(CCC1)c1nnc2CCCCCCn12 50377869C1CC(C1)(c1nnc2CCCCCCn12)c1ccccc1 50377870Cc1ccc(cc1)C1(CCCC1)c1nnc2CCCCCCn12 50377871Oc1cccc(c1)C1(CCCC1)c1nnc2CCCCCCn12 50377872Clc1ccc(cc1)C1(CCCC1)c1nnc2CCCCCCn12 50377873Fc1ccc(cc1)C1(CCCC1)c1nnc2CCCCCCn12 50377874C1CCC(C1)(c1nnc2CCCCCCn12)c1ccccc1 50377875Cc1ccc(cc1)C1(CCCCC1)c1nnc2CCCCCCn12 50377876Clc1ccc(cc1)C1(CCCCC1)c1nnc2CCCCCCn12 50377877C1CCC(CC1)(c1nnc2CCCCCCn12)c1ccccc1 50377878Cc1ccc(cc1)C1(CC1)c1nnc2CCCCCCn12 50377879FC(F)(F)c1ccccc1C1(CCC1)c1nnc2CCCCCCn12 50377880Cc1ccccc1C1(CCC1)c1nnc2CCCCCCn12 50377881Fc1ccccc1C1(CCC1)c1nnc2CCCCCCn12 50377882Cc1cccc(c1)C1(CCCC1)c1nnc2CCCCCCn12 50377883Fc1ccccc1C1(CCCC1)c1nnc2CCCCCCn12 50377884Clc1ccc(c(Cl)c1)C1(CC1)c1nnc2CCCCCCn12 50377885C1CC1(c1nnc2CCCCCCn12)c1ccccc1 50377886Clc1ccc(cc1)C1(CC1)c1nnc2CCCCCCn12 50377887F[C@H]1C[C@](C1)(c1nnc(C2CC2)n1C1CC1)c1ccc(Cl)cc1 50377888F[C@H]1C[C@@](C1)(c1nnc(C2CC2)n1C1CC1)c1ccc(Cl)cc1 50377889FC1(F)CC(C1)(c1nnc(C2CC2)n1C1CC1)c1ccc(Cl)cc1 50377890Fc1ccc(cc1)C1(CCCCC1)c1nnc2CCCCCCn12 50382382CC(C)[C@]1(C)SC(N[C@H]2C[C@H]3C[C@@H]2C[C@@H]3O)=NC1=O 50382383CC(C)[C@]1(C)SC(N[C@H]2C[C@H]3C[C@@H]2C[C@H]3O)=NC1=O 50382384CC(C)[C@]1(C)SC(N[C@H]2C[C@@H]3C[C@@H](O)[C@H]2C3)=NC1=O 50382385C[C@]1(SC(N[C@H]2C[C@@H]3CC[C@H]2C3)=NC1=O)[C@@H](O)CO 50382386C[C@]1(SC(N[C@H]2C[C@@H]3CC[C@H]2C3)=NC1=O)[C@H](O)CO 50382387CC(O)(O)[C@]1(C)SC(N[C@H]2C[C@@H]3CC[C@H]2C3)=NC1=O 50382388CC(=C)[C@]1(C)SC(N[C@H]2C[C@@H]3CC[C@H]2C3)=NC1=O 50382389CC(C)[C@]1(C)SC(N[C@H]2C[C@H]3C[C@@H]2CC3=O)=NC1=O 50382815CN(C(=O)c1ccc(CN2C(=O)Nc3ccc(Cl)cc3S2(=O)=O)cc1)C12CC3CC(CC(C3)C1)C2 50382816Clc1ccc2NC(=O)N(Cc3cccc(c3)C(=O)N(C3CC3)C3CCCCC3)S(=O)(=O)c2c1 50382817Clc1ccc2NC(=O)N(Cc3cccc(c3)C(=O)N(C3CC3)C3CCCCCC3)S(=O)(=O)c2c1 50382818CN(C1C2CC3CC(C2)CC1C3)C(=O)c1cccc(CN2C(=O)Nc3ccc(Cl)cc3S2(=O)=O)c1 50382819Clc1ccc2NC(=O)N(CC3CCN(CC3)C(=O)N(C3CC3)C3CCCCC3)S(=O)(=O)c2c1 50382820CN(C1CCCCCC1)C(=O)N1CCC(CN2C(=O)Nc3ccc(Cl)cc3S2(=O)=O)CC1 50382821Clc1ccc2NC(=O)N(CC3CCN(CC3)C(=O)N(C3CC3)C3CCCCCC3)S(=O)(=O)c2c1 50382822CN(C1C2CC3CC(C2)CC1C3)C(=O)N1CCC(CN2C(=O)Nc3ccc(Cl)cc3S2(=O)=O)CC1 50382823Clc1ccc2NC(=O)N(Cc3ccc(cc3)C(=O)NC3CCCCC3)S(=O)(=O)c2c1 50382824Clc1ccc2NC(=O)N(Cc3ccc(cc3)C(=O)NC3CCCCCC3)S(=O)(=O)c2c1 50382825Clc1ccc2NC(=O)N(Cc3ccc(cc3)C(=O)NC3CCCCCCC3)S(=O)(=O)c2c1 50382826Clc1ccc2NC(=O)N(Cc3ccc(cc3)C(=O)N(C3CC3)C3CCCCC3)S(=O)(=O)c2c1 50382827CN(C1CCCCCC1)C(=O)c1ccc(CN2C(=O)Nc3ccc(Cl)cc3S2(=O)=O)cc1 50382828Clc1ccc2NC(=O)N(Cc3ccc(cc3)C(=O)N(C3CC3)C3CCCCCC3)S(=O)(=O)c2c1 50382829Clc1ccc2NC(=O)N(Cc3ccc(cc3)C(=O)NC34CC5CC(CC(C5)C3)C4)S(=O)(=O)c2c1 50382830CN(C1CCCCCC1)C(=O)c1cccc(CN2C(=O)Nc3ccc(Cl)cc3S2(=O)=O)c1 50382831Clc1ccc2NC(=O)N(CC3CCN(CC3)C(=O)NC3CCCCCC3)S(=O)(=O)c2c1 50384518NC(=O)[C@@]12CC3CC(C1)[C@H](NC(=O)CN1CCCN(c4c(Cl)cc(Cl)cc4Cl)S1(=O)=O)C(C3)C2 50384519NC(=O)[C@@]12CC3CC(C1)[C@H](NC(=O)CN1CCCCN(c4c(Cl)cc(Cl)cc4Cl)S1(=O)=O)C(C3)C2 50384520CN(CC(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)C(N)=O)S(=O)(=O)N(C)c1c(Cl)cc(Cl)cc1Cl 50384521CC1CCN(c2c(Cl)cc(Cl)cc2Cl)S(=O)(=O)N1CC(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)C(N)=O 50384522CC1CN(CC(=O)N[C@H]2C3CC4CC2C[C@](C4)(C3)C(N)=O)S(=O)(=O)N(C1)c1c(Cl)cc(Cl)cc1Cl 50384523NC(=O)[C@@]12CC3CC(C1)[C@H](NC(=O)CN1CC(=C)CN(c4c(Cl)cc(Cl)cc4Cl)S1(=O)=O)C(C3)C2 50384524NC(=O)[C@@]12CC3CC(C1)[C@H](NC(=O)CN1CC4(CC4)CN(c4c(Cl)cc(Cl)cc4Cl)S1(=O)=O)C(C3)C2 50384525CC1(C)CN(CC(=O)N[C@H]2C3CC4CC2C[C@](C4)(C3)C(N)=O)S(=O)(=O)N(C1)c1c(Cl)cc(Cl)cc1Cl 50384526CC(C)(C)OC(=O)N1CCCN(CC(=O)NC2C3CC4CC(C3)CC2C4)S1(=O)=O 50384527O=C(CN1CCCN(Cc2ccccc2)S1(=O)=O)NC1C2CC3CC(C2)CC1C3 50384528O=C(CN1CCCN(CCc2ccccc2)S1(=O)=O)NC1C2CC3CC(C2)CC1C3 50384529O=C(CN1CCCN(c2ccccc2)S1(=O)=O)NC1C2CC3CC(C2)CC1C3 50384530O=C(CN1CCCN(c2ccccc2)S1(=O)=O)NC12CC3CC(CC(C3)C1)C2 50384531NC(=O)[C@@]12CC3CC(C1)[C@H](NC(=O)CN1CCCN(c4ccccc4)S1(=O)=O)C(C3)C2 50384532NC(=O)[C@@]12CC3CC(C1)[C@H](NC(=O)CN1CCCN(c4ccccc4F)S1(=O)=O)C(C3)C2 50384533NC(=O)[C@@]12CC3CC(C1)[C@H](NC(=O)CN1CCCN(c4cccc(F)c4)S1(=O)=O)C(C3)C2 50384535NC(=O)[C@@]12CC3CC(C1)[C@H](NC(=O)CN1CCCN(c4c(F)cc(F)cc4F)S1(=O)=O)C(C3)C2 50384536NC(=O)[C@@]12CC3CC(C1)[C@H](NC(=O)CN1CCN(c4c(Cl)cc(Cl)cc4Cl)S1(=O)=O)C(C3)C2 50384886C[C@H](CC[C@H](O)C(C)=C)[C@H]1CC[C@]2([C@@H]3CC[C@@H]4[C@]5(C[C@@]35CC[C@]12C)CCC(=O)C4(C)C)C(O)=O 50384887C[C@H](CC[C@@H](O)C(C)(C)O)[C@H]1CC[C@]2([C@@H]3CC[C@@H]4[C@]5(C[C@@]35CC[C@]12C)CC[C@H](O)C4(C)C)C(O)=O 50385022CC(C)N(c1ccc(cc1)C(C)(O)C(F)(F)F)S(=O)(=O)c1cccc(Cl)c1 50385023CC(O)(c1ccc(cc1)N(C1CCC1)S(=O)(=O)c1ccccc1Cl)C(F)(F)F 50385024CC(C)N(c1ccc(cc1)C(C)(O)C(F)(F)F)S(=O)(=O)c1cc(C)ccc1Cl 50385025CC(C)N(c1ccc(cc1)C(C)(O)C(F)(F)F)S(=O)(=O)c1cc(ccc1Cl)C(F)(F)F 50385026CC(C)N(c1ccc(cc1)C(C)(O)C(F)(F)F)S(=O)(=O)c1cc(ccc1Cl)C1CC1 50385027CC(O)(c1ccc(cc1)N(C1CC1)S(=O)(=O)c1ccccc1Cl)C(F)(F)F 50385028CC(C)(C)N(c1ccc(cc1)C(C)(O)C(F)(F)F)S(=O)(=O)c1ccccc1Cl 50385029CC(O)(c1ccc(cc1)N(C1CCCC1)S(=O)(=O)c1ccccc1Cl)C(F)(F)F 50385030CC(O)(c1ccc(cc1)N(CC1CC1)S(=O)(=O)c1ccccc1Cl)C(F)(F)F 50385031CC(C)CN(c1ccc(cc1)C(C)(O)C(F)(F)F)S(=O)(=O)c1ccccc1Cl 50385032CC(O)(c1ccc(cc1)N(C(CF)CF)S(=O)(=O)c1ccccc1Cl)C(F)(F)F 50385033CC(O)(c1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)c1ccccc1Cl)C(F)(F)F 50385034CC(O)(c1ccc(cc1)N(c1ccccc1)S(=O)(=O)c1ccccc1Cl)C(F)(F)F 50385035CC(C)N(c1ccc(cc1)[C@](C)(O)C(F)(F)F)S(=O)(=O)c1ccccc1Cl 50385036CC(C)N(c1ccc(cc1)[C@@](C)(O)C(F)(F)F)S(=O)(=O)c1ccccc1Cl 50385037CC(C)N(c1ccc(cc1)[C@](C)(O)C(F)(F)F)S(=O)(=O)c1cc(Cl)ccc1Cl 50385038CC(C)N(c1ccc(cc1)[C@@](C)(O)C(F)(F)F)S(=O)(=O)c1cc(Cl)ccc1Cl 50385039CC(C)N(c1ccc(cc1)C(C)(O)C(F)(F)F)S(=O)(=O)c1ccccc1Br 50385040CC(C)N(c1ccc(cc1)C(C)(O)C(F)(F)F)S(=O)(=O)c1ccccc1F 50385041CC(C)N(c1ccc(cc1)C(C)(O)C(F)(F)F)S(=O)(=O)c1ccccc1C#N 50385042CC(C)N(c1ccc(cc1)C(C)(O)C(F)(F)F)S(=O)(=O)c1ccccc1C(F)(F)F 50385043CC(C)N(c1ccc(cc1)C(C)(O)C(F)(F)F)S(=O)(=O)c1ccccc1[N+]([O-])=O 50385044CC(C)N(c1ccc(cc1)C(C)(O)C(F)(F)F)S(=O)(=O)c1ccccc1C1CC1 50385045CC(C)N(c1ccc(cc1)C(C)(O)C(F)(F)F)S(=O)(=O)c1ccccc1S(C)(=O)=O 50385046CC(C)N(c1ccc(cc1)C(C)(O)C(F)(F)F)S(=O)(=O)c1ccccc1C 50385047CC(C)N(c1ccc(cc1)C(C)(O)C(F)(F)F)S(=O)(=O)c1cccc(Cl)c1Cl 50385048CC(C)N(c1ccc(cc1)C(C)(O)C(F)(F)F)S(=O)(=O)c1cc(ccc1Cl)[N+]([O-])=O 50385049CC(C)N(c1ccc(cc1)C(C)(O)C(F)(F)F)S(=O)(=O)c1cc(N)ccc1Cl 50385050CC(C)N(c1ccc(cc1)C(C)(O)C(F)(F)F)S(=O)(=O)c1cc(NC(C)=O)ccc1Cl 50385051CC(C)N(c1ccc(cc1)C(C)(O)C(F)(F)F)S(=O)(=O)c1cc(Br)ccc1Cl 50385052CC(C)N(c1ccc(cc1)C(C)(O)C(F)(F)F)S(=O)(=O)c1ccccc1 50385054CCN(c1ccc(cc1)C(C)(O)C(F)(F)F)S(=O)(=O)c1ccccc1 50385055CC(C)N(c1ccc(cc1)C(C)(O)C(F)(F)F)S(=O)(=O)c1ccc(Cl)cc1 50385056CC(C)N(c1ccc(cc1)C(C)(O)C(F)(F)F)S(=O)(=O)c1ccc(Cl)cc1Cl 50385057CC(C)N(c1ccc(cc1)C(C)(O)C(F)(F)F)S(=O)(=O)c1c(Cl)cccc1Cl 50390692COc1ccc(C(=O)N2CCC(C2)c2c[nH]c3ccccc23)c(C)c1 50390693COc1ccc(C(=O)N2CCC(C2)c2c[nH]c3ccc(F)cc23)c(C)c1 50390694Fc1ccc2[nH]cc(C3CCN(C3)C(=O)C3CCCCC3)c2c1 50390695Cc1ccccc1C(=O)N1CCC(C1)c1c[nH]c2ccc(F)cc12 50390696O=C(N1CCC(C1)c1c[nH]c2ccccc12)C1(CC1)c1ccccc1 50390697Fc1ccc2[nH]cc(C3CCN(C3)C(=O)C3(CC3)c3ccccc3)c2c1 50390698Cc1ccccc1C(=O)N1CCC(C1)c1c[nH]c2ncccc12 50390699CC(C)(C(=O)N1CCC(C1)c1c[nH]c2ncccc12)c1ccccc1 50390700O=C(N1CCC(C1)c1c[nH]c2ncccc12)C1(CC1)c1ccccc1 50390701Clc1ccc(cc1)C1(CC1)C(=O)N1CCC(C1)c1c[nH]c2ncccc12 50390702CC(C)(C(=O)N1CCC(C1)c1c[nH]c2ncccc12)c1ccc(Cl)cc1 50390703Clc1ccc(cc1)C1(CCC1)C(=O)N1CCC(C1)c1c[nH]c2ncccc12 50390704CC(C)(Oc1ccccc1)C(=O)N1CCC(C1)c1c[nH]c2ncccc12 50390705Fc1ccc(OC2(CC2)C(=O)N2CCC(C2)c2c[nH]c3ncccc23)cc1 50390706Fc1ccc(cc1)C1(CC1)C(=O)N1CCC2(CC12)c1c[nH]c2ncccc12 50390707Fc1ccc(cc1)C1(CC1)C(=O)N1CC2CC2(C1)c1c[nH]c2ncccc12 50390708Cc1[nH]c2ncccc2c1C1CCN(C1)C(=O)C1(CC1)c1ccccn1 50390709Cc1[nH]c2ncccc2c1C1CCN(C1)C(=O)C(C)(C)c1ccc(Cl)cc1 50390710Cc1[nH]c2ncccc2c1C1CCN(C1)C(=O)C1(CC1)c1ccc(F)cc1 50390711Fc1ccc(cc1)C1(CC1)C(=O)N1CCC(C1)c1c[nH]c2ncc(F)cc12 50390712Fc1ccc(cc1)C1(CC1)C(=O)N1CCC(C1)c1c[nH]c2cnccc12 50390713Fc1ccc(cc1)C1(CC1)C(=O)N1CCC(C1)c1c[nH]c2ncccc12 50392216CCCSc1nc(ccc1C(=O)NC1CCCCC1)N1CCC[C@@H](CC(O)=O)C1 50392217CCCSc1ncccc1C(=O)NC1CCCCC1 50392218Fc1cccc(F)c1CS(=O)(=O)N1CCN(CC1)c1ncccc1C(F)(F)F 50392219CCCSc1ncccc1C(=O)N(C)C1CCCCC1 50392220CCCSc1ncccc1C(=O)NC1CCC(F)(F)CC1 50392221CCCSc1ncccc1C(=O)N(C)C1CCOCC1 50392222CCCSc1ncccc1C(=O)N[C@H]1[C@H]2CC3C[C@@H]1C[C@](O)(C3)C2 50392223CCCSc1ncccc1C(=O)N(C)[C@H]1[C@H]2CC3C[C@@H]1C[C@](O)(C3)C2 50392224CCCSc1ncccc1C(=O)N(C)[C@@H]1[C@H]2CC3C[C@@H]1C[C@](O)(C3)C2 50392225CCCSc1ncccc1C(=O)N1CCCC1c1ccncc1 50392227CCCSc1nc(N[C@H]2CC[C@@H](CC2)C(O)=O)ccc1C(=O)NC1CCCCC1 50392228CCCSc1nc(NC[C@H]2CC[C@@H](CC2)C(O)=O)ccc1C(=O)NC1CCCCC1 50392229CCCSc1nc(Oc2ccc(CC(O)=O)cc2)ccc1C(=O)NC1CCCCC1 50392230CCCSc1nc(Oc2cccc(CCC(O)=O)c2)ccc1C(=O)NC1CCCCC1 50392231CCCSc1nc(ccc1C(=O)NC1CCCCC1)N1CCCCC1C(O)=O 50392232CCCSc1nc(ccc1C(=O)NC1CCCCC1)N1CCCC(C1)C(O)=O 50392233CCCSc1nc(ccc1C(=O)NC1CCCCC1)N1CCC(CC1)C(O)=O 50392234CCCSc1nc(ccc1C(=O)NC1CCCCC1)N1CCC[C@H](CC(O)=O)C1 50392235CCCSc1nc(ccc1C(=O)NC1CCCCC1)N1CCC(CC(O)=O)CC1 50392236CCCOc1nc(ccc1C(=O)NC1CCCCC1)N1CCC[C@@H](CC(O)=O)C1 50392237CCCNc1nc(ccc1C(=O)NC1CCCCC1)N1CCC[C@@H](CC(O)=O)C1 50392238CCCN(C)c1nc(ccc1C(=O)NC1CCCCC1)N1CCC[C@@H](CC(O)=O)C1 50392239CCCCc1nc(ccc1C(=O)NC1CCCCC1)N1CCC[C@@H](CC(O)=O)C1 50392919Cc1c(Cl)cccc1S(=O)(=O)N1CCC[C@@H](C1)C(=O)N[C@H]1C[C@H]2CC[C@]1(C)C2(C)C 50392920Cc1c(Cl)cccc1S(=O)(=O)N1CCC[C@@H]1C(=O)NC1CCCCC1 50392921Cc1c(Cl)cccc1S(=O)(=O)N1CCC[C@]1(C)C(=O)NC1CCCCC1 50392922Cc1c(Cl)cccc1S(=O)(=O)N1CCC[C@]1(C)C(=O)N[C@H]1CC[C@H](O)CC1 50392923Cc1c(Cl)cccc1S(=O)(=O)N1CCC[C@]1(C)C(=O)NC1C2CC3CC(C2)CC1C3 50392924Cc1c(Cl)cccc1S(=O)(=O)N1CCC[C@]1(C)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50392925COC(=O)[C@H]1CC2COCC(C1)[C@H]2NC(=O)[C@@]1(C)CCCN1S(=O)(=O)c1cccc(Cl)c1C 50392926Cc1c(Cl)cccc1S(=O)(=O)N1CCC[C@@]1(C)C(=O)NC1CCCCC1 50392927Cc1c(Cl)cccc1S(=O)(=O)N1CCC[C@@]1(C)C(=O)N[C@H]1CC[C@H](O)CC1 50392928Cc1c(Cl)cccc1S(=O)(=O)N1CCC[C@@]1(C)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50392929COc1ccc(cc1OC)S(=O)(=O)N1CCC[C@]1(C)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50392930CC(C)(C)c1ccc(cc1)S(=O)(=O)N1CCC[C@]1(C)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50392931C[C@@]1(CCCN1S(=O)(=O)c1ccc(cc1Cl)C#N)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50392932C[C@@]1(CCCN1S(=O)(=O)c1ccccc1C#N)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50392933CC(=O)c1ccc(cc1)S(=O)(=O)N1CCC[C@]1(C)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50392934C[C@@]1(CCCN1S(=O)(=O)c1ccc(cc1)-c1ccccc1)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50392935C[C@@]1(CCCN1S(=O)(=O)c1cccnc1)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50392936C[C@@]1(CCCN1S(=O)(=O)c1cccs1)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50392937C[C@@]1(CCCN1S(=O)(=O)c1ccc(Br)s1)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50392938C[C@@]1(CCCN1S(=O)(=O)c1cccc2cccnc12)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50392939CN(C)c1cccc2c(cccc12)S(=O)(=O)N1CCC[C@]1(C)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50392940CC(O)(c1ccc(cc1)S(=O)(=O)N1CCC[C@]1(C)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2)C(F)(F)F 50392941CC(O)(c1ccc(cc1)S(=O)(=O)N1CCC[C@]1(C)C(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)C#N)C(F)(F)F 50392942COC(=O)[C@@]12CC3CC(C1)[C@H](NC(=O)[C@@]1(C)CCCN1S(=O)(=O)c1ccc(cc1)C(C)(O)C(F)(F)F)C(C3)C2 50392943CC[C@@]1(CCCN1S(=O)(=O)c1cccc2cccnc12)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50394000O[C@@]12CC3CC(C1)[C@H](NC(=O)c1ccc(nc1C1CC1)N1CCOCC1)C(C3)C2 50394001CCCOc1nc(ccc1C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2)N1CCOCC1 50394002Cc1nc(ncc1C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2)N1CCOCC1 50394003CC(C)(C)c1nc(ncc1C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2)N1CCOCC1 50394004O[C@@]12CC3CC(C1)[C@H](NC(=O)c1cnc(nc1C1CC1)N1CCOCC1)C(C3)C2 50394005O[C@@]12CC3CC(C1)[C@H](NC(=O)c1cnc(nc1C1CCC1)N1CCOCC1)C(C3)C2 50394006O[C@@]12CC3CC(C1)[C@H](NC(=O)c1cnc(nc1C1CCCC1)N1CCOCC1)C(C3)C2 50394007O[C@@]12CC3CC(C1)[C@H](NC(=O)c1cnc(nc1C1CCCCC1)N1CCOCC1)C(C3)C2 50394008CC1(CC1)c1nc(ncc1C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2)N1CCOCC1 50394009CCCOc1nc(ncc1C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2)N1CCOCC1 50394010CCCSc1ncncc1C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50394011CCCSc1nc(C)ccc1C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50394012CCCSc1nc(C)ncc1C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50394013CCCSc1nc(NC)ccc1C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50394014CCCSc1nc(NC)ncc1C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50394015CCCSc1nc(ccc1C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2)N(C)C 50394016CCCSc1nc(ncc1C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2)N(C)C 50394017CCCSc1nc(ccc1C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2)N1CCOCC1 50394018CCCSc1nc(ncc1C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2)N1CCOCC1 50394019CCCCc1nc(C)ncc1C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50394021CC(C)Cc1nc(C)ncc1C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50394022Cc1ncc(C(=O)N[C@H]2C3CC4CC2C[C@](O)(C4)C3)c(CC2CC2)n1 50394023Cc1ncc(C(=O)N[C@H]2C3CC4CC2C[C@](O)(C4)C3)c(CC2CCCC2)n1 50394025Cc1ncc(C(=O)N[C@H]2C3CC4CC2C[C@](O)(C4)C3)c(n1)C1CC1 50394026Cc1ncc(C(=O)N[C@H]2C3CC4CC2C[C@](O)(C4)C3)c(n1)C1CCCC1 50394027Cc1ccc(C(=O)N[C@H]2C3CC4CC2C[C@](O)(C4)C3)c(n1)C1CC1 50394421CN(Cc1cccs1)C(=O)C1(CCCC1)c1ccc(Cl)cc1 50394422CN(Cc1cccs1)C(=O)C1(CCC1)c1ccc(Cl)cc1 50394423CN(Cc1cccs1)C(=O)C1(CC1)c1ccc(Cl)cc1 50394424CN(Cc1cccs1)C(=O)C1(CC1)c1ccc(C)cc1 50394425CN(Cc1cccs1)C(=O)C1(C)CCCCC1 50394426CN(Cc1cccs1)C(=O)C12CC3CC1CC(C2)C3 50394427Cn1cccc1CNC(=O)CC12CC3CC(CC(C3)C1)C2 50394428CN(Cc1cccn1C)C(=O)CC12CC3CC(CC(C3)C1)C2 50394429CN(Cc1ccsc1)C(=O)CC12CC3CC(CC(C3)C1)C2 50394430CN(Cc1cccs1)C(=O)CC12CC3CC(CC(C3)C1)C2 50394431O=C(NCCc1ccccn1)C12CC3CC(CC(C3)C1)C2 50394432CN(CCc1ccccn1)C(=O)C12CC3CC(CC(C3)C1)C2 50394433O=C(NCCc1cccs1)C12CC3CC(CC(C3)C1)C2 50394434CN(CCc1cccs1)C(=O)C12CC3CC(CC(C3)C1)C2 50394435CN(Cc1cccc(N)c1)C(=O)C12CC3CC(CC(C3)C1)C2 50394436Cn1cccc1CNC(=O)C12CC3CC(CC(C3)C1)C2 50394437CN(Cc1cccn1C)C(=O)C12CC3CC(CC(C3)C1)C2 50394438CN(Cc1ccco1)C(=O)C12CC3CC(CC(C3)C1)C2 50394439CN(Cc1ccsc1)C(=O)C12CC3CC(CC(C3)C1)C2 50394440CN(Cc1sccc1C)C(=O)C12CC3CC(CC(C3)C1)C2 50394441O=C(NCc1cccs1)C12CC3CC(CC(C3)C1)C2 50394442CN(Cc1cccs1)C(=O)C12CC3CC(CC(C3)C1)C2 50399335CC(C)(C)c1c(cnn1-c1ccc(cc1)C(O)=O)C(=O)NC1C2CC3CC(C2)CC1C3 50399336CC1(CC1)c1c(cnn1-c1ccc(cc1)C(O)=O)C(=O)NC1C2CC3CC(C2)CC1C3 50399337OC(=O)c1ccc(cc1)-n1ncc(C(=O)NC2C3CC4CC(C3)CC2C4)c1C(F)(F)F 50399338OC(=O)c1ccc(cc1)-n1ncc(C(=O)NC2C3CC4CC(C3)CC2C4)c1C1CCCC1 50399339OC(=O)c1ccc(cc1)-n1ncc(C(=O)NC2C3CC4CC(C3)CC2C4)c1C1CCC1 50399340OC(=O)c1ccc(cc1)-n1ncc(C(=O)NC2C3CC4CC(C3)CC2C4)c1C1CC1 50399341CC(C)c1c(cnn1-c1ccc(cc1)C(O)=O)C(=O)NC1C2CC3CC(C2)CC1C3 50399342CCc1c(cnn1-c1ccc(cc1)C(O)=O)C(=O)NC1C2CC3CC(C2)CC1C3 50399343Cc1c(cnn1-c1ccc(cc1)C(O)=O)C(=O)NC1C2CC3CC(C2)CC1C3 50399344OC(=O)c1ccc(cc1)-n1cc(cn1)C(=O)NC1C2CC3CC(C2)CC1C3 50399345OC(=O)c1ccc(cc1)-n1ncc(C(=O)NC2C3CC4CC(C3)CC2C4)c1SC1CCCCC1 50399346OC(=O)c1ccc(cc1)-n1ncc(C(=O)NC2C3CC4CC(C3)CC2C4)c1SC1CCCC1 50399347CSc1c(cnn1-c1ccc(cc1)C(O)=O)C(=O)NC1C2CC3CC(C2)CC1C3 50399348CCSc1c(cnn1-c1ccc(cc1)C(O)=O)C(=O)NC1C2CC3CC(C2)CC1C3 50399349CCCSc1c(cnn1-c1ccc(cc1)C(O)=O)C(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)S(C)(=O)=O 50399350CCCSc1c(cnn1-c1ccc(cc1)C(O)=O)C(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)OC(F)F 50399351CCCSc1c(cnn1-c1ccc(cc1)C(O)=O)C(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)OC 50399352CCCSc1c(cnn1-c1ccc(cc1)C(O)=O)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50399353CCCSc1c(cnn1-c1ccc(cc1)C(O)=O)C(=O)NC1C2CC3CC(C2)CC1C3 50399354CCCSc1c(cnn1-c1ccc(cc1)C(O)=O)C(=O)N(C)C1CCCCC1 50399355CCCSc1c(cnn1-c1cccc(c1)C(O)=O)C(=O)NC1CCCCC1 50399356CCCSc1c(cnn1-c1ccc(cc1)C(O)=O)C(=O)NC1CCCCC1 50399357CCCSc1c(cnn1[C@H]1CC[C@@H](CC1)C(O)=O)C(=O)NC1CCCCC1 50399358CCCSc1c(cnn1[C@@H]1CC[C@@H](CC1)C(O)=O)C(=O)NC1CCCCC1 50399359CCCSc1c(cnn1C)C(=O)NC1CCCCC1 50400135O[C@@]12CC3CC(C1)[C@H](NC(=O)c1cnc(NC4CCS(=O)(=O)CC4)nc1C1CCC1)C(C3)C2 50400136O[C@@]12CC3CC(C1)[C@H](NC(=O)c1cnc(NC4CCOCC4)nc1C1CCC1)C(C3)C2 50400137O[C@@]12CC3CC(C1)[C@H](NC(=O)c1cnc(N[C@H]4CCOC4)nc1C1CCC1)C(C3)C2 50400138O[C@@]12CC3CC(C1)[C@H](NC(=O)c1cnc(N[C@@H]4CCOC4)nc1C1CCC1)C(C3)C2 50400139CC(C)(O)CNc1ncc(C(=O)N[C@H]2C3CC4CC2C[C@](O)(C4)C3)c(n1)C1CC1 50400140CC(C)(CO)Nc1ncc(C(=O)N[C@H]2C3CC4CC2C[C@](O)(C4)C3)c(n1)C1CC1 50400141O[C@@]12CC3CC(C1)[C@H](NC(=O)c1cnc(NC4CCOCC4)nc1C1CC1)C(C3)C2 50400142O[C@@]12CC3CC(C1)[C@H](NC(=O)c1cnc(N[C@H]4CCOC4)nc1C1CC1)C(C3)C2 50400143O[C@@]12CC3CC(C1)[C@H](NC(=O)c1cnc(N[C@@H]4CCOC4)nc1C1CC1)C(C3)C2 50400144O[C@@]12CC3CC(C1)[C@H](NC(=O)c1cnc(NC4COC4)nc1C1CC1)C(C3)C2 50400145O[C@@]12CC3CC(C1)[C@H](NC(=O)c1cnc(N[C@H]4CCNC4=O)nc1C1CCCC1)C(C3)C2 50400146O[C@@H]1CCC[C@@H]1Nc1ncc(C(=O)N[C@H]2C3CC4CC2C[C@](O)(C4)C3)c(n1)C1CCCC1 50400147O[C@@]12CC3CC(C1)[C@H](NC(=O)c1cnc(N[C@H]4CCOC4)nc1C1CCCC1)C(C3)C2 50400148O[C@@]12CC3CC(C1)[C@H](NC(=O)c1cnc(N[C@@H]4CCOC4)nc1C1CCCC1)C(C3)C2 50400149O[C@@]12CC3CC(C1)[C@H](NC(=O)c1cnc(NC4COC4)nc1C1CCCC1)C(C3)C2 50400150CC(C)(O)CNc1ncc(C(=O)N[C@H]2C3CC4CC2C[C@](O)(C4)C3)c(n1)C1CCC1 50400151OCCNc1ncc(C(=O)N[C@H]2C3CC4CC2C[C@](O)(C4)C3)c(n1)C1CCC1 50400152CC(C)(CO)Nc1ncc(C(=O)N[C@H]2C3CC4CC2C[C@](O)(C4)C3)c(OC2CCC2)n1 50400153OCCNc1ncc(C(=O)N[C@H]2C3CC4CC2C[C@](O)(C4)C3)c(OC2CCC2)n1 50400154O[C@@]12CC3CC(C1)[C@H](NC(=O)c1cnc(NC4CCS(=O)(=O)CC4)nc1OC1CCC1)C(C3)C2 50400155O[C@@]12CC3CC(C1)[C@H](NC(=O)c1cnc(NC4CCOCC4)nc1OC1CCC1)C(C3)C2 50400156O[C@@]12CC3CC(C1)[C@H](NC(=O)c1cnc(N[C@H]4CCOC4)nc1OC1CCC1)C(C3)C2 50400157O[C@@]12CC3CC(C1)[C@H](NC(=O)c1cnc(N[C@@H]4CCOC4)nc1OC1CCC1)C(C3)C2 50400158O[C@@]12CC3CC(C1)[C@H](NC(=O)c1cnc(NC4COC4)nc1OC1CCC1)C(C3)C2 50400159CC(C)Oc1nc(N[C@H]2CCOC2)ncc1C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50400160CC(C)Oc1nc(N[C@@H]2CCOC2)ncc1C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50400161CC(C)Oc1nc(NC2COC2)ncc1C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50400162CC(C)(O)CNc1ncc(C(=O)N[C@H]2C3CC4CC2C[C@](O)(C4)C3)c(n1)C1CCCC1 50400163CN(C)C(=O)CNc1ncc(C(=O)N[C@H]2C3CC4CC2C[C@](O)(C4)C3)c(n1)C1CCCC1 50400164CC(C)(CO)Nc1ncc(C(=O)N[C@H]2C3CC4CC2C[C@](O)(C4)C3)c(n1)C1CCCC1 50400165C[C@@H](O)CNc1ncc(C(=O)N[C@H]2C3CC4CC2C[C@](O)(C4)C3)c(n1)C1CCCC1 50400166C[C@H](O)CNc1ncc(C(=O)N[C@H]2C3CC4CC2C[C@](O)(C4)C3)c(n1)C1CCCC1 50400167COCCNc1ncc(C(=O)N[C@H]2C3CC4CC2C[C@](O)(C4)C3)c(n1)C1CCCC1 50400168OCCNc1ncc(C(=O)N[C@H]2C3CC4CC2C[C@](O)(C4)C3)c(n1)C1CCCC1 50400169O[C@@]12CC3CC(C1)[C@H](NC(=O)c1cnc(NC[C@@H]4CNC(=O)C4)nc1C1CCCC1)C(C3)C2 50400170O[C@@]12CC3CC(C1)[C@H](NC(=O)c1cnc(NC[C@H]4CCCO4)nc1C1CCCC1)C(C3)C2 50400171O[C@@]12CC3CC(C1)[C@H](NC(=O)c1cnc(NC[C@@H]4CCCO4)nc1C1CCCC1)C(C3)C2 50400172O[C@@]12CC3CC(C1)[C@H](NC(=O)c1cnc(N[C@@H]4CCC(=O)NC4)nc1C1CCCC1)C(C3)C2 50400173O[C@@]12CC3CC(C1)[C@H](NC(=O)c1cnc(NC4CCS(=O)(=O)CC4)nc1C1CCCC1)C(C3)C2 50400174CC(=O)N1CCC(CC1)Nc1ncc(C(=O)N[C@H]2C3CC4CC2C[C@](O)(C4)C3)c(n1)C1CCCC1 50400175O[C@@]12CC3CC(C1)[C@H](NC(=O)c1cnc(NC4CCOCC4)nc1C1CCCC1)C(C3)C2 50400176CC(=O)N1CC[C@H](C1)Nc1ncc(C(=O)N[C@H]2C3CC4CC2C[C@](O)(C4)C3)c(n1)C1CCCC1 50411920Fc1ccc(CNc2ccc(cc2)C(=O)N2CCC[C@H]3CCCC[C@H]23)cc1 50411921O=C(Cc1ccccc1)Nc1ccc(cc1)C(=O)N1CCC[C@H]2CCCC[C@H]12 50411922Clc1ccc(cc1)C(=O)Nc1ccc(cc1)C(=O)N1CCC[C@H]2CCCC[C@H]12 50411923CCC1CCCCN1C(=O)c1ccc(NC(=O)c2ccc(Cl)cc2Cl)cc1 50411924CC1CCCCN1C(=O)c1ccc(NC(=O)c2ccc(Cl)cc2Cl)cc1 50411925CC(C)(C(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)C(N)=O)c1ccc(nc1)N1CCOCC1 50411926CC(C)(C(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)C(N)=O)c1ccc(cn1)C#N 50411927CC(C)(Oc1ccc(cn1)-n1cccn1)C(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)C(N)=O 50411928CC(C)(Oc1ccc(cn1)N1CCOCC1)C(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)C(N)=O 50411929CC(C)(Oc1ccc(cn1)C#N)C(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)C(N)=O 50411930CC(C)(Oc1ccc(Br)cn1)C(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)C(N)=O 50411931CC(C)(Oc1ccc(Cl)cc1)C(=O)N[C@H]1C2CC3CC1C[C@](Cc1nnc(N)[nH]1)(C3)C2 50411932Cn1c(cnc1C12CCC(CC1)(CC2)c1nnc([nH]1)-c1ccc(F)cc1)-c1ccccc1C(F)(F)F 50411933Cn1c(cnc1C12CCC(CC1)(CC2)c1nc(c[nH]1)-c1ccc(F)cc1)-c1ccccc1C(F)(F)F 50411934Cn1c(nnc1C12CCC(CC1)(CC2)c1nc(no1)-c1ccc(F)cc1)-c1ccc(C=O)cc1Cl 50411935Cn1c(nnc1C12CCC(CC1)(CC2)c1nc(no1)-c1ccc(F)cc1)-c1ccc(OC(F)F)cc1 50411936CCCCCC12CCC(CC1)(CC2)c1nnc2CCCCCn12 50411937CCCCn1c(C)nnc1C12CC3CC(CC(C3)C1)C2 50411938O=C(N1CCC[C@H]2CCCC[C@H]12)c1ccc(cc1)C(=O)N1CCCc2ccccc12 50411939Clc1ccccc1C(=O)Nc1ccc(cc1)C(=O)N1CCC[C@H]2CCCC[C@H]12 50411940CNc1ccc(cn1)C(C)(C)C(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)C(N)=O 50411941CN1CCN(CC1)c1ccc(OC(C)(C)C(=O)N[C@H]2C3CC4CC2C[C@](C4)(C3)C(N)=O)nc1 50411942CC(C)(Oc1ccc(Cl)cc1)C(=O)N[C@H]1C2CC3CC1C[C@](Cc1ncc[nH]1)(C3)C2 50411943CC(C)(Oc1ccc(cn1)C#N)C(=O)N[C@@H]1C2COCC1C[C@H](C2)C(N)=O 50411944CC(C)(Oc1ccc(Cl)cc1)C(=O)N[C@@H]1C2CCCC1C[C@H](C2)C(N)=O 50411945CCCc1nnc(n1CC)C12CC3CC(CC(C3)C1)C2 50411946CCCn1c(CC)nnc1C12CC3CC(CC(C3)C1)C2 50413276C[C@@](O)(c1ccc(cc1)C(=C)N(C1CC1)[C@H]1CC[C@@H](CC1)c1ccccn1)C(F)(F)F 50413277C[C@@](O)(c1ccc(cc1)C(=C)N(C1CC1)[C@H]1CC[C@H](CC1)c1ccccn1)C(F)(F)F 50413278C[C@@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@](CC1)(C#N)c1ccc(F)cc1)C(F)(F)F 50413279C[C@@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@@](CC1)(C#N)c1ccc(F)cc1)C(F)(F)F 50413280C[C@@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@](CC1)(C#N)c1ccccn1)C(F)(F)F 50413281C[C@@](O)(c1ccc(cc1)C(=O)N(C1CC1)[C@H]1CC[C@@](CC1)(C#N)c1ccccn1)C(F)(F)F 50426475C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(s1)[C@@](C)(O)C(F)(F)F)c1ccc(F)cc1C(F)(F)F 50426476C[C@@H]1CN(CCN1S(=O)(=O)c1nc(n(C)n1)C(C)(O)C(F)(F)F)c1ccc(F)cc1C(F)(F)F 50426477C[C@@H]1CN(CCN1S(=O)(=O)c1cn(C)c(n1)C(C)(O)C(F)(F)F)c1ccc(F)cc1C(F)(F)F 50426478C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(s1)[C@@](O)(C(N)=O)C(F)(F)F)c1ccc(F)cc1C(F)(F)F 50426479C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(s1)C(O)(c1nnc[nH]1)C(F)(F)F)c1ccc(F)cc1C(F)(F)F 50426480C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(s1)[C@](O)(C(N)=O)C(F)(F)F)c1ccc(F)cc1C(F)(F)F 50426481C[C@@H]1CN(CCN1S(=O)(=O)c1ncc(s1)[C@](O)(C(N)=O)C(F)(F)F)c1ccc(F)cc1C(F)(F)F 50426482C[C@@H]1CN(CCN1S(=O)(=O)c1ncc(s1)[C@@](O)(C(N)=O)C(F)(F)F)c1ccc(F)cc1C(F)(F)F 50426483C[C@@H]1CN(CCN1S(=O)(=O)c1cccc(c1)[C@](O)(C(N)=O)C(F)(F)F)c1ccc(F)cc1C(F)(F)F 50426484C[C@@H]1CN(CCN1S(=O)(=O)c1cccc(c1)[C@@](O)(C(N)=O)C(F)(F)F)c1ccc(F)cc1C(F)(F)F 50426485C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(cc1)[C@](O)(C(N)=O)C(F)(F)F)c1ccc(F)cc1C(F)(F)F 50426486C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(cc1)[C@@](O)(C(N)=O)C(F)(F)F)c1ccc(F)cc1C(F)(F)F 50426487C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(s1)[C@](C)(O)C(F)(F)F)c1ccc(cc1C(F)(F)F)C(N)=O 50426488C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(s1)[C@@](C)(O)C(F)(F)F)c1ccc(cc1C(F)(F)F)C(N)=O 50426489C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(s1)[C@](C)(O)C(F)(F)F)c1ccc(F)cc1C(F)(F)F 50429300Cc1c(Cl)cccc1C(=O)N1CCC[C@@H](C1)c1nc(no1)-c1cccc(Br)c1 50429301Cc1c(Cl)cccc1C(=O)N1CCC[C@@H](C1)c1nc(no1)-c1ccccc1Br 50429302Cc1c(Cl)cccc1C(=O)N1CCC[C@@H](C1)c1nc(no1)-c1ccccc1Cl 50429303Cc1c(Cl)cccc1C(=O)N1CCC[C@@H](C1)c1nc(no1)-c1ccc(F)cc1 50429306Cc1c(Cl)cccc1C(=O)N1CCC[C@@H](C1)c1nc(no1)C1CCCCC1 50429307CC1(C)C(C(=O)N2CCC[C@@H](C2)c2nc(no2)-c2ccccc2)C1(C)C 50429308O=C(C1CC1)N1CCC[C@@H](C1)c1nc(no1)-c1ccccc1 50429309O=C(C1CCC1)N1CCC[C@@H](C1)c1nc(no1)-c1ccccc1 50429310O=C(C1CCCCC1)N1CCC[C@@H](C1)c1nc(no1)-c1ccccc1 50429311O=C(C1CCCCCC1)N1CCC[C@@H](C1)c1nc(no1)-c1ccccc1 50429312Cn1ccc2c(cccc12)C(=O)N1CCC[C@@H](C1)c1nc(no1)-c1ccccc1 50429313Cn1cccc1C(=O)N1CCC[C@@H](C1)c1nc(no1)-c1ccccc1 50429314O=C(N1CCC[C@@H](C1)c1nc(no1)-c1ccccc1)c1ccco1 50429315Cc1c(Br)cccc1C(=O)N1CCC[C@@H](C1)c1nc(no1)-c1ccccc1 50429316Cc1cccc(C(=O)N2CCC[C@@H](C2)c2nc(no2)-c2ccccc2)c1Cl 50429317Clc1ccc(cc1)C(=O)N1CCC[C@@H](C1)c1nc(no1)-c1ccccc1 50429318Clc1cccc(c1)C(=O)N1CCC[C@@H](C1)c1nc(no1)-c1ccccc1 50429319Clc1ccccc1C(=O)N1CCC[C@@H](C1)c1nc(no1)-c1ccccc1 50429320Cc1ccccc1C(=O)N1CCC[C@@H](C1)c1nc(no1)-c1ccccc1 50429321O=C(N1CCC[C@@H](C1)c1nc(no1)-c1ccccc1)c1ccccc1 50429322Cc1c(Cl)cccc1C(=O)N1CCC[C@@H](C1)c1nc(no1)-c1ccccc1 50429323Cc1c(Cl)cccc1C(=O)N1CCC[C@@H](C1)c1noc(n1)-c1ccccc1 50429324Cc1c(Cl)cccc1C(=O)N1CCC[C@@H](C1)n1nnc(n1)-c1ccccc1 50429325Cc1c(Cl)cccc1C(=O)N1CCC[C@@H](C1)c1nnc([nH]1)-c1ccccc1 50429326Cc1c(Cl)cccc1C(=O)N1CCC[C@@H](C1)c1nnc(o1)-c1ccccc1 50429327Cc1c(Cl)cccc1S(=O)(=O)N1CCC[C@@H](C1)C(=O)NC1CCCCC1 50430131CC1(C)CCN([C@H]2C3CC4CC2C[C@@](O)(C4)C3)C(=O)c2cnn(c12)-c1ccc(cc1)C(F)(F)F 50430132CC1(C)CCN([C@H]2C3CC4CC2C[C@@](O)(C4)C3)C(=O)c2cnn(c12)-c1cccc(c1)C(F)(F)F 50430134CC1(C)CCN([C@H]2C3CC4CC2C[C@@](O)(C4)C3)C(=O)c2cnn(c12)-c1cccc(Cl)c1 50430135CC1(C)CCN([C@H]2C3CC4CC2C[C@@](O)(C4)C3)C(=O)c2cnn(c12)-c1ccc(F)cc1 50430136CC1(C)CCN([C@H]2C3CC4CC2C[C@@](O)(C4)C3)C(=O)c2cnn(c12)-c1cccc(F)c1 50430137COc1ccc(cc1)-n1ncc2c1C(C)(C)CCN([C@H]1C3CC4CC1C[C@@](O)(C4)C3)C2=O 50430138COc1ccccc1-n1ncc2c1C(C)(C)CCN([C@H]1C3CC4CC1C[C@@](O)(C4)C3)C2=O 50430139Cc1ccc(cc1)-n1ncc2c1C(C)(C)CCN([C@H]1C3CC4CC1C[C@@](O)(C4)C3)C2=O 50430140Cc1cccc(c1)-n1ncc2c1C(C)(C)CCN([C@H]1C3CC4CC1C[C@@](O)(C4)C3)C2=O 50430142CC1(C)CCN([C@H]2C3CC4CC2C[C@@](O)(C4)C3)C(=O)c2cnn(c12)-c1ccccn1 50430143CC1(C)CCN([C@H]2C3CC4CC2C[C@@](O)(C4)C3)C(=O)c2cnn(C3CCCCC3)c12 50430144Cn1ncc2c1C(C)(C)CCN([C@H]1C3CC4CC1C[C@@](O)(C4)C3)C2=O 50430145CC1(C)CN([C@H]2C3CC4CC2C[C@@](O)(C4)C3)C(=O)c2cnn(c2C1)-c1ccccc1 50430146CC1CN([C@H]2C3CC4CC2C[C@@](O)(C4)C3)C(=O)c2cnn(c2C1)-c1ccccc1 50430147CC1(C)CCN([C@H]2C3CC4CC2C[C@@](O)(C4)C3)C(=O)c2cnn(c12)-c1ccccc1 50430148CC1CCN([C@H]2C3CC4CC2C[C@@](O)(C4)C3)C(=O)c2cnn(c12)-c1ccccc1 50430149O[C@]12CC3CC(C1)[C@@H](C(C3)C2)N1CCCc2c(cnn2-c2ccccn2)C1=O 50430150O[C@]12CC3CC(C1)[C@@H](C(C3)C2)N1CCCc2c(cnn2-c2ccccc2)C1=O 50430151O[C@]12CC3CC(C1)[C@@H](C(C3)C2)N1CCCc2c(cnn2C2CCCCC2)C1=O 50430152CC(C)(C)n1ncc2c1CCCN([C@H]1C3CC4CC1C[C@@](O)(C4)C3)C2=O 50430153CCn1ncc2c1CCCN([C@H]1C3CC4CC1C[C@@](O)(C4)C3)C2=O 50430155O[C@]12CC3CC(C1)[C@@H](C(C3)C2)N1CCCc2c(cnn2C2CCCCCC2)C1=O 50432927O=S(=O)(Nc1ccccn1)c1ccc(cc1)-c1ccc(cc1)C#N 50432928OCCc1cccc(NS(=O)(=O)c2ccc(cc2)-c2ccc(cc2)C#N)n1 50432929CC[C@H](O)c1cccc(NS(=O)(=O)c2ccc(cc2)-c2ccc(cc2)C#N)n1 50432930CC[C@@H](O)c1cccc(NS(=O)(=O)c2ccc(cc2)-c2ccc(cc2)C#N)n1 50432931C[C@H](O)c1cccc(NS(=O)(=O)c2ccc(cc2)-c2ccc(cc2)C#N)n1 50432932C[C@@H](O)c1cccc(NS(=O)(=O)c2ccc(cc2)-c2ccc(cc2)C#N)n1 50432933OCc1cccc(NS(=O)(=O)c2ccc(cc2)-c2ccc(cc2)C#N)n1 50432934Cc1cc(N)nc(NS(=O)(=O)c2ccc(cc2)-c2ccc(cc2)C#N)c1 50432935O=S(=O)(Nc1ccc2ncccc2n1)c1ccc(cc1)-c1ccc(cc1)C#N 50432936O=S(=O)(Nc1ccc2ccccc2n1)c1ccc(cc1)-c1ccc(cc1)C#N 50432937Cc1nc(NS(=O)(=O)c2ccc(cc2)-c2ccc(cc2)C#N)ccc1F 50432938Cc1ccc(F)c(NS(=O)(=O)c2ccc(cc2)-c2ccc(cc2)C#N)n1 50432939Cc1ccc(NS(=O)(=O)c2ccc(cc2)-c2ccc(cc2)C#N)nc1C 50432940Cc1cc(C)nc(NS(=O)(=O)c2ccc(cc2)-c2ccc(cc2)C#N)c1 50433400COc1ccc(cc1)-c1cnc(nc1)N1CCN(C(=O)N[C@H]2C3CC4CC2C[C@](O)(C4)C3)c2ccccc12 50433401COc1ccc(cc1)-c1cnc(nc1)N1CCN(C(=O)N[C@H]2C3CC4CC2C[C@@](O)(C4)C3)c2ccccc12 50433402COc1ccc(cc1)-c1cnc(nc1)N1CCN(C(=O)N[C@H]2C3CC4CC2C[C@](C4)(C3)C(N)=O)c2ccccc12 50433403COc1ccc(cc1)-c1cnc(nc1)N1CCN(C(=O)N[C@H]2C3CC4CC2C[C@](C4)(C3)OC(N)=O)c2ccccc12 50433404CS(=O)(=O)N1CCN(CC1)c1cnc(nc1)N1CCN(C(=O)N[C@H]2C3CC4CC2C[C@](O)(C4)C3)c2ccccc12 50433405CS(=O)(=O)N1CCN(CC1)c1ccc(nc1)N1CCN(C(=O)N[C@H]2C3CC4CC2C[C@](O)(C4)C3)c2ccccc12 50433406CS(=O)(=O)N1CCN(CC1)c1ccc(cc1)N1CCN(C(=O)N[C@H]2C3CC4CC2C[C@](O)(C4)C3)c2ccccc12 50433407CS(=O)(=O)N1CCN(CC1)c1ccc(cc1)N1CCN(C(=O)N[C@H]2C3CC4CC2C[C@](C4)(C3)C(N)=O)c2ccccc12 50433408CC(C)(C)N1CCN(CC1)c1ccc(nc1)N1CCN(C(=O)N[C@H]2C3CC4CC2C[C@](O)(C4)C3)c2ccccc12 50433409CC(=O)N1CCN(CC1)c1ccc(nc1)N1CCN(C(=O)N[C@H]2C3CC4CC2C[C@](O)(C4)C3)c2ccccc12 50433410O[C@@]12CC3CC(C1)[C@H](NC(=O)N1CCN(c4ccc(cn4)N4CCN(CC4)S(=O)(=O)C4CC4)c4ccccc14)C(C3)C2 50433411CC(C)(C)N1CCN(CC1)c1ccc(nc1)N1CCN(C(=O)N[C@H]2C3CC4CC2C[C@](C4)(C3)C(N)=O)c2ccccc12 50433412NC(=O)[C@@]12CC3CC(C1)[C@H](NC(=O)N1CCN(c4ccc(cn4)N4CCN(CC4)S(=O)(=O)C4CC4)c4ccccc14)C(C3)C2 50435691Cn1c(nnc1C12CCC(CC1)(CC2)c1noc(n1)C(C)(F)F)-c1ccccc1C(F)(F)F 50436974C[C@@]1(CO)CCC[C@@]2(C)[C@@H]3CC[C@H]4C[C@]3(CC4=C)CC[C@H]12 50436975C[C@@]12CCC[C@](C)([C@H]1CC[C@@]13C[C@H](CC[C@@H]21)[C@@](O)(CO)C3)C(O)=O 50436976C[C@@]1(CO)CCC[C@@]2(C)[C@@H]3CC[C@H]4C[C@]3(C[C@]4(O)CO)CC[C@H]12 50436977C[C@]1(CCC[C@@]2(C)[C@@H]3CC[C@H]4C[C@]3(CC4=C)CC[C@H]12)NC(=O)NC12CC3CC(CC(C3)C1)C2 50436978C[C@]1(CCC[C@@]2(C)[C@@H]3CC[C@H]4C[C@]3(CC4=C)CC[C@H]12)NC(=O)Nc1ccc(F)cc1 50436979CC(=O)O[C@H]1C[C@H]2C[C@@]3(CC[C@H]4[C@@](C)(CCC[C@@]4(C)C(O)=O)[C@H]13)[C@H](O)C2=C 50436980CSC(=S)O[C@H]1C[C@H]2C[C@@]3(CC[C@H]4[C@@](C)(CCC[C@@]4(C)C(O)=O)[C@H]13)[C@H](O)C2=C 50436982C[C@]1(CCC[C@]2(C)[C@@H]1CC[C@@]13C[C@H](C[C@H](O)[C@@H]21)C(=C)[C@H]3O)NC(=O)NC1CCCCC1 50436983C[C@]1(CCC[C@]2(C)[C@@H]1CC[C@@]13C[C@H](C[C@H](O)[C@@H]21)C(=C)[C@H]3O)NC(=O)Nc1cccc2ccccc12 50436984C[C@]1(CCC[C@]2(C)[C@@H]1CC[C@@]13C[C@H](C[C@H](O)[C@@H]21)C(=C)[C@H]3O)NC(=O)Nc1ccc(F)cc1 50436985C[C@]1(CCC[C@]2(C)[C@@H]1CC[C@@]13C[C@H](C[C@H](O)[C@@H]21)C(=C)[C@H]3O)NC(=O)Nc1ccccc1 50436987C[C@@H]1CC(C[C@@H](C)N1C(=O)c1cc(Cl)c(N)c(Cl)c1)n1c2ccccc2[nH]c1=O 50437197Fc1ccc(\C=C2/CC\C(=C/c3ccc(F)cc3)C2=O)cc1 50437199Fc1ccc(\C=C2/CCC\C(=C/c3ccc(F)cc3)C2=O)cc1 50437200Brc1ccccc1\C=C1/CC\C(=C/c2ccccc2Br)C1=O 50437202Brc1ccccc1\C=C1/CCC\C(=C/c2ccccc2Br)C1=O 50437203Brc1ccccc1\C=C\C(=O)\C=C\c1ccccc1Br 50437698CC(C)CC(=O)C(=O)[C@H](C)[C@@H]1CC[C@]2(C)C3=CC[C@H]4C(C)(C)[C@@H](O)CC[C@]4(C)[C@H]3C[C@@H](O)[C@@]12C 50437699CC(C)(O)[C@@H](O)[C@H]1C[C@@H]([C@@H]2CC[C@]3(C)C4=CC[C@H]5C(C)(C)[C@@H](O)CC[C@]5(C)[C@H]4CC[C@@]23C)C(=O)O1 50438063O=S1(=O)NC(O[C@@H]2CCCC[C@@H]12)=NC1CCCCC1 50438064O=S1(=O)NC(O[C@H]2CCCC[C@@H]12)=NC1CCCCC1 50438065CC(C)(O)C[C@H](N=C1NS(=O)(=O)C(C)(C)C(C)(C)O1)c1ccccc1Cl 50438066CC1(C)OC(NS(=O)(=O)C1(C)C)=N[C@@H](CCO)c1ccc(F)cc1 50438067CC1(C)OC(NS(=O)(=O)C1(C)C)=N[C@@H](CCO)c1cccc(c1)C#N 50438068CC1(C)OC(NS(=O)(=O)C1(C)C)=N[C@@H](CCO)c1ccccc1Cl 50438069CC1(C)OC(NS(=O)(=O)C1(C)C)=N[C@@H](CCO)c1ccccc1 50438070C[C@H](N=C1NS(=O)(=O)C(C)(C)C(C)(C)O1)c1ccccc1Cl 50438071C[C@H](N=C1NS(=O)(=O)C(C)(C)C(C)(C)O1)c1ccccc1 50438072CCC1OC(NS(=O)(=O)C11CC1)=NC1CCCCC1 50438073O=S1(=O)NC(OC2(CCC2)C11CC1)=NC1CCCCC1 50438074CC1(C)OC(NS(=O)(=O)C11CC1)=NC1CCCCC1 50438075CC1(C)OC(NS(=O)(=O)C1(C)C)=NC1CCCCC1 50438076OCCC[C@H](N=C1NS(=O)(=O)[C@@H]2CCCC[C@@H]2O1)c1ccccc1 50438077OCC[C@H](N=C1NS(=O)(=O)[C@@H]2CCCC[C@@H]2O1)c1ccccc1 50438078OC[C@H](N=C1NS(=O)(=O)[C@@H]2CCCC[C@@H]2O1)c1ccccc1 50438079CC(C)(N=C1NS(=O)(=O)[C@@H]2CCCC[C@@H]2O1)c1ccccc1 50438080O=S1(=O)NC(O[C@H]2CCCC[C@@H]12)=NC12CC3CC1CC(C2)C3 50438081O=S1(=O)NC(O[C@H]2CCCC[C@@H]12)=NCC12CC3CC(CC(C3)C1)C2 50438082OC12CC3CC(C1)CC(C3)(C2)N=C1NS(=O)(=O)[C@@H]2CCCC[C@@H]2O1 50438083O=S1(=O)NC(O[C@H]2CCCC[C@@H]12)=NC12CC3CC(CC(C3)C1)C2 50438084OC12CCC(CC1)(CC2)N=C1NS(=O)(=O)[C@@H]2CCCC[C@@H]2O1 50438085FC12CCC(CC1)(CC2)N=C1NS(=O)(=O)[C@@H]2CCCC[C@@H]2O1 50438086O=S1(=O)NC(O[C@H]2CCCC[C@@H]12)=NC12CCC(CC1)CC2 50438087O=S1(=O)NC(O[C@H]2CCCC[C@@H]12)=NC12CCCC1CCC2 50438088O=S1(=O)NC(O[C@H]2CCCC[C@@H]12)=NCc1ccccc1 50438089O=S1(=O)NC(O[C@H]2CCCC[C@@H]12)=NCC1CCCCC1 50438090CC1(C)CC(CC(C)(C)C1)N=C1NS(=O)(=O)[C@@H]2CCCC[C@@H]2O1 50438091CC1(C)CCC(CC1)N=C1NS(=O)(=O)[C@@H]2CCCC[C@@H]2O1 50438092O=S1(=O)NC(O[C@H]2CCCC[C@@H]12)=NC1CCCCCCC1 50438093O=S1(=O)NC(O[C@H]2CCCC[C@@H]12)=NC1CCCCCC1 50438094O=C(NC1CCCCC1)NS(=O)(=O)C1=CCCCC1 50438095O=S1(=O)NC(OC2(COC2)C11CC1)=NC1CCCCC1 50438096CNC(=O)C[C@H](N=C1NS(=O)(=O)[C@@H]2CCCC[C@@H]2O1)c1ccccc1 50438097NC(=O)C[C@H](N=C1NS(=O)(=O)[C@@H]2CCCC[C@@H]2O1)c1ccccc1 50438098NCC[C@H](N=C1NS(=O)(=O)[C@@H]2CCCC[C@@H]2O1)c1ccccc1 50438099OCC[C@@H](N=C1NS(=O)(=O)[C@@H]2CCCC[C@@H]2O1)c1ccccc1 50438101O=S1(=O)NC(O[C@H]2CCCC[C@@H]12)=Nc1ccccc1 50438102FC1(F)CCC(CC1)N=C1NS(=O)(=O)[C@@H]2CCCC[C@@H]2O1 50438103O=S1(=O)NC(O[C@H]2CCCC[C@@H]12)=NC1CCOCC1 50438104O=S1(=O)NC(O[C@H]2CCCC[C@@H]12)=NC1CCCC1 50438105C[C@]12CCCC[C@@]1(C)S(=O)(=O)NC(O2)=NC1CCCCC1 50438108O=S1(=O)NC(O[C@@H]2CCOC[C@@H]12)=NC1CCCCC1 50438109O=S1(=O)NC(O[C@H]2CCOC[C@@H]12)=NC1CCCCC1 50438110FC1(F)CC[C@@H]2OC(NS(=O)(=O)[C@@H]2C1)=NC1CCCCC1 50438111O=S1(=O)NC(O[C@H]2CCCC[C@H]12)=NC1CCCCC1 50438112O=S1(=O)NC(O[C@@H]2CCCC[C@H]12)=NC1CCCCC1 50440405COc1ccc(cc1)S(=O)(=O)N1CCN(CC1)c1nc2ccccc2n1C 50440406Cn1c(nc2ccccc12)N1CCN(CC1)S(=O)(=O)c1ccc(cc1)C(C)(C)C 50440407Cc1ccc(cc1)S(=O)(=O)N1CCN(CC1)c1nc2ccccc2n1C 50440408Cn1c(nc2ccccc12)N1CCN(CC1)S(=O)(=O)c1ccccc1 50442531CC(=O)[C@H]1CC[C@H]2[C@@H]3CCC4=CC(=O)CC[C@]4(C)[C@H]3[C@@H](O)C[C@]12C 50442535CCOC(=O)C(NO)C=N[C@H]1C[C@@]2(C)[C@@H](CC[C@@H]2C(C)=O)[C@@H]2CCC3=CC(=O)CC[C@]3(C)[C@@H]12 50442536CC(=O)[C@H]1CC[C@H]2[C@@H]3CCC4=CC(=O)CC[C@]4(C)[C@H]3[C@H](O)C[C@]12C 50445565OC1C2CC3CC1CC(C2)C3(Cc1nnn[nH]1)c1ccc(cc1)-c1ccc(F)cc1 50445566COc1ccc(cc1)-c1ccc(cc1)C1(Cc2nnn[nH]2)C2CC3CC1CC(C2)C3O 50445567OC1C2CC3CC1CC(C2)C3(Cc1nnn[nH]1)c1ccc(cc1)-c1cccc(c1)C(F)(F)F 50445568OC12CC3CC(C1)C(Cc1nnn[nH]1)(C(C3)C2)c1ccc(cc1)-c1ccccc1 50445569OC1C2CC3CC1CC(C2)C3(Cc1nnn[nH]1)c1ccc(cc1)-c1cccc(F)c1 50445570OC1C2CC3CC1CC(C2)C3(Cc1nnn[nH]1)c1ccc(cc1)-c1ccc(cc1)C#N 50445571C(c1nnn[nH]1)C1(C2CC3CC(C2)CC1C3)c1ccc(cc1)-c1ccccc1 50445572O[C@H]1C2CC3CC1CC(C2)C3(Cc1nnn[nH]1)c1ccc(cc1)-c1ccc(F)cc1 50445573Cc1ccc(cc1)-c1ccc(cc1)C1(Cc2nnn[nH]2)C2CC3CC1CC(C2)C3O 50445574OC1C2CC3CC1CC(C2)C3(Cc1nnn[nH]1)c1ccc(cc1)-c1ccc(cc1)C(F)(F)F 50445575OC1C2CC3CC1CC(C2)C3(Cc1nnn[nH]1)c1ccc(cc1)-c1ccccc1F 50445576COC12CC3CC(C1)C(Cc1nnn[nH]1)(C(C3)C2)c1ccc(cc1)-c1ccccc1 50445577OC1C2CC3CC1CC(C2)C3(Cc1nnn[nH]1)C#Cc1ccccc1 50445578OC1C2CC3CC1CC(C2)C3(Cc1nnn[nH]1)c1ccc(cc1)-c1cccnc1 50445579C(c1nnn[nH]1)C1(C2CC3CC(C2)CC1C3)c1ccccc1 50445580Fc1ccc(cc1)C1(Cc2nnn[nH]2)C2CC3CC(C2)CC1C3 50445581OC1C2CC3CC1CC(C2)C3(Cc1nnn[nH]1)c1ccc(Oc2ccccc2)cc1 50445582CS(=O)(=O)c1ccc(cc1)-c1ccc(cc1)C1(Cc2nnn[nH]2)C2CC3CC1CC(C2)C3O 50445583OC1C2CC3CC1CC(C2)C3(Cc1nnn[nH]1)c1ccc(cc1)-c1ccncc1 50445584OC1C2CC3CC1CC(C2)C3(Cc1nnn[nH]1)c1cccc(c1)-c1ccccc1 50445585OC12CC3CC(O)(CC(C1)C3(Cc1nnn[nH]1)c1ccc(cc1)-c1ccccc1)C2 50445586OC1C2CC3CC1CC(C2)C3(Cc1nnn[nH]1)Cc1ccccc1 50445587OC1C2CC3CC1CC(C2)C3(Cc1nnn[nH]1)c1ccc(nc1)-c1ccccc1 50445588OC1C2CC3CC1CC(C2)C3(Cc1nnn[nH]1)Cc1ccc(cc1)-c1ccccc1 50445589Clc1cccc(CC2(Cc3nnn[nH]3)C3CC4CC(C3)CC2C4)c1 50448221CC(C)(CC(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)C(N)=O)NS(=O)(=O)c1ccc(F)cc1 50448222CC(C)(CC(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)C(N)=O)NS(=O)(=O)c1cccc(F)c1 50448223CC(C)(CC(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)C(N)=O)NS(=O)(=O)c1ccccc1F 50448224CC(C)(CC(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)C(N)=O)NS(=O)(=O)c1cccc(Cl)c1 50448225CC(C)(CC(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)C(N)=O)NS(=O)(=O)c1c(F)cc(F)cc1F 50448226CC(C)(CC(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)C(N)=O)NS(=O)(=O)c1ccc(F)c(F)c1 50448227CC(C)(CC(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)C(N)=O)NS(=O)(=O)c1c(F)cccc1F 50448228CC(C)(CC(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)C(N)=O)NS(=O)(=O)c1cc(F)cc(F)c1 50448229CC(C)(CC(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)C(N)=O)NS(=O)(=O)c1cccc(F)c1F 50448230CC(C)(CC(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)C(N)=O)NS(=O)(=O)c1ccc(F)cc1F 50448231CC(C)(CC(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)C(N)=O)NS(=O)(=O)c1cccc(Cl)c1Cl 50448232CC(C)(CC(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)C(N)=O)NS(=O)(=O)c1cccc(Cl)c1F 50448233Cc1c(Cl)cccc1S(=O)(=O)NC1(CC(=O)NC2C3CC4CC(C3)CC2C4)CC1 50448234Cc1c(Cl)cccc1S(=O)(=O)NC(C)(C)CC(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)S(C)(=O)=O 50448235Cc1c(Cl)cccc1S(=O)(=O)NC(C)(C)CC(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)C(N)=O 50448236Cc1c(Cl)cccc1S(=O)(=O)NC(C)(C)CC(=O)N[C@H]1C2CC3CC1C[C@](C3)(C2)C(O)=O 50448237Cc1c(Cl)cccc1S(=O)(=O)NC(C)(C)CC(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50448238Cc1c(Cl)cccc1S(=O)(=O)NC(C)(C)CC(=O)NC1C2CC3CC(C2)CC1C3 50448239Cc1c(Cl)cccc1S(=O)(=O)NC(C)(C)CC(=O)NC12CC3CC(CC(C3)C1)C2 50448240C[C@H](CC(=O)NC1C2CC3CC(C2)CC1C3)NS(=O)(=O)c1cccc(Cl)c1C 50448241C[C@@H](CC(=O)NC1C2CC3CC(C2)CC1C3)NS(=O)(=O)c1cccc(Cl)c1C 50448243Cc1c(Cl)cccc1S(=O)(=O)NC(C)(C)CC(=O)NC1CCCCCC1 50448244Cc1c(Cl)cccc1S(=O)(=O)NC(C)(C)CC(=O)NC1CCCCC1 50448692C[C@H]1CN(C[C@@H](C)O1)c1ncc(C(=O)NC2C3CC4CC2CC(O)(C4)C3)c(n1)[C@H]1CCCO1 50448693OC12CC3CC(C1)C(NC(=O)c1sc(OC4CC(C4)C#N)nc1[C@H]1CCCO1)C(C3)C2 50448694C[C@H]1CN(C[C@@H](C)O1)c1ncc(C(=O)NC2C3CC4CC2CC(O)(C4)C3)c(n1)[C@@H]1CCCO1 50448696O[C@@]12CC3CC(C1)[C@H](NC(=O)c1sc(OCC4(CC4)C#N)nc1C1CC1)C(C3)C2 50448697O[C@@]12CC3CC(C1)[C@H](NC(=O)c1sc(OC4CCOCC4)nc1[C@H]1CCCO1)C(C3)C2 50448698COC[C@@H](C)Oc1nc(C2CC2)c(s1)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50448699COCCOc1nc(C2CC2)c(s1)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50448700OCCOc1nc(C2CC2)c(s1)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50448701CC(C)Oc1nc(C2CC2)c(s1)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50448702CCOc1nc(C2CC2)c(s1)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50448703COc1nc(C2CC2)c(s1)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50448704COC[C@H](C)Oc1nc([C@H]2CCCO2)c(s1)C(=O)NC1C2CC3CC1CC(O)(C3)C2 50448705COCCOc1nc([C@H]2CCCO2)c(s1)C(=O)NC1C2CC3CC1CC(O)(C3)C2 50448706COc1nc([C@H]2CCCO2)c(s1)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50448707CS(=O)(=O)Cc1nc([C@H]2CCCO2)c(s1)C(=O)NC1C2CC3CC1CC(O)(C3)C2 50448708CN(C)c1nc([C@H]2CCCO2)c(s1)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50448709CNc1nc([C@H]2CCCO2)c(s1)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50448710Nc1nc([C@H]2CCCO2)c(s1)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50448711COCCc1nc([C@H]2CCCO2)c(s1)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50448712COCc1nc([C@H]2CCCO2)c(s1)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50448713OC12CC3CC(C1)C(NC(=O)c1scnc1[C@H]1CCCO1)C(C3)C2 50448714CCc1nc([C@H]2CCCO2)c(s1)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50448715Cc1nc([C@H]2CCCO2)c(s1)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50448716Cc1nc([C@@H]2CCCO2)c(s1)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50448717Cc1nc(C2CC2)c(s1)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50448718Cc1nc(c(s1)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2)C(F)(F)F 50448719CCCSc1nc(C)sc1C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50448720Cc1nc(OC2COC2)c(s1)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50448721Cc1nc(OC2CCC2)c(s1)C(=O)NC1C2CC3CC1CC(O)(C3)C2 50448722CC(C)Oc1nc(C)sc1C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50448723Cc1nc(OCC(F)(F)F)c(s1)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50448724CCOc1nc(C)sc1C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50448725Cc1nc(C)c(s1)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50448727COc1ncsc1C(=O)NC1C2CC3CC1CC(O)(C3)C2 50448728COc1nc(C)sc1C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2 50448729COc1c(cnn1C)C(=O)NC1C2CC3CC1CC(O)(C3)C2 50448730C[C@H]1CN(C[C@@H](C)O1)c1ncc(C(=O)NC2C3CC4CC2CC(O)(C4)C3)c(n1)C1CCCC1 50448731O[C@@]12CC3CC(C1)[C@H](NC(=O)c1sc(OCC4CC4)nc1C1CC1)C(C3)C2 50448732O[C@@]12CC3CC(C1)[C@H](NC(=O)c1sc(OC4CCOCC4)nc1C1CC1)C(C3)C2 50448733O[C@@]12CC3CC(C1)[C@H](NC(=O)c1sc(O[C@@H]4CCCO4)nc1C1CC1)C(C3)C2 50448734COC[C@H](C)Oc1nc(C2CC2)c(s1)C(=O)N[C@H]1C2CC3CC1C[C@](O)(C3)C2