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139135Fc1ccc(cc1)-c1cc(NC[C@H]2CC[C@H](CC2)NC(=O)c2cc(ccc2Cl)C(F)(F)F)[nH]n1 139136Cc1ccncc1NC[C@H]1CC[C@H](CC1)NC(=O)c1cc(ccc1Cl)C(F)(F)F 139137CC(Nc1ccccc1)[C@H]1CC[C@@H](CC1)NC(=O)c1cc(ccc1Cl)C(F)(F)F 139138C[C@H]1CC(CNc2ccccc2)CCC1NC(=O)c1cc(ccc1Cl)C(F)(F)F 139140Cc1nn(C[C@H]2CC[C@@H](CC2)NC(=O)c2cc(Cl)cnc2C)c(C)c1C 139141Fc1cncc(NC[C@H]2CC[C@@H](CC2)NC(=O)c2cc(ccc2Cl)C(F)(F)F)c1 139142Fc1ccc(NC[C@H]2CC[C@@H](CC2)NC(=O)c2cc(ccc2Cl)C(F)(F)F)nc1 139143Cc1cc(NC[C@H]2CC[C@@H](CC2)NC(=O)c2cc(ccc2Cl)C(F)(F)F)ncc1F 139144FC(F)(F)c1ccc(Cl)c(c1)C(=O)N[C@H]1CC[C@H](CNc2n[nH]c3CCCCc23)CC1 139145CCc1cncc(NC[C@H]2CC[C@@H](CC2)NC(=O)c2cc(ccc2Cl)C(F)(F)F)c1 139146Cc1cc(NC[C@H]2CC[C@@H](CC2)NC(=O)c2cc(Cl)cnc2C)ncc1F 139147Cc1ncc(Cl)cc1C(=O)N[C@H]1CC[C@H](CNc2n[nH]c3CCCCc23)CC1 139148COc1ncc(C)cc1NC[C@H]1CC[C@@H](CC1)NC(=O)c1cc(ccc1Cl)C(F)(F)F 139149FC(F)(F)c1ccc(Cl)c(c1)C(=O)N[C@H]1CC[C@H](CNc2n[nH]c3ncccc23)CC1 139150Cc1ccc2[nH]nc(NC[C@H]3CC[C@@H](CC3)NC(=O)c3cc(ccc3Cl)C(F)(F)F)c2c1 139151Fc1ccc2[nH]nc(NC[C@H]3CC[C@@H](CC3)NC(=O)c3cc(ccc3Cl)C(F)(F)F)c2c1 139152Fc1cccc2[nH]nc(NC[C@H]3CC[C@@H](CC3)NC(=O)c3cc(ccc3Cl)C(F)(F)F)c12 139153Cc1cccc2[nH]nc(NC[C@H]3CC[C@@H](CC3)NC(=O)c3cc(ccc3Cl)C(F)(F)F)c12 139154FC(F)(F)c1ccc(Cl)c(c1)C(=O)N[C@H]1CC[C@H](CNc2n[nH]c3ccc(Cl)cc23)CC1 139155COc1ccc2c(NC[C@H]3CC[C@@H](CC3)NC(=O)c3cc(ccc3Cl)C(F)(F)F)n[nH]c2c1 139156Cc1cc(NC[C@H]2CC[C@@H](CC2)NC(=O)c2cc(ccc2Cl)C(F)(F)F)ncc1Cl 139157Cn1nc(NC[C@H]2CC[C@@H](CC2)NC(=O)c2cc(ccc2Cl)C(F)(F)F)c2ccccc12 139158Cc1n[nH]c(NC[C@H]2CC[C@@H](CC2)NC(=O)c2cc(ccc2Cl)C(F)(F)F)c1-c1ccccc1 139159Cc1ncc(Cl)cc1NC[C@H]1CC[C@@H](CC1)NC(=O)c1cc(ccc1Cl)C(F)(F)F 139160Cc1ccc2c(NC[C@H]3CC[C@@H](CC3)NC(=O)c3cc(ccc3Cl)C(F)(F)F)n[nH]c2n1 139162CCCc1[nH]nc(NC[C@H]2CC[C@@H](CC2)NC(=O)c2cc(ccc2Cl)C(F)(F)F)c1Br 139163Cc1c(NC[C@H]2CC[C@@H](CC2)NC(=O)c2cc(ccc2Cl)C(F)(F)F)n[nH]c1-c1ccccc1 139164FC(F)(F)c1ccc(Cl)c(c1)C(=O)N[C@H]1CC[C@H](CNc2n[nH]cc2-c2ccc(Cl)cc2)CC1 139165Cc1cc(NC[C@H]2CC[C@@H](CC2)NC(=O)c2cc(Cl)cnc2C)ncc1Cl 139166Cc1[nH]nc(NC[C@H]2CC[C@@H](CC2)NC(=O)c2cc(ccc2Cl)C(F)(F)F)c1-c1ccc(Cl)cc1 139167FC(F)(F)c1ccc(Cl)c(c1)C(=O)N[C@H]1CC[C@H](CNc2n[nH]c3cccnc23)CC1 139168FC(F)(F)c1ccc(Cl)c(c1)C(=O)N[C@H]1CC[C@H](CNc2n[nH]cc2-c2ccccc2)CC1 139169COc1ccc(Cl)c(NC[C@H]2CC[C@@H](CC2)NC(=O)c2cc(ccc2Cl)C(F)(F)F)n1 139170FC(F)(F)c1ccc(Cl)c(c1)C(=O)N[C@H]1CC[C@H](CNc2nnnn2-c2ccccc2)CC1 139171Cn1cc(c(NC[C@H]2CC[C@@H](CC2)NC(=O)c2cc(ccc2Cl)C(F)(F)F)n1)-c1ccccc1 139172Cc1noc(NC[C@H]2CC[C@@H](CC2)NC(=O)c2cc(ccc2Cl)C(F)(F)F)c1C 139173FC(F)(F)c1ccc(Cl)c(c1)C(=O)N[C@H]1CC[C@H](CNc2[nH]ncc2-c2cccnc2)CC1 139174Cc1ncc(Cl)cc1C(=O)N[C@H]1CC[C@H](CNc2cc(n[nH]2)C(F)(F)F)CC1 139175Cc1ncc(Cl)cc1C(=O)N[C@H]1CC[C@H](CNc2ccc(F)cn2)CC1 139176CCCc1cc(NC[C@H]2CC[C@@H](CC2)NC(=O)c2cc(Cl)cnc2C)n[nH]1 139177COc1ncc(Cl)cc1NC[C@H]1CC[C@@H](CC1)NC(=O)c1cc(ccc1Cl)C(F)(F)F 139178Cc1n[nH]c(NC[C@H]2CC[C@@H](CC2)NC(=O)c2cc(ccc2Cl)C(F)(F)F)c1Cl 139179Cc1cc(NC[C@H]2CC[C@@H](CC2)NC(=O)c2cc(ccc2Cl)C(F)(F)F)n(n1)-c1ccc(Cl)cc1 139180CCc1[nH]nc(NC[C@H]2CC[C@@H](CC2)NC(=O)c2cc(ccc2Cl)C(F)(F)F)c1C 139181FC(F)(F)c1ccc(Cl)c(c1)C(=O)N[C@H]1CC[C@H](Cn2ncc3ccccc23)CC1 139182FC(F)(F)c1ccc(Cl)c(c1)C(=O)N[C@H]1CC[C@H](Cn2cc3ccccc3n2)CC1 139183Cc1nc(C)n(C[C@H]2CC[C@@H](CC2)NC(=O)c2cc(ccc2Cl)C(F)(F)F)n1 139184Cc1cc(nn1C[C@H]1CC[C@@H](CC1)NC(=O)c1cc(ccc1Cl)C(F)(F)F)N1CCNC1=O 139185Cc1nn(C[C@H]2CC[C@@H](CC2)NC(=O)c2cc(ccc2Cl)C(F)(F)F)c(C)c1Cl 139186Cc1nn(C[C@H]2CC[C@@H](CC2)NC(=O)c2cc(ccc2Cl)C(F)(F)F)c(C)c1C 139187FC(F)(F)c1ccc(Cl)c(c1)C(=O)N[C@H]1CC[C@H](Cn2ccc(n2)-c2ccccc2)CC1 139188Cc1cc(nn1C[C@H]1CC[C@@H](CC1)NC(=O)c1cc(Cl)cnc1C)C(F)(F)F 50003909COCCN(CCOC)c1nc(C)nc(Nc2c(C)cc(C)cc2C)c1SC 50003910CCCN(CCC)c1nc(C)nc(Nc2c(C)cc(C)cc2C)c1SCC 50003911CCSc1c(Nc2c(C)cc(C)cc2C)nc(C)nc1N(CCOC)CCOC 50003912CCCN(CC1CC1)c1nc(C)nc(Nc2c(C)cc(C)cc2C)c1SCC 50054216CCCN(Cc1ccccc1)c1nc(C)nc(Nc2c(C)cc(C)cc2C)n1 50054219CCCCN(Cc1ccccc1)c1nc(C)nc(Nc2c(C)cc(C)cc2C)n1 50054221CCCCN(CCCC)c1nc(C)nc(Nc2c(C)cc(C)cc2C)n1 50054222CCc1cccc(CC)c1Nc1nc(C)nc(n1)N(CC=C)CC=C 50054223CCN(Cc1ccccc1)c1nc(C)nc(Nc2c(C)cc(C)cc2C)n1 50054225CCCN(CC1CC1)c1nc(C)nc(Nc2c(C)cc(C)cc2C)n1 50054226Cc1cc(C)c(Nc2nc(C)nc(n2)N(CC=C)CC=C)c(C)c1 50054229CCCN(CC1CC1)c1nc(C)nc(Nc2ccc(OC)cc2OC)n1 50054230CCCN(CCC)c1nc(C)nc(Nc2c(C)cc(C)cc2C)n1 50054234CN(CCc1ccccc1)c1nc(C)nc(Nc2c(C)cc(C)cc2C)n1 50054238CCN(Cc1ccccc1)c1nc(C)nc(Nc2c(CC)cccc2CC)n1 50054239Cc1cc(C)c(Nc2nc(C)nc(n2)N2CCC=CC2)c(C)c1 50054241Cc1cc(C)c(Nc2nc(C)nc(NCc3ccc(cc3)C(F)(F)F)n2)c(C)c1 50054244CCCN(CC1CC1)c1cc(Nc2cc(Cl)c(Cl)cc2Cl)nc(C)n1 50054245CCCN(CC1CC1)c1nc(C)nc(Nc2c(Cl)cc(Cl)cc2Cl)c1Cl 50054246CCCN(CC1CC1)c1cc(Nc2c(Cl)cc(Cl)cc2Cl)nc(C)n1 50054247CCCN(CC1CC1)c1nc(C)nc(N(C)c2c(Cl)cc(Cl)cc2Cl)c1C 50054248CCCN(CCC)c1nc(C)nc(Nc2c(Cl)cc(Cl)cc2Cl)c1C 50054249CCCN(CC1CC1)c1cc(C)nc(Nc2c(Cl)cc(Cl)cc2Cl)n1 50054250CCCN(CC1CC1)c1nc(C)nc(Nc2c(Cl)cc(Cl)cc2Cl)c1C 50054252CCCN(CC1CC1)c1nc(C)nc(Nc2c(Cl)cc(Cl)cc2Cl)c1Br 50054253CCCN(CC1CC1)c1nc(C)nc(Nc2c(Cl)cc(Cl)cc2Cl)c1CC 50054255CCCN(CC1CC1)c1cc(Nc2c(C)cc(C)cc2C)nc(C)n1 50058163CCCCN(CC)c1nc(C)nc2n(cc(C)c12)-c1c(C)cc(C)cc1C 50060874Cc1cc(O)c2c3c1c1c(C)cc(O)c4c1c1c3c3c(c(O)cc(O)c3c2=O)c2c(O)cc(O)c(c12)c4=O 50071226CCCCN(CC)c1cc(C)nc2c(cnn12)-c1ccc(Cl)cc1Cl 50071227CCCCN(OC)c1cc(C)nc2c(c(C)nn12)-c1ccc(Cl)cc1Cl 50071228CCCCNc1cc(C)nc2c(c(C)nn12)-c1ccc(Cl)cc1Cl 50071229CCN(CCOC)c1cc(C)nc2c(c(C)nn12)-c1ccc(Cl)cc1Cl 50071230CCCCN(CC)c1cc(C)nc2c(c(C)nn12)-c1c(Cl)cc(Cl)cc1Cl 50071231CCCCN(CC)c1cc(C)nc2c(c(C)nn12)-c1ccccc1 50071232Cc1nn2c(cc(C)nc2c1-c1ccc(Cl)cc1Cl)N1CCCCC1 50071233CCCCN(CC)c1cc(C)nc2c(c(C)nn12)-c1ccccc1Cl 50071234CCCCN(CC)c1cc(C)nc2c(c(C)nn12)-c1ccc(Cl)cc1Cl 50071235CCCN(CC1CC1)c1cc(C)nc2c(c(C)nn12)-c1ccc(Cl)cc1Cl 50071236Cc1nn2c(cc(C)nc2c1-c1ccc(Cl)cc1Cl)N1CCOCC1 50071237CCCCN(CC)c1cc(C)nc2c(c(C)nn12)-c1ccc(Cl)cc1 50071238CCCC1CCCCN1c1cc(C)nc2c(c(C)nn12)-c1ccc(Cl)cc1Cl 50074330CCCN(CCC#N)c1nc(C)nc(n1)N(CC)c1ccc(cc1C(F)(F)F)N(C)C 50074331CCCN(CCOC)c1cc(C)nc(n1)N(CC)c1ccc(cc1Br)C(C)C 50074332CCN(c1nc(C)nc(n1)N(CC=C)CC=C)c1ccc(OC(F)(F)F)cc1Br 50074333CCCN(C1CC1)c1cc(C)nc(n1)N(CC)c1ccc(cc1Br)C(C)C 50074334CCCCN(Cc1nnnn1C)c1cc(C)nc(n1)N(CC)c1ccc(cc1Br)C(C)C 50074335CCCN(CCC#N)c1nc(C)nc(n1)N(CC)c1ccc(cc1C)N(C)C 50074336CCN(CC)c1cc(C)nc(n1)N(CC)c1ccc(cc1Br)C(C)=O 50074337CCN(CC)c1cc(C)nc(n1)N(CC)c1c(Br)cc(cc1SC)C(C)C 50074338CCN(c1nc(C)cc(C)n1)c1c(Br)cc(cc1OC)N(C)C 50074339CCN(CC)c1nc(C)nc(n1)N(CC)c1ccc(cc1Br)N(C)C 50074340CCN(CC)c1cc(C)nc(n1)N(CC)c1c(Br)cc(Br)cc1OC 50074342CCN(CC)c1cc(C)nc(n1)N(CC)c1c(Cl)cc(OC)cc1Cl 50074343CCN(c1nc(C)nc(NCC=C)n1)c1ccc(cc1Br)C(C)C 50074344CCN(CC)c1nc(C)nc(n1)N(CC)c1ccc(cc1Br)C(C)=O 50074345CCN(CC)c1cc(C)nc(n1)N(CC)c1ccc(cc1Br)S(C)(=O)=O 50074347CCCCN(CC#N)c1nc(C)nc(n1)N(CC)c1ccc(cc1C(F)(F)F)N(C)C 50074349CCC(CC)c1cc(C)nc(n1)N(CC)c1ccc(cc1Br)C(C)C 50074352CCN(c1nc(C)cc(C)n1)c1c(Br)cc(cc1SC)C(C)C 50074353CCN(c1nc(C)nc(n1)N1CCOCC1)c1c(Br)cc(OC)cc1OC 50074354CCN(c1nc(C)nc(n1)N(CC=C)CC=C)c1ccc(cc1Br)N(C)C 50074356CCN(c1nc(C)cc(C)n1)c1ccc(cc1SC)N(C)C 50074357CCN(c1nc(C)cc(n1)N1CCCCC1)c1ccc(cc1Br)C(C)C 50074358CCN(c1nc(C)cc(C)n1)c1ccc(cc1C(F)(F)F)N(C)C 50074359CCN(Cc1ccccc1)c1cc(C)nc(n1)N(CC)c1ccc(cc1Br)C(C)C 50074360CCN(CC)c1cc(C)nc(n1)N(CC)c1c(Cl)cc(OC)cc1OC 50074361CCC(CC)CNc1cc(C)nc(n1)N(CC)c1ccc(cc1Br)C(C)C 50074362CCN(CC)c1cc(C)nc(n1)N(CC)c1ccc(SC)cc1Br 50074363CCN(c1nc(C)cc(n1)N(CCOC)Cc1ccccc1)c1ccc(cc1Br)C(C)C 50074364CCCCN(CC)c1cc(C)nc(n1)N(CC)c1ccc(cc1Br)C(C)C 50074365CCN(CC)c1cc(C)nc(n1)N(CC)c1c(Br)cc(OC)cc1OC 50074366CCCN(CCC)c1cc(C)nc(n1)N(CC)c1ccc(cc1Br)C(C)C 50074367CCCCN(CC)c1nc(C)nc(n1)N(CC)c1c(C)cc(C)cc1C 50074368CCCCN(CC)c1cc(C)nc(n1)N(CC)c1ccc(cc1Br)C(C)=O 50074369CCN(CC)c1cc(C)nc(n1)N(CC)c1c(Cl)cc(Br)cc1Cl 50074371CCN(c1nc(C)cc(C)n1)c1ccc(OC)cc1SC 50074372CCN(c1nc(C)cc(n1)N1CCOCC1)c1ccc(cc1Br)C(C)C 50074373CCN(c1nc(C)cc(C)n1)c1ccc(OC)cc1Br 50074374CCN(c1nc(C)nc(n1)N(CCOC)CCOC)c1ccc(cc1Br)C(C)C 50074375CCN(c1nc(C)nc(n1)N(CC1CC1)CC1CC1)c1ccc(cc1C(F)(F)F)N(C)C 50074377CCC(CC)Nc1nc(C)nc(n1)N(CC)c1ccc(cc1Br)C(C)C 50074378CCN(CC)c1nc(C)nc(n1)N(CC)c1ccc(cc1C(F)(F)F)N(C)C 50074379CCCCN(CC)c1cc(C)nc(n1)N(CC)c1ccc(I)cc1Br 50074380CCN(c1nc(C)cc(C)n1)c1ccc(cc1SC)C(C)C 50074381CCCN(CCC)c1nc(C)nc(n1)N(CC)c1ccc(cc1C)N(C)C 50074382CCN(CC)c1nc(C)nc(n1)N(CC)c1ccc(cc1Br)C(C)C 50074383CCCN(CC1CC1)c1cc(C)nc(n1)N(CC)c1ccc(cc1Br)C(C)C 50074384CCCN(CC1CC1)c1nc(C)nc(n1)N(CC)c1ccc(cc1C(F)(F)F)N(C)C 50074385CCN(c1nc(C)nc(n1)N(CCOC)CC1CC1)c1c(C)cc(C)cc1C 50074387CCN(CC)c1cc(C)nc(n1)N(CC)c1ccc(cc1Br)C(C)C 50074388CCCN(CCC)c1nc(C)nc(n1)N(CC)c1ccc(cc1C(F)(F)F)N(C)C 50074389CCN(CC)c1cc(C)nc(n1)N(CC)c1c(Br)cc(cc1OC)C(C)=O 50074390CCN(c1ccc(cc1C)N(C)C)c1nc(C)cc(C)n1 50074391CCN(c1nc(C)nc(n1)N(CC=C)CC=C)c1ccc(cc1Br)C(C)C 50074392CCN(c1nc(C)cc(C)n1)c1c(Br)cc(cc1OC)C(C)C 50074393CCN(CC)c1cc(C)nc(n1)N(CC)c1ccc(I)cc1Br 50074394CCCCN(CCC#N)c1nc(C)nc(n1)N(CC)c1ccc(cc1C)N(C)C 50074397CCCCN(CC)c1nc(C)nc(n1)N(CC)c1ccc(cc1Br)C(C)C 50074399CCCCN(CC)c1nc(C)nc(n1)N(CC)c1ccc(OC(F)(F)F)cc1Br 50074400CCN(CC)c1nc(C)nc(n1)N(CC)c1c(Br)cc(OC)cc1OC 50074401CCN(c1nc(C)nc(n1)N(CC=C)C1CC1)c1ccc(cc1Br)C(C)C 50074402CCN(c1nc(C)cc(C)n1)c1ccc(cc1SC)C(C)=O 50074403CCCCN(CCOC)c1nc(C)nc(n1)N(CC)c1c(C)cc(C)cc1C 50074404CCCN(CCC)c1nc(C)nc(n1)N(CC)c1ccc(cc1Br)C(C)C 50074406CCN(CCOC)c1nc(C)nc(n1)N(CC)c1c(C)cc(C)cc1C 50074407CCCCN(CC#N)c1nc(C)nc(n1)N(CC)c1ccc(cc1C)N(C)C 50074410CCN(c1nc(C)cc(n1)N(CCOC)CCOC)c1ccc(cc1Br)C(C)C 50074411CCN(c1nc(C)cc(C)n1)c1c(Br)cc(OC)cc1OC 50074412CCN(CC)c1cc(C)nc(n1)N(CC)c1ccc(cc1Br)N(C)C 50074413CCN(CC)c1cc(C)nc(n1)N(CC)c1ccc(cc1C(F)(F)F)N(C)C 50074414CCN(CCOC)c1cc(C)nc(n1)N(CC)c1ccc(cc1Br)C(C)C 50074443CCC(COC)Nc1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074444CCC(CCOC)Nc1nc(C)nc2n(cnc12)-c1ccc(cc1Br)C(C)C 50074445CCC(Nc1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C)C(=O)OC 50074446COCC(Cc1ccccc1)Nc1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074447CCCCN(CC)c1nc(C)nc2n(nnc12)-c1c(Cl)cc(OC)cc1OC 50074448COCCN(CCOC)c1nc(C)nc2n(nnc12)-c1ccc(cc1SC)C(C)C 50074449COCCN(CCOC)c1cc(C)nc2n(nnc12)-c1ccc(cc1SC)C(C)C 50074450CCCCN(CC)c1nc(C)nc2n(nnc12)-c1ccc(SC)cc1Br 50074451CCCC(Nc1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C)C(=O)N(C)C 50074452CCCCC(CC)Nc1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074453CCCCN(CC)c1cc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074454CCCCC(CCCC)Nc1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074455COCCN(CCOC)c1nc(C)nc2n(c(C)c(C)c12)-c1c(C)cc(C)cc1C 50074456COCCN(CCOC)c1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074457COCCN(CC1CC1)c1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074458CCCCN(CC)c1nc(C)nc2n(nnc12)-c1c(Br)cc(OC)cc1OC 50074459CCCCC(CC)Oc1nc(C)nc2n(cnc12)-c1ccc(cc1Br)C(C)C 50074460CCN(CCOC)c1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074461CCCCN(CC)c1nc(C)nc2n(nnc12)-c1c(C)cc(C)nc1C 50074462CCCCC(CC)Nc1nc(C)nc2n(nnc12)-c1c(C)cc(C)cc1C 50074463COCCN(CCOC)c1ncnc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074464COCCN(CCOC)c1nc(C)nc2n(c(C)nc12)-c1ccc(cc1Br)C(C)C 50074465CCCCN(CC)c1nc(C)nc2n(c(nc12)C(F)(F)F)-c1ccc(cc1Br)C(C)C 50074466CCCCNc1nc(C)nc2n(c(C)c(C)c12)-c1c(C)cc(C)cc1C 50074467COCCCNc1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074468CCCCN(CC)c1cc(C)nc2n(nnc12)-c1ccc(cc1SC)C(C)C 50074469COCCN(CCOC)c1nc(C)nc2n(nnc12)-c1c(C)cc(C)cc1C 50074470CCC(CC)Oc1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074471Cc1c(C)c2c(nc(C)nc2n1-c1c(C)cc(C)cc1C)N1CCOCC1 50074472CCCCN(CC)c1nc(C)nc2n(cnc12)-c1ccc(cc1Br)C(C)C 50074473CCN(C(COC)COC)c1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074474CCCC(CC)Nc1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074475COCCN(CCOC)c1nc(C)nc2n(cnc12)-c1c(Br)cc(OC)cc1OC 50074476COCCNc1nc(C)nc2n(nnc12)-c1c(C)cc(C)cc1C 50074477CCCCN(CCCC)c1nc(C)nc2n(cnc12)-c1ccc(cc1Br)C(C)C 50074478CCCCNc1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074479COCC(COC)Nc1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074480CCN(CCOC)c1nc(C)nc2n(cnc12)-c1ccc(cc1Br)C(C)C 50074481COCCN(CCOC)c1nc(C)nc2n(nnc12)-c1c(Br)cc(OC)cc1N(C)C 50074482CCC(COC)Oc1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074483COCC(Cc1ccccc1)Nc1nc(C)nc2n(nnc12)-c1c(C)cc(C)cc1C 50074484COCC(C)(C)Nc1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074485CC(C)c1ccc(c(Br)c1)-n1nnc2c(nc(C)nc12)N1CCCC1 50074486COCCN(CCOC)c1nc(C)nc2n(nnc12)-c1ccc(Br)cc1Br 50074487COCCN(Cc1cccnc1)c1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074488COCCN(CCOC)c1nc(C)nc2n(cnc12)-c1ccc(cc1Br)C(C)C 50074489CCCCN(CC)c1nc(C)nc2n(nnc12)-c1ccc(cc1Br)S(C)(=O)=O 50074490COCCN(Cc1ccccc1)c1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074491CCC(COC)Oc1nc(C)nc2n(cnc12)-c1ccc(cc1Br)C(C)C 50074492CCCCN(CC)c1nc(C)nc2n(c(C)nc12)-c1ccc(cc1Br)C(C)C 50074493CCOCC(COCC)Oc1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074494CCCCN(CC)c1cc(C)nc2n(nnc12)-c1ccc(cc1S(C)(=O)=O)C(C)C 50074495CCCCN(CC)c1cc(C)nc2n(c(C)nc12)-c1ccc(cc1Br)C(C)C 50074496CCCCN(CC)c1nc(C)nc2n(c(C)nc12)-c1c(Cl)cc(OC)cc1OC 50074497CC(C)c1ccc(c(Br)c1)-n1nnc2c(nc(C)nc12)N(CCO)CCO 50074498COCC(COC)Oc1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074499COCC(COC)N(C)c1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074500CCCCC(CC)Oc1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074501CCCCN(CC)c1nc(C)nc2n(c(C)c(C)c12)-c1c(C)cc(C)cc1C 50074502CCCCN(CC)c1ncnc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074503COCCN(CCOC)c1cc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074504COCCN(CCOC)c1nc(C)nc2n(cnc12)-c1c(C)cc(C)cc1C 50074505CCCCC(CC)Nc1nc(C)nc2n(cnc12)-c1ccc(cc1Br)C(C)C 50074506CCC(CO)Nc1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074507COCCN(CCO)c1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074508COCCN(CCOC)c1nc(C)nc2n(nnc12)-c1c(Cl)cc(OC)cc1OC 50074509CCCC(CCC)Nc1nc(C)nc2n(nnc12)-c1ccc(Br)cc1Br 50074510CCC(COC)Nc1nc(C)nc2n(nnc12)-c1c(C)cc(C)cc1C 50074511CCCCN(CCCC)c1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074512CCCCN(CC)c1nc(C)nc2n(cnc12)-c1c(Cl)cc(OC)cc1OC 50074513COCCN(CCOC)c1nc(C)nc2n(nnc12)-c1ccc(cc1)C(C)C 50074514CCCCN(CC)c1nc(C)nc2n(nnc12)-c1c(C)cc(C)cc1C 50074515CCN(CCOC)c1nc(C)nc2n(nnc12)-c1c(C)cc(C)cc1C 50074516CC(C)c1ccc(c(Br)c1)-n1nnc2c(NC3CCCC3)nc(C)nc12 50074517CCCCN(CC)c1nc(C)nc2n(nnc12)-c1ccc(Br)cc1Br 50074518COCCN(CCOC)c1nc(C)nc2n(nnc12)-c1ccc(cc1C(F)(F)F)N(C)C 50074519CCCCN(CC)c1nc(C)nc2n(nnc12)-c1ccc(cc1C(F)(F)F)N(C)C 50074520COCCN(CC=C)c1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074521CCN(CCN(C)C)c1nc(C)nc2n(cnc12)-c1ccc(cc1Br)C(C)C 50074522CCCCN(CC)c1nc(C)nc2n(cnc12)-c1c(Br)cc(OC)cc1OC 50074523CCCCN(CC)c1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074524CCCC(C)Nc1nc(C)nc2n(nnc12)-c1c(C)cc(C)cc1C 50074525CCCC(CCC)Nc1nc(C)nc2n(nnc12)-c1c(C)cc(C)cc1C 50074526CCCC(CN(C)C)Nc1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074527COCCN(CCOC)c1cc(C)nc2n(c(C)nc12)-c1ccc(cc1Br)C(C)C 50074528CCC(CC)Nc1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074529COCCN(CCOC)c1nc(C)nc2n(nnc12)-c1c(Br)cc(OC)cc1OC 50074530COCCN(CCOC)c1nc(C)nc2n(nnc12)-c1ccc(cc1Br)N(C)C 50074531COCCCN(CCOC)c1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074532CCCCN(CC)c1nc(C)nc2n(cnc12)-c1c(C)cc(C)cc1C 50074533CC(C)c1ccc(c(Br)c1)-n1nnc2c(nc(C)nc12)N1CCCCC1 50074534CCCC(CC)Nc1nc(C)nc2n(cnc12)-c1ccc(cc1Br)C(C)C 50074535CCC(CO)Nc1nc(C)nc2n(c(C)c(C)c12)-c1c(C)cc(C)cc1C 50074536CCC(CC)Nc1nc(C)nc2n(nnc12)-c1c(C)cc(C)cc1C 50074537COCCN(CCOC)c1nc(C)nc2n(nnc12)-c1ccc(OC(F)(F)F)cc1Br 50074538COCCN(CCOC)c1cc(C)nc2n(nnc12)-c1ccc(cc1S(C)(=O)=O)C(C)C 50074539COCCNc1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074540CCN(CC)c1nc(C)nc2n(cnc12)-c1ccc(cc1Br)C(C)C 50074541COCCN(CCOC)c1nc(C)nc2n(nnc12)-c1ccc(cc1S(C)(=O)=O)C(C)C 50074542CCC(CC)Oc1nc(C)nc2n(cnc12)-c1ccc(cc1Br)C(C)C 50074543CCCCN(CC)c1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)=O 50074544CCCCN(CC)c1nc(C)nc2n(c(nc12)-c1ccccc1)-c1c(Cl)cc(OC)cc1OC 50074545COCCN(CCOC)c1nc(C)nc2n(nnc12)-c1c(C)cc(C)nc1C 50074546CCCC(CCC)Nc1nc(C)nc2n(cnc12)-c1ccc(cc1Br)C(C)C 50074547CCCCN(CC)c1nc(C)nc2n(c(CCCC)nc12)-c1c(Cl)cc(OC)cc1OC 50074548CCN(CC)c1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074549CCC(COC)N(C)c1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C 50074550COCCCN(CCOC)c1nc(C)nc2n(cnc12)-c1c(Cl)cc(OC)cc1OC 50074551COCCNc1nc(C)nc2n(cnc12)-c1ccc(cc1Br)C(C)C 50076602CCCCN(CC)c1nc(C)nc2n(c(Cl)nc12)-c1ccc(cc1Br)C(C)C 50076603CCCCN(CC)c1nc(C)nc2n(c(OCC3CC3)nc12)-c1ccc(cc1Br)C(C)C 50076604CCCCC(CC)Nc1nc(C)nc2n(-c3c(C)cc(C)cc3C)c(=O)n(C)c12 50076605CCCCN(CC)c1nc(C)nc2n(-c3ccc(cc3Br)C(C)C)c(=O)[nH]c12 50076606COCCN(CCOC)c1nc(C)nc2n(-c3ccc(cc3Br)C(C)C)c(=O)n(C)c12 50076607CCC(COC)Nc1nc(C)nc2n(-c3ccc(cc3Br)C(C)C)c(=O)n(C)c12 50076608CCCCN(CC)c1cc(C)nc2n(-c3ccc(cc3Br)C(C)C)c(=O)n(C)c12 50076609CCCCN(CC)c1nc(C)nc2n(-c3c(C)cc(C)cc3C)c(=O)n(C)c12 50076610CCCCN(CC)c1nc(C)nc2n(-c3c(C)cc(C)nc3C)c(=O)n(C)c12 50076611CCCCN(CC)c1nc(C)nc2n(-c3ccc(cc3Br)C(C)C)c(=O)n(CC3CC3)c12 50076612COCCNc1nc(C)nc2n(-c3ccc(cc3Br)C(C)C)c(=O)n(C)c12 50076613CCCCN(CC)c1nc(C)nc2n(c(OC)nc12)-c1ccc(cc1Br)C(C)C 50076614COCCN(Cc1ccccc1)c1nc(C)nc2n(-c3ccc(cc3Br)C(C)C)c(=O)n(C)c12 50076615CCCN(CCC)c1nc(C)nc2n(-c3ccc(cc3Br)C(C)C)c(=O)n(C)c12 50076616CCCN(CC1CC1)c1nc(C)nc2n(-c3ccc(cc3Br)C(C)C)c(=O)n(C)c12 50076617CCCCN(CC)c1nc(C)cc2n(-c3ccc(cc3Br)C(C)C)c(=O)n(C)c12 50076618CCCN(CC1CC1)c1nc(C)nc2n(-c3c(C)cc(C)nc3C)c(=O)n(C)c12 50076619CCCCN(CC)c1nc(C)nc2n(-c3ccc(cc3Br)C(C)C)c(=O)n(C)c12 50076620CCCCC(CC)Nc1nc(C)nc2n(-c3ccc(cc3Br)C(C)C)c(=O)n(C)c12 50076621COCCN(CCOC)c1nc(C)nc2n(-c3c(C)cc(C)cc3C)c(=O)n(C)c12 50076622CCCN(CCC)c1nc(C)nc2n(-c3c(C)cc(C)nc3C)c(=O)n(C)c12 50076623COCCN(CC1CC1)c1nc(C)nc2n(-c3ccc(cc3Br)C(C)C)c(=O)n(C)c12 50076624CCCN(CC1CC1)c1nc(C)nc2n(-c3c(C)cc(C)cc3C)c(=O)n(C)c12 50076625CCN(CCOC)c1nc(C)nc2n(-c3ccc(cc3Br)C(C)C)c(=O)n(C)c12 50076626CCCCN(CC)c1nc(C)nc2n(c(nc12)N1CCOCC1)-c1ccc(cc1Br)C(C)C 50076746CCN(c1nc(C)cc(n1)-c1ccccc1C(F)(F)F)c1ccc(cc1Br)C(C)=O 50076747CCN(c1nc(C)cc(n1)-c1ccccc1C#N)c1ccc(cc1Br)C(C)C 50076748CCN(c1nc(C)cc(n1)-c1cccnc1)c1c(Br)cc(OC)cc1OC 50076749CCN(c1nc(C)cc(n1)-c1ccccc1OC)c1c(Br)cc(OC)cc1OC 50076750CCN(c1nc(C)cc(n1)-c1ccccn1)c1c(Br)cc(OC)cc1OC 50076751CCN(c1nc(C)cc(n1)-c1ccccc1Cl)c1c(Br)cc(OC)cc1OC 50076752CCN(c1nc(C)cc(n1)-c1ccccc1N(C)C)c1ccc(cc1Br)C(C)C 50076753CCN(c1nc(C)cc(n1)-c1c(C)cc(C)cc1C)c1ccc(cc1Br)C(C)C 50076754CCN(c1nc(C)cc(n1)-c1ccccc1C(F)(F)F)c1ccc(cc1Br)C(C)C 50076755CCN(c1nc(C)cc(n1)-c1ccccc1C(O)=O)c1ccc(cc1Br)C(C)C 50076756CCN(c1nc(C)cc(n1)-c1ccccc1-c1ccccc1)c1ccc(cc1Br)C(C)C 50076757CCN(c1nc(C)cc(n1)-c1ccccc1C)c1ccc(cc1Br)C(C)C 50076758CCN(c1nc(C)cc(n1)-c1ccccc1C(F)(F)F)c1c(Br)cc(cc1OC)N(C)C 50076759CCN(c1nc(C)cc(n1)-c1ccccc1Cl)c1ccc(cc1Br)C(C)C 50076760CCN(c1nc(C)cc(n1)-c1cccc(c1)-c1ccccc1)c1ccc(cc1Br)C(C)C 50076761CCN(c1nc(C)cc(n1)-c1ccccc1C(F)(F)F)c1c(Br)cc(OC)cc1OC 50076762CCN(c1nc(C)cc(n1)-c1ccccc1)c1c(Br)cc(OC)cc1OC 50076763CCN(c1nc(C)cc(n1)-c1ccccc1F)c1ccc(cc1Br)C(C)C 50076764CCN(c1nc(C)cc(n1)-c1ccccc1C(F)(F)F)c1ccc(SC)cc1Br 50076765CCN(c1nc(C)cc(n1)-c1ccccc1[N+]([O-])=O)c1ccc(cc1Br)C(C)C 50076766CCN(c1nc(C)cc(n1)-c1cccc2ccccc12)c1ccc(cc1Br)C(C)C 50076767CCN(c1nc(C)cc(n1)-c1ccccc1NC)c1ccc(cc1Br)C(C)C 50076768CCN(c1nc(C)cc(n1)-c1ccccc1C(F)(F)F)c1ccc(Br)cc1Br 50076769CCN(c1nc(C)cc(n1)-c1ccccc1N)c1ccc(cc1Br)C(C)C 50076770CCN(c1nc(C)cc(n1)-c1ccccc1-c1nnn[nH]1)c1ccc(cc1Br)C(C)C 50076771CCN(c1nc(C)cc(n1)-c1ccccc1C(F)(F)F)c1ccc(cc1Br)S(C)(=O)=O 50076772CCN(c1nc(C)cc(n1)-c1cccc(c1)C(F)(F)F)c1ccc(cc1Br)C(C)C 50076773CCN(c1nc(C)cc(n1)-c1c(C)cc(C)nc1C)c1c(C)cc(cc1Br)C(C)C 50076774CCN(c1nc(C)cc(n1)-c1ccccc1)c1ccc(cc1Br)C(C)C 50076775CCN(c1nc(C)cc(n1)-c1c(Cl)cccc1Cl)c1ccc(cc1Br)C(C)C 50076776CCN(c1nc(C)cc(n1)-c1ccccc1Br)c1ccc(cc1Br)C(C)C 50076777COc1cc(Br)c(c(OC)c1)-n1c(C)nc2c(nc(C)nc12)-c1ccccc1C(F)(F)F 50076778Cc1cc(C)c(c(C)c1)-n1nnc2c(nc(C)nc12)-c1ccccc1C(F)(F)F 50076779CCN(c1nc(C)nc(n1)-c1ccccc1C(F)(F)F)c1ccc(cc1Br)C(C)C 50076780COc1cc(Br)c(Nc2nc(C)nc(-c3ccccc3C(F)(F)F)c2[N+]([O-])=O)c(OC)c1 50076781COc1cc(Br)c(c(OC)c1)-n1c2nc(C)nc(-c3ccccc3C(F)(F)F)c2[nH]c1=O 50076782CCN(CC1CC1)c1nc(C)nc(Nc2c(Cl)cc(Cl)cc2Cl)c1C 50076783CSc1nn(-c2c(Cl)cc(Cl)cc2Cl)c2nc(C)nc(-c3ccccc3C(F)(F)F)c12 50076784COc1cc(Br)c(Nc2nc(C)nc(c2N)-c2ccccc2C(F)(F)F)c(OC)c1 50076785Cc1c(C)c2c(nc(C)nc2n1-c1c(C)cc(C)cc1C)-c1ccccc1C(F)(F)F 50076786COc1cc(Br)c(c(OC)c1)-n1nnc2c(nc(C)nc12)-c1ccccc1C(F)(F)F 50076787COc1cc(Br)c(c(OC)c1)-n1c2nc(C)nc(-c3ccccc3C(F)(F)F)c2n(C)c1=O 50076892CCN(CC)c1nc(C)nc2n(-c3c(C)cc(C)cc3C)c(=O)sc12 50076893CCCN(CC1CC1)c1nc(C)nc2n(-c3ccc(cc3Br)C(C)C)c(=S)sc12 50076894COCCN(CCOC)c1nc(C)nc2n(-c3ccc(cc3Br)C(C)C)c(=O)sc12 50076895CC(C)c1ccc(c(Br)c1)-n1c2nc(C)nc(N3CCOCC3)c2sc1=S 50076896CCCCN(CC)c1nc(C)nc2n(-c3ccc(cc3Br)C(C)C)c(=S)sc12 50076897CCCN(CC1CC1)c1nc(C)nc2n(-c3c(C)cc(C)cc3C)c(=S)sc12 50076898CCCN(CC1CC1)c1nc(C)nc2n(-c3c(C)cc(C)cc3C)c(=O)sc12 50076899COCCN(CCOC)c1nc(C)nc2n(-c3ccc(cc3Br)C(C)C)c(=S)sc12 50076900CCN(CC)c1nc(C)nc2n(-c3ccc(cc3Br)C(C)C)c(=O)sc12 50076901CCN(CC)c1nc(C)nc2n(-c3c(C)cc(C)cc3C)c(=S)sc12 50076902COCCN(CCOC)c1nc(C)nc2n(-c3c(C)cc(C)cc3C)c(=O)sc12 50076903CCCN(CC1CC1)c1nc(C)nc2n(-c3ccc(cc3Br)C(C)C)c(=O)sc12 50076904CCC(C)N(C(C)CC)c1nc(C)nc2n(-c3ccc(cc3Br)C(C)C)c(=S)sc12 50076905CCN(CC)c1nc(C)nc2n(-c3ccc(cc3Br)C(C)C)c(=S)sc12 50076906COCCN(CCOC)c1nc(C)nc2n(-c3c(C)cc(C)cc3C)c(=S)sc12 50078345CCCN(CC1CC1)c1nc(C)nc(Nc2c(OC)cc(OC)cc2OC)n1 50084868CCOCC(COCC)Nc1nc(C)nc2c(c(C)nn12)-c1ccc(Cl)cc1Cl 50084869CCN(CC)c1nc(C)nc2c(c(C)nn12)-c1ccc(Cl)cc1Cl 50084870CCCCC(CC)Nc1nc(C)nc2c(c(C)nn12)-c1ccc(Cl)cc1Cl 50084871CN(c1ccccc1)c1nc(C)nc2c(c(C)nn12)-c1ccc(Cl)cc1Cl 50084872CCC(COC)Nc1nc(C)nc2c(c(C)nn12)-c1ccc(Cl)cc1Cl 50084873CCC(CC)Nc1nc(C)nc2c(c(C)nn12)-c1ccc(Cl)cc1Cl 50084874CCCCN(CC)c1nc(C)nc2c(c(C)nn12)-c1ccc(Cl)cc1Cl 50084875COCC(COC)Nc1nc(C)nc2c(c(C)nn12)-c1ccc(Cl)cc1Cl 50084876CCCN(CCC)c1nc(C)nc2c(c(C)nn12)-c1ccc(Cl)cc1Cl 50084877CCCC(CC)Nc1nc(C)nc2c(c(C)nn12)-c1ccc(Cl)cc1Cl 50084878CCCCN(CC)c1nc(C)nc2c(c(C)nn12)-c1ccc(Cl)cc1Cl 50084879COCCN(CCOC)c1nc(C)nc2c(c(C)nn12)-c1ccc(Cl)cc1Cl 50084880CCCN(CC1CC1)c1nc(C)nc2c(c(C)nn12)-c1ccc(Cl)cc1Cl 50084881CCCC(CCC)Nc1nc(C)nc2c(c(C)nn12)-c1ccc(Cl)cc1Cl 50087702COCC(COC)n1nnc2c(Nc3c(C)cc(C)cc3Cl)nc(C)cc12 50087703NA 50087704NA 50087706NA 50087707CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ccc(OC)cc1OC 50087709NA 50087711CC[C@H](C)[C@H](NC(=O)[C@@H](NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](NC(=O)[C@H](CCSC)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(O)=O)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@H]1CCCN1C(=O)CNC(=O)[C@@H](N)CCC(N)=O)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)O)C(N)=O 50087713CCC(CC)Nc1cc(C)nc2c(c(C)nn12)-c1ccc(OC)cc1C 50087714CCCN(CCOC)c1cc(C)nc2c(c(C)nn12)-c1ccc(OC)c(OC)c1 50087719CCC(CC)n1nnc2c(nc(C)cc12)N1CCc2cc(Cl)cc(Cl)c12 50087722NA 50107068CCCN(C(C1CC1)C1CC1)c1nnc([nH]1)-c1c(C)cc(C)cc1C 50107069CCCN(C(C1CC1)C1CC1)c1nc(-c2ccc(Cl)cc2OC)n(C)n1 50107070CCCN(C(C1CC1)C1CC1)c1nc(-c2c(C)cc(C)cc2C)n(CC=C)n1 50107071CCCN(C(C1CC1)C1CC1)c1nc(-c2c(C)cc(C)cc2C)n(C)n1 50107072CCCN(C(C1CC1)C1CC1)c1nc(-c2c(C)cc(C)cc2C)n(CC)n1 50107073CCCN(c1nc(-c2ccc(Cl)cc2Cl)n(C)n1)c1ccccc1OC 50107074CCCN(C(C1CC1)C1CC1)c1nc(-c2ccc(Cl)cc2C)n(C)n1 50107075CCCN(C(C1CC1)C1CC1)c1nnc([nH]1)-c1ccc(Cl)cc1Cl 50107076CCCN(C(C1CC1)C1CC1)c1nc(-c2ccc(C)cc2C)n(C)n1 50107078CCCN(CCC)c1nc(-c2ccc(Cl)cc2Cl)n(CCO)n1 50107079CCCN(CCC)c1nc(-c2ccc(Cl)cc2Cl)n(C)n1 50107080CCCN(C(C1CC1)C1CC1)c1nc(-c2ccc(Cl)cc2)n(C)n1 50107081CCCN(C(C1CC1)C1CC1)c1nc(-c2c(C)cc(C)cc2C)n(CC(F)(F)F)n1 50107083CCCN(C(C1CC1)C1CC1)c1nc(-c2ccc(Cl)cc2Cl)n(C)n1 50107084CCCN(C(C1CC1)C1CC1)c1nc(-c2ccc(Cl)cc2Cl)n(CC)n1 50107085CCCN(C(C1CC1)C1CC1)c1nc(-c2cc(F)c(Cl)cc2Cl)n(C)n1 50107086CCCN(C(C1CC1)C1CC1)c1nc(-c2ccc(Br)cc2C)n(C)n1 50113150CC(=O)C(Nc1cccc(Cl)c1)=NNc1ccc(Br)cc1 50113152CC(=O)C(Nc1ccc(Cl)cc1)=NNc1ccccc1C 50113153CC(=O)C(Nc1cccc(C)c1)=NNc1ccccc1C 50113154CC(=O)C(Nc1cccc(c1)C(F)(F)F)=NNc1ccccc1C 50113155CC(=O)C(Nc1ccccc1)=NNc1ccccc1C 50113158CN(C(=NNc1ccccc1[N+]([O-])=O)C(C)=O)c1cccc(Cl)c1 50113159CC(=O)C(Nc1cccc(Cl)c1)=NNc1ccccc1Cl 50113162CC(=O)C(Nc1cccc(Cl)c1)=NNc1ccccc1C#N 50113163CC(=O)C(Nc1cccc(Cl)c1)=NNc1ccccc1 50113166CC(=O)C(Oc1ccc(Cl)cc1)=NNc1ccccc1C#N 50113168CC(=O)C(Nc1ccccc1)=NNc1ccccc1C#N 50113171CC(=O)C(Nc1ccc(Cl)cc1)=NNc1ccccc1Cl 50113172CC(=O)C(Nc1cccc(Cl)c1)=NNc1ccc(C)cc1 50113174CC(=O)C(Nc1ccccc1)=NNc1ccccc1C(F)(F)F 50113180CC(=O)C(Nc1cccc(C)c1)=NNc1ccccc1C(F)(F)F 50113181CC(=O)C(Nc1cccc(c1)C#C)=NNc1ccccc1C 50113182CC(=O)C(Nc1ccccc1)=NNc1ccccc1 50113184CC(=O)C([N-]c1cccc(Cl)c1)=[NH+]Nc1ccccc1[N+]([O-])=O 50113187COc1cccc(NC(=NNc2ccccc2C(F)(F)F)C(C)=O)c1 50113188CC(=O)C(Nc1cccc(c1)C#C)=NNc1ccccc1C(F)(F)F 50113189CC(=O)C(Nc1cccc(F)c1)=NNc1ccccc1Cl 50113190CC(=O)C(Nc1ccccc1)=NNc1ccccc1Cl 50113191CC(=O)C(Nc1cccc(C)c1)=NNc1ccccc1 50113196COc1cccc(OC(=NNc2ccccc2C#N)C(C)=O)c1 50113199CC(=O)C(Nc1cccc(Cl)c1)=NNc1ccccc1C 50113200COc1cccc(NC(=NNc2ccccc2C)C(C)=O)c1 50113201CC(=O)C(Nc1cccc(F)c1)=NNc1ccccc1C 50113203CC(=O)C(Nc1cccc(Cl)c1)=NNc1ccccc1C(F)(F)F 50113205CC(=O)C(Oc1cccc(C)c1)=NNc1ccccc1C#N 50113206CC(=O)C(Nc1cccc(C)c1)=NNc1ccccc1Cl 50113208CC(=O)C(Nc1cccc(F)c1)=NNc1ccccc1C(F)(F)F 50113209CC(=O)C(Nc1cccc(c1)C#C)=NNc1ccccc1Cl 50113210COc1cccc(NC(=NNc2ccccc2Cl)C(C)=O)c1 50116092CCCN(CCC)c1nc(C)nc2c(-c3c(C)cc(C)cc3C)n(CC)nc12 50116093CCCN(CC)c1nc(C)nc2c(-c3ccc(Cl)cc3Cl)n(C)nc12 50116094CCC(CC)Nc1nc(C)nc2c(-c3ccc(Cl)cc3Cl)n(C)nc12 50116095CCCN(CCC)c1nc(C)nc2c(-c3ccc(Cl)cc3Cl)n(C)nc12 50116096CCCCCNc1nc(C)nc2c(-c3ccc(Cl)cc3Cl)n(C)nc12 50116097CCCN(CCC)c1nc(C)nc2c(n[nH]c12)-c1c(C)cc(C)cc1C 50116098CCCN(CCN1CCCC1)c1nc(C)nc2c(-c3ccc(Cl)cc3Cl)n(C)nc12 50116099CCCN(CCC)c1nc(C)nc2c(-c3c(C)cc(C)cc3C)n(CCC)nc12 50116100CCNc1nc(C)nc2c(-c3ccc(Cl)cc3Cl)n(C)nc12 50116101CCCN(CCC)c1nc(C)nc2c(nn(CC)c12)-c1c(C)cc(C)cc1C 50116103CCCN(CCC)c1nc(C)nc2c(-c3ccc(OC)cc3OC)n(C)nc12 50116104CCCN(CCC)c1nc(C)nc2c(-c3c(C)cc(C)cc3C)n(C)nc12 50116105CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1cnc(cc1C)N(C)C 50116106CCCN(CCC)c1nc(C)nc2c(-c3c(Cl)cccc3Cl)n(C)nc12 50116107CCCCNc1nc(C)nc2c(-c3ccc(Cl)cc3Cl)n(C)nc12 50116108CCCCCCNc1nc(C)nc2c(-c3ccc(Cl)cc3Cl)n(C)nc12 50116109CCCN(CCC)c1nc(C)nc2c(-c3ccc(Cl)cc3C)n(C)nc12 50116110CCCN(CCN1CCCCC1)c1nc(C)nc2c(-c3ccc(Cl)cc3Cl)n(C)nc12 50116112CCCN(CCC)c1nc(C)nc2c(nn(C)c12)-c1c(C)cc(C)cc1C 50116113CCCCCCN(CC)c1nc(C)nc2c(-c3ccc(Cl)cc3Cl)n(C)nc12 50116115Cc1nc(NC2CCCCC2)c2nn(C)c(-c3ccc(Cl)cc3Cl)c2n1 50116117CCCN(CCC)c1nc(C)nc2c(nn(CCC)c12)-c1c(C)cc(C)cc1C 50116118COCCN(CCOC)c1nc(C)nc2c(-c3ccc(Cl)cc3Cl)n(C)nc12 50116119CCCN(CCC)c1nc(C)nc2c(-c3ccccc3Cl)n(C)nc12 50116120CCCNc1nc(C)nc2c(-c3ccc(Cl)cc3Cl)n(C)nc12 50116121Cc1nc(NC2CCCC2)c2nn(C)c(-c3ccc(Cl)cc3Cl)c2n1 50116122CCCN(CCN(C)C)c1nc(C)nc2c(-c3ccc(Cl)cc3Cl)n(C)nc12 50116123CCCCN(CC)c1nc(C)nc2c(-c3ccc(Cl)cc3Cl)n(C)nc12 50119593NA 50119598NA 50119599NA 50119600NA 50119602CCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(O)=O)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)C1CCCN1C(=O)C1CCCN1C(=O)CNC(=O)[C@@H](N)CCC(O)=O)C(C)CC)C(C)CC)C(=O)N[C@@H](C(C)CC)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](C(C)CC)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@H]1CCC(=O)NCCCC[C@H](NC(=O)[C@@H](C)NC(=O)[C@H](CCC(N)=O)NC1=O)C(=O)N(C)[C@@H](CC(N)=O)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](C(C)O)C(=O)N[C@@H](C(C)CC)C(N)=O 50119607NA 50119611NA 50119614NA 50119615NA 50119616NA 50130959CCCN(CCC)c1c(C)nc(-c2ccc(Cl)cc2Cl)n(CC)c1=O 50130960CCCN(CCC)c1c(C)nc(-c2c(C)cc(C)cc2C)n(CC)c1=O 50130961CCCN(CCC)c1c(C)nc(-c2ccc(OC)cc2OC)n(C)c1=O 50130962CCCN(CCC)c1c(C)nc(-c2ccc(OC)cc2OC)n(CCC)c1=O 50130963CCCN(CCC)c1c(C)nc(-c2ccc(OC)cc2OC)n(CC)c1=O 50130964CCCN(CCC)c1c(C)nc(-c2c(C)cc(C)cc2OC)n(CCF)c1=O 50130965CCCN(CCC)c1c(C)nc(-c2c(OC)cccc2OC)n(CC)c1=O 50130966CCCN(CCC)c1c(C)nc(-c2c(C)cc(C)cc2OC)n(CC(F)(F)F)c1=O 50130967CCCN(CCC)c1c(C)nc(-c2c(OC)cccc2OC(F)F)n(CC)c1=O 50130968CCCN(CCC)c1c(C)nc(-c2ccc(OC)cc2OC)n(CCOC)c1=O 50130969CCCN(CCC)c1c(C)nc(-c2c(C)cc(C)cc2C)n(C)c1=O 50130970CCCN(CCC)c1c(C)nc(-c2c(C)cc(C)cc2OC)n(C)c1=O 50130971CCCN(CCC)c1c(C)nc(-c2c(C)cc(C)cc2OC)n(CC)c1=O 50130972CCCN(CCC)c1c(C)nc(-c2ccc(OC)cc2OC)n(CC2CC2)c1=O 50130973CCCN(CCC)c1c(CC)nc(-c2c(C)cc(C)cc2OC)n(CC)c1=O 50130974CCCN(CCC)c1c(CC)nc([nH]c1=O)-c1c(C)cc(C)cc1OC 50130975CCCN(CCC)c1c(CC)nc(-c2c(C)cc(C)cc2OC)n(C)c1=O 50130976CCCN(CCC)c1c(C)nc(-c2c(OC)cccc2OC)n(C)c1=O 50130977CCCN(CCC)c1c(C)nc(-c2c(C)cc(C)cc2OC)n(C(C)C)c1=O 50130978CCCN(CCC)c1c(C)nc(-c2c(C)cc(C)cc2OC)n(CCC)c1=O 50130979CCCN(CCC)c1c(C)nc([nH]c1=O)-c1c(C)cc(C)cc1OC 50132884CCCCN(CCCC)c1cc(C)nc2c(-c3ccc(Cl)cc3Cl)n(CCC)nc12 50132885CCCCN(CCCC)c1cc(C)nc2c(nn(C(C)C)c12)-c1ccc(Cl)cc1Cl 50132886CCCCN(CC)c1cc(C)nc2c(n[nH]c12)-c1ccc(Cl)cc1Cl 50132887CCCCN(CCCC)c1cc(C)nc2c(-c3c(C)cc(C)cc3C)n(C)nc12 50132888CCCCN(CC)c1cc(C)nc2c(-c3ccc(Cl)cc3Cl)n(CC)nc12 50132889CCCCN(CCCC)c1cc(C)nc2c(-c3ccc(Cl)cc3Cl)n(C)nc12 50132890CCCN(CC1CC1)c1cc(C)nc2c(n[nH]c12)-c1ccc(Cl)cc1Cl 50132891CCCN(CCC)c1cc(C)nc2c(-c3ccccc3)n(C)nc12 50132892CCCCN(CC)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132893CCCCN(CCCC)c1cc(C)nc2c(n[nH]c12)-c1ccc(Cl)cc1Cl 50132894CCCN(CC1CC1)c1cc(C)nc2c(-c3ccc(Cl)cc3Cl)n(C)nc12 50132895CCCN(CC1CC1)c1cc(C)nc2c(-c3ccc(Cl)cc3Cl)n(CC)nc12 50132896CCCN(CCC)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132897CCCCN(CCc1ccc(OC)cc1)c1cc(C)nc2c(-c3ccc(Cl)cc3Cl)n(C)nc12 50132898CCCCN(CCCC)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132899CCCN(CCC)c1cc(C)nc2c(-c3ccc(Cl)cc3Cl)n(C)nc12 50132900CCCN(CC1CC1)c1cc(C)nc2c(-c3ccc(C)cc3Cl)n(CC)nc12 50132901CCCN(CC1CC1)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132902CCCCN(CCCC)c1cc(C)nc2c(nn(CC)c12)-c1ccc(Cl)cc1Cl 50132903CCCCN(CCCC)c1cc(C)nc2c(-c3ccc(OC)cc3Cl)n(C)nc12 50132904CCCCN(CC)c1cc(C)nc2c(nn(CC)c12)-c1ccc(Cl)cc1Cl 50132905CCCCN(CCCC)c1cc(C)nc2c(-c3ccc(Cl)cc3Cl)n(nc12)C(C)C 50132906CCCCN(CC)c1cc(C)nc2c(-c3ccc(Cl)cc3Cl)n(C)nc12 50132907CCCN(CC1CC1)c1cc(C)nc2c(nn(CC)c12)-c1ccc(Cl)cc1Cl 50132908CCCCN(CCCC)c1cc(C)nc2c(nn(CCC)c12)-c1ccc(Cl)cc1Cl 50132909CCCN(CCC)c1cc(C)nc2c(-c3ccc(Cl)cc3)n(C)nc12 50132910CCCCN(CCCC)c1cc(C)nc2c(-c3ccc(Cl)cc3Cl)n(CC)nc12 50132911CCCCN(CCCC)c1cc(C)nc2c(-c3ccc(C)cc3Cl)n(CC)nc12 50132912CCCCN(CCCC)c1cc(C)nc2c(nn(C)c12)-c1ccc(C)cc1Cl 50132913CCCCCN(CCC)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132914CCCCN(CCSC)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132915CCCN(CCCOC)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132916CCCN(CCOC)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132917COCCN(C(C)C)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132918CCCCN(CC1CCCO1)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132919CCCCN(CCCOC)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132920CCCCN(CCc1ccccn1)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132921CCCCCN(CC)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132922CCCCN(C(CC)CC)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132923CCCCCN(CC1CC1)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132924CCCCCCN(CC1CC1)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132925CCN(CCCOC)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132926CCN(CCOC)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132927CCCCN(CC1CC1)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132928CCCCCN(CCOC)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132929CCCCNc1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132930COCCN(CCOC)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132931CCCCN(Cc1ccncc1)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132932CCN(CC1CC1)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132933CCCCN(CCCC)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1 50132934CCCCN(CCCC)c1cc(C)nc2c(nn(C)c12)-c1c(C)cc(C)cc1Cl 50132935CCCCN(CCCC)c1cc(C)nc2c(nn(C)c12)-c1c(C)cc(C)cc1C 50132936CCCCN(CCOC)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132937COCCN(C)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132938CCCN(CC)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132940CCCC(CO)Nc1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132941CCCCN(CCc1ccncc1)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132942CCCN(CCO)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132943CC(C)CN(CC1CC1)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132944CCCCCCN(CCOC)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132945COCCN(CC(C)C)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132946CCCN(Cc1ccc(O)cc1)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132947CCCCN(CC1CCCN1C)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132948CCCCN(CCCC)c1cc(C)nc2c(nn(C)c12)-c1ccc(OC)cc1Cl 50132949CCCN(C)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132950CCCCCN(CCCC)c1cc(C)nc2c(nn(C)c12)-c1ccc(Cl)cc1Cl 50132951CCCN(CCC)c1cc(C)nc2c(cccc12)-c1ccc(Cl)cc1Cl 50132952COCCN(CCOC)c1cc(C)nc2c(cccc12)-c1ccc(Cl)cc1Cl 50132953CCCN(Cc1ccccc1)c1cc(C)nc2c(cccc12)-c1ccc(Cl)cc1Cl 50132954CSc1cc(C)nc2c(cccc12)-c1ccc(Cl)cc1Cl 50132955CCCCN(CC)c1cc(C)nc2c(cccc12)-c1ccc(Cl)cc1Cl 50132956Cc1cc(C)c2cccc(-c3ccc(Cl)cc3Cl)c2n1 50132957CCCN(CCC)c1cc(C)nc2c(cccc12)-c1ccccc1 50132958COCCN(CCOC)c1cc(C)nc2c(c(C)ccc12)-c1ccc(Cl)cc1Cl 50132959CCCN(CCC)c1cc(C)nc2c(cccc12)-c1ccc(C)cc1 50132960Cc1cc(Cl)c2cccc(-c3ccc(Cl)cc3Cl)c2n1 50132961CCCCN(CC)c1cc(C)nc2c(cccc12)-c1c(C)cc(C)cc1C 50132962CCCN(CCC)c1cc(C)nc2c(c(OC)ccc12)-c1ccc(Cl)cc1 50132963CCCN(CCC)c1cc(C)nc2c(cccc12)-c1ccc(OC)cc1 50132964CCCN(Cc1ccccc1)c1cc(C)nc2c(cccc12)-c1c(C)cc(C)cc1C 50132965CCCN(CC1CC1)c1cc(C)nc2c(cccc12)-c1ccc(Cl)cc1Cl 50132966CCCN(CC1CC1)c1cc(C)nc2c(c(C)ccc12)-c1ccc(Cl)cc1Cl 50132967CCCN(CCC)c1cc(C)nc2c(c(C)ccc12)-c1ccc(Cl)cc1Cl 50132968COc1cc(C)nc2c(cccc12)-c1ccc(Cl)cc1Cl 50132969CCCN(CCC)c1cc(C)nc2c(cccc12)-c1c(C)cc(C)cc1C 50132971CCCCN(CCC)c1cc(C)nc2c(cccc12)-c1c(C)cc(C)cc1C 50132972COCCN(CCOC)c1cc(C)nc2c(cccc12)-c1c(C)cc(C)cc1C 50132973CCCN(CC1CC1)c1cc(C)nc2c(cccc12)-c1c(C)cc(C)cc1C 50132974CCCN(CCC)c1cc(C)nc2c(cccc12)-c1ccc(OC)cc1OC 50132975CCCN(CCC)c1cc(C)nc2c(cccc12)-c1ccc(Cl)cc1 50135327CCCN(CC1CC1)Cc1sc(Nc2ccc(cc2Br)C(C)C)nc1C(F)(F)F 50135328CCCN(CC1CC1)Cc1sc(Nc2c(Cl)cc(cc2Cl)C(F)(F)F)nc1C(F)(F)F 50135329CCCN(CC1CC1)Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F 50135330CCCN(CC1CC1)Cc1sc(Nc2ccc(OC)cc2OC)nc1C(F)(F)F 50135333CCCN(CC1CC1)Cc1oc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F 50135334CCCN(CC1CC1)Cc1sc(nc1C(F)(F)F)N(CC)c1ccc(cc1Br)C(C)C 50135336CCCN(CC1CC1)Cc1sc(nc1C(F)(F)F)N(C)c1c(C)cc(C)cc1Cl 50135337CCCN(CC1CC1)Cc1sc(Nc2c(Br)cc(C)cc2Br)nc1C(F)(F)F 50135338CCCN(CC1CC1)Cc1sc(Nc2c(C)cc(Cl)cc2C)nc1C(F)(F)F 50135339CCCN(CC1CC1)Cc1sc(Nc2c(C)cc(Cl)cc2Cl)nc1C(F)(F)F 50135340CCCN(CC1CC1)Cc1sc(Nc2c(C)cc(C)cc2Br)nc1C(F)(F)F 50135341CCCN(CCC)C(=O)c1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C 50135343CCCN(CC1CC1)Cc1sc(Nc2c(C)cc(C)cc2C)nc1C(F)(F)F 50135344CCCCN(CC)C(=O)c1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C 50135345CCCN(CC1CC1)Cc1sc(Nc2c(C)cc(C)cc2Cl)nc1C(F)(F)F 50135346CCCN(CC1CC1)C(=O)c1sc(Nc2c(C)cc(C)cc2C)nc1C 50135347CCCN(CC1CC1)C(=O)c1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C 50135349CCCN(CC1CC1)Cc1sc(Nc2c(Br)cc(Br)cc2Br)nc1C(F)(F)F 50135350CCN(CC)C(=O)c1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C 50135351CCCN(CC1CC1)Cc1sc(Nc2ccc(Cl)cc2Cl)nc1C(F)(F)F 50135352CCCN(CC1CC1)Cc1sc(nc1C(F)(F)F)N(CC)c1c(C)cc(C)cc1Cl 50139901CC[C@H](C)[C@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)C(CCCCC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](CCCCN)NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H]1CCCCNC(=O)CC[C@@H](NC(C)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](Cc2cnc[nH]2)C(=O)N1)C(C)C)[C@@H](C)CC)C(N)=O 50139904CC[C@H](C)[C@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)C(CCCCC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H]1CCCCNC(=O)CC[C@@H](N(C)C(C)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N1)C(C)C)[C@@H](C)CC)C(N)=O 50139905CC[C@H](C)[C@H](NC(=O)[C@@H](NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CC1CCCCC1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H]1CCCCNC(=O)CC[C@@H](NC(C)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(O)=O)C(=O)N1)[C@@H](C)CC)C(N)=O 50139906NA 50139907CC[C@H](C)[C@H](NC(=O)[C@@H](NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CC1CCCCC1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H]1CCCCNC(=O)CC[C@@H](NC(C)=O)C(=O)N[C@H](C)C(=O)N[C@@H](CCC(O)=O)C(=O)N1)[C@@H](C)CC)C(N)=O 50139908CC[C@H](C)[C@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)C(CCCCC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H]1CCCCNC(=O)CC[C@@H](NC(C)=O)C(=O)N[C@H](C)C(=O)N[C@@H](Cc2cnc[nH]2)C(=O)N1)C(C)C)[C@@H](C)CC)C(N)=O 50139909CC[C@H](C)[C@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)C(CCCCC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H]1CCCCNC(=O)CC[C@@H](N(C)C(C)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCCN)C(=O)N1)C(C)C)[C@@H](C)CC)C(N)=O 50139910CC[C@H](C)[C@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)C(CCCCC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](C)NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H]1CCCCNC(=O)CC[C@@H](NC(C)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](Cc2cnc[nH]2)C(=O)N1)C(C)C)[C@@H](C)CC)C(N)=O 50139913CC[C@H](C)[C@H](NC(=O)[C@@H](NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)=O)NC(=O)[C@@H]1CCCCNC(=O)CC[C@@H](NC(C)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(O)=O)C(=O)N1)[C@@H](C)CC)C(N)=O 50139914CC[C@H](C)[C@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)C(CCCCC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H]1CCCCNC(=O)CC[C@@H](N(C)C(C)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(O)=O)C(=O)N1)C(C)C)[C@@H](C)CC)C(N)=O 50139915CC[C@H](C)[C@H](NC(=O)[C@@H](NC(=O)[C@H](CC(O)=O)NC(=O)C(CCCCC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H]1CCCCNC(=O)CC[C@@H](NC(C)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(O)=O)C(=O)N1)C(C)C)[C@@H](C)CC)C(N)=O 50139920CC[C@H](C)[C@H](NC(=O)[C@@H](NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)=O)NC(=O)[C@@H]1CCCCNC(=O)CC[C@@H](NC(C)=O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N1)[C@@H](C)CC)C(N)=O 50144189CCCN(C1CCCC1)c1nccc(n1)-c1c(OC)cc(OC)cc1OC 50144190CCCN(c1nccc(n1)-c1c(OC)cc(OC)cc1OC)C1(CC1)c1cccs1 50144191CCCN(C(C1CC1)C1CC1)c1ncc(C)c(n1)-c1c(C)cc(OC)cc1OC 50144192COc1cc(Cl)c(cc1C)-c1nc(sc1C)N(CC#C)[C@@H](CC1CC1)c1ccc(C)c(F)c1 50144193CCCN(C(C1CC1)C1CC1)c1nccc(n1)-c1c(OC)cc(OC)cc1OC 50144194CCCN(C(C1CC1)C1CC1)c1ncc(C)c(n1)-c1ccc(OC)cc1OC 50144195CCCN(C(C1CC1)C1CC1)c1ncc(CC)c(n1)-c1ccc(OC)cc1OC 50144196CCCN(C(C1CC1)C1CC1)c1ncc(C)c(n1)-c1ccc(Br)cc1 50144197CCCN(C(C1CC1)C1CC1)c1ncc(C)c(n1)-c1ccc(Br)cc1C 50144198CCCN(c1nccc(n1)-c1c(OC)cc(OC)cc1OC)C1(CC1)c1ccsc1 50144199CCCN(c1nccc(n1)-c1c(OC)cc(OC)cc1OC)C1(CC1)c1ccoc1 50144200CCCN(C(C1CC1)C1CC1)c1nccc(n1)-c1c(F)cc(OC)cc1OC 50144201CCCN(C(C1CC1)C1CC1)c1nccc(n1)-c1ccc(OC)cc1OC 50144202CCCN([C@H](C1CC1)c1ccccc1)c1nccc(n1)-c1c(OC)cc(OC)cc1OC 50144203COc1cc(OC)c(c(OC)c1)-c1ccnc(n1)N(CC=C)C(C1CC1)C1CC1 50144204CCCN(C(C1CC1)C1CC1)c1nccc(n1)-c1c(Cl)cc(OC)cc1OC 50145728CC(C)c1ccccc1C(Nc1ccc(C)cc1Cl)C(=O)CCc1ccncc1 50145729Cc1ccc(NC(C(=O)CCc2ccncc2)c2ccccc2C)c(Cl)c1 50145730Cc1ccc(NC(C(=O)CCc2ccncc2)c2ccccc2Br)c(Cl)c1 50145731Cc1cccc(C)c1C(Nc1ccc(Cl)cc1Cl)C(=O)CCc1ccncc1 50145732COc1ccc(cc1O)C(=O)C(Nc1ccc(Cl)cc1Cl)c1ccccc1C 50145733Cc1cc(F)ccc1C(Nc1ccc(Cl)cc1Cl)C(=O)CCc1ccncc1 50145735Clc1ccc(NC(C(=O)CCc2ccncc2)c2ccccc2Br)c(Cl)c1 50145737COc1ccc(cc1O)C(=O)C(Nc1ccc(C)cc1Cl)c1ccccc1Br 50145739CC(=O)Nc1cccc(c1)C(=O)C(Nc1ccc(Cl)cc1Cl)c1ccccc1Br 50145740Cc1ccc(NC(C(=O)CCc2ccncc2)c2ccccc2C=C)c(Cl)c1 50145741Cc1ccc(N[C@@H](C(=O)CCc2ccncc2)c2ccccc2Br)c(Cl)c1 50145742Cc1ccccc1[C@@H](Nc1ccc(Cl)cc1Cl)C(=O)CCc1ccncc1 50145745Cc1ccc(NC(C(=O)CCc2ccncc2)c2ccccc2C)c(F)c1 50145749Cc1ccccc1C(Nc1ccc(Cl)cc1Cl)C(=O)CCc1ccncc1 50145751Cc1ccc(N[C@@H](C(=O)CCc2ccncc2)c2ccccc2C)c(Cl)c1 50145752Cc1ccc(NC(C(=O)CCc2ccncc2)c2ccccc2Cl)c(Cl)c1 50145754CCc1ccccc1C(Nc1ccc(Cl)cc1Cl)C(=O)CCc1ccncc1 50145755Cc1ccc(NC(C(=O)CCc2ccncc2)c2ccccc2C)c(c1)C(F)(F)F 50145758Cc1ccccc1C(Nc1ccc(Cl)cc1C(F)(F)F)C(=O)CCc1ccncc1 50145759FC(F)(F)c1ccccc1C(Nc1ccc(Cl)cc1Cl)C(=O)CCc1ccncc1 50145761Cc1ccccc1[C@H](Nc1ccc(Cl)cc1Cl)C(=O)CCc1ccncc1 50145763Clc1ccccc1NC(C(=O)CCc1ccncc1)c1ccccc1Br 50145764CNC(=O)c1cccc(c1)C(=O)C(Nc1ccc(C)cc1Cl)c1ccccc1Br 50148883CCC(CC)Nc1cc(C)nc2c(c(C)nn12)-c1ccc(OC)cc1OC 50148884CCCN(CCC)c1cc(CC)nc2c(c(C)nn12)-c1ccc(Cl)cc1 50148885CCCN(CCC)c1cc(C)nc2c(c(CO)nn12)-c1ccc(Cl)cc1 50148887CCCN(CC1CC1)c1cc(C)nc2c(c(C)nn12)-c1ccc(OC)cc1OC 50148888CCCN(CCO)c1cc(C)nc2c(c(C)nn12)-c1ccc(OC)cc1OC 50148889CCCN(CCOC)c1cc(C)nc2c(c(C)nn12)-c1ccc(OC)cc1OC 50148890CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1cccc(OC)c1 50148892CCCCN(CC)c1cc(C)nc2n(c(C)c(C)c12)-c1c(C)cc(C)cc1C 50148893CCCN(CC1CC1)c1cc(C)nc2c(c(C)nn12)-c1ccc(OC)cc1 50148895CCCCN(CC)c1cc(C)nc2c(c(C)nn12)-c1ccc(OC)cc1OC 50148897CCCN(CC1CC1)c1cc(SC)nc2c(c(C)nn12)-c1ccc(Cl)cc1Cl 50148898CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ccc(Cl)cc1 50148899COCCN(CCOC)c1cc(C)nc2c(c(C)nn12)-c1ccc(OC)cc1OC 50148901CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ccccc1OC 50148902CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ccc(OC)cc1 50148903CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ccc(OC)c(OC)c1 50148904CCCN(CC1CC1)c1cc(nc2c(c(C)nn12)-c1ccc(Cl)cc1Cl)S(C)=O 50148906CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ccccc1 50148907CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ccc(cc1)C#N 50148908CCCN(CC1CC1)c1cc(nc2c(c(C)nn12)-c1ccc(Cl)cc1Cl)S(C)(=O)=O 50149513CCC(CC)Nc1nc(C)nc(C(=O)c2c(C)cc(C)cc2C)c1C 50149515CCCN(CC1CC1)c1nc(C)nc(C(=O)c2c(C)cc(C)cc2C)c1C 50149517CCCN(CC1CC1)c1cc(nc(C)n1)C(=C)c1c(OC)cc(OC)cc1OC 50149518CCCN(CC1CC1)c1nc(C)nc(C(=O)c2c(CC)cc(CC)cc2CC)c1C 50149519COC[C@@H]1CCCN1c1nc(C)nc(C(=O)c2c(C)cc(C)cc2C)c1C 50149520CCCN(c1ccccc1)c1nc(C)nc(C(=O)c2c(C)cc(C)cc2C)c1C 50149521CCCN(CC1CC1)c1nc(C)nc(C(=O)c2c(OC)cc(OC)cc2OC)c1C 50149522CCCN(CCC)c1nc(C)nc(C(=O)c2c(C)cc(C)cc2C)c1C 50149524CCCN(CC1CC1)c1cc(nc(C)n1)C(O)c1c(OC)cc(OC)cc1OC 50149525COCCN(CCOC)c1nc(C)nc(C(=O)c2c(C)cc(C)cc2C)c1C 50149526Cc1cc(C)c(C(=O)c2nc(C)nc(N(CC=C)CC=C)c2C)c(C)c1 50149527CCCN(CC1CC1)c1nc(C)nc(C(=O)c2ccc(OC)cc2OC)c1C 50149528CCCN(CC1CC1)c1cc(Cc2c(OC)cc(OC)cc2OC)nc(C)n1 50149529CCCN(CC1CC1)c1nc(C)nc(C(=O)c2c(C)cc(C)cc2C)c1CC=C 50149530CCCN(CC1CC1)c1cc(nc(C)n1)C(C)c1c(OC)cc(OC)cc1OC 50149531CCCN(CC1CC1)c1cc(nc(C)n1)C(=O)c1c(OC)cc(OC)cc1OC 50149532CCCN(CC1CC1)c1cc(nc(C)n1)C(OC)c1c(CC)cc(CC)cc1CC 50149533CCCN(CC1CC1)c1nc(C)nc(C(=O)c2c(C)cc(C)cc2C)c1CC 50149534CCN(c1ccccc1)c1nc(C)nc(C(=O)c2c(C)cc(C)cc2C)c1C 50149535CCCN(CC1CC1)c1cc(nc(C)n1)C(C)(O)c1c(OC)cc(OC)cc1OC 50149536CCCN(CCO)c1nc(C)nc(C(=O)c2c(C)cc(C)cc2C)c1C 50149537CCCN(CC1CC1)c1nc(C)nc(C(=O)c2ccccc2C)c1C 50149538CCCN(CC1CC1)c1cc(C)nc(n1)C(=O)c1c(OC)cc(OC)cc1OC 50149539CCCN(CC1CC1)c1cc(nc(C)n1)C(O)c1c(CC)cc(CC)cc1CC 50149540CCCN(CC1CC1)c1cc(nc(C)n1)C(=O)c1c(C)cc(C)cc1C 50149541CCCN(CC1CC1)c1cc(nc(C)n1)C(O)c1c(C)cc(C)cc1C 50149542CCCN(CC1CC1)c1nc(C)nc(C(=O)c2c(C)c(C)c(C)c(C)c2C)c1C 50149652COCCN(CCOC)c1cc(C)nc2c(c(C)nn12)-c1ncc(cc1Cl)C(F)(F)F 50149653CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ncc(N)cc1C 50149654CCCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ncc(cc1Cl)C(F)(F)F 50149655CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ncc(cc1C)N1CCCCC1 50149656CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ncc(C)cc1N(C)C 50149657CCCN(Cc1ccccc1)c1cc(C)nc2c(c(C)nn12)-c1ncc(cc1Cl)C(F)(F)F 50149658CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ncc(Cl)cc1Cl 50149659CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ncc(C)cc1[N+]([O-])=O 50149660CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ncc(cc1C)N=O 50149661CCCN(CC1CC1)c1cc(C)nc2c(c(C)nn12)-c1ncc(Cl)cc1Cl 50149662CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ncc(cc1C)N(CC)CC 50149663CCCCN(CCCC)c1cc(C)nc2c(c(C)nn12)-c1ncc(cc1Cl)C(F)(F)F 50149664CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ncc(C)cc1OC 50149665CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ncc(O)cc1C 50149666CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ncc(NC)cc1C 50149667CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ncc(Cl)cc1C 50149668CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ncc(I)cc1C 50149669CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ncc(cc1C)[N+]([O-])=O 50149670CCCN(CC1CC1)c1cc(C)nc2c(c(C)nn12)-c1ncc(cc1Cl)C(F)(F)F 50149671CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ncc(cc1Cl)C(F)(F)F 50149672CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ncc(cc1C)N(C)C 50149673CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ccc(Cl)cn1 50149675CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ncc(OC)cc1C 50149676CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ncc(F)cc1C 50149677CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ncc(C)cc1NC 50149679COCCN(CCOC)c1cc(C)nc2c(c(C)nn12)-c1ncc(Cl)cc1Cl 50149680CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ncc(C)cc1N 50149681CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ncccc1C 50149682CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ncc(C)cc1Cl 50149683CCCN(CCOC)c1cc(C)nc2c(c(C)nn12)-c1ncc(Cl)cc1Cl 50152159CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1cnc(C)cc1C 50152160CCN(Cc1ccccc1F)c1cc(C)nc2c(c(C)nn12)-c1cnc(cc1C)N(C)C 50152161CCCN(CCC)c1cc(C)nc2c(cnn12)-c1c(C)cc(nc1C)N(C)C 50152162CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ccc(nc1)N(C)C 50152163CCCN(CCC)c1c(F)c(C)nc2c(c(C)nn12)-c1cnc(cc1C)N(C)C 50152164CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ccc(nc1C)N(C)C 50152165CCC(CC)Nc1cc(C)nc2c(c(C)nn12)-c1cnc(cc1C)N(C)C 50152166CC(C)N(Cc1ccccc1)c1cc(C)nc2c(c(C)nn12)-c1cnc(cc1C)N(C)C 50152167CC(C)C(C)Nc1cc(C)nc2c(c(C)nn12)-c1cnc(cc1C)N(C)C 50152168CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1ccc(C)nc1 50152169CCCN(CC1CC1)c1cc(C)nc2c(c(C)nn12)-c1cnc(cc1C)N(C)C 50152170CCCCN(Cc1ccccc1)c1cc(C)nc2c(c(C)nn12)-c1cnc(cc1C)N(C)C 50152171CCCN(CCC)c1c(Br)c(C)nc2c(c(C)nn12)-c1cnc(cc1C)N(C)C 50152172CCCN(Cc1ccccc1)c1cc(C)nc2c(c(C)nn12)-c1cnc(cc1C)N(C)C 50152173CCCCN(CC)c1cc(C)nc2c(c(C)nn12)-c1cnc(cc1C)N(C)C 50152174CCCN(CCC)c1c(Cl)c(C)nc2c(c(C)nn12)-c1cnc(cc1C)N(C)C 50152175CCC(COC)Nc1cc(C)nc2c(c(C)nn12)-c1cnc(cc1C)N(C)C 50152176CCN(Cc1ccc(Cl)c(Cl)c1)c1cc(C)nc2c(c(C)nn12)-c1cnc(cc1C)N(C)C 50152177CCCN(CCC)c1cc(C)nc2c(c(C)nn12)-c1c(C)cc(nc1C)N(C)C 50152178CCN(Cc1ccccc1C)c1cc(C)nc2c(c(C)nn12)-c1cnc(cc1C)N(C)C 50152179CCN(Cc1cccc(C)c1)c1cc(C)nc2c(c(C)nn12)-c1cnc(cc1C)N(C)C 50152180COCC(Cc1ccccc1)Nc1cc(C)nc2c(c(C)nn12)-c1cnc(cc1C)N(C)C 50152181CCCN(Cc1cccc(OC)c1)c1cc(C)nc2c(c(C)nn12)-c1cnc(cc1C)N(C)C 50152182CCCN(c1ccccc1)c1cc(C)nc2c(c(C)nn12)-c1cnc(cc1C)N(C)C 50152183CCN(Cc1ccc(C)cc1)c1cc(C)nc2c(c(C)nn12)-c1cnc(cc1C)N(C)C 50152184CC(C)CCC(C)Nc1cc(C)nc2c(c(C)nn12)-c1cnc(cc1C)N(C)C 50152185CCCCN(CCCC)c1cc(C)nc2c(c(C)nn12)-c1cnc(cc1C)N(C)C 50152186CCCC(CCC)Nc1cc(C)nc2c(c(C)nn12)-c1cnc(cc1C)N(C)C 50152187CCCN(Cc1ccc2ccccc2c1)c1cc(C)nc2c(c(C)nn12)-c1cnc(cc1C)N(C)C 50152188CCN(Cc1ccc(Cl)cc1)c1cc(C)nc2c(c(C)nn12)-c1cnc(cc1C)N(C)C 50158102CC(C)N(Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F)C(C)C 50158103COC[C@@H]1CCCN1Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F 50158104CSc1snnc1NCc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F 50158105CCCN(CC)Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F 50158106FC(F)(F)c1nc(Nc2c(Cl)cc(Cl)cc2Cl)sc1CN1CC=CC1 50158108Fc1cccc(CN(CCC(F)(F)F)Cc2sc(Nc3c(Cl)cc(Cl)cc3Cl)nc2C(F)(F)F)c1 50158110CCCN(CC1CCC1)Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F 50158111CCc1nccn1Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F 50158112CCCN(CCC)Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F 50158113CCCCN(CC)Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F 50158114CCN(CC1CC1)Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F 50158115FC(F)(F)CN(Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F)Cc1ccccc1 50158116CCCN(Cc1cccs1)Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F 50158117FC(F)(F)CCN(Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F)Cc1ccc(Cl)cc1 50158120CCCN(CCc1ccccc1)Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F 50158122CCCN(Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F)Cc1ccccc1 50158123FC(F)(F)CCN(Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F)Cc1ccccc1 50158124CCN(CCc1ccccc1)Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F 50158125CCN(CCC1CC1)Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F 50158126FC(F)(F)c1nc(Nc2c(Cl)cc(Cl)cc2Cl)sc1CN(CC=C)CC=C 50158127CCCN(CCC1CC1)Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F 50158128CCCN(CC=C)Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F 50158129FC(F)(F)CCN(CCc1ccccc1)Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F 50158130CCN(Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F)Cc1ccccc1 50158131CCCN(Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F)Cc1ccncc1 50158132CN(CCc1ccccc1)Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F 50158133FC(F)(F)CN(CCc1ccccc1)Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F 50158134Fc1ccc(CN(CCC(F)(F)F)Cc2sc(Nc3c(Cl)cc(Cl)cc3Cl)nc2C(F)(F)F)cc1 50158135CCCN(Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F)Cc1ccccn1 50158136CCCN(Cc1ccco1)Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F 50158137CCCN(Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F)Cc1ccc(Cl)cc1 50158139CCCN(CC1CCCCC1)Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F 50158141FC(F)(F)c1nc(Nc2c(Cl)cc(Cl)cc2Cl)sc1CN(CC1CC1)CC1CC1 50158142CCCN(Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F)Cc1ccccc1F 50158143CCCN(Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F)Cc1ccc(F)cc1 50158144CCCN(Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F)Cc1ccc(OC)cc1 50158145FC(F)(F)CCN(CC1CC1)Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F 50158146CCCN(Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F)Cc1cccnc1 50158148CCCN(CC(C)C)Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F 50158149FC(F)(F)CN(CC1CC1)Cc1sc(Nc2c(Cl)cc(Cl)cc2Cl)nc1C(F)(F)F 50158983CC[C@H](C)[C@H](NC(=O)[C@@H](NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](NC(=O)[C@H](CCSC)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(O)=O)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@@H]1CCC(=O)N1)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)O)C(O)=O 50162451CCC(N(CC)c1nc(-c2ccc(Cl)cc2OC)n(C)n1)c1ccccc1 50162452CCCCC(N(CCC)c1nc(-c2ccc(OC)cc2C)n(C)n1)c1ccccc1 50162453CCCN(C(C)CC)c1nc(-c2ccc(Cl)cc2OC)n(C)n1 50162454CCCC(N(CCC)c1nc(-c2cc(OC)c(OC)cc2Cl)n(C)n1)c1ccccc1 50162457CCCC(N(CCC)c1nc(-c2ccc(OC)cc2OC)n(C)n1)c1ccccc1 50162458CCCC(N(CCC)c1nc(-c2ccc(Cl)cc2OC)n(C)n1)c1ccccc1 50162459CCCCC(CC)N(CCC)c1nc(-c2ccc(Cl)cc2OC)n(C)n1 50162462CCCCC(N(CCC)c1nc(-c2ccc(Cl)cc2OC)n(C)n1)c1ccc(F)cc1 50162463CCCC(N(CCC)c1nc(-c2ccc(OC)cc2C)n(C)n1)c1ccccc1 50162465CCCN(C(CC)c1ccccc1)c1nc(-c2ccc(Cl)cc2OC)n(C)n1 50162466CCCN(C(C(C)C)C(C)C)c1nc(-c2ccc(Cl)cc2OC)n(C)n1 50162467CCCCC(CC)N(CC1CC1)c1nc(-c2ccc(Cl)cc2OC)n(C)n1 50162469CCCCC(CC)N(OCCC)c1nc(-c2ccc(Cl)cc2OC)n(C)n1 50162470CCCN(C(CC)c1ccc(cc1)C(F)(F)F)c1nc(-c2ccc(OC)cc2C)n(C)n1 50162472CCCCC(N(CCC)c1nc(-c2ccc(Cl)cc2OC)n(C)n1)c1ccccc1 50162473CCCN(CC1CC1)c1nc(-c2ccc(Cl)cc2OC)n(C)n1 50162474CCCCC(N(CCC)c1nc(-c2ccc(OC)cc2OC)n(C)n1)c1ccc(F)cc1 50162476CCCN(C(CC)c1ccc(cc1)C(F)(F)F)c1nc(-c2ccc(Cl)cc2OC)n(C)n1 50168460CCCC(CCC)N1CCc2cn(-c3ccccc3OC)c3nc(C)cc1c23 50168461CCCCN1CCc2cn(-c3ccc(Cl)cc3C#N)c3nc(C)cc1c23 50168462CCCC(CCC)N1CCc2nn(-c3ccc(Cl)cc3Cl)c3nc(C)cc1c23 50168463CCCC(CCC)N1CCc2cn(-c3ccc(OC)nc3OC)c3nc(C)cc1c23 50168464CCCC(CCC)N1CCc2cn(-c3ccc(OC)cc3C)c3nc(C)cc1c23 50168465CCCC(CCC)N1CCc2cn(-c3ccc(Cl)cc3C#N)c3nc(C)cc1c23 50168466CCCC(CCC)N1CCc2cn(-c3ccc(Cl)cc3Cl)c3nc(C)cc1c23 50168467CCC(CC)N1CCc2cn(-c3ccc(Cl)cc3C#N)c3nc(C)cc1c23 50168468CCCC(CCC)N1CCc2cn(-c3cccc(OC)c3)c3nc(C)cc1c23 50168469CCC(COC)N1CCc2cn(-c3c(C)cc(Cl)cc3C)c3nc(C)cc1c23 50168470CCCC(CCC)N1CCc2cn(Cc3ccc(Cl)cc3C)c3nc(C)cc1c23 50168473CCCC(CCC)N1CCc2cn(-c3ccc(cc3Cl)C#N)c3nc(C)cc1c23 50168474CCC(CC)N1CCc2cn(-c3ccc(OC(F)(F)F)cc3C)c3nc(C)cc1c23 50168475CCCC(CCC)N1CCc2cn(-c3ccc(C)cc3Cl)c3nc(C)cc1c23 50168476CCCC(CCC)N1CCc2cn(CCCOC(C)C)c3nc(C)cc1c23 50168477CCCC(CCC)N1CCc2cn(-c3ccc(cc3Cl)S(C)(=O)=O)c3nc(C)cc1c23 50168478CCCC(CCC)N1CCc2cn(-c3ccc(C)cc3)c3nc(C)cc1c23 50168479COCC(COC)N1CCc2cn(-c3ccc(Cl)cc3C#N)c3nc(C)cc1c23 50168480CCC(COC)N1CCc2cn(-c3ccc(Cl)cc3C#N)c3nc(C)cc1c23 50169498Cc1cc(C)c(c(C)c1)-n1c2ccccc2n2c(CN(CC3CCC3)CC(F)(F)F)c(nc12)C(F)(F)F 50169499CN(Cc1c(nc2n(-c3c(C)cc(C)cc3C)c3ccccc3n12)C(F)(F)F)Cc1ccccc1 50169500CCCCN(CC)Cc1c(nc2n(-c3c(C)cc(C)cc3C)c3ccccc3n12)C(F)(F)F 50169501CCCN(CCC1CC1)Cc1c(nc2n(-c3c(C)cc(C)cc3C)c3ccccc3n12)C(F)(F)F 50169502Cc1cc(C)c(c(C)c1)-n1c2ccccc2n2c(CN(CCC3CC3)CC(F)(F)F)c(nc12)C(F)(F)F 50169503CCN(Cc1c(nc2n(-c3c(C)cc(C)cc3C)c3ccccc3n12)C(F)(F)F)Cc1ccccc1 50169504Cc1cc(C)c(c(C)c1)-n1c2ccccc2n2c(CN(CCC3CC3)CCC(F)(F)F)c(nc12)C(F)(F)F 50169505CCCN(CC1CC1)Cc1c(nc2n(-c3ccc(cc3Br)C(C)C)c3ccccc3n12)C(F)(F)F 50169506Cc1cc(C)c(c(C)c1)-n1c2ccccc2n2c(CN(CCC(F)(F)F)Cc3ccccc3)c(nc12)C(F)(F)F 50169507Cc1cc(C)c(c(C)c1)-n1c2ccccc2n2c(CN(CC=C)CC=C)c(nc12)C(F)(F)F 50169508CCCN(CC1CC1)Cc1c(C)nc2n(-c3c(C)cc(C)cc3C)c3ccccc3n12 50169509CCCN(CC1CC1)Cc1c(CC)nc2n(-c3c(C)cc(C)cc3C)c3ccc(F)cc3n12 50169510CCCN(CC1CC1)Cc1c(nc2n(-c3ccc(Cl)cc3Cl)c3ccccc3n12)C(F)(F)F 50169511CCCN(Cc1c(nc2n(-c3c(C)cc(C)cc3C)c3ccccc3n12)C(F)(F)F)CC(F)(F)C(F)(F)F 50169512Cc1cc(C)c(c(C)c1)-n1c2ccccc2n2c(CN(CCc3ccccc3)CCc3ccccc3)c(nc12)C(F)(F)F 50169513CCCN(Cc1c(nc2n(-c3c(C)cc(C)cc3C)c3ccccc3n12)C(F)(F)F)Cc1ccccc1 50169514CCCN(CC1CC1)C(=O)c1c(CC)nc2n(-c3c(C)cc(C)cc3C)c3ccc(F)cc3n12 50169515CCCN(Cc1c(nc2n(-c3c(C)cc(C)cc3C)c3ccccc3n12)C(F)(F)F)CC(F)(F)F 50169516Cc1cc(C)c(c(C)c1)-n1c2ccccc2n2c(CN(CCc3ccccc3)CCC(F)(F)F)c(nc12)C(F)(F)F 50169517Cc1cc(C)c(c(C)c1)-n1c2ccccc2n2c(CN(CCC(F)(F)F)CC3CC3)c(nc12)C(F)(F)F 50169518Cc1cc(C)c(c(C)c1)-n1c2ccccc2n2c(CN(CCC(F)(F)F)CC(F)(F)F)c(nc12)C(F)(F)F 50169519CCCN(CC1CC1)C(=O)c1c(C)nc2n(-c3c(C)cc(C)cc3C)c3ccccc3n12 50169520CCCN(CC1CCC1)Cc1c(nc2n(-c3c(C)cc(C)cc3C)c3ccccc3n12)C(F)(F)F 50169521CCCCN(Cc1c(nc2n(-c3c(C)cc(C)cc3C)c3ccccc3n12)C(F)(F)F)Cc1ccccc1 50169522CCCN(CCc1ccccc1)Cc1c(nc2n(-c3c(C)cc(C)cc3C)c3ccccc3n12)C(F)(F)F 50169523Cc1cc(C)c(c(C)c1)-n1c2ccccc2n2c(CN(CC3CC3)CC(F)(F)C(F)(F)F)c(nc12)C(F)(F)F 50169524CCCN(CC1CC1)Cc1c(nc2n(-c3c(C)cc(C)cc3C)c3ccccc3n12)C(F)(F)F 50169525Cc1cc(C)c(c(C)c1)-n1c2ccccc2n2c(CN(CCc3ccccc3)CC(F)(F)F)c(nc12)C(F)(F)F 50169526CCCN(CCC(F)(F)F)Cc1c(nc2n(-c3c(C)cc(C)cc3C)c3ccccc3n12)C(F)(F)F 50169527CCCN(CC1CC1)C(=O)c1c(CC)nc2n(-c3c(C)cc(C)cc3C)c3ccccc3n12 50169528CCCN(CCc1ccccc1)Cc1c(nc2n(-c3ccc(Cl)cc3Cl)c3ccccc3n12)C(F)(F)F 50169529CCCN(CC1CC1)Cc1c(C)nc2n(-c3c(C)cc(C)cc3C)c3ccc(F)cc3n12 50169530CCCN(CC1CC1)C(=O)c1c(C)nc2n(-c3c(C)cc(C)cc3C)c3ccc(F)cc3n12 50169531CCCN(CC1CC1)Cc1c(CC)nc2n(-c3c(C)cc(C)cc3C)c3ccccc3n12 50169532CCCN(CC1CC1)C(=O)c1c(nc2n(-c3c(C)cc(C)cc3C)c3ccccc3n12)C(F)(F)F 50169533CCN(CC1CC1)Cc1c(nc2n(-c3c(C)cc(C)cc3C)c3ccccc3n12)C(F)(F)F 50169534CCN(CCc1ccccc1)Cc1c(nc2n(-c3c(C)cc(C)cc3C)c3ccccc3n12)C(F)(F)F 50169535Cc1cc(C)c(c(C)c1)-n1c2ccccc2n2c(CN(CC3CC3)CC3CC3)c(nc12)C(F)(F)F 50169536CCCN(CCc1ccccc1)Cc1c(nc2n(-c3ccc(cc3Br)C(C)C)c3ccccc3n12)C(F)(F)F 50169537CC(C)c1ccc(c(Br)c1)-n1c2ccccc2n2c(CN(CC3CC3)CC3CC3)c(nc12)C(F)(F)F 50169538CCN(CCC1CC1)Cc1c(nc2n(-c3c(C)cc(C)cc3C)c3ccccc3n12)C(F)(F)F 50169539FC(F)(F)c1nc2n(-c3ccc(Cl)cc3Cl)c3ccccc3n2c1CN(CC1CC1)CC1CC1 50169540Cc1cc(C)c(c(C)c1)-n1c2ccccc2n2c(CN(CC3CC3)CC(F)(F)F)c(nc12)C(F)(F)F 50169556CCCN(CC=C)C(=O)c1c(CC)nc2N(CCn12)c1c(C)cc(C)cc1C 50169557CCCN(CCC)C(=O)c1c(CC)nc2N(CCn12)c1c(C)cc(C)cc1C 50169558CCN(CC1CC1)C(=O)c1c(CC)nc2N(CCn12)c1c(C)cc(C)cc1C 50169559CCCN(CC1CC1)C(=O)c1c(CC)nc2N(CCn12)c1c(C)cc(C)cc1C 50169560CCCCN(CC)C(=O)c1c(CC)nc2N(CCn12)c1c(C)cc(C)cc1C 50169562CCCN(Cc1ccccc1)C(=O)c1c(CC)nc2N(CCn12)c1c(C)cc(C)cc1C 50169563CCc1nc2N(CCn2c1C(=O)N(CC1CC1)CC(F)(F)F)c1c(C)cc(C)cc1Br 50169564CCCN(Cc1cccc(F)c1)C(=O)c1c(CC)nc2N(CCn12)c1c(C)cc(C)cc1C 50169565CCCN(CCC1CC1)C(=O)c1c(CC)nc2N(CCn12)c1c(C)cc(C)cc1C 50169566CCCN(Cc1ccc(Cl)cc1)C(=O)c1c(CC)nc2N(CCn12)c1c(C)cc(C)cc1C 50169567CCc1nc2N(CCn2c1C(=O)N(CCC(F)(F)F)Cc1ccccc1)c1c(C)cc(C)cc1C 50169569CCc1nc2N(CCn2c1C(=O)N(CC1CC1)CC(F)(F)F)c1c(C)cc(Cl)cc1Cl 50169571CCCN(CC1CC1)Cc1c(C)nc2N(CCn12)c1c(C)cc(C)cc1C 50169572CCCN(CC1CC1)C(=O)c1c(CC)nc2N(CCn12)c1ccc(cc1Br)C(C)C 50169573CCCN(CC1CC1)C(=O)c1c(CC)nc2N(CCn12)c1c(C)cc(C)cc1Br 50169574CCc1nc2N(CCn2c1C(=O)N(CC=C)CC=C)c1c(C)cc(C)cc1C 50169575CCc1nc2N(CCn2c1C(=O)N(CC1CC1)CC(F)(F)F)c1c(C)cc(C)cc1Cl 50169576CCCN(CC(F)(F)F)C(=O)c1c(CC)nc2N(CCn12)c1c(C)cc(C)cc1C 50169578CCCN(CCc1ccccc1)C(=O)c1c(CC)nc2N(CCn12)c1c(C)cc(C)cc1C 50169579CCc1nc2N(CCn2c1C(=O)N(CC1CC1)CC1CC1)c1c(C)cc(C)cc1C 50169581CCCN(CC1CC1)C(=O)c1c(CC)nc2N(CCn12)c1c(C)cc(Cl)cc1Cl 50169582CCc1nc2N(CCn2c1C(=O)N(CC1CC1)CC(F)(F)F)c1ccc(cc1Br)C(C)C 50169584CCc1nc2N(CCn2c1C(=O)N(CC1CC1)CC(F)(F)F)c1c(C)cc(C)cc1C 50169585CCCN(CC1CC1)C(=O)c1c(C)nc2N(CCn12)c1c(C)cc(C)cc1C 50169587CCc1nc2N(CCn2c1C(=O)N(CCC1CC1)CCC(F)(F)F)c1c(C)cc(C)cc1C 50169588CCc1nc2N(CCn2c1C(=O)N(CCC(F)(F)F)CC1CC1)c1c(C)cc(C)cc1C 50169589CCc1nc2N(CCn2c1C(=O)N(CC1CC1)CC(F)(F)C(F)(F)F)c1c(C)cc(C)cc1C 50169590CCc1nc2N(CCn2c1C(=O)N(CCC(F)(F)F)Cc1ccc(Cl)cc1)c1c(C)cc(C)cc1C 50169591CCCN(CC1CC1)C(=O)c1c(CC)nc2N(CCn12)c1c(C)cc(C)cc1Cl 50169592CCN(CCC1CC1)C(=O)c1c(CC)nc2N(CCn12)c1c(C)cc(C)cc1C 50169593CCCN(CCC(F)(F)F)C(=O)c1c(CC)nc2N(CCn12)c1c(C)cc(C)cc1C 50171314CCCC(CCC)N1CCn2c3c1cc(C)nc3n(-c1cccc(OC)c1)c2=O 50171315CCCC(CCC)N1CCn2c3c1cc(C)nc3n(-c1ccc(Cl)cn1)c2=O 50171316CCC(CC)N1CCn2c3c1cc(C)nc3n(-c1ccc(OC)cc1)c2=O 50171317CCC(CC)N1CCn2c3c1cc(C)nc3n(-c1ccc(cc1)C(F)(F)F)c2=O 50171318CCCC(CCC)N1CCn2c3c1cc(C)nc3n(-c1ccc(OC)cc1)c2=O 50171319CCC(CC)N1CCn2c3c1cc(C)nc3n(-c1ccc(Cl)cc1)c2=O 50171320CCCC(CCC)N1CCn2c3c1cc(C)nc3n(-c1ccccc1OC)c2=O 50171321CCC(CC)N1CCn2c3c1cc(C)nc3n(-c1ccc(OC)cc1C)c2=O 50171322CCCC(CCC)N1CCn2c3c1cc(C)nc3n(-c1ccc(Cl)cc1Cl)c2=O 50171324CCCCN1CCn2c3c1cc(C)nc3n(-c1ccc(OC)cc1)c2=O 50171325CCCC(CCC)N1CCn2nc(-c3ccc(Cl)cc3Cl)c3nc(C)cc1c23 50171326CCCC(OC)N1CCn2c3c1cc(C)nc3n(-c1ccc(Cl)cc1)c2=O 50171327CCCC(CCC)N1CCn2c3c1cc(C)nc3n(-c1ccc(cc1)C(=O)OC)c2=O 50171328CCCC(CCC)N1CCn2c3c1cc(C)nc3n(-c1ccc(Cl)cc1)c2=O 50171329CCCC(OC)N1CCn2c3c1cc(C)nc3n(-c1ccc(OC)cc1C)c2=O 50171330CCCC(CCC)N1CCn2c3c1cc(C)nc3n(-c1ccc(cc1)S(C)(=O)=O)c2=O 50171331CCCC(CCC)N1CCn2c3c1cc(C)nc3n(-c1ccc(OC)nc1)c2=O 50171332CCCC(CCC)N1CCn2c3c1cc(C)nc3n(-c1ccc(cc1Br)C(C)C)c2=O 50171333CCCC(CCC)N1CCn2c3c1cc(C)nc3n(-c1ccc(OCC)cc1)c2=O 50171334CCCC(CCC)N1CCn2c3c1cc(C)nc3n(-c1ccc(cc1)C(F)(F)F)c2=O 50171335CCCC(OC)N1CCn2c3c1cc(C)nc3n(-c1ccc(cc1)C(F)(F)F)c2=O 50171336CCCC(OC)N1CCn2c3c1cc(C)nc3n(-c1ccc(OC)cc1)c2=O 50203587CCN(CCc1ccccc1)Cc1c(C)nc2n(-c3c(C)cc(C)cc3Cl)c3ncccc3n12 50203588CCN(CC1CC1)Cc1c(C)nc2n(-c3c(C)cc(C)cc3Cl)c3ncccc3n12 50203589CCCN(CC1CC1)Cc1c(C)nc2n(-c3c(C)cc(C)cc3C)c3ncccc3n12 50203590CCCN(CC1CC1)Cc1c(C)nc2n(-c3c(C)cc(C)cc3Cl)c3ncccc3n12 50203591CN(CCc1ccccn1)Cc1c(C)nc2n(-c3c(C)cc(C)cc3Cl)c3ncccc3n12 50203592Cc1nc2n(-c3c(C)cc(C)cc3Cl)c3ncccc3n2c1CN1CCC(Cc2ccccc2)C1 50203593CN(Cc1c(C)nc2n(-c3c(C)cc(C)cc3Cl)c3ncccc3n12)Cc1cccnc1 50203594Cc1nc2n(-c3c(C)cc(C)cc3C)c3ncccc3n2c1CN(CC1CC1)CC1CC1 50203595COCC(COC)NCc1c(C)nc2n(-c3c(C)cc(C)cc3Cl)c3ncccc3n12 50203596CCN(CC)Cc1c(C)nc2n(-c3c(C)cc(C)cc3Cl)c3ncccc3n12 50203597CCCCN(CCCC)Cc1c(C)nc2n(-c3c(C)cc(C)cc3Cl)c3ncccc3n12 50203598CCCN(CC1CCC1)Cc1c(C)nc2n(-c3c(C)cc(C)cc3C)c3ncccc3n12 50203599CCN(CC1CCC1)Cc1c(C)nc2n(-c3c(C)cc(C)cc3Cl)c3ncccc3n12 50203600CCCN(Cc1c(C)nc2n(-c3c(C)cc(C)cc3Cl)c3ncccc3n12)Cc1ccccc1 50203601COCCN(CCOC)Cc1c(C)nc2n(-c3c(C)cc(C)cc3Cl)c3ncccc3n12 50203602Cc1nc2n(-c3c(C)cc(C)cc3Cl)c3ncccc3n2c1CN(CC=C)CC=C 50203603CN(CCc1ccncc1)Cc1c(C)nc2n(-c3c(C)cc(C)cc3Cl)c3ncccc3n12 50203604CCCN(CC=C)Cc1c(C)nc2n(-c3c(C)cc(C)cc3C)c3ncccc3n12 50203605CCN(CC1CC1)Cc1c(C)nc2n(-c3c(C)cc(C)cc3C)c3ncccc3n12 50203606CCCCN(CC)Cc1c(C)nc2n(-c3c(C)cc(C)cc3Cl)c3ncccc3n12 50203607Cc1nc2n(-c3c(C)cc(C)cc3Cl)c3ncccc3n2c1CN1CCCC1CCc1ccccc1 50203608CCCN(CC1CC1)Cc1c(nc2n(-c3c(C)cc(C)cc3C)c3ncccc3n12)C(F)(F)F 50203609CCCN(CC=C)Cc1c(C)nc2n(-c3c(C)cc(C)cc3Cl)c3ncccc3n12 50203610CCCN(CCC1CC1)Cc1c(C)nc2n(-c3c(C)cc(C)cc3Cl)c3ncccc3n12 50203611CCCN(CC1CCC1)Cc1c(C)nc2n(-c3c(C)cc(C)cc3Cl)c3ncccc3n12 50203612CCCN(CCC1CC1)Cc1c(C)nc2n(-c3c(C)cc(C)cc3C)c3ncccc3n12 50203613CN(CCc1cccnc1)Cc1c(C)nc2n(-c3c(C)cc(C)cc3Cl)c3ncccc3n12 50203614CCN(CCC1CC1)Cc1c(C)nc2n(-c3c(C)cc(C)cc3Cl)c3ncccc3n12 50203615Cc1nc2n(-c3c(C)cc(C)cc3Cl)c3ncccc3n2c1CN1CCCC1Cc1ccccc1 50203616Cc1nc2n(-c3c(C)cc(C)cc3Cl)c3ncccc3n2c1CN1CCC(CCc2ccccc2)C1 50203617CCCN(CC1CCC1)Cc1c(CC)nc2n(-c3c(C)cc(C)cc3C)c3ncccc3n12 50203619Cc1nc2n(-c3c(C)cc(C)cc3C)c3ncccc3n2c1CN(CC=C)CC=C 50203620Cc1nc2n(-c3c(C)cc(C)cc3Cl)c3ncccc3n2c1CN1CCOCC1 50203621Cc1nc2n(-c3c(C)cc(C)cc3Cl)c3ncccc3n2c1CN1CCC(C1)c1ccccc1 50203622Cc1nc2n(-c3c(C)cc(C)cc3Cl)c3ncccc3n2c1CN1CCCC1c1ccccc1 50203623CCCC(C)NCc1c(C)nc2n(-c3c(C)cc(C)cc3Cl)c3ncccc3n12 50203624CCCN(CCC)Cc1c(C)nc2n(-c3c(C)cc(C)cc3Cl)c3ncccc3n12 50203625CCN(CCc1ccccc1)Cc1c(C)nc2n(-c3c(C)cc(C)cc3C)c3ncccc3n12 50203626CCCN(CCc1ccccc1)Cc1c(C)nc2n(-c3c(C)cc(C)cc3Cl)c3ncccc3n12 50203627CN(Cc1c(C)nc2n(-c3c(C)cc(C)cc3Cl)c3ncccc3n12)Cc1ccncc1 50222975CCc1nc(Oc2cc(C)ccn2)c(CC)nc1N[C@H]1[C@H](Cc2ccccc12)OC 50222976CC(C)C(Nc1nc(C)c(Oc2cc(C)ccn2)nc1C)c1ccccc1 50222977CCc1nc(Oc2cc(C)ccn2)c(CC)nc1N[C@H]1[C@H](Cc2ccccc12)OC1CCCC1 50222978CCC(CC)Nc1nc(C)c(Oc2cc(C)ccn2)nc1C 50222979CCc1nc(Oc2cc(C)ccn2)c(CC)nc1NC(C)c1ccccc1 50222980CCc1nc(Oc2cc(C)ccn2)c(CC)nc1N[C@H]1[C@H](Cc2ccccc12)OC(C)C 50222982CCCN(CCC)c1nc(CC)c(Oc2cc(C)ccn2)nc1CC 50222983CCO[C@H]1Cc2ccccc2[C@@H]1Nc1nc(CC)c(Oc2cc(C)ccn2)nc1CC 50222984CCc1nc(Oc2cc(C)ccn2)c(CC)nc1NC(CO)c1ccccc1 50222985CCc1nc(Oc2cc(C)ccn2)c(CC)nc1N[C@H]1[C@H](Cc2ccccc12)OCCF 50222986CCc1nc(Oc2cc(C)ccn2)c(CC)nc1N[C@H]1[C@H](Cc2ccccc12)OC1CC1 50222988CCC(CC)Nc1nc(CC)c(Nc2c(Cl)cc(Cl)cc2Cl)nc1CC 50222989CCC(CC)Nc1nc(C)c(Nc2ncc(Cl)cc2Cl)nc1C 50222991CCc1nc(Oc2ccccn2)c(CC)nc1N[C@H]1[C@H](Cc2ccccc12)OCCF 50222994CCC(CC)Nc1nc(CC)c(Nc2cccc(C)n2)nc1CC 50222995CCc1nc(Nc2ncc(Cl)cc2Cl)c(CC)nc1N[C@H]1[C@H](Cc2ccccc12)OCCF 50222998CCc1nc(Oc2cc(C)ccn2)c(CC)nc1NC(COC(C)C)c1ccccc1 50223002CCO[C@H]1Cc2ccccc2[C@H]1Nc1nc(CC)c(Oc2cc(C)ccn2)nc1CC 50223003CCC(Nc1nc(C)c(Oc2cc(C)ccn2)nc1C)c1ccccc1 50223004CCCO[C@H]1Cc2ccccc2[C@H]1Nc1nc(CC)c(Oc2cc(C)ccn2)nc1CC 50223005CCc1nc(Oc2cc(C)ccn2)c(CC)nc1NC(C(C)C)c1ccccc1 50223007CCOCC(Nc1nc(CC)c(Oc2cc(C)ccn2)nc1CC)c1ccccc1 50223010CCO[C@H]1Cc2ccccc2[C@H]1Nc1nc(CC)c(Oc2ncccc2C)nc1CC 50223013CCCN(CC1CC1)c1nc(C)c(Oc2cc(C)ccn2)nc1C 50223014CCO[C@H]1Cc2ccccc2[C@H]1Nc1nc(C)c(Oc2cc(C)ccn2)nc1C 50223015CCC(Nc1nc(CC)c(Oc2cc(C)ccn2)nc1CC)c1ccccc1 50223016CCc1nc(Oc2cc(C)ccn2)c(CC)nc1N[C@H]1[C@H](Cc2ccccc12)OC(C)=O 50223017CCc1nc(Oc2cc(C)ccn2)c(CC)nc1N[C@H]1[C@H](Cc2ccccc12)OCCO 50223019CCCN(CCC)c1nc(C)c(Oc2cc(C)ccn2)nc1C 50223020CCO[C@H]1Cc2ccccc2[C@H]1Nc1nc(CC)c(Oc2cc(CC)ccn2)nc1CC 50223023CCO[C@H]1Cc2ccccc2[C@H]1Nc1nc(CC)c(Oc2cc(C)cc(C)n2)nc1CC 50223024CCC(CC)Nc1nc(CC)c(Nc2ccc(Cl)cc2)nc1CC 50223025CCc1nc(N(C)c2ncc(Cl)cc2Cl)c(CC)nc1N[C@H]1[C@H](Cc2ccccc12)OCCF 50223027CCO[C@H]1Cc2ccccc2[C@H]1Nc1nc(CC)c(Oc2cccc(C)n2)nc1CC 50223028CCC(CC)Nc1nc(CC)c(Nc2ncc(Cl)cc2Cl)nc1CC 50223030CCCO[C@H]1Cc2ccccc2[C@H]1Nc1nc(CC)c(Oc2cc(C)cc(C)n2)nc1CC 50223031CCc1nc(N(C)[C@H]2[C@H](Cc3ccccc23)OC)c(CC)nc1Oc1cc(C)ccn1 50223032CCO[C@H]1Cc2ccccc2[C@H]1Nc1nc(CC)c(Oc2ccc(C)cn2)nc1CC 50223033CCc1nc(Oc2cc(C)ncn2)c(CC)nc1N[C@H]1[C@H](Cc2ccccc12)OCCF 50223034CCC(Nc1nc(CC)c(Oc2ncccc2C)nc1CC)c1ccccc1 50223035CCO[C@H]1Cc2ccccc2[C@H]1Nc1nc(CC)c(Oc2cccc(C)c2)nc1CC 50231903CCCN(CCC)c1c(C)nc(-c2ccc(Cl)cc2)c2ccccc12 50231904CCCNc1c(C)nc(-c2c(C)cc(C)cc2OC)c2ccccc12 50231905CCCN(CCC)c1c(C)nc(-c2ccc(Cl)cc2Cl)c2ccccc12 50231906CCCN(CCC)c1c(C)nc(-c2c(C)cc(C)cc2OCCN2CCCCC2)c2ccccc12 50231907CCCN(CCC)c1c(C)nc(-c2c(CC(F)F)cc(CC(F)F)cc2OC)c2ccccc12 50231908CCCN(CCC)c1c(C)nc(-c2c(C)cc(C)cc2OCCN2CCCC2)c2ccccc12 50231909CCCN(CCC)c1c(C)nc(-c2ccc(OC)cc2C)c2ccccc12 50231910CCCN(CCC)c1c(C)nc(-c2c(C)cc(OC)cc2C)c2ccccc12 50231911CCCN(CCn1ccnc1)c1c(C)nc(-c2c(C)cc(C)cc2OC)c2ccccc12 50231912CCCN(CCC)c1c(C)nc(-c2c(C)cc(C)cc2OCCN2CCCC(O)C2)c2ccccc12 50231914CCCN(CCC)c1c(C)nc(-c2ccccc2Cl)c2ccccc12 50231915CCCN(CCC)c1cnc(-c2c(C)cc(C)cc2OC)c2ccccc12 50231916CCCN(CC1CC1)c1c(C)nc(-c2c(C)cc(C)cc2OC)c2ccccc12 50231917CCCN(CCC)c1c(C)nc(-c2c(C)cc(C)cc2OCCN2CCN(C)CC2)c2ccccc12 50231918CCCN(CCN1CCCC1)c1c(C)nc(-c2c(C)cc(C)cc2OC)c2ccccc12 50231919CCCN(CCC)c1c(C)nc(-c2ccc(OC(F)F)cc2OC)c2ccccc12 50231921CCCN(CCC)c1c(C)nc(-c2c(C)cc(C)cc2OC)c2ccccc12 50231922CCCN(CCC)c1c(C)nc(-c2c(C)cc(C)cc2OCCN(C)C)c2ccccc12 50231923CCCN(CCC)c1c(C)nc(-c2ccc(OC)cc2CC)c2ccccc12 50231924CCCN(CCC)c1c(C)nc(-c2c(C)cc(C)cc2OCCN2CCC(O)CC2)c2ccccc12 50231925COc1cc(C)cc(C)c1-c1nc(C)c(N(CC2CC2)CC2CC2)c2ccccc12 50231926CCCN(CCC)c1c(C)nc(-c2c(C)cc(C)cc2OCCN2CCOCC2)c2ccccc12 50231927CCCN(CCC)c1c(CC)nc(-c2c(C)cc(C)cc2OC)c2ccccc12 50231928CCCN(CCC)c1c(C)nc(-c2ccc(OC)cc2OC)c2ccccc12 50231930CCCN(CCC)c1c(C)nc(-c2ccc(Cl)cc2C)c2ccccc12 50272635CCCN(CCC)c1c(C)nc(nc1OCCO)-c1c(C)cc(C)cc1OC 50272636CCCN(CCC)c1c(CC)nc(nc1OC)-c1c(C)cc(C)cc1OC 50272637CCCN(CCC)c1c(CCC)nc(nc1OC)-c1c(C)cc(C)cc1OC 50272638CCCN(CCC)c1c(C)nc(nc1OC)-c1c(OC)cc(Cl)cc1OC 50272640CCC(CC)Nc1c(C)nc(nc1OC)-c1c(C)cc(C)cc1OC 50272695CCC(CC)c1cc(C)nn2c(c(C)nc12)-c1sc(nc1Cl)N1CCOCC1 50272696CCCN(CCC)c1cnc(nc1C)-c1c(C)cc(C)cc1OC 50272697CCCN(CCC)c1c(C)nc(nc1OC)-c1c(OC)cccc1OC 50272698CCCN(CCC)c1c(CC(C)O)nc(nc1OC)-c1c(C)cc(C)cc1OC 50272699CCCN(CCC)c1c(CC(C)(C)O)nc(nc1OC)-c1c(C)cc(C)cc1OC 50272701CCCN(CCC)c1c(C)nc(nc1OC)-c1ccc(OC)cc1OC 50272702CCCN(CCC)c1c(C)nc(nc1OC)-c1c(OC)cc(cc1C(F)(F)F)C(F)(F)F 50272703CCC(CC)Oc1c(C)nc(nc1OC)-c1c(C)cc(C)cc1OC 50272704CCC(CC)Oc1c(C)nc(nc1OC)-c1c(OC)cc(Cl)cc1OC 50272705CCC(CC)Oc1c(C)nc(nc1OC)-c1c(OC)cc(cc1OC)C(F)F 50272750CCCN(CCC)c1c(C)nc(nc1OC)-c1c(C)cc(C)cc1OC 50272751CCCN(CCC)c1c(C)nc(nc1Cl)-c1c(C)cc(C)cc1OC 50272752CCCN(CCC)c1c(C)nc(nc1OC)-c1c(C)cc(C)cc1C 50272753CCCN(CCC)c1c(C)nc(nc1OCC)-c1c(C)cc(C)cc1OC 50272754CCCOc1nc(nc(C)c1N(CCC)CCC)-c1c(C)cc(C)cc1OC 50293910C[C@@H](C1CC1)n1cc(Cl)nc(Nc2c(Cl)cc(OC(F)F)cc2Cl)c1=O 50293912COC[C@@H](C1CC1)n1cc(Cl)nc(Nc2cc(C)c(OC)cc2C)c1=O 50300147COC[C@H](C1CC1)n1cc(Cl)nc(Nc2cc(C#N)c(OC(F)F)nc2C)c1=O 50302573CCCC(CCC)Nc1nc(C)nc2n(ncc12)-c1ccc(OC)cc1C 50302574CCCCN(CC)c1nc(C)nc2n(nc(C)c12)-c1c(C)cc(C)cc1C 50302575CC[C@@H](COC)Nc1nc(C)nc2n(nc(C)c12)-c1ccc(OC)cc1C 50302576CC[C@H](COC)Nc1nc(C)nc2n(nc(C)c12)-c1ccc(OC)cc1C 50302577CCC[C@H](CO)Nc1nc(C)nc2n(nc(C)c12)-c1ccc(OC)cc1C 50302578CCC[C@@H](CO)Nc1nc(C)nc2n(nc(C)c12)-c1ccc(OC)cc1C 50302579CC[C@@H](CO)Nc1nc(C)nc2n(nc(C)c12)-c1ccc(OC)cc1C 50302580CC[C@H](CO)Nc1nc(C)nc2n(nc(C)c12)-c1ccc(OC)cc1C 50302581CCC(CC)Nc1nc(C)nc2n(nc(C)c12)-c1ccc(OC)cc1C 50302582CCCC(CCC)Nc1nc(C)nc2n(nc(C)c12)-c1ccc(OC)cc1C 50302583CCCC(CCOC)Nc1nc(C)nc2n(ncc12)-c1ccc(OC)cc1C 50302584CCC(CC)Nc1nc(C)nc2n(ncc12)-c1ccc(OC)cc1C 50302585COCCN(CCOC)c1nc(C)nc2n(nc(C)c12)-c1ccc(OC)cc1C 50302586CCCN(CCO)c1nc(C)nc2n(nc(C)c12)-c1ccc(OC)cc1C 50302587CCCN(CC(=O)N(C)C)c1nc(C)nc2n(nc(C)c12)-c1ccc(OC)cc1C 50302588CCCNCc1nnc(Nc2nc(C)nc3n(nc(C)c23)-c2ccc(OC)cc2C)o1 50302589CCCNCc1noc(Nc2nc(C)nc3n(nc(C)c23)-c2ccc(OC)cc2C)n1 50302590CCCNCc1nc(Nc2nc(C)nc3n(nc(C)c23)-c2ccc(OC)cc2C)no1 50302591CCCNCc1nccn1Nc1nc(C)nc2n(nc(C)c12)-c1ccc(OC)cc1C 50302592CCCNCc1cncn1Nc1nc(C)nc2n(nc(C)c12)-c1ccc(OC)cc1C 50302593CCCN(CCOC)c1nc(C)nc2n(nc(C)c12)-c1ccc(OC)cc1C 50302594CCCN(CCOC)c1nc(C)nc2n(nc(C)c12)-c1ccc(OC)cc1OC 50302595CCCN(CCOC)c1nc(C)nc2n(nc(C)c12)-c1ccc(cc1C)C#N 50302596CCCN(CCOC)c1nc(C)nc2n(nc(C)c12)-c1ccc(cc1C#N)C#N 50302597CCCN(CCOC)c1nc(C)nc2n(nc(C)c12)-c1ccc(cc1C)C(N)=O 50302598CCCN(CCOC)c1nc(C)nc2n(nc(C)c12)-c1ccc(OC)nc1C 50302599CCCN(CCOC)c1nc(C)nc2n(nc(C)c12)-c1ccc(OC)nc1OC 50302600CCCN(CCOC)c1nc(C)nc2n(nc(C)c12)-c1cnc(cc1C)N(C)C 50302601CCCN(CCOC)c1nc(C)nc2n(nc(C)c12)-c1ccc(nc1C)C(N)=O 50302602CCN(CCOC)c1nc(C)nc2n(nc(C)c12)-c1ccc(OC)cc1C 50313989Cc1nc2N(CCCn2c1C(=O)N(CC1CC1)CC1CC1)c1c(C)cc(C)cc1C 50313990CCCN(CC1CCC1)C(=O)c1c(C)nc2N(CCCn12)c1c(C)cc(C)cc1C 50313991CCCN(CCc1ccccc1)C(=O)c1c(C)nc2N(CCCn12)c1c(C)cc(C)cc1C 50313995CCCN(CC1CC1)C(=O)c1c(CC)nc2N(CCCn12)c1c(C)cc(C)cc1C 50313996CCCN(CC1CC1)C(=O)c1c(nc2N(CCCn12)c1c(C)cc(C)cc1C)C(F)(F)F 50314007CCCN(CC1CC1)Cc1c(nc2N(CCCn12)c1c(C)cc(C)cc1C)C(F)(F)F 50314008Cc1cc(C)c(N2CCCn3c(CN(CC4CC4)CC(F)(F)F)c(nc23)C(F)(F)F)c(C)c1 50314009Cc1cc(C)c(N2CCCn3c(CN(CC4CC4)CC(F)(F)C(F)(F)F)c(nc23)C(F)(F)F)c(C)c1 50314010Cc1cc(C)c(N2CCCn3c2nc(c3C(=O)N(CC=C)CC=C)C(F)(F)F)c(C)c1 50314011CCCN(CC1CCC1)Cc1c(nc2N(CCCn12)c1c(C)cc(C)cc1C)C(F)(F)F 50314012Cc1cc(C)c(N2CCCn3c(CN(CC4CCC4)CC(F)(F)F)c(nc23)C(F)(F)F)c(C)c1 50314013CCN(CC1CC1)Cc1c(nc2N(CCCn12)c1c(C)cc(C)cc1C)C(F)(F)F 50314014CCCN(CCc1ccccc1)Cc1c(nc2N(CCCn12)c1c(C)cc(C)cc1C)C(F)(F)F 50314015Cc1cc(C)c(N2CCCn3c(CN(CCc4ccccc4)CC(F)(F)F)c(nc23)C(F)(F)F)c(C)c1 50314016CCCN(CC=C)Cc1c(nc2N(CCCn12)c1c(C)cc(C)cc1C)C(F)(F)F 50314017CCCN(CCC(F)(F)F)Cc1c(nc2N(CCCn12)c1c(C)cc(C)cc1C)C(F)(F)F 50314018Cc1cc(C)c(N2CCCn3c(CN4CCCCC4)c(nc23)C(F)(F)F)c(C)c1 50314019Cc1cc(C)c(N2CCCn3c(CN4CCC=CC4)c(nc23)C(F)(F)F)c(C)c1 50314020Cc1cc(C)c(N2CCCn3c(CN4CCOCC4)c(nc23)C(F)(F)F)c(C)c1 50314021Cc1cc(C)c(N2CCCn3c(CN4CCSCC4)c(nc23)C(F)(F)F)c(C)c1 50319848CCCN(CC1CC1)Cc1c(nc2n(c(Cl)cn12)-c1ccc(OC)cc1C)C(F)(F)F 50319849CCCN(CC1CC1)Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1Cl)C(F)(F)F 50319850CCCN(CC1CC1)Cc1c(nc2n(ccn12)-c1c(C)cc(C)cc1C)C(F)(F)F 50319851CCCN(CC1CC1)C(=O)c1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F 50319852CCCN(CC1CC1)C(=O)c1c(C)nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C 50319853Cc1cc(C)c(c(C)c1)-n1c(Cl)cn2c(CN3CCSCC3)c(nc12)C(F)(F)F 50319854Cc1cc(C)c(c(C)c1)-n1c(Cl)cn2c(CN3CCOCC3)c(nc12)C(F)(F)F 50319855Cc1cc(C)c(c(C)c1)-n1c(Cl)cn2c(CN3CCC=CC3)c(nc12)C(F)(F)F 50319856CC1CCN(Cc2c(nc3n(c(Cl)cn23)-c2c(C)cc(C)cc2C)C(F)(F)F)CC1 50319857CC1CCCN(Cc2c(nc3n(c(Cl)cn23)-c2c(C)cc(C)cc2C)C(F)(F)F)C1 50319858CC1CCCCN1Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F 50319859Cc1cc(C)c(c(C)c1)-n1c(Cl)cn2c(CN3CCCCC3)c(nc12)C(F)(F)F 50319860Cc1cc(C)c(c(C)c1)-n1c(Cl)cn2c(CN3CCC(C3)c3ccccc3)c(nc12)C(F)(F)F 50319861Cc1cc(C)c(c(C)c1)-n1c(Cl)cn2c(CN3CCCC3Cc3ccccc3)c(nc12)C(F)(F)F 50319863Cc1cc(C)c(c(C)c1)-n1c(Cl)cn2c(CN(CCc3ccccc3)CCC(F)(F)F)c(nc12)C(F)(F)F 50319864Cc1cc(C)c(c(C)c1)-n1c(Cl)cn2c(CN(CCc3ccccc3)CC(F)(F)F)c(nc12)C(F)(F)F 50319865CN(CCc1ccncc1)Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F 50319866CN(CCc1cccnc1)Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F 50319867CN(CCc1ccccn1)Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F 50319868CN(CCc1ccccc1)Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F 50319869CCN(CCc1ccccc1)Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F 50319870CCCN(CCc1ccccc1)Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F 50319871CN(Cc1ccco1)Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F 50319872CCN(Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F)Cc1ccccc1C 50319873CCN(Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F)Cc1ccc(Cl)c(Cl)c1 50319874CCN(Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F)Cc1ccccc1 50319875CCCN(Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F)Cc1ccc(F)cc1 50319876CCCN(Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F)Cc1cccc(F)c1 50319877CCCN(Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F)Cc1ccc(cc1)[N+]([O-])=O 50319878CCCN(Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F)Cc1ccc(Cl)cc1 50319879CCCN(Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F)Cc1ccccc1 50319880CN(Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F)Cc1ccccc1 50319881CCCCN(Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F)Cc1ccccc1 50319882Cc1cc(C)c(c(C)c1)-n1c(Cl)cn2c(CN(CCC(F)(F)F)Cc3ccc(Cl)cc3)c(nc12)C(F)(F)F 50319883Cc1cc(C)c(c(C)c1)-n1c(Cl)cn2c(CN(Cc3ccc(F)cc3)CC(F)(F)F)c(nc12)C(F)(F)F 50319884Cc1cc(C)c(c(C)c1)-n1c(Cl)cn2c(CN(CCC(F)(F)F)Cc3ccc(F)cc3)c(nc12)C(F)(F)F 50319885Cc1cc(C)c(c(C)c1)-n1c(Cl)cn2c(CN(CCC(F)(F)F)Cc3cccc(F)c3)c(nc12)C(F)(F)F 50319886Cc1cc(C)c(c(C)c1)-n1c(Cl)cn2c(CN(CCC(F)(F)F)Cc3ccccc3)c(nc12)C(F)(F)F 50319887Cc1cc(C)c(c(C)c1)-n1c(Cl)cn2c(CN(CCC3CC3)CCC(F)(F)F)c(nc12)C(F)(F)F 50319888CCCN(CCC1CC1)Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F 50319889CCN(CCC1CC1)Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F 50319890Cc1cc(C)c(c(C)c1)-n1c(Cl)cn2c(CN(CCC3CC3)CC(F)(F)F)c(nc12)C(F)(F)F 50319891CCN(CC1CCC1)Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F 50319892Cc1cc(C)c(c(C)c1)-n1c(Cl)cn2c(CN(CC3CCC3)CC(F)(F)F)c(nc12)C(F)(F)F 50319893CCCN(CC1CCC1)Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F 50319894CCN(CC(C)=C)Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F 50319895Cc1cc(C)c(c(C)c1)-n1c(Cl)cn2c(CN(CC=C)CC=C)c(nc12)C(F)(F)F 50319896CCCN(CC=C)Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F 50319897CCCCN(C)Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F 50319898CCCCN(CC)Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F 50319899CCCN(Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F)CC(F)(F)C(F)(F)F 50319900CCCN(CCC)Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F 50319901CCCN(CCOC)Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F 50319902CCCN(CCC(F)(F)F)Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F 50319903CCCN(Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F)CC(F)(F)F 50319904Cc1cc(C)c(c(C)c1)-n1c(Cl)cn2c(CN(CCC(F)(F)F)CC3CC3)c(nc12)C(F)(F)F 50319905CCN(CC1CC1)Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F 50319906Cc1cc(C)c(c(C)c1)-n1c(Cl)cn2c(CN(CC3CC3)CC(F)(F)F)c(nc12)C(F)(F)F 50319907CCCN(CC1CC1)Cc1c(nc2n(c(Cl)cn12)-c1c(C)cc(C)cc1C)C(F)(F)F 50340208CCN(CC)c1nc2n(C)cc(-c3c(C)cc(C)cc3C)c2c(=O)n1C 50340209CCCN(CCC)c1nc2n(C)cc(-c3c(C)cc(C)cc3C)c2c(=O)n1C 50340210CCCCN(CCCC)c1nc2n(C)cc(-c3c(C)cc(C)cc3C)c2c(=O)n1C 50340211Cc1cc(C)c(-c2cn(C)c3nc(N(CC4CC4)CC4CC4)n(C)c(=O)c23)c(C)c1 50340212Cc1cc(C)c(-c2cn(C)c3nc(N4CCCCC4)n(C)c(=O)c23)c(C)c1 50340213CCCN(CCC)c1nc2n(C)c(C)c(-c3c(C)cc(C)cc3C)c2c(=O)n1C 50340214CCCN(CCC)c1nc2n(C)c(C)c(-c3ccc(C)cc3C)c2c(=O)n1C 50340215CCCN(CCC)c1nc2n(C)cc(-c3ccc(C)cc3C)c2c(=O)n1C 50340216CCCN(CCC)c1nc2n(C)cc(-c3c(OC)cc(OC)cc3OC)c2c(=O)n1C 50340217CCCN(CCC)c1nc2n(C)cc(-c3ccc(OC)cc3OC)c2c(=O)n1C 50340218CCCN(CCC)c1nc2n(C)cc(-c3ccc(cc3C(F)(F)F)C(F)(F)F)c2c(=O)n1C 50342734CCN(CCN)c1nc(C)nc2n(-c3c(C)cc(C)cc3C)c3ccccc3c12 50348777CCC(CC)Nc1nc(OC)c(nc1CC)-c1ccc(OC(F)F)cc1Cl 50348778CCC(CC)Nc1nc(OC)c(nc1CC)-c1ccc(OC)cc1Cl 50348779CCC(CC)Nc1nc(OC)c(nc1CC)-c1ccc(OC(F)(F)F)cc1OC 50348780CCOc1ccc(c(Cl)c1)-c1nc(OC)c(NC(CC)CC)nc1C 50348781CCC(CC)Nc1nc(C)c(nc1OC)-c1ccc(OC(F)F)cc1Cl 50348782CCC(CC)Nc1nc(C)c(nc1OC)-c1ccc(OC(F)(F)F)cc1OC 50348783CCC(CC)Nc1nc(CC)c(nc1OC)-c1ccc(OC(F)F)cc1Cl 50348784CCC(CC)Nc1nc(CC)c(nc1OC)-c1ccc(OC)cc1C(F)(F)F 50348785CCC(CC)Nc1nc(CC)c(nc1OC)-c1ccc(cc1OC)C(F)(F)F 50348786CCC(CC)Nc1nc(CC)c(nc1OC)-c1ccc(OC)cc1CC 50348787CCC(CC)Nc1nc(OC)c(nc1CC)-c1ccc(Cl)cc1Cl 50348788CCC(CC)Nc1nc(OC)c(nc1C)-c1ccc(Cl)cc1Cl 50348789CCC(CC)Nc1nc(OC)c(nc1OC)-c1ccc(Cl)cc1Cl 50348790CCC(CC)Nc1nc(C)c(nc1OC)-c1ccc(Cl)cc1Cl 50348791CCC(CC)Nc1nc(C)c(nc1C)-c1ccc(Cl)cc1Cl 50348792CCC(CC)Nc1nc(C)c(nc1CC)-c1ccc(Cl)cc1Cl 50348793CCC(CC)Nc1nc(CC)c(nc1C)-c1ccc(Cl)cc1Cl 50348794CCCCc1nc(c(CC)nc1NC(CC)CC)-c1ccc(Cl)cc1Cl 50348795CCOc1nc(c(CC)nc1NC(CC)CC)-c1ccc(Cl)cc1Cl 50348796CCC(CC)Nc1nc(CC)c(nc1OC)-c1ccc(Cl)cc1Cl 50348797CCC(CC)Nc1nc(CC)c(nc1I)-c1ccc(Cl)cc1Cl 50348798CCC(CC)Nc1nc(CC)c(nc1Cl)-c1ccc(Cl)cc1Cl 50348799CCC(CC)Nc1nc(CC)c(nc1F)-c1ccc(Cl)cc1Cl 50348800CCC(CC)Nc1cnc(c(CC)n1)-c1ccc(Cl)cc1Cl 50348801CCC(CC)Cc1nc(CC)c(nc1CC)-c1ccc(Cl)cc1Cl 50348802CCC(C)Sc1nc(CC)c(nc1CC)-c1ccc(Cl)cc1Cl 50348803CCC(CC)Oc1nc(CC)c(nc1CC)-c1ccc(Cl)cc1Cl 50348804CCCN(CCN(C)C)c1nc(CC)c(nc1CC)-c1ccc(Cl)cc1Cl 50348805CCc1nc(c(CC)nc1N(CCOC)CCOC)-c1ccc(Cl)cc1Cl 50348806CCCN(CC1CC1)c1nc(CC)c(nc1CC)-c1ccc(Cl)cc1Cl 50348807CCc1nc(c(CC)nc1N(CC1CC1)CC1CC1)-c1ccc(Cl)cc1Cl 50348808CCc1nc(c(CC)nc1NC(C)CN(C)C)-c1ccc(Cl)cc1Cl 50348809CCc1nc(c(CC)nc1NC(COC)COC)-c1ccc(Cl)cc1Cl 50348810CCc1nc(c(CC)nc1NC(C1CC1)C1CC1)-c1ccc(Cl)cc1Cl 50348811CCC(CC)Nc1nc(CC)c(nc1CC)-c1cnc(OC)nc1OC 50348812CCC(CC)Nc1nc(CC)c(nc1CC)-c1ccc(OC)nc1OC 50348813CCC(CC)Nc1nc(CC)c(nc1CC)-c1cnc(C)cc1N(C)C 50348814CCC(CC)Nc1nc(CC)c(nc1CC)-c1ccc(OC)cc1C(F)(F)F 50348815CCC(CC)Nc1nc(CC)c(nc1CC)-c1ccc(OC)cc1OC(F)(F)F 50348816CCC(CC)Nc1nc(CC)c(nc1CC)-c1ccc(OC)cc1O 50348817CCC(CC)Nc1nc(CC)c(nc1CC)-c1ccc(cc1OC)C(F)(F)F 50348818CCC(CC)Nc1nc(CC)c(nc1CC)-c1ccc(C)cc1OC 50348819CCC(CC)Nc1nc(CC)c(nc1CC)-c1ccc(OC(C)C)cc1OC 50348820CCOc1ccc(c(OC)c1)-c1nc(CC)c(NC(CC)CC)nc1CC 50348821CCC(CC)Nc1nc(CC)c(nc1CC)-c1ccc(OC(F)(F)F)cc1OC 50348822CCC(CC)Nc1nc(CC)c(nc1CC)-c1ccc(OC)cc1OC 50348823CCC(CC)Nc1nc(CC)c(nc1CC)-c1ccc(Cl)cc1Cl 50348827CCCN(CCC)c1c(C)ncc2c(cccc12)-c1ccc(Cl)cc1Cl 50348828COc1cc(Cl)c(cc1C)-c1nc(sc1C)N(CC#C)[C@@H](CC1CC1)c1ccc(C)c(F)c1 50348829CCC(CC)Nc1nc(C)c(nc1OC)-c1ccc(cc1OC)C(F)(F)F 50351370CCC(CC)Nc1c2CCCc2nc2c(c(C)nn12)-c1ccc(OC)cc1C 50351371CCC(CC)Nc1c2OCCc2nc2c(c(C)nn12)-c1ccc(OC)cc1C 50351372CCC(CC)Nc1c2SCCc2nc2c(c(C)nn12)-c1ccc(OC)cc1C 50351373CCC(CC)Nc1c2NCCc2nc2c(c(C)nn12)-c1ccc(OC)cc1C 50351374CCC(CC)Nc1c2COCc2nc2c(c(C)nn12)-c1ccc(OC)cc1C 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50398572COCc1cc(OC)c(-c2csc3c(N(C(C)C)C4CCOCC4)c(OC)nn23)c(OC)c1 50398573CCCCN(C1CCOCC1)c1c(OC)nn2c(csc12)-c1c(OC)cc(COC)cc1OC 50398574COCc1cc(OC)c(-c2csc3c(N(CCC4CC4)C4CCOCC4)c(OC)nn23)c(OC)c1 50398575CCCN(C1CCOCC1)c1c(OC)nn2c(csc12)-c1c(OC)cc(COC)cc1OC 50398576CCN(C1CCOCC1)c1c(OC)nn2c(csc12)-c1c(OC)cc(COC)cc1OC 50398577COCc1cc(OC)c(-c2csc3c(N(CC4CC4)C4CCOCC4)c(OC)nn23)c(OC)c1 50398578COCCN(CC1CC1)c1c(OC)nn2c(csc12)-c1c(OC)cc(COC)cc1OC 50398579COCc1cc(OC)c(-c2csc3c(N(CC4CC4)CC4CCCO4)c(OC)nn23)c(OC)c1 50398580COCc1cc(OC)c(-c2csc3c(N(CC4CC4)CC4CCOC4)c(OC)nn23)c(OC)c1 50398581COCc1cc(OC)c(-c2csc3c(N(CC4CC4)CC4CCCCO4)c(OC)nn23)c(OC)c1 50398582COCc1cc(OC)c(-c2csc3c(N(CC4CC4)CC4CCCOC4)c(OC)nn23)c(OC)c1 50398583COCc1cc(OC)c(-c2csc3c(N(CC4CC4)CC4(F)CCOCC4)c(OC)nn23)c(OC)c1 50398584COCc1cc(OC)c(-c2csc3c(N(CC4CC4)CC4(O)CCOCC4)c(OC)nn23)c(OC)c1 50398585COCc1cc(OC)c(-c2csc3c(N(CC4CC4)CC4CCOCC4)c(OC)nn23)c(OC)c1 50398586COCc1cc(OC)c(-c2c(C)sc3c(N(CC4CC4)CC4CCOCC4)c(C)nn23)c(OC)c1 50398587COCc1cc(OC)c(-c2csc3c(N(CC4CC4)CC4CCOCC4)c(C)nn23)c(OC)c1 50410275CCCN([C@H](CC)c1ccc(cc1)C(F)(F)F)c1nc(-c2ccc(Cl)cc2OC)n(C)n1 50410276CCCC[C@@H](N(CCC)c1nc(-c2ccc(OC)cc2C)n(C)n1)c1ccccc1 50410277CCC[C@@H](N(CCC)c1nc(-c2ccc(OC)cc2C)n(C)n1)c1ccccc1 50410278CCCC[C@H](N(CCC)c1nc(-c2ccc(OC)cc2C)n(C)n1)c1ccccc1 50410279CCC[C@H](N(CCC)c1nc(-c2ccc(OC)cc2C)n(C)n1)c1ccccc1 50410280CCCN([C@@H](CC)c1ccc(cc1)C(F)(F)F)c1nc(-c2ccc(Cl)cc2OC)n(C)n1 50410281CCCC[C@H](N(CCC)c1nc(-c2ccc(Cl)cc2OC)n(C)n1)c1ccc(F)cc1 50410282CCCC[C@@H](N(CCC)c1nc(-c2ccc(Cl)cc2OC)n(C)n1)c1ccc(F)cc1 50412798COc1ccc(N2CCc3c2nc(C)cc3-n2ccc(n2)N2CCNC2=O)c(C)c1 50412799COc1ccc(N2CCc3c2nc(C)cc3-n2ccc(n2)N2CCCC2=O)c(C)c1 50412800COc1ccc(N2CCc3c2nc(C)cc3-n2ccc(n2)N2CCN(C)C2=O)c(C)c1 50412801COc1ccc(N2CCc3c2nc(C)cc3-n2ccc(n2)N2CCOC2=O)c(C)c1 50412802COc1ccc(N2CCc3c2nc(C)cc3-n2ccc(n2)-n2cc[nH]c2=O)c(C)c1 50412803COc1ccc(N2CCc3c2nc(C)cc3-n2ccc(n2)N2CCCNC2=O)c(C)c1 50412804COc1ccc(N2CCc3c2nc(C)cc3-n2ccc(n2)N2CCNS2(=O)=O)c(C)c1 50412805COc1ccc(N2CCc3c2nc(C)cc3-n2ccc(n2)N2CCCS2(=O)=O)c(C)c1 50412806CCOc1ccc(N2CCc3c2nc(C)cc3-n2ccc(n2)N2CCNC2=O)c(C)c1 50412807CC(C)Oc1ccc(N2CCc3c2nc(C)cc3-n2ccc(n2)N2CCNC2=O)c(C)c1 50412808Cc1cc(c2CCN(c2n1)c1ccc(OC(F)(F)F)cc1C)-n1ccc(n1)N1CCNC1=O 50412809Cc1cc(c2CCN(c2n1)c1ccc(cc1C)C#N)-n1ccc(n1)N1CCNC1=O 50412810Cc1cc(c2CCN(c2n1)c1ccc(cc1C)-n1cccn1)-n1ccc(n1)N1CCNC1=O 50412811Cc1cc(c2CCN(c2n1)c1ccc(cc1C(F)(F)F)C#N)-n1ccc(n1)N1CCNC1=O 50412812COc1ccc(N2CCc3c2nc(C)cc3-n2ccc(n2)N2CCNC2=O)c(c1)C(F)F 50412813Cc1cc(c2CCN(c2n1)c1ccc(cc1OC(F)(F)F)C#N)-n1ccc(n1)N1CCNC1=O 50412814CCc1cc(ccc1N1CCc2c1nc(C)cc2-n1ccc(n1)N1CCNC1=O)C#N 50412815COc1cc(ccc1N1CCc2c1nc(C)cc2-n1ccc(n1)-n1cc[nH]c1=O)-n1cccn1 50412816Cc1cc(c2CCN(c2n1)c1ccc(Cl)cc1Cl)-n1ccc(n1)-n1cc[nH]c1=O 50412817Cc1cc(c2CCN(c2n1)c1ccc(cc1C(F)(F)F)C(F)(F)F)-n1ccc(n1)-n1cc[nH]c1=O 50413195FC(F)(F)c1ccc(N2CCc3c2nccc3-n2ccc(n2)-c2nccs2)c(c1)C(F)(F)F 50413196[O-][N+](=O)c1ccc(N2CCc3c2nccc3-n2ccc(n2)-c2nccs2)c(c1)C(F)(F)F 50413197FC(F)(F)c1cc(ccc1N1CCc2c1nccc2-n1ccc(n1)-c1nccs1)C#N 50413198COc1ccc(N2CCc3c2nccc3-n2ccc(n2)-c2nccs2)c(C)c1 50413199Cc1cc(ccc1N1CCc2c1nccc2-n1ccc(n1)-c1nccs1)C#N 50413200Cc1cc(ccc1N1CCc2c1nccc2-n1ccc(n1)-c1nccs1)-n1cccn1 50413201Cc1cc(F)ccc1N1CCc2c1nccc2-n1ccc(n1)-c1nccs1 50413202Cc1cc(O)ccc1N1CCc2c1nccc2-n1ccc(n1)-c1nccs1 50413204Cc1cc(OC(F)(F)F)ccc1N1CCc2c1nccc2-n1ccc(n1)-c1nccs1 50413205CCc1cc(ccc1N1CCc2c1nccc2-n1ccc(n1)-c1nccs1)C#N 50413206COc1ccc(N2CCc3c2nccc3-n2ccc(n2)-c2nccs2)c(OC)c1 50413207FC(F)(F)Oc1cc(ccc1N1CCc2c1nccc2-n1ccc(n1)-c1nccs1)C#N 50413208COc1ccc(N2CCc3c2nccc3-n2ccc(n2)-c2nccs2)c(Cl)c1 50413209Clc1cc(ccc1N1CCc2c1nccc2-n1ccc(n1)-c1nccs1)C#N 50413210CS(=O)(=O)c1ccc(N2CCc3c2nccc3-n2ccc(n2)-c2nccs2)c(Cl)c1 50413211N#Cc1cc(ccc1N1CCc2c1nccc2-n1ccc(n1)-c1nccs1)-c1cccs1 50413212N#Cc1ccc(N2CCc3c2nccc3-n2ccc(n2)-c2nccs2)c(c1)C#N 50413217CS(=O)(=O)c1ccc(N2CCc3c2nccc3-n2ccc(n2)-c2nccs2)c(c1)S(C)(=O)=O 50413218COc1ccc(N2CCc3c2nccc3-n2ccc(n2)-c2nccs2)c(c1)C(F)F 50413219COc1ccc(cc1)N1CCc2c1nccc2-n1ccc(n1)-c1nccs1 50413220Fc1cc(ccc1N1CCc2c1nccc2-n1ccc(n1)-c1nccs1)C#N 50413221COc1ccc(N2CCc3c2nccc3-n2ccc(n2)-c2nccs2)c(C)n1 50413222COc1ccc(N2CCc3c2nccc3-n2ccc(n2)-c2nccs2)c(OC)n1 50413223COc1ccc(N2CCc3c2nccc3-n2ccc(n2)-c2nccs2)c(n1)C(F)(F)F 50413224CN(C)c1ccc(N2CCc3c2nccc3-n2ccc(n2)-c2nccs2)c(C)n1 50413225Clc1cc(ccc1N1CCc2c1nccc2-n1ccc(n1)-c1ccccn1)C#N 50413226Cc1cc(ccc1N1CCc2c1nccc2-n1ccc(n1)-c1ccccn1)C#N 50413227FC(F)(F)c1cc(ccc1N1CCc2c1nccc2-n1ccc(n1)-c1ccccn1)C#N 50413228Cc1cc(ccc1N1CCc2c1nccc2-n1ccc(n1)-n1cccn1)C#N 50413229Clc1cc(ccc1N1CCc2c1nccc2-n1ccc(n1)-n1cccn1)C#N 50413230FC(F)(F)c1cc(ccc1N1CCc2c1nccc2-n1ccc(n1)-n1cccn1)C#N 50413231COc1ccc(c(C)c1)-n1ccc2c(cc(C)nc12)-n1ccc(n1)-c1nccs1 50413232Cc1cc(-n2ccc(n2)-c2nccs2)c2cnn(-c3ccc(cc3C)C#N)c2n1 50413236Cc1cc(-n2ccc(n2)-c2nccs2)c2[nH]c(=O)n(-c3ccc(cc3C(F)(F)F)C(F)(F)F)c2n1 50417499COc1ccc(-c2c(C)nn3c(NCc4nc(C)no4)cc(C)nc23)c(C)c1 50417500CCN(Cc1nc(C)no1)c1cc(C)nc2c(c(C)nn12)-c1ccc(OC)cc1C 50417501CCC(Nc1cc(C)nc2c(c(C)nn12)-c1ccc(OC)cc1C)c1nc(C)no1 50417502CC[C@@H](Nc1cc(C)nc2c(c(C)nn12)-c1ccc(OC)cc1C)c1nc(C)no1 50417503CC[C@H](Nc1cc(C)nc2c(c(C)nn12)-c1ccc(OC)cc1C)c1nc(C)no1 50417504COc1ccc(-c2c(C)nn3c(NC4(CC4)c4nc(C)no4)cc(C)nc23)c(C)c1 50417505COc1ccc(-c2c(C)nn3c(NC4(CCC4)c4nc(C)no4)cc(C)nc23)c(C)c1 50417506COc1ccc(-c2c(C)nn3c(NC(C)Cc4nc(C)no4)cc(C)nc23)c(C)c1 50417507CCC(Nc1cc(C)nc2c(c(C)nn12)-c1ccc(OC)cc1C)c1nnc(C)o1 50417508COc1ccc(-c2c(C)nn3c(NC(C)Cc4nnc(C)o4)cc(C)nc23)c(C)c1 50417509COc1ccc(-c2c(C)nn3c(NC(C)Cc4noc(C)n4)cc(C)nc23)c(C)c1 50417510CCC(Nc1cc(C)nc2c(c(C)nn12)-c1cnc(cc1C)N(C)C)c1nc(C)no1 50417511CCC(Nc1cc(C)nc2c(c(C)nn12)-c1ccc(OC)cc1OC)c1nc(C)no1 50417512COc1ccc(-c2c(C)nn3c(NC(C)c4nc(C)no4)cc(C)nc23)c(C)c1 50420904CCc1nn2c(cccc2c1N(CC1CC1)CC1CC1)-c1ccc(OC)cc1Cl 50420905CCc1nn2c(cccc2c1N(CC1CC1)CC1CC1)-c1ccc(OC)cc1C 50420906CCc1nn2c(cccc2c1N(CC1CC1)CC1CC1)-c1ccc(C)cc1OC 50420907CCc1nn2c(cccc2c1N(CC1CC1)CC1CC1)-c1c(C)cc(C)cc1OC 50420908CCc1nn2c(cccc2c1N(CC1CC1)CC1CC1)-c1c(C)cc(OC)cc1C 50420909CCCN(CCC)c1c(CC)nn2c(cccc12)-c1ccc(OC)cc1Cl 50420910CCCN(CCC)c1c(CC)nn2c(cccc12)-c1ccc(OC)cc1C 50420911CCc1nn2c(cccc2c1N(CCOC)CC1CC1)-c1c(C)cc(C)cc1OC 50420912CCc1nn2c(cccc2c1N(CCCF)CC1CC1)-c1c(C)cc(C)cc1OC 50420913CCc1nn2c(cccc2c1N(CC1CC1)CC1CCOC1)-c1c(C)cc(C)cc1OC 50420914CCc1nn2c(cccc2c1N(CC1CC1)CC1CCCO1)-c1c(C)cc(C)cc1OC 50420915CCc1nn2c(cccc2c1N(CC1CC1)CC1CCOCC1)-c1c(C)cc(C)cc1OC 50420916CCc1nn2c(cccc2c1N(CC1CC1)CC1CCOCC1)-c1c(OC)cc(C)cc1OC 50420917CCc1nn2c(cccc2c1N(CC1CC1)CC1CCOCC1)-c1c(C)cc(OC)cc1OC 50420918CCc1nn2c(cccc2c1N(CC1CC1)CC1CCOCC1)-c1cc(OC)c(OC)cc1OC 50420919CCc1nn2c(cccc2c1N(CC1CC1)CC1CCOCC1)-c1c(OC)cc(CO)cc1OC 50420920CCc1nn2c(cccc2c1N(CC1CC1)CC1CCOCC1)-c1c(OC)cc(COC)cc1OC 50420921CCc1nn2c(cccc2c1N(CC1CC1)CC1CCOCC1)-c1c(COC)cc(OC)cc1OC 50420922CCOCc1cc(OC)c(c(OC)c1)-c1cccc2c(N(CC3CC3)CC3CCOCC3)c(CC)nn12 50420923CCc1nn2c(cccc2c1N(CC1CC1)CC1CCOCC1)-c1c(OC)cccc1OC 50420924CCCN(CC1CCOCC1)c1c(CC)nn2c(cccc12)-c1c(OC)cc(C)cc1OC 50420925CCCN(CC1CCOCC1)c1c(CC)nn2c(cccc12)-c1c(OC)cc(COC)cc1OC 50420926COCc1cc(OC)c(c(OC)c1)-c1cccc2c(N(CC3CC3)CC3CCOCC3)c(OC)nn12 50420927COCc1cc(OC)c(c(OC)c1)-c1cccc2c(N(CC3CC3)CC3CCOCC3)c(SC)nn12 50420928COCc1cc(OC)c(c(OC)c1)-c1cccc2c(N(CC3CC3)CC3CCOCC3)c(C)nn12 50420929COCc1cc(OC)c(c(OC)c1)-c1cccc2c(N(CC3CC3)CC3CCOCC3)c(nn12)C#N 50420930COc1nn2c(cccc2c1N(CC1CC1)CC1CCOCC1)-c1c(OC)cc(C)cc1OC 50420931COc1cc(C)cc(OC)c1-c1cccc2c(N(CC3CC3)CC3CCOCC3)c(SC)nn12 50420933COCc1cc(OC)c(c(OC)c1)-c1cccc2c(N(CC3CCOCC3)CC3(O)CC3)c(SC)nn12 50420934COCc1cc(OC)c(c(OC)c1)-c1cccc2c(N(CC3CCOCC3)CC3(CC3)C#N)c(SC)nn12 50420935COCc1cc(OC)c(c(OC)c1)-c1cccc2c(N(CC3CC3)CC3COCCO3)c(SC)nn12 50420936COCc1cc(OC)c(c(OC)c1)-c1cccc2c(N(CC3CC3)CC3OCCCO3)c(SC)nn12 50420937COCCN(CC1CCOCC1)c1c(SC)nn2c(cccc12)-c1c(OC)cc(COC)cc1OC 50420938CCc1nn2c(cccc2c1N(CC1CC1)CC1CCOCC1)-c1c(OC)cc(OC)cc1OC 50422737CC[C@H]1Cn2nc(-c3ccc(Cl)cc3Cl)c3nc(C)cc(N1CC1CC1)c23 50423371CCCC(CCC)n1cc2CCN(c3ccc(cc3C)C#N)c3nc(C)nc1c23 50423372CCCC(CCC)n1cc2CCN(c3ccc(cc3C(F)(F)F)C(F)(F)F)c3nc(C)cc1c23 50423373CCCC(CCC)n1cc2CCN(c3ccc(cc3C(F)(F)F)C(F)(F)F)c3nc(C)nc1c23 50423374CCC(COC)n1cc2CCN(c3ccc(cc3C)C#N)c3nc(C)cc1c23 50423375CCC(CC)n1cc2CCN(c3ccc(cc3C(F)(F)F)C(F)(F)F)c3nc(C)nc1c23 50423376CCC(COC)n1cc2CCN(c3ccc(OC)cc3C)c3nc(C)cc1c23 50423377CCC(CC)n1cc2CCN(c3ccc(cc3C(F)(F)F)C(F)(F)F)c3nc(C)cc1c23 50423378CCC(CC)n1cc2CCN(c3ccc(OC(F)(F)F)cc3C)c3nc(C)cc1c23 50423379CCCC(CCC)N1CCC2CN(c3nc(C)nc1c23)c1ccc(Cl)cc1Cl 50423380CCC(CC)n1cc2CCN(c3ccc(cc3C)C#N)c3nc(C)cc1c23 50423381CCC(CC)n1cc2CCN(c3ccc(OC)c(F)c3)c3nc(C)cc1c23 50423382CCCC(CCC)n1cc2CCN(c3ccc(cc3C)C#N)c3nc(C)cc1c23 50423383CCCC(CCC)n1cc2CCN(c3ccc(OC)c(F)c3)c3nc(C)cc1c23 50423384CCCC(CCC)n1cc2CCN(c3ccc(OC)cc3C)c3nc(C)cc1c23 50423385CCC(CC)n1cc2CCN(c3ccc(OC)cc3C)c3nc(C)cc1c23 50423386CCC(CC)n1cc2CCN(c3ccc(OC)cc3)c3nc(C)cc1c23