4552COc1cc(Nc2c(cnc3cc(OCCCN4CCN(C)CC4)c(OC)cc23)C#N)c(Cl)cc1Cl
4779Fc1ccc(Nc2ncnc3cc(OCCCN4CCOCC4)c(NC(=O)C=C)cc23)cc1Cl
4814CCN(CC)CCNC(=O)c1c(C)[nH]c(\C=C2/C(=O)Nc3ccc(F)cc23)c1C
5446COCCOc1cc2ncnc(Nc3cccc(c3)C#C)c2cc1OCCOC
5655CN1CC[C@@H]([C@H](O)C1)c1c(O)cc(O)c2c1oc(cc2=O)-c1ccccc1Cl
6568CSc1cccc(Nc2ncc3cc(-c4c(Cl)cccc4Cl)c(=O)n(C)c3n2)c1
14028C[C@H]1CNCCCN1S(=O)(=O)c1cccc2cncc(C)c12
15138Cc1n[nH]c2ccc(cc12)-c1cncc(OC[C@@H](N)Cc2ccccc2)c1
17055CN(C)C[C@@H]1CCn2cc(C3=C(C(=O)NC3=O)c3cn(CCO1)c1ccccc31)c1ccccc21
25117CNC(=O)c1ccccc1Sc1ccc2c(\C=C\c3ccccn3)n[nH]c2c1
25118CN1CCN(CC1)c1ccc2nc([nH]c2c1)-c1c(N)c2c(F)cccc2[nH]c1=O
27817CNC(=O)c1c(F)cccc1Nc1nc(Nc2cc3N(CCc3cc2OC)C(=O)CN(C)C)nc2[nH]ccc12
31085CCN1CCN(Cc2ccc(NC(=O)Nc3ccc(Oc4cc(NC)ncn4)cc3)cc2C(F)(F)F)CC1
31095Cc1[nH]c(\C=C2/C(=O)Nc3ccc(F)cc23)c(C)c1C(=O)NC[C@H](O)CN1CCOCC1
36409CC(C)n1nc(-c2cc3cc(O)ccc3[nH]2)c2c(N)ncnc12
41571Cn1cc(\C=C\c2n[nH]c3ccnc(OC4CCCCC4)c23)cn1
41572CC(C)Oc1nccc2[nH]nc(-c3cc(C(=O)N4CCOCC4)n(c3)C(C)C)c12
41573CN1CCc2c1cccc2-c1n[nH]c2ccnc(OC3CCOCC3)c12
41574CNC(=O)c1cccc(c1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105061C[C@H]1CCCN(C1)C(=O)CCc1[nH]nc2ccnc(NC3CCOCC3)c12
105062O=C(CCc1[nH]nc2ccnc(OC3CCCCC3)c12)N1CCC[C@@H](C1)c1ccccc1
105063O=C(CCc1[nH]nc2ccnc(NC3CCCCC3)c12)N1CCN(CC1)C1CC1
105064C1CC(CCO1)Nc1nccc2[nH]nc(-c3ccnc(c3)N3CCOCC3)c12
105065CN1CCN(CC1)c1cc(ccn1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105066C1CC1c1[nH]nc2ccnc(OC3CCCCC3)c12
105067C1CC1c1[nH]nc2ccnc(OC3CCOCC3)c12
105068CCC(C)Oc1nccc2n[nH]c(C3CC3)c12
105069Cc1[nH]nc2ccnc(OC3CCOC3)c12
105070C1CC(CCO1)Oc1nccc2[nH]nc(-c3ccco3)c12
105071C1CCC(C1)n1cc(cn1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105072C(C1CCC1)n1cc(cn1)-c1n[nH]c2ccnc(OC3CCCCC3)c12
105073CC(C)Oc1nccc2[nH]nc(-c3cc(C(=O)N(C)C)n(c3)C(C)C)c12
105074CC(C)Oc1nccc2[nH]nc(-c3cc(C(=O)N4CCCCC4)n(c3)C(C)C)c12
105075CC(C)Oc1nccc2[nH]nc(-c3cc(C(=O)NC4COC4)n(c3)C(C)C)c12
105076COc1nccc2[nH]nc(-c3cc(C(=O)N(C)C)n(c3)C(C)C)c12
105077COc1nccc2[nH]nc(-c3cc(C(=O)NC4COC4)n(c3)C(C)C)c12
105078CC(C)n1cc(cc1C(=O)N1CCOCC1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105079CC(C)n1cc(cc1C(=O)N(C)C)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105080CC(C)n1cc(cc1C(=O)NC1COC1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105081O=C(N1CCOCC1)c1cc(ccn1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105082FC(F)(F)COc1nccc2[nH]nc(-c3ccnc(c3)N3CCOCC3)c12
105083CC(C)n1cc(cn1)-c1n[nH]c2ccnc(OCC(F)(F)F)c12
105084CC(C)n1cc(cn1)-c1n[nH]c2ccnc(OC(C)C(F)(F)F)c12
105085C1CC(CCO1)Oc1nccc2[nH]nc(-c3ccnc(n3)N3CCOCC3)c12
105086COc1nccc2[nH]nc(-c3cnn(c3)C3COC3)c12
105088COc1nccc2[nH]nc(-c3cnn(CC(F)(F)F)c3)c12
105089COc1nccc2[nH]nc(-c3cnn(CC4(C)COC4)c3)c12
105090C(C1CCOCC1)n1cc(cn1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105091FC(F)(F)Cn1cc(cn1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105092C1CC(CO1)n1cc(cn1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105093Cc1cc(cc(C)n1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105094COc1cc(ccn1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105095Fc1c(ccnc1N1CCOCC1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105096COc1cc(ccn1)-c1n[nH]c2ccnc(OC)c12
105097COc1nccc2[nH]nc(-c3ccnc(c3)N3CCOCC3)c12
105098COc1nccc2[nH]nc(-c3ccnc(c3)C(F)(F)F)c12
105099COc1nccc2n[nH]c(-c3ccc(C(=O)N4CCOCC4)c(Cl)c3)c12
105100C1CCN(C1)c1cc(ccn1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105101CC1CCCN(C1)c1cc(ccn1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105102C1OCC1Nc1cc(ccn1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105103C1CN(C1)c1cc(ccn1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105104Cn1cc(cn1)-c1cc(ccn1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105105COc1nccc2[nH]nc(-c3ccnc(c3)N3[C@H]4CC[C@@H]3COC4)c12
105106COc1nccc2[nH]nc(-c3ccnc(c3)N3C[C@@H]4C[C@H]3CO4)c12
105107COc1nccc2[nH]nc(-c3ccnc(c3)N3CCCC3)c12
105108COc1nccc2[nH]nc(-c3ccnc(c3)-c3cnn(C)c3)c12
105109CC(C)n1cnc2ccc(cc12)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105110C1OCC1n1cnc2cc(ccc12)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105111C1OCC1n1cnc2ccc(cc12)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105112FC1(F)CC1Cn1cnc2ccc(cc12)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105113C1CC(CO1)n1cnc2ccc(cc12)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105114C1CC(CO1)n1cnc2cc(ccc12)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105115Clc1ccccc1C#Cc1[nH]nc2ccnc(OC3CCOCC3)c12
105116O=C(N1CCOCC1)c1ccc(cc1)-c1[nH]nc2ccnc(OC3CCOCC3)c12
105117CN(C)C(=O)c1ccc(cc1F)-c1[nH]nc2ccnc(OC3CCOCC3)c12
105118C1CC(CCO1)Oc1nccc2[nH]nc(-c3ccc4cn[nH]c4c3)c12
105119C1CC(CCO1)Oc1nccc2[nH]nc(-c3ccc4nc[nH]c4c3)c12
105120Cn1ncc2cc(ccc12)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105121CC(C)n1cc2ccc(cc2n1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105123Cn1cnc2cc(ccc12)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105124C1C[C@H](CO1)n1cc(cn1)-c1c[nH]c2ccnc(OC3CCOCC3)c12
105125C1C[C@@H](CO1)n1cc(cn1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105126Cc1[nH]nc2cc(nc(OC3CCCCC3)c12)C1CC1
105128C1CC(CCO1)Oc1nccc2[nH]nc(-c3cnc4ccccc4c3)c12
105129N#CCc1cccc(c1)-c1[nH]nc2ccnc(OC3CCOCC3)c12
105130CN(C)c1cccc(c1)-c1[nH]nc2ccnc(OC3CCOCC3)c12
105131CC(C)NC(=O)c1cccc(c1)-c1[nH]nc2ccnc(OC3CCOCC3)c12
105132O=C(NC1CC1)c1cccc(c1)-c1[nH]nc2ccnc(OC3CCOCC3)c12
105133N#Cc1cncc(c1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105134C1CC(CCO1)Oc1nccc2[nH]nc(-c3cccc4[nH]ccc34)c12
105137C(N1CCOCC1)c1cccc(c1)-c1[nH]nc2ccnc(OC3CCOCC3)c12
105138COc1cc(Nc2[nH]nc3ccnc(OC4CCOCC4)c23)ccn1
105139C1CC(CCO1)Oc1nccc2n[nH]c(Nc3ccncc3)c12
105140CC(C)n1cc(Nc2[nH]nc3ccnc(OC4CCOCC4)c23)cn1
105141CS(=O)(=O)c1cccc(c1)-c1[nH]nc2ccnc(OC3CCOCC3)c12
105142COc1nccc2n[nH]c(-c3cccc(c3)S(C)(=O)=O)c12
105143CC(C)c1nc(n[nH]1)-c1n[nH]c2ccnc(NC3CCOCC3)c12
105144CNC(=O)c1cccc(c1)-c1[nH]nc2cc(C)nc(OC3CCOCC3)c12
105145Cc1cc2[nH]nc(-c3ccnc(c3)N3CCOCC3)c2c(OC2CCOCC2)n1
105146COc1nccc2n[nH]c(-c3ccc(cc3)S(C)(=O)=O)c12
105147N#Cc1cc(ccn1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105148Cn1cccc(Nc2n[nH]c3ccnc(OC4CCOCC4)c23)c1=O
105150CC(Oc1nccc2[nH]nc(-c3ccnc(c3)N3CCOCC3)c12)C(F)(F)F
105151COCCOc1nccc2[nH]nc(-c3ccnc(c3)N3CCOCC3)c12
105152O=C1OCCN1CCOc1nccc2[nH]nc(-c3ccnc(c3)N3CCOCC3)c12
105153CC(C)n1cc(cn1)-c1n[nH]c2ccnc(OCCN3CCOC3=O)c12
105154COc1nccc2[nH]nc(-c3cnn(c3)C3CCOCC3)c12
105155COC(=O)c1[nH]nc2ccnc(NC3CCOCC3)c12
105156C1CC(CCO1)Oc1nccc2[nH]nc(-c3cnn(c3)C3CCOCC3)c12
105157Cc1[nH]nc2ccnc(NC3CCOCC3)c12
105158C1CC(CO1)Oc1nccc2[nH]nc(-c3ccnc(c3)N3CCOCC3)c12
105159Cc1[nH]nc2ccnc(OC3CCCC3)c12
105160C1CC(CCO1)Oc1nccc2[nH]nc(-c3ccnc(c3)-c3cccnc3)c12
105161C1CC(CCO1)Oc1nccc2[nH]nc(-c3ccnc(c3)-c3ccncc3)c12
105162C1CC(CCO1)Oc1nccc2[nH]nc(-c3ccnc(c3)-c3cncnc3)c12
105163N#Cc1cccc(c1)-c1cc(ccn1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105164N#Cc1ccc(cc1)-c1cc(ccn1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105165CN(C)C(=O)c1cccc(c1)-c1cc(ccn1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105166C1CC(CCO1)Oc1nccc2[nH]nc(-c3ccnc(c3)-c3cn[nH]c3)c12
105168CC(=O)Nc1ccccc1-c1cc(ccn1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105169CC(=O)Nc1ccc(cn1)-c1cc(ccn1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105171CC(=O)Nc1cccc(c1)-c1cc(ccn1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105172CC(=O)Nc1ccc(cc1)-c1cc(ccn1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105173CNC(=O)c1cccc(c1)-c1cc(ccn1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105174CN(C)C(=O)c1ccc(cc1)-c1cc(ccn1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105175CCn1cc(cn1)-c1cc(ccn1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105176CC(C)Oc1nccc2[nH]nc(-c3cc(C(=O)N4CCCC4)n(c3)C(C)C)c12
105177CC(C)n1cc(cc1C(=O)N1CCC1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105178CC(C)Oc1nccc2[nH]nc(-c3ccnc(c3)C(=O)N3C[C@@H]4C[C@H]3CO4)c12
105179O=C(N1CCCC1)c1cc(ccn1)-c1n[nH]c2ccnc(OC3CCOCC3)c12
105180CC(C)n1cc(cn1)-c1n[nH]c2ccnc(OC3CCOC3)c12
105181COc1nccc2[nH]nc(-c3cnn(c3)C3CCOC3)c12
105182CNC(=O)c1cccc(c1)-c1[nH]nc2cc(C)nc(OC)c12
105183COc1nccc2[nH]nc(-c3ccnc(c3)N3C[C@H](C)O[C@H](C)C3)c12
127872CNc1nc(Nc2ccc(cc2Cl)-c2nnn[nH]2)ncc1C(F)(F)F
127873CNc1nc(Nc2ccc(cc2Cl)-c2nnn(C)n2)ncc1C(F)(F)F
127874CNc1nc(Nc2ccc(cc2OC)-n2cncn2)ncc1C(F)(F)F
127875CNc1nc(Nc2ccc(cc2OC)-c2cnn(C)c2)ncc1C(F)(F)F
127876CNc1nc(Nc2cc(F)c(cc2OC)-c2nc(C)no2)ncc1C(F)(F)F
127877CNc1nc(Nc2cc(OC)c(cc2Cl)-c2nnc(C)o2)ncc1C(F)(F)F
127878CNc1nc(Nc2ccc(cc2OC)-c2cncn2C)ncc1C(F)(F)F
127880CNc1nc(Nc2ccc(cc2OC)-c2nnnn2C)ncc1Cl
127881CNc1nc(Nc2cc(OC)c(cc2Cl)-c2cnnn2C)ncc1C(F)(F)F
127884CNc1nc(Nc2ccc(cc2OC)-c2cnoc2)ncc1Cl
127885CNc1nc(Nc2ccc(cc2OC)-c2nccn2C)ncc1Cl
127886CNc1nc(Nc2ccc(cc2OC)-c2cncn2C)ncc1Cl
127887CNc1nc(Nc2ccc(cc2OC)-c2cnnn2C)ncc1C(F)(F)F
127888CNc1nc(Nc2ccc(cc2OC)-c2nnn(C)n2)ncc1C(F)(F)F
127889CNc1nc(Nc2cc(OC)c(cc2Cl)-c2nccn2C)ncc1C(F)(F)F
127890CNc1nc(Nc2ccc(cc2OC)-c2nnnn2C)ncc1C(F)(F)F
127891CNc1nc(Nc2cc(OC)c(cc2Cl)-c2cncn2C)ncc1C(F)(F)F
127892CNc1nc(Nc2cc(F)c(cc2OC)-c2nnnn2C)ncc1C(F)(F)F
127893CNc1nc(Nc2ccc(cc2OC)-c2cnnn2C)ncc1Cl
127894CNc1nc(Nc2cc(OC)c(cc2Cl)-c2c(C)nn(C)c2C)ncc1C(F)(F)F
127895CNc1nc(Nc2ccc(cc2OC)-c2ccnn2C)ncc1C(F)(F)F
127896CNc1nc(Nc2ccc(cc2OC)-c2c(C)noc2C)ncc1C(F)(F)F
127897CNc1nc(Nc2ccc(cc2OC)-n2cnnn2)ncc1C(F)(F)F
127898CNc1nc(Nc2cc(OC)c(cc2Cl)-c2ccnn2C)ncc1C(F)(F)F
127899CCNc1nc(Nc2cc(F)c(cc2OC)-c2nnc(C)o2)ncc1C(F)(F)F
127900CNc1nc(Nc2cc(F)c(cc2OC)-c2nnc(C)o2)ncc1C(F)(F)F
127901CNc1nc(Nc2cc(OC)c(cc2Cl)-c2nc(C)no2)ncc1C(F)(F)F
127902CNc1nc(Nc2cc(OC)c(cc2Cl)-c2cnn(C)c2)ncc1C(F)(F)F
127903CNc1nc(Nc2ccc(cc2Cl)-c2nnc(C)o2)ncc1Cl
127904CNc1nc(Nc2ccc(cc2Cl)-c2nc(C)no2)ncc1Cl
127905CNc1nc(Nc2ccc(cc2OC)-c2cnn(C)c2)ncc1Cl
127906CNc1nc(Nc2cc(OC)c(cc2Cl)-c2nc(C)no2)ncc1Cl
127907CNc1nc(Nc2cc(OC)c(cc2Cl)-c2nnc(C)o2)ncc1Cl
127908CNc1nc(Nc2ccc(cc2OC)-c2cn(C)nc2C)ncc1C(F)(F)F
127909CNc1nc(Nc2ccc(cc2OC)-c2cnn(C)c2C)ncc1C(F)(F)F
127910CNc1nc(Nc2ccc(cc2OC)-c2nncn2C)ncc1C(F)(F)F
127911CNc1nc(Nc2cc(F)c(cc2OC)-c2cnn(C)c2C(=O)N(C)C)ncc1C(F)(F)F
127912CNc1nc(Nc2cc(F)c(cc2OC)-n2nnnc2C)ncc1C(F)(F)F
127913CNc1nc(Nc2cc(F)c(cc2OC)-c2cnnn2C)ncc1C(F)(F)F
127914CNc1nc(Nc2cc(F)c(cc2OC)-c2cnn(c2)C2COC2)ncc1C(F)(F)F
127915CNc1nc(Nc2cc(C)c(cc2OC)-n2nnnc2C)ncc1C(F)(F)F
127916CNc1nc(Nc2cc(C)c(cc2OC)-n2nnnc2COC)ncc1C(F)(F)F
127917CNc1nc(Nc2cc(F)c(cc2OC)-n2nc(C)cc2COC)ncc1C(F)(F)F
127918CNc1nc(Nc2ccc(cc2OC)-n2nc(C)cc2COC)ncc1C(F)(F)F
127919CNc1nc(Nc2cc(F)c(cc2OC)-n2nnnc2COC)ncc1C(F)(F)F
128246CNc1nc(Nc2cc3OCCN(C)C(=O)c3cc2Cl)ncc1C(F)(F)F
128247CNc1nc(Nc2cc3OC(C)(C)C(=O)N(C)c3cc2OC)ncc1Cl
128248CNc1nc(Nc2cc3oc(cc3cc2OC)C(=O)N(C)C)ncc1C(F)(F)F
128249CNc1nc(Nc2cc3n(C)c(=O)n(C)c3cc2Cl)ncc1C(F)(F)F
128250CNc1nc(Nc2cc3oc(=O)n(C)c3cc2Cl)ncc1C(F)(F)F
128251CNc1nc(Nc2cc3nc(C)oc3cc2Cl)ncc1C(F)(F)F
128252CNc1nc(Nc2cc3C(=O)N(C)Cc3cc2OC)ncc1C(F)(F)F
128253CNc1nc(Nc2cc3CN(C)C(=O)c3cc2Cl)ncc1Cl
128254CNc1nc(Nc2cc3CN(C)C(=O)c3cc2Cl)ncc1C(F)(F)F
128255CNc1nc(Nc2ccc3C(=O)N(Cc3c2OC)C2CC2)ncc1C(F)(F)F
128256CNc1nc(Nc2ccc3C(=O)N(C)Cc3c2OC)ncc1C(F)(F)F
128257CNc1nc(Nc2cc3OC(C)(C)C(=O)N(C)c3cc2OC)ncc1C(F)(F)F
128258CNc1nc(Nc2cc3oc(=O)[nH]c3cc2Cl)ncc1Cl
128260CNc1nc(Nc2cc3CCN(C)C(=O)c3cc2OC)ncc1C(F)(F)F
128261CNc1nc(Nc2cc3CCN(C)C(=O)c3cc2OC)ncc1C#N
128262CNc1nc(Nc2cc3cnn(C)c(=O)c3cc2OC)ncc1C(F)(F)F
128263CCN1Cc2c(ccc(Nc3ncc(c(NC)n3)C(F)(F)F)c2OC)C1=O
128264CNc1nc(Nc2ccc3C(=O)N(Cc3c2OC)C(C)(C)O)ncc1C(F)(F)F
128265CNc1nc(Nc2ccc3C(=O)N(Cc3c2OC)C2COC2)ncc1C(F)(F)F
128266CNc1nc(Nc2cc3CN(C)C(=O)c3cc2OC)ncc1C(F)(F)F
128267CNc1nc(Nc2cc3n(C)cc(C(=O)N4CCOCC4)c3cc2Cl)ncc1C(F)(F)F
128268CNc1nc(Nc2cc3CN(CC(C)(C)O)C(=O)c3cc2OC)ncc1C(F)(F)F
128269CNc1nc(Nc2cc3CN(C4COC4)C(=O)c3cc2OC)ncc1C(F)(F)F
128270CCNc1nc(Nc2cc3CN(C4COC4)C(=O)c3cc2OC)ncc1C(F)(F)F
128271CNc1nc(Nc2cc3n(C)cc(C(=O)N(C)C)c3cc2Cl)ncc1C(F)(F)F
128272CNc1nc(Nc2cc3n(C)cc(C(=O)N4CCNCC4)c3cc2Cl)ncc1C(F)(F)F
128273CCNc1nc(Nc2cc3n(C)cc(C(=O)N4CCOCC4)c3cc2Cl)ncc1C(F)(F)F
128274CNc1nc(Nc2cc3n(C)cc(C(=O)N4CCOCC4)c3cc2OC)ncc1C(F)(F)F
128275CNc1nc(Nc2cc3n(C)cc(C(=O)N4CCN(C)CC4)c3cc2Cl)ncc1C(F)(F)F
128276CCN1CCN(CC1)C(=O)c1cn(C)c2cc(Nc3ncc(c(NC)n3)C(F)(F)F)c(Cl)cc12
128277CNc1nc(Nc2cc3n(C)cc(C(=O)N4C[C@@H]5C[C@H]4CO5)c3cc2Cl)ncc1C(F)(F)F
129008CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCC(O)CC2)ncc1F
129009CNc1nc(Nc2ccc(cc2OC)C(=O)N(C)C)ncc1Cl
129010CNc1nc(Nc2ccc(cc2OC)C(=O)NC2CC2)ncc1Cl
129012CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCN3CCCCC3C2)ncc1Cl
129013CNc1nc(Nc2ccc(cc2OC)C(=O)N2CC(C)CC(C)C2)ncc1Cl
129014CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCCCC2)ncc1Cl
129015CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCC2)ncc1Cl
129016CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCC(F)(F)CC2)ncc1Cl
129017CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCN(CC2)C(C)=O)ncc1Cl
129018CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCCC(C2)C(F)(F)F)ncc1Cl
129019CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCCC2C)ncc1Cl
129020CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCCC2)ncc1Cl
129021CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCN(CC2)S(C)(=O)=O)ncc1Cl
129022CCC1(CC)CN(CCO1)C(=O)c1ccc(Nc2ncc(Cl)c(NC)n2)c(OC)c1
129023CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCOCC2CO)ncc1Cl
129024CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCOC(CC(C)C)C2)ncc1Cl
129025CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCNCC2)ncc1Cl
129026CCOc1cc(ccc1Nc1ncc(Cl)c(NC)n1)C(=O)N1CCOCC1
129027CNc1nc(Nc2ccc(cc2OC)C(N)=O)ncc1Cl
129028CNc1nc(Nc2ccc(cc2OC)C(=O)NC(C)C)ncc1Cl
129029CNc1nc(Nc2ccc(cc2OC)C(=O)N2C3CCC2COC3)ncc1Cl
129030COc1cc(ccc1Nc1ncc(Cl)c(OC(C)C)n1)C(=O)N1CCOCC1
129031CNc1nc(Nc2ccc(cc2OC)C(=O)N2CC3CC2CO3)ncc1Cl
129032CNc1nc(Nc2ccc(cc2OC)C(=O)N2CC3CCC(C2)O3)ncc1Cl
129033CNc1nc(Nc2ccc(cc2OC)C(=O)NCCCN)ncc1Cl
129034CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCOCC2)ncc1C1CC1
129035COc1cc(ccc1Nc1ncc(Cl)c(NCC(C)C)n1)C(=O)N1CCOCC1
129036CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCN(CC2)C(=O)C2CC2)ncc1Cl
129037CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCC(CC2)C(C)(C)O)ncc1Br
129038CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCC(C2)C(F)(F)F)ncc1Br
129039CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCC(CC2)C#N)ncc1Br
129040CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCN(CC2)C2CCC2)ncc1Br
129041CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCN(CC(F)(F)F)CC2)ncc1Br
129042CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCC(CC2)OC)ncc1Br
129043CNc1nc(Nc2ccc(cc2OC)C(=O)N2CC[C@@H](O)C2)ncc1Br
129044CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCN(CC2)C2COC2)ncc1Br
129045CNc1nc(Nc2ccc(cc2OC(C)C)C(=O)N2CCOCC2)ncc1Cl
129046COc1cc(ccc1Nc1ncc(Cl)c(NCC2CC2)n1)C(=O)N1CCOCC1
129047COc1cc(ccc1Nc1ncc(Cl)c(NC2CCC2)n1)C(=O)N1CCOCC1
129048CNc1nc(Nc2ccc(cc2O)C(=O)N2CCOCC2)ncc1Cl
129049CCN1CCN(CC1)C(=O)c1ccc(Nc2ncc(Br)c(OC)n2)c(OC)c1
129050COc1nc(Nc2ccc(cc2OC2CCC2)C(=O)N2CCOCC2)ncc1Br
129051CCNc1nc(Nc2cc(F)c(cc2OC)C(=O)N2CCOCC2)ncc1Cl
129052COc1cc(ccc1Nc1ncc(Br)c(OC)n1)C(=O)N1CC(C1)N1CCOCC1
129053CNc1nc(Nc2ccc(cc2OC)C(=O)N2CC(C2)N2CCOCC2)ncc1Cl
129054COc1cc(ccc1Nc1ncc(Cl)c(NC2(C)CCC2)n1)C(=O)N1CCOCC1
129055COc1cc(ccc1Nc1ncc(Cl)c(NCC2CCOC2)n1)C(=O)N1CCOCC1
129056COc1cc(ccc1Nc1ncc(I)c(OC)n1)C(=O)N1CCOCC1
129058COc1cc(ccc1Nc1ncc(Cl)c(NCCC2CC2)n1)C(=O)N1CCOCC1
129059COCCNc1nc(Nc2ccc(cc2OC)C(=O)N2CCOCC2)ncc1Cl
129060COCCNc1nc(Nc2ccc(cc2OCC(F)(F)F)C(=O)N2CCOCC2)ncc1Cl
129061CNc1nc(Nc2ccc(cc2Cl)C(=O)N2CCOCC2)ncc1Cl
129062CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCOCC2)ncc1OC
129063COCCOc1nc(Nc2ccc(cc2OC)C(=O)N2CCOCC2)ncc1Br
129064CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)N(C)C)ncc1Cl
129065CNc1nc(Nc2cc(OC)c(cc2Cl)C(N)=O)ncc1Cl
129066CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)NCCO)ncc1Cl
129067CNC(=O)c1cc(Cl)c(Nc2ncc(Cl)c(NC)n2)cc1OC
129068CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)N2CCC(F)(F)CC2)ncc1Cl
129069CCNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)NC2CC2)ncc1C(F)(F)F
129070CCNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)NCCOC)ncc1C(F)(F)F
129071CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)N2CCNCC2)ncc1Cl
129072CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)N2CCC(CC2)N(C)C)ncc1Cl
129073CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)N2CCC(O)C2)ncc1Cl
129074CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)NC2COC2)ncc1Cl
129075CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)NC2CC2)ncc1C(F)(F)F
129076CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)NC2CCN(C)CC2)ncc1Cl
129077CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)N2CCCC2)ncc1Cl
129078CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)NC(C)(C)C)ncc1Cl
129079CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)N(C)C)ncc1C(F)(F)F
129080CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)N2CCC(O)CC2)ncc1Cl
129081CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)N2CCOC(CO)C2)ncc1Cl
129082CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)N(C)CCO)ncc1Cl
129083CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)N2CCCOCC2)ncc1Cl
129084CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)N2CCC(CC2)C#N)ncc1Cl
129085CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)N2CC(O)C2)ncc1Cl
129086CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)NC2(CC2)C#N)ncc1Cl
129087CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)N2CCC(C2)C#N)ncc1Cl
129088CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)N2C[C@H](C)N[C@H](C)C2)ncc1Cl
129089CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)NC2CCN(C)CC2)ncc1C(F)(F)F
129090CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)NC2COC2)ncc1C(F)(F)F
129091CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)NCC(C)(C)O)ncc1C(F)(F)F
129092CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)N2CCNCC2)ncc1C(F)(F)F
129093CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)N2CCC(C2)C#N)ncc1C(F)(F)F
129094CNc1nc(Nc2cc(F)c(cc2OC)C(=O)N2CCC(C2)C#N)ncc1C(F)(F)F
129095CNC(=O)c1cc(OC)c(Nc2ncc(c(NC)n2)C(F)(F)F)cc1F
129096CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)N(C)CC(C)(C)O)ncc1C(F)(F)F
129097COc1cc(ccc1Nc1ncc(C2CC2)c(OC)n1)C(=O)N1CCOCC1
129098CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCOCC2)ncc1C(C)=O
129099COCCNc1nc(Nc2cc(F)c(cc2OC)C(=O)N2CCOCC2)ncc1Br
129100COCCNc1nc(Nc2ccc(cc2OC(C)C)C(=O)N2CCOCC2)ncc1Br
129101COCCOc1nc(Nc2ccc(cc2OC2CCC2)C(=O)N2CCOCC2)ncc1Cl
129102CNc1nc(Nc2ccc(cc2OC2CCCC2)C(=O)N2CC3(COC3)C2)ncc1Cl
129103CNc1nc(Nc2ccc(cc2OC)C(=O)N2CC3(COC3)C2)ncc1Cl
129104CNc1nc(Nc2ccc(cc2OC)C(=O)N2CC(F)(F)OC(F)(F)C2)ncc1C#N
129105CNc1nc(Nc2ccc(cc2C2CC2)C(=O)N2CCOCC2)ncc1Cl
129106CNc1nc(Nc2ccc(cc2OC)C(=O)NC2CC(F)(F)C2)ncc1C#N
129107CNc1nc(Nc2ccc(cc2OC)C(=O)NCC2CC2)ncc1C#N
129108CNc1nc(Nc2ccc(cc2OC)C(=O)N2CC[C@H](F)C2)ncc1C#N
129109CNC(=O)c1ccc(Nc2ncc(C#N)c(NC)n2)c(OC)c1
129110CCN(CC)C(=O)c1ccc(Nc2ncc(C#N)c(NC)n2)c(OC)c1
129111CNc1nc(Nc2ccc(cc2OC)C(=O)NC(C)C)ncc1C#N
129112CCNC(=O)c1ccc(Nc2ncc(C#N)c(NC)n2)c(OC)c1
129113CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCCCC2)ncc1C#N
129114CNc1nc(Nc2ccc(cc2OC)C(=O)NCC(F)F)ncc1C#N
129115CNc1nc(Nc2ccc(cc2OC)C(=O)NC(C)(C)C)ncc1C#N
129116CCN(C(C)C)C(=O)c1ccc(Nc2ncc(C#N)c(NC)n2)c(OC)c1
129117CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCC(F)(F)C2)ncc1C#N
129119CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCC2)ncc1C#N
129120CNc1nc(Nc2ccc(cc2OC)C(=O)N(C)C(C)C)ncc1C#N
129121COc1cc(ccc1Nc1ncc(Cl)c(NC2CCOC2)n1)C(=O)N1CCOCC1
129122CNc1nc(Nc2ccc(cc2OC(C)C)C(=O)N2CCOCC2)ncc1C(F)(F)F
129123CCOc1cc(ccc1Nc1ncc(c(NC)n1)C(F)(F)F)C(=O)N1CCOCC1
129124CNc1nc(Nc2ccc(cc2OC2CC2)C(=O)N2CCOCC2)ncc1Cl
129125CNc1nc(Nc2ccc(cc2OC2CC2)C(=O)N2CCOCC2)ncc1Br
129126COc1cc(ccc1Nc1ncc(Cl)c(NCCS(C)(=O)=O)n1)C(=O)N1CCOCC1
129127CNc1nc(Nc2cc(OC)c(CC(=O)N3CCOCC3)cc2OC)ncc1Br
129128CNc1nc(Nc2cc(OC)c(CC(=O)N3CCOCC3)cc2OC)ncc1Cl
129129CNc1nc(Nc2ccc(CC(=O)N3CCOCC3)cc2OC)ncc1Cl
129130CNc1nc(Nc2ccc(CC(=O)N3CCOCC3)cc2OC)ncc1C(F)(F)F
129131COc1cc(CC(=O)N2CCOCC2)ccc1Nc1ncc(Br)c(OC)n1
129132CNc1nc(Nc2cc(OC)c(CC(=O)N3CCOCC3)cc2OC)ncc1C(F)(F)F
129133CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)NCCCN)ncc1Cl
129134COCCNc1nc(Nc2ccc(cc2OC)C(=O)N2CCOCC2)ncc1Br
129135COC(C)CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCOCC2)ncc1Cl
129136CNc1nc(Nc2ccc(cc2C)C(=O)N2CCC(O)CC2)ncc1Cl
129137CCNc1nc(Nc2ccc(cc2OC(F)(F)F)C(=O)N2CCOCC2)ncc1C(F)(F)F
129138CNc1nc(Nc2ccc(cc2OC(F)(F)F)C(=O)N2CCOCC2)ncc1C(F)(F)F
129139CCNc1nc(Nc2cc(OC)c(cc2F)C(=O)N2CCOCC2)ncc1C(F)(F)F
129140CCNc1nc(Nc2cc(F)c(cc2OC)C(=O)N(C)C)ncc1C#N
129141CCNc1nc(Nc2ccc(C(=O)N3CCOCC3)c(F)c2OC)ncc1C(F)(F)F
129142CCNc1nc(Nc2ccc(C(=O)N3C[C@@H]4C[C@H]3CO4)c(F)c2OC)ncc1C(F)(F)F
129143CNc1nc(Nc2ccc(cc2OC)C(=O)N2C[C@H](F)[C@@H](F)C2)ncc1C#N
129144CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)N2CCC(C2)OC)ncc1C(F)(F)F
129145CNc1nc(Nc2cc(F)c(cc2OC)C(=O)N2CCC(C2)OC)ncc1C(F)(F)F
129146CNc1nc(Nc2cc(F)c(cc2OC)C(=O)N(C)CC(C)(C)O)ncc1C(F)(F)F
129147CNc1nc(Nc2cc(F)c(cc2OC)C(=O)N2C[C@H](C)O[C@H](C)C2)ncc1C(F)(F)F
129148CCNc1nc(Nc2ccc(cc2OC(C)C)C(=O)N2CCOCC2)ncc1C(F)(F)F
129149COc1cc(ccc1Nc1ncc(Cl)c(n1)N1CCCCC1)C(=O)N1CCOCC1
129150COc1cc(ccc1Nc1ncc(Cl)c(n1)N1CCCC1)C(=O)N1CCOCC1
129152CCNc1nc(Nc2ccc(cc2OC)C(=O)N2CCOCC2)ncc1C(F)(F)F
129153CCNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)N2CCOCC2)ncc1Cl
129154COc1cc(C(=O)N2CCOCC2)c(F)cc1Nc1ncc(c(OC)n1)C(F)(F)F
129155COc1cc(Nc2ncc(Cl)c(OC)n2)c(Cl)cc1C(=O)N1CCOCC1
129156COc1nc(Nc2ccc(cc2Cl)C(=O)N2CCOCC2)ncc1Cl
129157COc1cc(C(=O)N2CCOCC2)c(Cl)cc1Nc1ncc(c(OC)n1)C(F)(F)F
129158COc1cc(ccc1Nc1ncc(c(OC)n1)C(F)(F)F)C(=O)N1CCOCC1
129159COc1cc(ccc1Nc1ncc(Cl)c(OC2CCOCC2)n1)C(=O)N1CCOCC1
129161CNc1nc(Nc2ccc(cc2OCCF)C(=O)N2CCOCC2)ncc1C(F)(F)F
129162CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)NC2(CC2)C#N)ncc1C(F)(F)F
129163CNC(=O)c1cc(Cl)c(Nc2ncc(c(NC)n2)C(F)(F)F)cc1OC
129164CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)N2CC(C)OC(C)C2)ncc1C(F)(F)F
129165FC(F)(F)c1cnc(Nc2ccc(cc2Br)C(=O)N2CCOCC2)nc1N1CCCC1
129166CNc1nc(Nc2ccc(cc2OC2CCC2)C(=O)N2CCOCC2)ncc1C(F)(F)F
129167CNc1nc(Nc2ccc(cc2OC)C(=O)N2CC(F)(F)C2)ncc1C(F)(F)F
129168CNc1nc(Nc2ccc(cc2OC)C(=O)NC2COC2)ncc1C(F)(F)F
129169CNc1nc(Nc2ccc(cc2OC)C(=O)N2CC3CCC(C2)O3)ncc1C(F)(F)F
129170CNc1nc(Nc2ccc(cc2OC)C(=O)N2CC3CC(C2)O3)ncc1C(F)(F)F
129171CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCCC2)ncc1C(F)(F)F
129172CCN(CC)C(=O)c1ccc(Nc2ncc(c(NC)n2)C(F)(F)F)c(OC)c1
129173CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCC(CC2)N(C)C)ncc1C(F)(F)F
129174CNc1nc(Nc2ccc(cc2OC)C(=O)N2CC(C)OC(C)C2)ncc1C(F)(F)F
129175CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCC(CC2)C#N)ncc1C(F)(F)F
129176CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCN(CC(F)(F)F)CC2)ncc1C(F)(F)F
129177CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCC(CC2)OC)ncc1C(F)(F)F
129178CNc1nc(Nc2ccc(cc2OC)C(=O)NCCOC)ncc1C(F)(F)F
129179CNc1nc(Nc2ccc(cc2OC)C(=O)NC2CCN(C)CC2)ncc1C(F)(F)F
129180CNc1nc(Nc2ccc(cc2OC)C(=O)NC2CCC(F)(F)CC2)ncc1C(F)(F)F
129181CNc1nc(Nc2ccc(cc2OC2COC2)C(=O)N2CCOCC2)ncc1Cl
129182CNc1nc(Nc2ccc(cc2OCC2CC2)C(=O)N2CCOCC2)ncc1C(F)(F)F
129183CNc1nc(Nc2ccc(cc2OCC2CCC2)C(=O)N2CCOCC2)ncc1C(F)(F)F
129184CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)N2CCOCC2)ncc1Br
129185CNc1nc(Nc2ccc(cc2C2CC2)C(=O)N2CCOCC2)ncc1C(F)(F)F
129186CNc1nc(Nc2ccc(cc2Br)C(=O)N2CCOCC2)ncc1C(F)(F)F
129187CNc1nc(Nc2ccc(cc2Cl)C(=O)N2CCOCC2)ncc1C(F)(F)F
129188CNc1nc(Nc2cc(Cl)c(cc2OC)C(=O)N2CCOCC2)ncc1Cl
129189COc1cc(C(=O)N2CCOCC2)c(Cl)cc1Nc1ncc(Br)c(OC)n1
129190CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)N2CCOCC2)ncc1Cl
129192COc1cc(ccc1Nc1ncc(Cl)c(OC)n1)C(=O)N1CCCC1
129193CCOc1cc(C(=O)N2CCOCC2)c(F)cc1Nc1ncc(c(NC)n1)C(F)(F)F
129194CNc1nc(Nc2ccc(cc2OC)C(=O)N(C)CCOC)ncc1C(F)(F)F
129195CCNc1nc(Nc2ccc(cc2OC)C(=O)N(C)CCOC)ncc1C(F)(F)F
129196CNc1nc(Nc2cc(F)c(cc2OC)C(=O)N(C)CCOC)ncc1C(F)(F)F
129197CCNc1nc(Nc2cc(F)c(cc2OC)C(=O)N(C)CCOC)ncc1C(F)(F)F
129198CNc1nc(Nc2cc(F)c(cc2OC)C(=O)N2CCC[C@H]2COC)ncc1C(F)(F)F
129199CCNc1nc(Nc2cc(F)c(cc2OC)C(=O)N2CCC[C@H]2COC)ncc1C(F)(F)F
129200CCNc1nc(Nc2cc(F)c(cc2OC)C(=O)N(CC)CCOC)ncc1C(F)(F)F
129201CCN(CCOC)C(=O)c1cc(OC)c(Nc2ncc(c(NC)n2)C(F)(F)F)cc1F
129202CCNc1nc(Nc2cc(F)c(cc2OCC)C(=O)N2CCOCC2)ncc1C(F)(F)F
129206COc1cc(ccc1Nc1ncc(C#N)c(OC)n1)C(=O)N1CCOCC1
129207CCNc1nc(Nc2cc(F)c(cc2OC)C(=O)N2CCOCC2)ncc1C#N
129208CNc1nc(Nc2cc(F)c(cc2OC)C(=O)N2CCOCC2)ncc1C#N
129209CNc1nc(Nc2cc(F)c(cc2OC)C(=O)N2C[C@H](C)O[C@H](C)C2)ncc1C#N
129210CCNc1nc(Nc2cc(F)c(cc2OC)C(=O)N2C[C@H](C)O[C@H](C)C2)ncc1C#N
129211CNc1nc(Nc2cc(F)c(cc2OC)C(=O)N(C)C)ncc1C#N
50059889CN[C@@H]1CC2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13
50132420O=C1Nc2ccc(cc2\C1=C\c1ccc[nH]1)-c1cccnc1
50193995C[C@@H]1CCN(C[C@@H]1N(C)c1ncnc2[nH]ccc12)C(=O)CC#N
50222572CS(=O)(=O)c1ccc(cc1)-c1ccc2c(Nc3ccccc3)c(cnc2c1)C(N)=O
50242742COc1cc(ccc1Nc1ncc(Cl)c(Nc2ccccc2S(=O)(=O)C(C)C)n1)N1CCC(CC1)N1CCN(C)CC1
50249542COc1cc(Nc2ncc(F)c(Nc3ccc4OC(C)(C)C(=O)Nc4n3)n2)cc(OC)c1OC
50332294Cc1cnc(Nc2ccc(OCCN3CCCC3)cc2)nc1Nc1cccc(c1)S(=O)(=O)NC(C)(C)C
50355496O=C(N1CCNCC1)c1ccc(\C=C\c2n[nH]c3ccccc23)cc1
50355499CN(C)CC(=O)N1CCC(CC1)c1ccc(NC(=O)c2ncc([nH]2)C#N)c(c1)C1=CCCCC1
50355501N#CC[C@H](C1CCCC1)n1cc(cn1)-c1ncnc2[nH]ccc12
50355502CN(C(=O)CN1CCN(C)CC1)c1ccc(cc1)N=C(C1C(=O)Nc2ccccc12)c1ccccc1
50360301C[C@@H]1CCNC(=O)c2cc3ccc(cc3n12)C(=O)Nc1nc2ccccc2n1CCCN(C)C
50379529COc1cc(ccc1Nc1ncc2N(C)C(=O)c3ccccc3N(C)c2n1)C(=O)N1CCC(CC1)N1CCN(C)CC1
50393038Cn1cc(C=Cc2[nH]nc3ccnc(OC4CCCCC4)c23)cn1
50396041CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCOCC2)ncc1Cl
50396147CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCOCC2)ncc1C#N
50396148CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCOCC2)ncc1C(F)(F)F
50396149CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCOCC2)ncc1F
50396150CNc1nc(Nc2ccc(cc2OC)C(=O)N2CCOCC2)ncc1Br
50396151CNc1nc(Nc2ccc(cc2Br)C(=O)N2CCOCC2)ncc1Cl
50396152CNc1nc(Nc2ccc(cc2C)C(=O)N2CCOCC2)ncc1Cl
50396153CNc1nc(Nc2ccccc2OC(F)F)ncc1Cl
50396154CNc1nc(Nc2ccccc2Br)ncc1Cl
50396155CNc1nc(Nc2ccccc2OC)ncc1Cl
50396156CNc1nc(Nc2ccccc2C)ncc1Cl
50396157CNc1nc(Nc2ccccc2)ncc1Cl
50396158CNc1nc(Nc2ccc(cc2)C(=O)N2CCOCC2)ncc1Cl
50396159Cc1cc(cc(C)c1C)-c1ccc2nc(Nc3ccccc3)nn2c1
50396160Cc1ccccc1Nc1nc2ccc(cn2n1)-c1cc(C)c(O)c(C)c1
50398659COc1cc(ccc1Nc1ncc(Br)c(OC)n1)C(=O)N1CCOCC1
50398660COc1cc(ccc1Nc1ncc(Cl)c(OC)n1)C(=O)N1CCOCC1
50398661CCNc1nc(Nc2cc3CN(CC(C)(C)O)C(=O)c3cc2OC)ncc1C(F)(F)F
50398662CCNc1nc(Nc2cc(F)c(cc2OC)C(=O)NCC(C)(C)O)ncc1C(F)(F)F
50398663CNc1nc(Nc2cnc(cc2OC)C2CCOCC2)ncc1C(F)(F)F
50398664CCNc1nc(Nc2cnc(cc2OC)C(=O)N2CCOCC2)ncc1C(F)(F)F
50398665CNc1nc(Nc2cc(F)c(cc2OC)S(C)(=O)=O)ncc1C(F)(F)F
50398666CNc1nc(Nc2ccc(cc2Cl)-c2nnnn2C)ncc1C(F)(F)F
50398667COc1cc(C(=O)N2CCOCC2)c(F)cc1Nc1ncc(c(NC2CC2)n1)C(F)(F)F
50398668CCNc1nc(Nc2cc(F)c(cc2OC)C(=O)N2CCOCC2)ncc1C(F)(F)F
50398669CNc1nc(Nc2cc(F)c(cc2OC)C(=O)N2CCOCC2)ncc1C(F)(F)F
50398670CNc1nc(Nc2ccc(C(=O)N3CCOCC3)c(F)c2OC)ncc1C(F)(F)F
50398671CNc1nc(Nc2cc(OC)c(cc2F)C(=O)N2CCOCC2)ncc1C(F)(F)F
50398672CNc1nc(Nc2cc(C)c(cc2OC)C(=O)N2CCOCC2)ncc1C(F)(F)F
50398673CNc1nc(Nc2cc(C)c(cc2Cl)C(=O)N2CCOCC2)ncc1C(F)(F)F
50398674CCNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)N2CCOCC2)ncc1C(F)(F)F
50398675CNc1nc(Nc2cc(OC)c(cc2Cl)C(=O)N2CCOCC2)ncc1C(F)(F)F
50398676CNc1nc(Nc2cc(OC)c(cc2OC)C(=O)N2CCOCC2)ncc1C(F)(F)F
50398677CNc1nc(Nc2cc(Cl)c(cc2OC)C(=O)N2CCOCC2)ncc1C(F)(F)F
50401284Fc1cc(ccn1)-c1ccc(OCc2ccccc2)c(c1)C(=O)Nc1cccnc1
50423656CO[C@H]1[C@@H](C[C@H]2O[C@@]1(C)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13)N(C)C(=O)c1ccccc1
50423773C[C@]12O[C@@H](C[C@@]1(O)CO)n1c3ccccc3c3c4C(=O)NCc4c4c5ccccc5n2c4c13
50426395CNc1nc(Nc2cn(C)nc2C)ncc1C(F)(F)F
50426396CNc1nc(Nc2cnn(C)c2)ncc1C(F)(F)F
50426397CNc1nc(Nc2ccnn2C)ncc1C(F)(F)F
50426398CNc1nc(Nc2ccn(C)n2)ncc1C(F)(F)F
50426401CNc1nc(Nc2cnn(C)c2Cl)ncc1C(F)(F)F
50426402CNc1nc(Nc2cnn(C)c2C)ncc1C(F)(F)F
50426403CNc1nc(Nc2cnn(CC(C)(C)O)c2Cl)ncc1C(F)(F)F
50428692CC(C)Nc1c(nnc2c(C)c(ccc12)-c1ccncc1)C(N)=O
50428693CNC(=O)c1nnc2cc(ccc2c1N[C@H](C)C1CC1)-c1ccc(cc1)S(C)(=O)=O
50428694CNC(=O)c1nnc2cc(ccc2c1NC(C)C)-c1ccc(cc1)S(C)(=O)=O
50428695CC(C)Nc1c(nnc2cc(ccc12)-c1cnsc1)C(N)=O
50428696CC(C)Nc1c(nnc2cc(ccc12)N1CCOCC1)C(N)=O
50428697CC(C)Nc1c(nnc2cc(ccc12)N1CCN(C)CC1)C(N)=O
50428698CC(C)Nc1c(nnc2cc(ccc12)-c1cnn(C)c1)C(N)=O
50428699CC(C)Nc1c(nnc2ccc(cc12)-c1cnn(C)c1)C(N)=O
50428700CC(C)Nc1c(nnc2cc(ccc12)-c1cn[nH]c1)C(N)=O
50428701CC(C)Nc1c(nnc2ccc(cc12)-c1cn[nH]c1)C(N)=O
50428702CC(C)Nc1c(nnc2ccc(cc12)-c1ccncc1)C(N)=O
50428703C[C@@H](Nc1c(nnc2cc(ccc12)-c1ccncc1)C(N)=O)C1CC1
50428704CC(C)Nc1c(nnc2cc(ccc12)-c1ccncc1)C(N)=O
50428705NC(=O)c1nnc2cc(ccc2c1NCCO)-c1ccncc1
50428706NC(=O)c1nnc2cc(ccc2c1NCCCO)-c1ccncc1
50428707C[C@@H](Nc1c(nnc2cc(ccc12)-c1ccc(cc1)S(C)(=O)=O)C(N)=O)c1ccccc1
50428708CS(=O)(=O)c1ccc(cc1)-c1ccc2c(N)c(nnc2c1)C(N)=O
50428709CNc1c(nnc2cc(ccc12)-c1ccc(cc1)S(C)(=O)=O)C(N)=O
50428710CS(=O)(=O)c1ccc(cc1)-c1ccc2c(NC3CCOC3)c(nnc2c1)C(N)=O
50428711CS(=O)(=O)c1ccc(cc1)-c1ccc2c(NC3CC3)c(nnc2c1)C(N)=O
50428712CS(=O)(=O)c1ccc(cc1)-c1ccc2c(NC3CCOCC3)c(nnc2c1)C(N)=O
50428713CCNc1c(nnc2cc(ccc12)-c1ccc(cc1)S(C)(=O)=O)C(N)=O
50428714CS(=O)(=O)c1ccc(cc1)-c1ccc2c(NCC3CC3)c(nnc2c1)C(N)=O
50428715CS(=O)(=O)c1ccc(cc1)-c1ccc2c(NC3CCC3)c(nnc2c1)C(N)=O
50428716C[C@@H](Nc1c(nnc2cc(ccc12)-c1ccc(cc1)S(C)(=O)=O)C(N)=O)C1CC1
50428717CC[C@@H](C)Nc1c(nnc2cc(ccc12)-c1ccc(cc1)S(C)(=O)=O)C(N)=O
50428718CC(C)Nc1c(nnc2cc(ccc12)-c1ccc(cc1)S(C)(=O)=O)C(N)=O
50428719CC(C)Nc1c(cnc2cc(ccc12)-c1ccc(cc1)S(C)(=O)=O)C(N)=O
50431895CC(C)Nc1c(cnc2cc(ccc12)-c1ccc(cc1)S(C)(=O)=O)-c1nccs1
50431896CC(C)Nc1c(cnc2cc(ccc12)-c1ccc(cc1)S(C)(=O)=O)C(C)=O
50431897C[C@@H](Nc1c(cnc2cc(ccc12)-c1ccc(cc1)-n1ccoc1=O)C#N)C1CC1
50431898C[C@@H](Nc1c(cnc2cc(ccc12)-c1ccc(cc1)S(C)(=O)=O)C#N)C1CC1
50431899CN(C(C)=O)c1c(cnc2cc(ccc12)-c1ccc(cc1)S(C)(=O)=O)C#N
50431900CS(=O)(=O)c1ccc(cc1)-c1ccc2c(c(cnc2c1)C#N)-n1ccnc1
50431901CN(c1ccccc1)c1c(cnc2cc(ccc12)-c1ccc(cc1)S(C)(=O)=O)C#N
50431902CN1CCN(CC1)c1c(cnc2cc(ccc12)-c1ccc(cc1)S(C)(=O)=O)C#N
50431903CS(=O)(=O)c1ccc(cc1)-c1ccc2c(N3CCCCC3)c(cnc2c1)C#N
50431904CN(C)c1c(cnc2cc(ccc12)-c1ccc(cc1)S(C)(=O)=O)C#N
50431905CS(=O)(=O)c1ccc(cc1)-c1ccc2c(N3CCC3)c(cnc2c1)C#N
50431906Cn1cc(cn1)-c1ccc2c(N3CCC3)c(cnc2c1)C#N
50431907CC(C)Nc1c(cnc2ccccc12)C#N
50431908CC(C)Nc1c(cnc2cc(ccc12)-c1ccc(Cl)s1)C#N
50431909CC(C)Nc1c(cnc2cc(ccc12)-c1ccc(nc1)S(C)(=O)=O)C#N
50431910CC(C)Nc1c(cnc2cc(ccc12)-c1ccc(cc1)S(=O)(=O)N(C)C)C#N
50431911CC(C)Nc1c(cnc2cc(ccc12)-c1ccc(cc1)S(=O)(=O)N1CCCC1)C#N
50431912CC(C)Nc1c(cnc2cc(ccc12)-c1cnc(C)s1)C#N
50431913CC(C)Nc1c(cnc2cc(ccc12)-c1ccc(cc1)S(=O)(=O)N1CCOCC1)C#N
50431914CNS(=O)(=O)c1ccc(cc1)-c1ccc2c(NC(C)C)c(cnc2c1)C#N
50431915CC(C)Nc1c(cnc2cc(ccc12)-c1cnn(C)c1)C#N
50431916CC(C)Nc1c(cnc2cc(ccc12)-c1ccc(cc1)S(C)(=O)=O)-c1cnn(C)c1
50431917CC(C)Nc1c(cnc2cc(ccc12)-c1ccc(cc1)S(C)(=O)=O)C#N
50432020FC(F)(F)c1cccc(c1)S(=O)(=O)c1ccc2nnc(-c3ccccc3)n2n1
50432021FC(F)(F)c1cccc(c1)S(=O)c1ccc2nnc(-c3ccccc3)n2n1
50432030CC(Sc1ccc2nnc(-c3cccc(Cl)c3)n2n1)c1ccn[nH]1
50432031CC(Sc1ccc2nnc(-c3cccs3)n2n1)c1nnco1
50432032CC(C)(Sc1ccc2nnc(-c3cccs3)n2n1)C(N)=O
50432033CC(C)C(Sc1ccc2nnc(-c3cccs3)n2n1)C(N)=O
50432034CCC(Sc1ccc2nnc(-c3cccs3)n2n1)C(=O)OC
50432035COC(=O)[C@@H](C)Sc1ccc2nnc(-c3cccs3)n2n1
50432036COC(=O)[C@H](C)Sc1ccc2nnc(-c3cccs3)n2n1
50432037CC(Sc1ccc2nnc(-c3cccs3)n2n1)C(N)=O
50432038S(c1ccccc1)c1ccc2nnc(-c3cncs3)n2n1
50432039FC(F)(F)c1ccnc(Sc2ccc3nnc(-c4cncs4)n3n2)n1
50432040S(c1ccc2nnc(-c3cncs3)n2n1)c1ncccn1
50432041FC(F)(F)Oc1cccc(Sc2ccc3nnc(-c4cncs4)n3n2)c1
50432042CC(C)(C)c1cccc(Sc2ccc3nnc(-c4cncs4)n3n2)c1
50432043COc1cccc(Sc2ccc3nnc(-c4cncs4)n3n2)c1
50432044Fc1cccc(Sc2ccc3nnc(-c4cncs4)n3n2)c1
50432045Clc1cccc(Sc2ccc3nnc(-c4cncs4)n3n2)c1
50432046Brc1cccc(Sc2ccc3nnc(-c4cncs4)n3n2)c1
50432047FC(F)(F)c1ccccc1Sc1ccc2nnc(-c3ccccc3)n2n1
50432048FC(F)(F)c1ccc(Sc2ccc3nnc(-c4ccccc4)n3n2)cc1
50432051FC(F)(F)c1cccc(Sc2ccc3nnc(C4CCOCC4)n3n2)c1
50432052FC(F)(F)c1cccc(Sc2ccc3nnc(C4CCCC4)n3n2)c1
50432053FC(F)(F)c1cccc(Sc2ccc3nnc(C4CC4)n3n2)c1
50432054Fc1ccc(cc1)-c1nnc2ccc(Sc3cccc(c3)C(F)(F)F)nn12
50432055FC(F)(F)c1cccc(Sc2ccc3nnc(-c4cccc(c4)N4CCNCC4)n3n2)c1
50432056FC(F)(F)c1cccc(Sc2ccc3nnc(-c4cccc(Cl)c4)n3n2)c1
50432057FC(F)(F)c1cccc(Sc2ccc3nnc(-c4ccccc4Cl)n3n2)c1
50432058FC(F)(F)c1cccc(Sc2ccc3nnc(-c4ccncc4)n3n2)c1
50432059FC(F)(F)c1cccc(Sc2ccc3nnc(-c4cccnc4)n3n2)c1
50432060FC(F)(F)c1cccc(Sc2ccc3nnc(-c4ccccn4)n3n2)c1
50432061FC(F)(F)c1cccc(Sc2ccc3nnc(-c4sccc4Br)n3n2)c1
50432062FC(F)(F)c1cccc(Sc2ccc3nnc(-c4cscn4)n3n2)c1
50432063FC(F)(F)c1cccc(Sc2ccc3nnc(-c4nccs4)n3n2)c1
50432064FC(F)(F)c1cccc(Sc2ccc3nnc(-c4cncs4)n3n2)c1
50432065FC(F)(F)c1cccc(Sc2ccc3nnc(-c4ccn[nH]4)n3n2)c1
50432066COC(=O)C(C)Sc1ccc2ncc(-c3cccs3)n2n1
50432067FC(F)(F)c1cccc(Sc2cn3c(cnc3cn2)-c2cccs2)c1
50432068FC(F)(F)c1cccc(Sc2ccc3ncc(-c4cccs4)n3c2)c1
50432070FC(F)(F)c1cccc(Sc2ccc3ncc(-c4cccs4)n3n2)c1
50432071FC(F)(F)c1cccc(Sc2ccc3nnc(-c4cccs4)n3n2)c1
50432072FC(F)(F)c1cccc(Sc2ccc3nnc(-c4ccccc4)n3n2)c1
50436423COc1cc(ccc1Nc1ncc(F)c(Nc2ccccc2NS(C)(=O)=O)n1)N1CCOCC1
50437051CC(C)Oc1ccc2NC(=O)\C(=C/c3cc4CN(CCc4[nH]3)C(C)=O)c2c1
50437052CC(=O)Nc1ccc2NC(=O)\C(=C/c3cc4CN(CCc4[nH]3)C(=O)N3CCOCC3)c2c1
50437055COc1ccc2NC(=O)\C(=C/c3cc4CN(CCc4[nH]3)C(=O)N3CCOCC3)c2c1
50437056COc1ccc2NC(=O)\C(=C/c3cc4CN(CCc4[nH]3)C(=O)N3CCN(C)CC3)c2c1
50437057COc1ccc2NC(=O)\C(=C/c3cc4CN(CCc4[nH]3)C(=O)c3cnoc3C)c2c1
50437058COc1ccc2NC(=O)\C(=C/c3cc4CN(CCc4[nH]3)C(C)=O)c2c1
50437059COc1ccc2NC(=O)\C(=C/c3cc4CN(CCc4[nH]3)C(=O)CCN)c2c1
50437061CC(=O)N1CCc2[nH]c(\C=C3/C(=O)Nc4ccc(cc34)C#N)cc2C1
50437062CC(=O)N1CCc2[nH]c(\C=C3/C(=O)Nc4ccc(cc34)C(F)(F)F)cc2C1
50437063COc1ccc2NC(=O)\C(=C/c3[nH]c4CCN(Cc4c3Cl)C(C)=O)c2c1
50437064COc1ccc2N(C)C(=O)\C(=C/c3cc4CN(CCc4[nH]3)C(=O)N3CCOCC3)c2c1
50437065COc1ccc2NC(=O)\C(=C/c3[nH]c(C)c(C(=O)NCCCN)c3C)c2c1
50441567CN1CCN(Cc2ccc(cc2)-c2cnc3[nH]cc(-c4ccc5[nH]ccc5c4)c3c2)CC1
50441569Nc1ccc(cn1)-c1cnc2[nH]cc(-c3ccc4[nH]ccc4c3)c2c1
50441571COc1cc(cc(OC)c1OC)-c1cnc2[nH]cc(-c3ccc(N)nc3)c2c1
50441572COc1cc(cc(OC)c1OC)-c1cnc2[nH]cc(-c3ccc4[nH]ccc4c3)c2c1
50441573COc1cc(cc(OC)c1OC)-c1cnc2[nH]c(=O)n(-c3ccc4[nH]ccc4c3)c2n1
50442139CCc1ccc2nc(Nc3cc(Cc4ccccc4)nc(N[C@H]4CC[C@H](O)CC4)n3)sc2c1
50448110CNc1nc(Nc2cnn([C@H]3CCN(C[C@@H]3F)C3COC3)c2Cl)ncc1C(F)(F)F
50448111CNc1nc(Nc2cn(nc2C)[C@H]2CCN(C[C@H]2F)C2COC2)ncc1C(F)(F)F
50448112CNc1nc(Nc2cnn(C3CCN(CC3)C3COC3)c2C)ncc1C(F)(F)F
50448113CNc1nc(Nc2cnn(C3CCOCC3)c2C)ncc1C(F)(F)F
50448114CNc1nc(Nc2cnn(C3COC3)c2C)ncc1C(F)(F)F
50448115CNc1nc(Nc2cnn(c2Cl)C2(CC2)C#N)ncc1C(F)(F)F
50448116CNc1nc(Nc2cn(nc2C)C2(CC2)C#N)ncc1C(F)(F)F
50448117CNc1nc(Nc2cnn(c2C)C(C)(C)C#N)ncc1C(F)(F)F
50448118CNc1nc(Nc2cn(nc2C)C(C)(C)C#N)ncc1C(F)(F)F
50448119CNc1nc(Nc2cn(nc2C)C(C)(C)C(=O)NCC(F)(F)F)ncc1C(F)(F)F
50448120CNc1nc(Nc2cn(nc2C)C(C)(C)C(=O)NC(C)C)ncc1C(F)(F)F
50448121CCNC(=O)C(C)(C)n1cc(Nc2ncc(c(NC)n2)C(F)(F)F)c(C)n1
50448122CNC(=O)C(C)(C)n1cc(Nc2ncc(c(NC)n2)C(F)(F)F)c(C)n1
50448123CNc1nc(Nc2cnn3CCOC(C)c23)ncc1C(F)(F)F
50448124CNc1nc(Nc2cnn3C[C@H](C)OC(C)c23)ncc1C(F)(F)F
50448125CNc1nc(Nc2cnn3CCOCc23)ncc1C(F)(F)F
50448126CNc1nc(Nc2cnn3CC(C)(C)OCc23)ncc1C(F)(F)F
50448127CCNc1nc(Nc2cc(nn2C)C(C)(C)C#N)ncc1C(F)(F)F